PL2326621T3 - Podstawione pochodne kwasu1,2,3,4-tetrahydrocyklopenta[b]indol- 3-ilo)octowego użyteczne w leczeniu zaburzeń autoimmunologicznych i zapalnych - Google Patents

Podstawione pochodne kwasu1,2,3,4-tetrahydrocyklopenta[b]indol- 3-ilo)octowego użyteczne w leczeniu zaburzeń autoimmunologicznych i zapalnych

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Publication number
PL2326621T3
PL2326621T3 PL09788983.6T PL09788983T PL2326621T3 PL 2326621 T3 PL2326621 T3 PL 2326621T3 PL 09788983 T PL09788983 T PL 09788983T PL 2326621 T3 PL2326621 T3 PL 2326621T3
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PL
Poland
Prior art keywords
tetrahydrocyclopenta
indol
autoimmune
substituted
treatment
Prior art date
Application number
PL09788983.6T
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English (en)
Inventor
Robert M. Jones
Daniel J. Buzard
Sangdon Han
Sun Hee Kim
Juerg Lehmann
Brett Ullman
Jeanne V. Moody
Xiuwen Zhu
Scott Stirn
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Publication of PL2326621T3 publication Critical patent/PL2326621T3/pl

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    • C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/56—Ring systems containing three or more rings
    • C07D209/80—[b, c]- or [b, d]-condensed
    • C07D209/94—[b, c]- or [b, d]-condensed containing carbocyclic rings other than six-membered
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    • A61K31/13—Amines
    • A61K31/135—Amines having aromatic rings, e.g. ketamine, nortriptyline
    • A61K31/137—Arylalkylamines, e.g. amphetamine, epinephrine, salbutamol, ephedrine or methadone
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    • A61K31/19—Carboxylic acids, e.g. valproic acid
    • A61K31/195—Carboxylic acids, e.g. valproic acid having an amino group
    • A61K31/197—Carboxylic acids, e.g. valproic acid having an amino group the amino and the carboxyl groups being attached to the same acyclic carbon chain, e.g. gamma-aminobutyric acid [GABA], beta-alanine, epsilon-aminocaproic acid or pantothenic acid
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    • A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A61K31/403—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with carbocyclic rings, e.g. carbazole
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PL09788983.6T 2008-07-23 2009-07-22 Podstawione pochodne kwasu1,2,3,4-tetrahydrocyklopenta[b]indol- 3-ilo)octowego użyteczne w leczeniu zaburzeń autoimmunologicznych i zapalnych PL2326621T3 (pl)

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US13567208P 2008-07-23 2008-07-23
US20937409P 2009-03-06 2009-03-06

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PL2326621T3 true PL2326621T3 (pl) 2016-12-30

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EP (1) EP2326621B1 (pl)
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