PL365009A1 - Sposób wytwarzania 9-aminopodstawionych 9,10-dihydropirolo-[2,1-b] [1,3] benzotiazepin - Google Patents

Sposób wytwarzania 9-aminopodstawionych 9,10-dihydropirolo-[2,1-b] [1,3] benzotiazepin

Info

Publication number: PL365009A1
Authority: PL; Poland
Prior art keywords: preparation; sub; benzotiazepines; dihydropyrrolo; amino substituted
Prior art date: 2000-08-01

Application number

PL01365009A

Other languages

English (en)

Other versions

PL202400B1 (pl

Inventor

Patrizia Minetti

Domenico Mastroianni

Original Assignee

Sigma-Tau Industrie Farmaceutiche Riunite S.P.A.

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2000-08-01

Filing date

2001-07-20

Publication date

2004-12-27

2001-07-20 Application filed by Sigma-Tau Industrie Farmaceutiche Riunite S.P.A. filed Critical Sigma-Tau Industrie Farmaceutiche Riunite S.P.A.

2004-12-27 Publication of PL365009A1 publication Critical patent/PL365009A1/pl

2009-06-30 Publication of PL202400B1 publication Critical patent/PL202400B1/pl

Links

238000000034 method Methods 0.000 title abstract 3
150000001412 amines Chemical class 0.000 abstract 2
150000001875 compounds Chemical class 0.000 abstract 2
150000002081 enamines Chemical class 0.000 abstract 1
QLZNAQUHVSHPNB-UHFFFAOYSA-N pyrrolo[2,3-i][1,2]benzothiazepin-9-one Chemical compound C1=CC=NSC2=C1C=CC1=NC(=O)C=C21 QLZNAQUHVSHPNB-UHFFFAOYSA-N 0.000 abstract 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
- C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D495/04—Ortho-condensed systems
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
- C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
- C07D513/04—Ortho-condensed systems
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia

Landscapes

Organic Chemistry (AREA)
Chemical & Material Sciences (AREA)
Health & Medical Sciences (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Neurosurgery (AREA)
General Health & Medical Sciences (AREA)
Biomedical Technology (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Veterinary Medicine (AREA)
Pharmacology & Pharmacy (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
Neurology (AREA)
Public Health (AREA)
Psychiatry (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)
Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
Macromolecular Compounds Obtained By Forming Nitrogen-Containing Linkages In General (AREA)
Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)

PL365009A 2000-08-01 2001-07-20 Sposób wytwarzania 9-aminopodstawionych 9,10-dihydropirolo-[2,1-b] [1,3] benzotiazepin PL202400B1 (pl)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
IT2000RM000434A IT1317886B1 (it)	2000-08-01	2000-08-01	Procedimento per la preparazione di 9,10-diidro-pirrolo (2,1-b)(1,3)benzotiazepine 9-ammino sostituite.
PCT/IT2001/000391 WO2002010174A1 (en)	2000-08-01	2001-07-20	Process for the preparation of 9-amino substituted 9,10-dihydropyrrolo [2,1-b][1,3]benzotiazepines

Publications (2)

Publication Number	Publication Date
PL365009A1 true PL365009A1 (pl)	2004-12-27
PL202400B1 PL202400B1 (pl)	2009-06-30

Family

ID=11454867

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
PL365009A PL202400B1 (pl)	2000-08-01	2001-07-20	Sposób wytwarzania 9-aminopodstawionych 9,10-dihydropirolo-[2,1-b] [1,3] benzotiazepin

Country Status (22)

Country	Link
US (1)	US7078521B2 (pl)
EP (1)	EP1305318B1 (pl)
JP (1)	JP2004505089A (pl)
KR (1)	KR100801269B1 (pl)
CN (1)	CN100354281C (pl)
AT (1)	ATE261977T1 (pl)
AU (2)	AU7768701A (pl)
BR (1)	BR0112974A (pl)
CA (1)	CA2415050C (pl)
CZ (1)	CZ294502B6 (pl)
DE (1)	DE60102385T2 (pl)
DK (1)	DK1305318T3 (pl)
ES (1)	ES2215922T3 (pl)
HU (2)	HUP0301648A3 (pl)
IT (1)	IT1317886B1 (pl)
MX (1)	MXPA03000917A (pl)
PL (1)	PL202400B1 (pl)
PT (1)	PT1305318E (pl)
SI (1)	SI1305318T1 (pl)
SK (1)	SK287190B6 (pl)
TR (1)	TR200400821T4 (pl)
WO (1)	WO2002010174A1 (pl)

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
IT1301965B1 (it) *	1998-07-28	2000-07-20	Sigma Tau Ind Farmaceuti	Pirrolo (2,1-b)(1,3) benzotiazepine con attivita' antipsicoticaatipica.

2000
- 2000-08-01 IT IT2000RM000434A patent/IT1317886B1/it active
2001
- 2001-07-20 PT PT01955529T patent/PT1305318E/pt unknown
- 2001-07-20 WO PCT/IT2001/000391 patent/WO2002010174A1/en not_active Ceased
- 2001-07-20 HU HU0301648A patent/HUP0301648A3/hu unknown
- 2001-07-20 AU AU7768701A patent/AU7768701A/xx active Pending
- 2001-07-20 DE DE60102385T patent/DE60102385T2/de not_active Expired - Lifetime
- 2001-07-20 PL PL365009A patent/PL202400B1/pl not_active IP Right Cessation
- 2001-07-20 AU AU2001277687A patent/AU2001277687B2/en not_active Ceased
- 2001-07-20 EP EP01955529A patent/EP1305318B1/en not_active Expired - Lifetime
- 2001-07-20 JP JP2002515903A patent/JP2004505089A/ja not_active Withdrawn
- 2001-07-20 SI SI200130086T patent/SI1305318T1/xx unknown
- 2001-07-20 DK DK01955529T patent/DK1305318T3/da active
- 2001-07-20 US US10/343,629 patent/US7078521B2/en not_active Expired - Fee Related
- 2001-07-20 TR TR2004/00821T patent/TR200400821T4/xx unknown
- 2001-07-20 BR BR0112974-0A patent/BR0112974A/pt not_active Application Discontinuation
- 2001-07-20 HU HU0301647A patent/HUP0301647A3/hu unknown
- 2001-07-20 CN CNB018131433A patent/CN100354281C/zh not_active Expired - Fee Related
- 2001-07-20 CZ CZ200311A patent/CZ294502B6/cs not_active IP Right Cessation
- 2001-07-20 SK SK126-2003A patent/SK287190B6/sk not_active IP Right Cessation
- 2001-07-20 ES ES01955529T patent/ES2215922T3/es not_active Expired - Lifetime
- 2001-07-20 CA CA002415050A patent/CA2415050C/en not_active Expired - Fee Related
- 2001-07-20 MX MXPA03000917A patent/MXPA03000917A/es active IP Right Grant
- 2001-07-20 AT AT01955529T patent/ATE261977T1/de not_active IP Right Cessation
- 2001-07-20 KR KR1020037000134A patent/KR100801269B1/ko not_active Expired - Fee Related

Also Published As

Publication number	Publication date
EP1305318A1 (en)	2003-05-02
SI1305318T1 (en)	2004-08-31
MXPA03000917A (es)	2003-09-05
CN1443188A (zh)	2003-09-17
ES2215922T3 (es)	2004-10-16
HUP0301647A2 (hu)	2003-11-28
JP2004505089A (ja)	2004-02-19
DK1305318T3 (da)	2004-07-26
SK1262003A3 (en)	2004-03-02
ITRM20000434A0 (it)	2000-08-01
DE60102385D1 (de)	2004-04-22
WO2002010174A1 (en)	2002-02-07
PL202400B1 (pl)	2009-06-30
PT1305318E (pt)	2004-08-31
ITRM20000434A1 (it)	2002-02-01
HUP0301648A2 (hu)	2003-08-28
IT1317886B1 (it)	2003-07-15
TR200400821T4 (tr)	2004-07-21
CZ200311A3 (cs)	2003-05-14
SK287190B6 (sk)	2010-02-08
CA2415050C (en)	2009-10-27
CA2415050A1 (en)	2002-02-07
AU2001277687B2 (en)	2006-10-05
HK1059775A1 (en)	2004-07-16
CZ294502B6 (cs)	2005-01-12
US7078521B2 (en)	2006-07-18
CN100354281C (zh)	2007-12-12
KR20030013525A (ko)	2003-02-14
BR0112974A (pt)	2003-07-08
HUP0301647A3 (en)	2009-08-28
HUP0301648A3 (en)	2004-06-28
US20030181437A1 (en)	2003-09-25
EP1305318B1 (en)	2004-03-17
DE60102385T2 (de)	2005-02-17
KR100801269B1 (ko)	2008-02-04
AU7768701A (en)	2002-02-13
ATE261977T1 (de)	2004-04-15

Legal Events

Date	Code	Title	Description
2012-09-28	LAPS	Decisions on the lapse of the protection rights	Effective date: 20110720

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EP1092720A3 (en)	2001-09-19	Process for the preparation of pyrazolo [4,3-d] pyrimidin-7-ones-3-pyridylsulphonyl compounds and intermediates thereof
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MXPA03008727A (es)	2004-07-30	Procedimiento para la preparacion de derivados de imidazol tetrasubstituidos y estructuras cristalinas novedosas de los mismos.