PL358481A1 - Pochodne 6-hydroksy-indazolu do leczenia jaskry - Google Patents

Pochodne 6-hydroksy-indazolu do leczenia jaskry

Info

Publication number
PL358481A1
PL358481A1 PL00358481A PL35848100A PL358481A1 PL 358481 A1 PL358481 A1 PL 358481A1 PL 00358481 A PL00358481 A PL 00358481A PL 35848100 A PL35848100 A PL 35848100A PL 358481 A1 PL358481 A1 PL 358481A1
Authority
PL
Poland
Prior art keywords
hydroxy
treating glaucoma
indazole derivatives
indazole
derivatives
Prior art date
Application number
PL00358481A
Other languages
English (en)
Inventor
Jesse A. May
Anura P. Dantanarayana
Zixia Feng
Original Assignee
Alcon Inc.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Alcon Inc. filed Critical Alcon Inc.
Publication of PL358481A1 publication Critical patent/PL358481A1/pl

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D231/00Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/54Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings condensed with carbocyclic rings or ring systems
    • C07D231/56Benzopyrazoles; Hydrogenated benzopyrazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00Drugs for disorders of the senses
    • A61P27/02Ophthalmic agents
    • A61P27/06Antiglaucoma agents or miotics

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Ophthalmology & Optometry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
PL00358481A 2000-03-17 2000-11-14 Pochodne 6-hydroksy-indazolu do leczenia jaskry PL358481A1 (pl)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US19038000P 2000-03-17 2000-03-17

Publications (1)

Publication Number Publication Date
PL358481A1 true PL358481A1 (pl) 2004-08-09

Family

ID=22701093

Family Applications (1)

Application Number Title Priority Date Filing Date
PL00358481A PL358481A1 (pl) 2000-03-17 2000-11-14 Pochodne 6-hydroksy-indazolu do leczenia jaskry

Country Status (14)

Country Link
EP (1) EP1268438A1 (pl)
JP (1) JP2003528085A (pl)
KR (1) KR20030065304A (pl)
CN (1) CN1450994A (pl)
AR (1) AR032138A1 (pl)
AU (1) AU2001216072A1 (pl)
BR (1) BR0017157A (pl)
CA (1) CA2402403A1 (pl)
GC (1) GC0000155A (pl)
MX (1) MXPA02008547A (pl)
PL (1) PL358481A1 (pl)
TW (1) TWI221839B (pl)
WO (1) WO2001070702A1 (pl)
ZA (1) ZA200206851B (pl)

Families Citing this family (20)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6960579B1 (en) 1998-05-19 2005-11-01 Alcon Manufacturing, Ltd. Serotonergic 5HT7 receptor compounds for treating ocular and CNS disorders
TW593302B (en) 2001-12-20 2004-06-21 Alcon Inc Novel benzodifuranimidazoline and benzofuranimidazoline derivatives and their use for the treatment of glaucoma
AU2002360819A1 (en) * 2001-12-28 2003-07-24 Bayer Corporation Cyclohexano- and cycloheptapyrazole derivative compounds, for use in diseases associated with the 5-ht2c receptor
US7196082B2 (en) 2002-11-08 2007-03-27 Merck & Co. Inc. Ophthalmic compositions for treating ocular hypertension
CA2505127A1 (en) 2002-11-08 2004-05-27 James B. Doherty Ophthalmic compositions for treating ocular hypertension
CN100384827C (zh) * 2002-11-08 2008-04-30 默克公司 用于治疗高眼压症的眼用组合物
US7053085B2 (en) 2003-03-26 2006-05-30 Merck & Co. Inc. EP4 receptor agonist, compositions and methods thereof
CA2506204A1 (en) 2002-12-13 2004-07-01 Alcon, Inc. Novel benzopyran analogs and their use for the treatment of glaucoma
JP2004262812A (ja) * 2003-02-28 2004-09-24 Rohto Pharmaceut Co Ltd 眼圧低下剤
CN1845914A (zh) 2003-09-02 2006-10-11 默克公司 用于治疗眼压过高的眼用组合物
KR20060090801A (ko) 2003-09-04 2006-08-16 머크 앤드 캄파니 인코포레이티드 고안압증 치료용 안용 조성물
WO2005025568A1 (en) 2003-09-04 2005-03-24 Merck & Co., Inc. Ophthalmic compositions for treating ocular hypertension
US7129257B1 (en) 2003-12-15 2006-10-31 Alcon, Inc. Pyrazolo[3,4- e]benzoxazoles for the treatment of glaucoma
WO2005058911A2 (en) 2003-12-15 2005-06-30 Alcon, Inc. Substituted [1,4]oxazino[2,3-g]indazoles for the treatment of glaucoma
US7338972B1 (en) 2003-12-15 2008-03-04 Alcon, Inc. Substituted 1-alkylamino-1H-indazoles for the treatment of glaucoma
CN1988903A (zh) 2004-07-20 2007-06-27 默克公司 用于治疗高眼压症的眼用组合物
KR20070094747A (ko) 2004-11-29 2007-09-21 워너-램버트 캄파니 엘엘씨 치료용 피라졸로[3,4-b]피리딘 및 인다졸
WO2006062839A1 (en) 2004-12-08 2006-06-15 Alcon, Inc. Use of dioxindoindazoles and dioxoloindazoles for treating glaucoma
CN101704785B (zh) * 2009-11-16 2012-02-29 东南大学 有机二羧酸和其盐及其制备方法
CN105884687B (zh) * 2016-04-14 2018-06-22 梯尔希(南京)药物研发有限公司 一种5-苄基苄达明的制备方法

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2002515408A (ja) * 1998-05-19 2002-05-28 アルコン ラボラトリーズ, インコーポレーテッド 眼および中枢神経系疾患治療用セロトニン作動性5ht7受容体化合物
ATE247963T1 (de) * 1998-05-26 2003-09-15 Pfizer Prod Inc Medikament zur behandlung von glaukoma und ischämischer retinopathie
GB9819032D0 (en) * 1998-09-01 1998-10-28 Cerebrus Ltd Chemical compounds IV
ATE310566T1 (de) * 1998-09-18 2005-12-15 Alcon Mfg Ltd 5ht2-agoniste zur behandlung des glaukoms
GB9820767D0 (en) * 1998-09-23 1998-11-18 Cerebrus Ltd Chemical compounds VIII

Also Published As

Publication number Publication date
CA2402403A1 (en) 2001-09-27
CN1450994A (zh) 2003-10-22
GC0000155A (en) 2005-06-29
AU2001216072A1 (en) 2001-10-03
ZA200206851B (en) 2003-10-21
WO2001070702A1 (en) 2001-09-27
BR0017157A (pt) 2002-11-26
EP1268438A1 (en) 2003-01-02
KR20030065304A (ko) 2003-08-06
MXPA02008547A (es) 2003-03-12
AR032138A1 (es) 2003-10-29
JP2003528085A (ja) 2003-09-24
TWI221839B (en) 2004-10-11

Similar Documents

Publication Publication Date Title
AU2001219185A1 (en) 2-acylaminobenzimidazole derivatives for treating glaucoma
EG22695A (en) Novel phenyl-propargylether derivatives
HUP0201111A3 (en) Shunt device for treating glaucoma
AU6053701A (en) 2-aminocarbonyl-9h-purine derivatives
HRP20030055A2 (en) 4-phenyl-pyridine derivatives
IL150841A0 (en) 1h-imidazopyridine derivatives
EP1414464A4 (en) METHOD OF TREATING GLAUCOMA
PL358481A1 (pl) Pochodne 6-hydroksy-indazolu do leczenia jaskry
AU2042301A (en) 1-aminoalkyl-1H-indoles for treating glaucoma
AU1397802A (en) Substituted c-cyclohexylmethylamine derivatives
AU2001237939A1 (en) Methods for treating glaucoma
AU1918001A (en) 5-hydroxy indazole derivatives for treating glaucoma
AU4498201A (en) Quinolinyl-piperidin-4-ylidene-methyl-benzamide derivatives for the treatment ofpain
PL356565A1 (pl) Pochodne aminosulfonylobifenylu
HUP0300562A3 (en) Hydroxyphenyl-piperazinyl-methyl-benzamide derivatives for the
IL150557A0 (en) Substituted aminomethyl-phenyl-cyclohexane derivatives
AU2002241670A1 (en) Method for treating glaucoma IB
PL361632A1 (pl) Podstawione pochodne 1-aminobutan-3-olu
AU1603401A (en) Pyranoindoles for treating glaucoma
IL150558A0 (en) Aminomethyl-phenyl-cyclohexanone derivatives
AU2163202A (en) 5-amino-1-pentene-3-ol substituted derivatives
IL151598A0 (en) 2-phenylpyran-4-one derivatives
HK1050196A (en) 6-hydroxy-indazole derivatives for treating glaucoma
HK1051979A (en) Methods for treating glaucoma
GB0019872D0 (en) Glaucoma treatment

Legal Events

Date Code Title Description
REFS Decisions on refusal to grant patents (taken after the publication of the particulars of the applications)