PL2683708T3 - Postacie stałe 3-(5-amino-2-metylo-4-okso-4h-chinazolin-3-ylo)-piperydyno-2,6-dionu oraz ich kompozycje farmaceutyczne i zastosowania - Google Patents

Postacie stałe 3-(5-amino-2-metylo-4-okso-4h-chinazolin-3-ylo)-piperydyno-2,6-dionu oraz ich kompozycje farmaceutyczne i zastosowania

Info

Publication number
PL2683708T3
PL2683708T3 PL12710834T PL12710834T PL2683708T3 PL 2683708 T3 PL2683708 T3 PL 2683708T3 PL 12710834 T PL12710834 T PL 12710834T PL 12710834 T PL12710834 T PL 12710834T PL 2683708 T3 PL2683708 T3 PL 2683708T3
Authority
PL
Poland
Prior art keywords
quinazolin
dione
piperidine
oxo
amino
Prior art date
Application number
PL12710834T
Other languages
English (en)
Inventor
George W. Muller
Hon-Wah Man
Benjamin M. Cohen
Ying Li
Jean Xu
William W. Leong
Original Assignee
Celgene Corporation
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=45888486&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=PL2683708(T3) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Celgene Corporation filed Critical Celgene Corporation
Publication of PL2683708T3 publication Critical patent/PL2683708T3/pl

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/517—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with carbocyclic ring systems, e.g. quinazoline, perimidine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B2200/00—Indexing scheme relating to specific properties of organic compounds
    • C07B2200/13—Crystalline forms, e.g. polymorphs

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Medicinal Preparation (AREA)
PL12710834T 2011-03-11 2012-03-09 Postacie stałe 3-(5-amino-2-metylo-4-okso-4h-chinazolin-3-ylo)-piperydyno-2,6-dionu oraz ich kompozycje farmaceutyczne i zastosowania PL2683708T3 (pl)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201161451806P 2011-03-11 2011-03-11
EP12710834.8A EP2683708B1 (en) 2011-03-11 2012-03-09 Solid forms of 3-(5-amino-2-methyl-4-oxo-4h-quinazolin-3-yl)-piperidine-2,6-dione, and their pharmaceutical compositions and uses
PCT/US2012/028419 WO2012125438A1 (en) 2011-03-11 2012-03-09 Solid forms of 3-(5-amino-2methyl-4-oxo-4h-quinazolin-3-yl)-piperidine-2,6-dione, and their pharmaceutical compositions and uses

Publications (1)

Publication Number Publication Date
PL2683708T3 true PL2683708T3 (pl) 2018-03-30

Family

ID=45888486

Family Applications (1)

Application Number Title Priority Date Filing Date
PL12710834T PL2683708T3 (pl) 2011-03-11 2012-03-09 Postacie stałe 3-(5-amino-2-metylo-4-okso-4h-chinazolin-3-ylo)-piperydyno-2,6-dionu oraz ich kompozycje farmaceutyczne i zastosowania

Country Status (36)

Country Link
US (5) US8802685B2 (pl)
EP (2) EP2683708B1 (pl)
JP (1) JP5959543B2 (pl)
KR (1) KR20140014221A (pl)
CN (2) CN106083812A (pl)
AR (1) AR085650A1 (pl)
AU (2) AU2012229279B2 (pl)
BR (1) BR112013023279A2 (pl)
CA (3) CA2829570C (pl)
CL (1) CL2013002593A1 (pl)
CO (1) CO6821939A2 (pl)
CR (2) CR20130458A (pl)
CY (1) CY1119974T1 (pl)
DK (1) DK2683708T3 (pl)
EA (1) EA026100B1 (pl)
EC (1) ECSP13012877A (pl)
ES (1) ES2656855T3 (pl)
HR (1) HRP20180133T1 (pl)
HU (1) HUE037955T2 (pl)
LT (1) LT2683708T (pl)
MX (1) MX2013010360A (pl)
NI (1) NI201300080A (pl)
NO (1) NO2683708T3 (pl)
PE (1) PE20140983A1 (pl)
PH (1) PH12013501821A1 (pl)
PL (1) PL2683708T3 (pl)
PT (1) PT2683708T (pl)
RS (1) RS56770B1 (pl)
RU (1) RU2611007C2 (pl)
SG (1) SG192946A1 (pl)
SI (1) SI2683708T1 (pl)
SM (1) SMT201800032T1 (pl)
TW (2) TWI540127B (pl)
UA (1) UA113512C2 (pl)
WO (1) WO2012125438A1 (pl)
ZA (1) ZA201306234B (pl)

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WO2017205622A1 (en) * 2016-05-25 2017-11-30 Savant Neglected Diseases, Llc Method of making benznidazole
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RU2695326C1 (ru) * 2018-06-05 2019-07-23 Федеральное государственное бюджетное научное учреждение "Научно-исследовательский институт биомедицинской химии имени В.Н. Ореховича" (ИБМХ) Противоопухолевое средство для лечения рака предстательной железы в форме саше
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