PL1989182T3 - Postać krystaliczna soli peryndoprylu z argininą, sposób jej wytwarzania i kompozycje farmaceutyczne ją zawierające - Google Patents

Postać krystaliczna soli peryndoprylu z argininą, sposób jej wytwarzania i kompozycje farmaceutyczne ją zawierające

Info

Publication number: PL1989182T3
Authority: PL; Poland
Prior art keywords: perindopril; preparing; pharmaceutical compositions; crystalline form; arginine salt
Prior art date: 2006-02-28

Application number

PL07731039.9T

Other languages

English (en)

Inventor

Gérard Coquerel

Loïc Lefebvre

Jean-Claude Souvie

Pascale Authouart

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2006-02-28

Filing date

2007-02-26

Publication date

2016-09-30

Family has litigation

First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=37022969&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=PL1989182(T3) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.

2007-02-26 Application filed filed Critical

2016-09-30 Publication of PL1989182T3 publication Critical patent/PL1989182T3/pl

Links

125000000637 arginyl group Chemical class N[C@@H](CCCNC(N)=N)C(=O)* 0.000 title 1
238000004519 manufacturing process Methods 0.000 title 1
IPVQLZZIHOAWMC-QXKUPLGCSA-N perindopril Chemical compound C1CCC[C@H]2C[C@@H](C(O)=O)N(C(=O)[C@H](C)N[C@@H](CCC)C(=O)OCC)[C@H]21 IPVQLZZIHOAWMC-QXKUPLGCSA-N 0.000 title 1
229960002582 perindopril Drugs 0.000 title 1
239000008194 pharmaceutical composition Substances 0.000 title 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
- C07D209/04—Indoles; Hydrogenated indoles
- C07D209/30—Indoles; Hydrogenated indoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to carbon atoms of the hetero ring
- C07D209/42—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
- A61K31/403—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with carbocyclic rings, e.g. carbazole
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/10—Antioedematous agents; Diuretics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/04—Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Life Sciences & Earth Sciences (AREA)
Public Health (AREA)
Medicinal Chemistry (AREA)
Pharmacology & Pharmacy (AREA)
Veterinary Medicine (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Cardiology (AREA)
Heart & Thoracic Surgery (AREA)
Vascular Medicine (AREA)
Urology & Nephrology (AREA)
Diabetes (AREA)
Hematology (AREA)
Hospice & Palliative Care (AREA)
Epidemiology (AREA)
Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Peptides Or Proteins (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Indole Compounds (AREA)
Medicinal Preparation (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

PL07731039.9T 2006-02-28 2007-02-26 Postać krystaliczna soli peryndoprylu z argininą, sposób jej wytwarzania i kompozycje farmaceutyczne ją zawierające PL1989182T3 (pl)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
FR0601748A FR2897866B1 (fr)	2006-02-28	2006-02-28	Forme cristalline alpha du sel d'arginine du perindopril, son procede de preparation, et les compositions pharmaceutiques qui la contiennent

Publications (1)

Publication Number	Publication Date
PL1989182T3 true PL1989182T3 (pl)	2016-09-30

Family

ID=37022969

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
PL07731039.9T PL1989182T3 (pl)	2006-02-28	2007-02-26	Postać krystaliczna soli peryndoprylu z argininą, sposób jej wytwarzania i kompozycje farmaceutyczne ją zawierające

Country Status (27)

Country	Link
US (1)	US7846961B2 (pl)
EP (1)	EP1989182B1 (pl)
JP (1)	JP5255454B2 (pl)
KR (2)	KR20120001818A (pl)
CN (1)	CN101389603B (pl)
AU (1)	AU2007220435B2 (pl)
BR (1)	BRPI0708278B8 (pl)
CA (1)	CA2644467C (pl)
CY (1)	CY1117753T1 (pl)
DK (1)	DK1989182T3 (pl)
EA (1)	EA014716B1 (pl)
ES (1)	ES2581982T3 (pl)
FR (1)	FR2897866B1 (pl)
GE (1)	GEP20125433B (pl)
HR (1)	HRP20160644T1 (pl)
HU (1)	HUE027898T2 (pl)
MA (1)	MA30276B1 (pl)
ME (1)	ME02456B (pl)
MY (1)	MY151035A (pl)
NO (1)	NO20083535L (pl)
NZ (1)	NZ570367A (pl)
PL (1)	PL1989182T3 (pl)
RS (1)	RS54754B1 (pl)
SI (1)	SI1989182T1 (pl)
UA (1)	UA89905C2 (pl)
WO (1)	WO2007099217A1 (pl)
ZA (1)	ZA200807024B (pl)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
DK2318365T3 (en)	2008-06-24	2015-11-23	Mylan Lab Ltd	NOVEL polymorphic forms of perindopril (L) -arginine AND PROCESS FOR PREPARATION THEREOF
AU2009212902A1 (en)	2008-09-03	2010-03-18	Apotex Pharmachem Inc.	Amorphous form of an L-arginine salt of perindopril and processes of preparation thereof
SI23149A (sl)	2009-09-21	2011-03-31	Silverstone Pharma	Nove benzatinske soli ACE inhibitorjev, postopek za njihovo pripravo in njihova uporaba za zdravljenje kardiovaskularnih bolezni
FR2985511B1 (fr) *	2012-01-05	2014-01-03	Servier Lab	Forme cristalline delta du sel d'arginine du perindopril, son procede de preparation, et les compositions pharmaceutiques qui la contiennent
FR2985512B1 (fr) *	2012-01-05	2014-06-20	Servier Lab	Procede de preparation du sel de l-arginine du perindopril
CN103172696B (zh) *	2012-12-19	2014-12-17	宁波美诺华药业股份有限公司	一种γ晶型的培哚普利精氨酸盐的制备方法
PH12018502155B1 (en)	2016-04-20	2024-03-27	Servier Lab	Pharmaceutical composition comprising a beta blocker, a converting enzyme inhibitor and an antihypertensive or an nsaid
EP3842035A1 (en)	2019-12-23	2021-06-30	KRKA, d.d., Novo mesto	Composition for the preparation of perindopril arginine granules, a method for their preparation and pharmaceutical composition comprising the granules
SI26268A (sl)	2021-11-18	2023-05-31	Zupet Rok	Postopek za pripravo hidratirane oblike perindopril l-arginina
CN114149357B (zh) *	2021-12-29	2024-06-25	江苏嘉逸医药有限公司	一种γ晶型培哚普利精氨酸盐的制备方法

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
FR2503155A2 (fr) *	1980-10-02	1982-10-08	Science Union & Cie	Nouveaux imino diacides substitues, leurs procedes de preparation et leur emploi comme inhibiteur d'enzyme
FR2811319B1 (fr) *	2000-07-06	2002-08-23	Adir	Nouvelle forme cristalline beta du sel de tert-butylamine du perindopril, son procede de preparation et les compositions pharmaceutiques qui la contiennent
FR2811318B1 (fr) *	2000-07-06	2002-08-23	Adir	Nouvelle forme cristalline gamma du sel de tert-butylamine du perindopril, son procede de preparation et les compositions pharmaceutiques qui la contiennent
FR2811320B1 (fr) *	2000-07-06	2002-08-23	Adir	Nouvelle forme cristalline alpha du sel de tert-butylamine du perindopril, son procede de preparation et les compositions pharmaceutiques qui la contiennent
FR2838648B1 (fr) *	2002-04-18	2004-05-21	Servier Lab	Nouveau sel de perindopril et les compositions pharmaceutiques qui le contiennent
FR2897865B1 (fr)	2006-02-28	2008-04-18	Servier Lab	Forme cristalline beta du sel d'arginine du perindopril, son procede de preparation, et les compositions pharmaceutiques qui la contiennent
DK2318365T3 (en)	2008-06-24	2015-11-23	Mylan Lab Ltd	NOVEL polymorphic forms of perindopril (L) -arginine AND PROCESS FOR PREPARATION THEREOF

2006
- 2006-02-28 FR FR0601748A patent/FR2897866B1/fr not_active Expired - Lifetime
2007
- 2007-02-26 WO PCT/FR2007/000335 patent/WO2007099217A1/fr not_active Ceased
- 2007-02-26 DK DK07731039.9T patent/DK1989182T3/en active
- 2007-02-26 MY MYPI20082991 patent/MY151035A/en unknown
- 2007-02-26 RS RS20160321A patent/RS54754B1/sr unknown
- 2007-02-26 JP JP2008556812A patent/JP5255454B2/ja active Active
- 2007-02-26 ME MEP-2016-140A patent/ME02456B/me unknown
- 2007-02-26 SI SI200731781A patent/SI1989182T1/sl unknown
- 2007-02-26 GE GEAP200710918A patent/GEP20125433B/en unknown
- 2007-02-26 ZA ZA200807024A patent/ZA200807024B/xx unknown
- 2007-02-26 UA UAA200811436A patent/UA89905C2/ru unknown
- 2007-02-26 CN CN2007800061889A patent/CN101389603B/zh active Active
- 2007-02-26 NZ NZ570367A patent/NZ570367A/en unknown
- 2007-02-26 US US12/224,369 patent/US7846961B2/en active Active
- 2007-02-26 HR HRP20160644TT patent/HRP20160644T1/hr unknown
- 2007-02-26 EA EA200801777A patent/EA014716B1/ru unknown
- 2007-02-26 PL PL07731039.9T patent/PL1989182T3/pl unknown
- 2007-02-26 EP EP07731039.9A patent/EP1989182B1/fr not_active Revoked
- 2007-02-26 BR BRPI0708278A patent/BRPI0708278B8/pt active IP Right Grant
- 2007-02-26 AU AU2007220435A patent/AU2007220435B2/en active Active
- 2007-02-26 HU HUE07731039A patent/HUE027898T2/en unknown
- 2007-02-26 ES ES07731039.9T patent/ES2581982T3/es active Active
- 2007-02-26 KR KR1020117028452A patent/KR20120001818A/ko not_active Ceased
- 2007-02-26 CA CA2644467A patent/CA2644467C/fr not_active Expired - Fee Related
- 2007-02-26 KR KR1020087023638A patent/KR20080106948A/ko not_active Ceased
2008
- 2008-08-14 NO NO20083535A patent/NO20083535L/no not_active Application Discontinuation
- 2008-09-11 MA MA31232A patent/MA30276B1/fr unknown
2016
- 2016-07-11 CY CY20161100654T patent/CY1117753T1/el unknown

Also Published As

Publication number	Publication date
BRPI0708278B1 (pt)	2021-03-02
HRP20160644T1 (hr)	2016-07-01
BRPI0708278A2 (pt)	2011-05-24
CA2644467C (fr)	2011-07-26
SI1989182T1 (sl)	2016-07-29
NZ570367A (en)	2011-03-31
GEP20125433B (en)	2012-03-26
ZA200807024B (en)	2010-04-28
CY1117753T1 (el)	2017-05-17
HUE027898T2 (en)	2016-10-28
KR20120001818A (ko)	2012-01-04
MA30276B1 (fr)	2009-03-02
CA2644467A1 (fr)	2007-09-07
EA200801777A1 (ru)	2009-02-27
KR20080106948A (ko)	2008-12-09
UA89905C2 (ru)	2010-03-10
MY151035A (en)	2014-03-31
RS54754B1 (sr)	2016-10-31
EP1989182A1 (fr)	2008-11-12
CN101389603A (zh)	2009-03-18
BRPI0708278B8 (pt)	2021-05-25
DK1989182T3 (en)	2016-07-25
JP5255454B2 (ja)	2013-08-07
US20090203758A1 (en)	2009-08-13
EA014716B1 (ru)	2011-02-28
EP1989182B1 (fr)	2016-04-13
ME02456B (me)	2017-02-20
HK1129669A1 (en)	2009-12-04
AU2007220435A1 (en)	2007-09-07
NO20083535L (no)	2008-08-14
FR2897866A1 (fr)	2007-08-31
FR2897866B1 (fr)	2008-04-18
JP2009534295A (ja)	2009-09-24
CN101389603B (zh)	2012-07-04
US7846961B2 (en)	2010-12-07
ES2581982T3 (es)	2016-09-08
AU2007220435B2 (en)	2010-11-04
WO2007099217A1 (fr)	2007-09-07

Publication	Publication Date	Title
SI1989182T1 (sl)	2016-07-29	Kristalinična oblika argininske soli perindoprila, postopek za njeno pripravo in farmacevtski sestavki, ki jo vsebujejo
SI1752443T1 (sl)	2012-10-30	Nova kristalinična oblika V agomelatina, postopek za njeno pripravo in farmacevtski sestavki, ki jo vsebujejo
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PL2210872T3 (pl)	2017-07-31	Nowa postać krystaliczna III agomelatyny, sposób jej wytwarzania i kompozycje farmaceutyczne ją zawierające
IL218539A (en)	2015-09-24	Annotated 4,1-Androsteadian-3-Oxo-9,6-Dihlo-16-Isoxazolidine-17-Noble N-Converted
IL188069A0 (en)	2008-03-20	Process for preparing new tiotropium salts, new tiotropium salts as such and pharmaceutical compositions thereof
HUP0600809A2 (en)	2008-08-28	New phenylsulfamoyl-benzamide derivatives as bradykinin antagonists, process and intermediates for their preparation and pharmaceutical compositions containing them
SI2231598T1 (sl)	2011-11-30	Novi derivati diazeniumdiolata postopek pripravele teh in njihovi farmacevtski sestavki
IL205082A0 (en)	2010-11-30	Process for the preparation of tetranorlabdane derivatives
HUP0600808A3 (en)	2008-09-29	New benzamide derivatives as bradykinin antagonists, process for their preparation and pharmaceutical compositions containing them
HUP0600293A2 (en)	2007-12-28	Zinc salt of rosuvastatine, process for its preparation and pharmaceutical compositions containing it
PL2612850T3 (pl)	2014-01-31	Postać krystaliczna delta soli argininy peryndoprylu, sposób jej wytwarzania oraz kompozycje farmaceutyczne, które ją zawierają
ZA200902414B (en)	2010-07-28	Indole derivatives, process for the preparation thereof and pharmaceutical compositions containing them
SI1707564T1 (sl)	2007-12-31	Indanil-piperazinski derivati, postopek za njihovo pripravo in farmacevtski sestavki, ki jih vsebujejo
PL1979321T3 (pl)	2009-10-30	Nowe pirydynyloaminoalkileno- i pirydynyloksyalkileno- cyklopropanoaminy, sposób ich wytwarzania i zawierające je kompozycje farmaceutyczne
ZA200902413B (en)	2010-07-28	Novel indole derivatives, process for the preparation thereof and pharmaceutical compositions containing them
PL1753720T3 (pl)	2014-09-30	Proces wytwarzania peryndoprylu i jego soli
IL192963A0 (en)	2009-02-11	Rimonabant monohydrate, process for the preparation thereof and pharmaceutical compositions containing same
WO2009000909A3 (en)	2010-03-18	Salts of perindopril