PH26465A - Piperidine compounds and their use - Google Patents

Piperidine compounds and their use Download PDF

Info

Publication number
PH26465A
PH26465A PH40049A PH40049A PH26465A PH 26465 A PH26465 A PH 26465A PH 40049 A PH40049 A PH 40049A PH 40049 A PH40049 A PH 40049A PH 26465 A PH26465 A PH 26465A
Authority
PH
Philippines
Prior art keywords
mmol
thiadiazol
solution
added
pyridine
Prior art date
Application number
PH40049A
Other languages
English (en)
Inventor
Per Sauerberg
Preben Houlberg Olesen
Original Assignee
Ferrosan As
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from DK82589A external-priority patent/DK82589A/da
Priority claimed from DK231589A external-priority patent/DK231589D0/da
Application filed by Ferrosan As filed Critical Ferrosan As
Publication of PH26465A publication Critical patent/PH26465A/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/02—Drugs for disorders of the nervous system for peripheral neuropathies
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A61P27/02—Ophthalmic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A61P27/02—Ophthalmic agents
    • A61P27/06—Antiglaucoma agents or miotics
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Veterinary Medicine (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Ophthalmology & Optometry (AREA)
  • Pain & Pain Management (AREA)
  • Hospice & Palliative Care (AREA)
  • Psychiatry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
PH40049A 1989-02-22 1990-02-14 Piperidine compounds and their use PH26465A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DK82589A DK82589A (da) 1989-02-22 1989-02-22 Piperidinforbindelser, deres fremstilling og anvendelse
DK231589A DK231589D0 (da) 1989-05-12 1989-05-12 Piperidinforbindelser og deres fremstilling og anvendelse

Publications (1)

Publication Number Publication Date
PH26465A true PH26465A (en) 1992-07-27

Family

ID=26064725

Family Applications (1)

Application Number Title Priority Date Filing Date
PH40049A PH26465A (en) 1989-02-22 1990-02-14 Piperidine compounds and their use

Country Status (22)

Country Link
US (5) US5043345A (de)
EP (2) EP0384285A3 (de)
JP (2) JP2921578B2 (de)
KR (1) KR0163763B1 (de)
CN (1) CN1028105C (de)
AR (1) AR247565A1 (de)
AT (1) ATE123030T1 (de)
AU (2) AU629302B2 (de)
CA (2) CA2010578C (de)
DE (1) DE69019550T2 (de)
DK (1) DK0384288T3 (de)
ES (1) ES2072323T3 (de)
FI (2) FI900887A7 (de)
GR (1) GR3017062T3 (de)
HU (2) HU221623B1 (de)
IE (1) IE69672B1 (de)
IL (2) IL93352A (de)
NO (2) NO900831L (de)
NZ (1) NZ232615A (de)
PH (1) PH26465A (de)
PT (2) PT93242A (de)
RU (1) RU2042676C1 (de)

Families Citing this family (93)

* Cited by examiner, † Cited by third party
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US5328925A (en) * 1989-02-22 1994-07-12 Novo Nordisk A/S Piperidine compounds and their use
US5264444A (en) * 1989-02-22 1993-11-23 Novo Nordisk A/S Piperidine compounds and use
US5260311A (en) * 1989-02-22 1993-11-09 Novo Nordisk A/S Piperidine compounds and their use
EP0459568A3 (en) * 1990-05-31 1992-09-30 Merck Sharp & Dohme Ltd. Substituted oxadiazoles and thiadiazoles for use in the treatment of glaucoma and novel compounds having such use
USRE35822E (en) * 1990-08-21 1998-06-09 Novo Nordisk A/S Heterocyclic compounds
DK198590D0 (da) * 1990-08-21 1990-08-21 Novo Nordisk As Heterocykliske forbindelser, deres fremstilling og anvendelse
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US5376668A (en) * 1990-08-21 1994-12-27 Novo Nordisk A/S Heterocyclic compounds
US5418240A (en) * 1990-08-21 1995-05-23 Novo Nordisk A/S Heterocyclic compounds and their preparation and use
US5527813A (en) * 1990-08-21 1996-06-18 Novo Nordisk A/S Heterocyclic compounds and their preparation and use
DK198390D0 (da) * 1990-08-21 1990-08-21 Novo Nordisk As Heterocykliske forbindelser, deres fremstilling og anvendelse
HUT65880A (en) * 1990-11-29 1994-07-28 Allergan Inc Process for preparation of ophtalmological medicaments containing pyridine derivatives usefules for treatment of ocular hypertension
EP0492903A1 (de) * 1990-12-21 1992-07-01 MERCK SHARP & DOHME LTD. Substituierte Pyrazine, Pyrimidine und Pyridazine zur Anwendung in der Behandlung von Glaukoma
IE922270A1 (en) * 1991-07-26 1993-01-27 Akzo Nv Pyrazole derivatives
US5641791A (en) * 1991-08-13 1997-06-24 Novo Nordisk A.S Heterocyclic compounds and their preparation and use
US5175166A (en) * 1991-08-27 1992-12-29 The University Of Toledo Muscarinic agonists
WO1993014089A1 (en) * 1992-01-13 1993-07-22 Novo Nordisk A/S Heterocyclic compounds and their preparation and use
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AU678186B2 (en) * 1992-10-23 1997-05-22 Merck Sharp & Dohme Limited Dopamine receptor subtype ligands
FI955829L (fi) * 1993-06-04 1995-12-04 Novo Nordisk As Heterosyklinen kemia
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IL112024A (en) * 1993-12-21 1999-07-14 Novo Nordisk As Pharmaceutical compositions comprising tetrahydropyridine derivatives substituted with oxadiazole or thiadiazole for treating gastrointestinal motility disorders
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Family Cites Families (15)

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NZ219646A (en) * 1986-03-27 1990-10-26 Merck Sharp & Dohme Oxadiazole derivatives of azacyclics for treating cns disorders
IL83275A (en) * 1986-09-08 1994-02-27 Novo Nordisk As Substituted 1, 2, 4- oxadiazolyl piperidine compounds, their preparation and pharmaceutical compositions containing them
US5017618A (en) * 1987-03-16 1991-05-21 University Of Florida Labile derivatives of ketone analogs of 3-substituted-1-alkylamino-2-propanols and their use as beta-adrenergic blockers
GB8714789D0 (en) * 1987-06-24 1987-07-29 Lundbeck & Co As H Heterocyclic compounds
NZ225999A (en) * 1987-09-10 1992-04-28 Merck Sharp & Dohme Azacyclic- or azabicyclic-substituted thiadiazole derivatives and pharmaceutical compositions
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DK162892C (da) * 1988-07-04 1992-05-11 Novo Nordisk As 1,2,5,6-tetrahydropyridinforbindelser, deres fremstilling og farmaceutiske praeparater indeholdende disse
US5264444A (en) * 1989-02-22 1993-11-23 Novo Nordisk A/S Piperidine compounds and use
US5043345A (en) * 1989-02-22 1991-08-27 Novo Nordisk A/S Piperidine compounds and their preparation and use
US5328925A (en) * 1989-02-22 1994-07-12 Novo Nordisk A/S Piperidine compounds and their use
US5260311A (en) * 1989-02-22 1993-11-09 Novo Nordisk A/S Piperidine compounds and their use
DK198490D0 (da) * 1990-08-21 1990-08-21 Novo Nordisk As Heterocykliske forbindelser, deres fremstilling og anvendelse
DK198390D0 (da) * 1990-08-21 1990-08-21 Novo Nordisk As Heterocykliske forbindelser, deres fremstilling og anvendelse
US5175166A (en) * 1991-08-27 1992-12-29 The University Of Toledo Muscarinic agonists

Also Published As

Publication number Publication date
EP0384288B1 (de) 1995-05-24
CA2010578C (en) 2000-05-23
NO179639B (no) 1996-08-12
US5712297A (en) 1998-01-27
AU4999790A (en) 1990-08-30
CA2010578A1 (en) 1990-08-22
AU4999690A (en) 1990-08-30
NZ232615A (en) 1992-06-25
HU211705A9 (en) 1995-12-28
US5041455A (en) 1991-08-20
NO179639C (no) 1996-11-20
CN1028105C (zh) 1995-04-05
PT93241A (pt) 1990-08-31
AU629302B2 (en) 1992-10-01
EP0384285A3 (de) 1991-04-24
HU221623B1 (hu) 2002-12-28
KR910015569A (ko) 1991-09-30
DE69019550T2 (de) 1995-10-05
EP0384288A2 (de) 1990-08-29
PT93241B (pt) 1996-01-31
RU2042676C1 (ru) 1995-08-27
IL93352A (en) 1994-08-26
CN1045104A (zh) 1990-09-05
DK0384288T3 (da) 1995-10-02
JPH02255679A (ja) 1990-10-16
JPH02255680A (ja) 1990-10-16
US5043345A (en) 1991-08-27
HU900884D0 (en) 1990-05-28
FI900887A7 (fi) 1990-08-23
NO900831D0 (no) 1990-02-21
JP2921578B2 (ja) 1999-07-19
US5559138A (en) 1996-09-24
HUT58326A (en) 1992-02-28
EP0384288A3 (de) 1991-04-10
AR247565A1 (es) 1995-01-31
FI95704B (fi) 1995-11-30
FI900886A0 (fi) 1990-02-22
ATE123030T1 (de) 1995-06-15
FI95704C (fi) 1996-03-11
FI900887A0 (fi) 1990-02-22
CA2010579A1 (en) 1990-08-22
ES2072323T3 (es) 1995-07-16
IE900504L (en) 1990-08-22
NO900830D0 (no) 1990-02-21
PT93242A (pt) 1990-08-31
IE69672B1 (en) 1996-10-02
NO900830L (no) 1990-08-23
EP0384285A2 (de) 1990-08-29
IL93423A0 (en) 1990-11-29
DE69019550D1 (de) 1995-06-29
US5284859A (en) 1994-02-08
KR0163763B1 (ko) 1998-12-01
NO900831L (no) 1990-08-23
IL93352A0 (en) 1990-11-29
GR3017062T3 (en) 1995-11-30

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