PT93324A - Processo para a preparacao de fosfatos de {3-alcano-sulfinil- e sulfonil-2-meto-ximetil-propil}-(2-tirmetilamonio-etilo) cujo grupo alcano possui 16 a 18 atomos de carbono, e de composicoes farmaceuticas que os contem - Google Patents
Processo para a preparacao de fosfatos de {3-alcano-sulfinil- e sulfonil-2-meto-ximetil-propil}-(2-tirmetilamonio-etilo) cujo grupo alcano possui 16 a 18 atomos de carbono, e de composicoes farmaceuticas que os contemInfo
- Publication number
- PT93324A PT93324A PT93324A PT9332490A PT93324A PT 93324 A PT93324 A PT 93324A PT 93324 A PT93324 A PT 93324A PT 9332490 A PT9332490 A PT 9332490A PT 93324 A PT93324 A PT 93324A
- Authority
- PT
- Portugal
- Prior art keywords
- alcano
- phosphates
- tyethymmethylamyl
- contem
- sulfinyl
- Prior art date
Links
- OKTJSMMVPCPJKN-UHFFFAOYSA-N Carbon Chemical compound [C] OKTJSMMVPCPJKN-UHFFFAOYSA-N 0.000 title 1
- 229910019142 PO4 Inorganic materials 0.000 title 1
- 229910052799 carbon Inorganic materials 0.000 title 1
- 239000008194 pharmaceutical composition Substances 0.000 title 1
- NBIIXXVUZAFLBC-UHFFFAOYSA-K phosphate Chemical compound [O-]P([O-])([O-])=O NBIIXXVUZAFLBC-UHFFFAOYSA-K 0.000 title 1
- 230000000259 anti-tumor effect Effects 0.000 abstract 1
- 150000001875 compounds Chemical class 0.000 abstract 1
- 239000003814 drug Substances 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
- -1 sulphonyl-2-methoxymethylpropyl (2-trimethylammonioethyl)phosphates Chemical class 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
- C07F9/02—Phosphorus compounds
- C07F9/06—Phosphorus compounds without P—C bonds
- C07F9/08—Esters of oxyacids of phosphorus
- C07F9/09—Esters of phosphoric acids
- C07F9/10—Phosphatides, e.g. lecithin
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Biochemistry (AREA)
- Molecular Biology (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Steroid Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE3906952A DE3906952A1 (de) | 1989-03-04 | 1989-03-04 | (3-(c(pfeil abwaerts)1(pfeil abwaerts)(pfeil abwaerts)6(pfeil abwaerts)-c(pfeil abwaerts)1(pfeil abwaerts)(pfeil abwaerts)8(pfeil abwaerts))alkansulfinyl- und sulfonyl-2-methoxymethyl-propyl)-(2-trimethylammonio-ethyl) phosphate, verfahren zu deren herstellung diese verbindungen enthaltende arzneimittel |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| PT93324A true PT93324A (pt) | 1990-11-07 |
| PT93324B PT93324B (pt) | 1996-02-29 |
Family
ID=6375519
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| PT93324A PT93324B (pt) | 1989-03-04 | 1990-03-02 | Processo para a preparacao de fosfatos de {3-alcano-sulfinil- e sulfonil-2-meto-ximetil-propil}-(2-tirmetilamonio-etilo) cujo grupo alcano possui 16 a 18 atomos de carbono, e de composicoes farmaceuticas que os contem |
Country Status (19)
| Country | Link |
|---|---|
| US (1) | US5543402A (pt) |
| EP (1) | EP0395849B1 (pt) |
| JP (1) | JPH0341027A (pt) |
| KR (1) | KR900014412A (pt) |
| AT (1) | ATE121409T1 (pt) |
| AU (1) | AU633304B2 (pt) |
| CA (1) | CA2011209A1 (pt) |
| DD (1) | DD292259A5 (pt) |
| DE (2) | DE3906952A1 (pt) |
| FI (1) | FI93122C (pt) |
| HU (1) | HU204057B (pt) |
| IE (1) | IE900743L (pt) |
| IL (1) | IL93598A (pt) |
| MX (1) | MX19722A (pt) |
| NO (1) | NO901008L (pt) |
| NZ (1) | NZ232692A (pt) |
| PT (1) | PT93324B (pt) |
| RU (1) | RU2035466C1 (pt) |
| ZA (1) | ZA901601B (pt) |
Families Citing this family (18)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE3929217A1 (de) * | 1989-09-02 | 1991-03-07 | Boehringer Mannheim Gmbh | Verwendung von phospholipid-derivaten als antivirale arzneimittel und neue phospholipide |
| GB8928580D0 (en) * | 1989-12-19 | 1990-02-21 | Scras | 3-(n-methyl-n-alkylamino)-methoxymethyl-propanol phosphocholine derivatives |
| US6172050B1 (en) | 1992-07-11 | 2001-01-09 | Asta Medica Aktiengesellschaft | Phospholipid derivatives |
| DE4222910A1 (de) * | 1992-07-11 | 1994-01-13 | Asta Medica Ag | Neue Phospholipidderivate |
| WO1994002153A1 (en) * | 1992-07-22 | 1994-02-03 | Boehringer Mannheim Gmbh | Use of sulphur containing phospholipids for treating leishmaniasis |
| JP5048201B2 (ja) | 2000-08-04 | 2012-10-17 | ディーエムアイ バイオサイエンシズ インコーポレイテッド | ジケトピペラジン類の使用方法とジケトピペラジン類を含む組成物 |
| KR100469556B1 (ko) * | 2001-11-17 | 2005-02-02 | 주식회사 건축사사무소다인그룹 | 도어 잠금장치 |
| EP1448579A1 (de) * | 2001-11-21 | 2004-08-25 | Heidelberg Pharma Holding GmbH | Phospholipid-derivate von nucleosiden als antitumorale arzneimittel |
| DK1571970T3 (da) * | 2002-10-02 | 2011-11-28 | Dmi Biosciences Inc | Diagnose og monitorering af sygdomme |
| CN102210852B (zh) | 2003-05-15 | 2016-10-19 | 安皮奥制药股份有限公司 | T-细胞介导的疾病的治疗 |
| JP5856843B2 (ja) * | 2008-05-27 | 2016-02-10 | アンピオ ファーマシューティカルズ,インコーポレイテッド | ジケトピペラジンを用いた医薬組成物 |
| EP2613786A4 (en) | 2010-09-07 | 2013-10-23 | Dmi Acquisition Corp | TREATMENT OF DISEASES |
| PH12014500685B1 (en) | 2011-10-10 | 2018-10-03 | Ampio Pharmaceuticals Inc | Treatment of degenerative joint disease |
| JP2014530063A (ja) | 2011-10-10 | 2014-11-17 | アンピオ ファーマシューティカルズ,インコーポレイテッド | 免疫寛容が高められた埋込み型医療用デバイス、ならびに製造方法および埋込み方法 |
| HK1198812A1 (en) | 2011-10-28 | 2015-06-12 | Ampio Pharmaceuticals, Inc. | Treatment of rhinitis |
| CA2906864A1 (en) | 2013-03-15 | 2014-09-18 | Ampio Pharmaceuticals, Inc. | Compositions for the mobilization, homing, expansion and differentiation of stem cells and methods of using the same |
| EP4066836A1 (en) | 2014-08-18 | 2022-10-05 | Ampio Pharmaceuticals, Inc. | Treatment of joint conditions |
| EP3310375A4 (en) | 2015-06-22 | 2019-02-20 | Ampio Pharmaceuticals, Inc. | USE OF LOW-MOLECULAR FRACTIONS OF HUMAN SERUMALBUMINE IN THE TREATMENT OF ILLNESSES |
Family Cites Families (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE2009341C3 (de) * | 1970-02-27 | 1979-06-21 | Max-Planck-Gesellschaft Zur Foerderung Der Wissenschaften E.V., 3400 Goettingen | 3-Octadecyloxy-propanol-(l)-phosphorsäure-monocholinester und Verfahren zu dessen Herstellung |
| DE2619686C2 (de) * | 1976-05-04 | 1986-08-07 | Max-Planck-Gesellschaft zur Förderung der Wissenschaften e.V., 3400 Göttingen | Verwendung eines Lysolecithins zur Tumorbehandlung |
| DE2619715A1 (de) * | 1976-05-04 | 1977-11-24 | Max Planck Gesellschaft | Tumor-antigen und verfahren zu dessen herstellung |
| GB2046092B (en) * | 1979-03-05 | 1983-11-02 | Toyama Chemical Co Ltd | Pharmaceutical composition containing a lysophospholid and a phospholipid |
| US4444766A (en) * | 1980-10-21 | 1984-04-24 | Boehringer Mannheim Gmbh | Sulfur-containing phospholipid compounds and therapeutic compositions |
| DE3127503A1 (de) * | 1981-07-11 | 1983-02-17 | Boehringer Mannheim Gmbh, 6800 Mannheim | Neue phospholipide, verfahren zu deren herstellung und diese verbindungen enthaltende arzneimittel |
| DE3304870A1 (de) * | 1983-02-12 | 1984-08-16 | Boehringer Mannheim Gmbh, 6800 Mannheim | Neue phospholipide, verfahren zu deren herstellung und diese verbindungen enthaltende arzneimittel |
-
1989
- 1989-03-04 DE DE3906952A patent/DE3906952A1/de not_active Withdrawn
-
1990
- 1990-02-26 EP EP90103661A patent/EP0395849B1/de not_active Expired - Lifetime
- 1990-02-26 AT AT90103661T patent/ATE121409T1/de not_active IP Right Cessation
- 1990-02-26 DE DE59008915T patent/DE59008915D1/de not_active Expired - Fee Related
- 1990-02-27 NZ NZ232692A patent/NZ232692A/en unknown
- 1990-02-28 DD DD90338238A patent/DD292259A5/de not_active IP Right Cessation
- 1990-02-28 AU AU50596/90A patent/AU633304B2/en not_active Ceased
- 1990-03-01 IL IL9359890A patent/IL93598A/en not_active IP Right Cessation
- 1990-03-01 MX MX1972290A patent/MX19722A/es unknown
- 1990-03-02 FI FI901096A patent/FI93122C/fi not_active IP Right Cessation
- 1990-03-02 ZA ZA901601A patent/ZA901601B/xx unknown
- 1990-03-02 IE IE900743A patent/IE900743L/xx unknown
- 1990-03-02 PT PT93324A patent/PT93324B/pt not_active IP Right Cessation
- 1990-03-02 JP JP2051584A patent/JPH0341027A/ja active Pending
- 1990-03-02 HU HU901280A patent/HU204057B/hu not_active IP Right Cessation
- 1990-03-02 NO NO90901008A patent/NO901008L/no unknown
- 1990-03-02 RU SU904743486A patent/RU2035466C1/ru active
- 1990-03-05 CA CA002011209A patent/CA2011209A1/en not_active Abandoned
- 1990-03-05 KR KR1019900002942A patent/KR900014412A/ko not_active Withdrawn
-
1993
- 1993-07-23 US US08/095,478 patent/US5543402A/en not_active Expired - Fee Related
Also Published As
| Publication number | Publication date |
|---|---|
| NO901008L (no) | 1990-09-05 |
| IL93598A (en) | 1994-06-24 |
| CA2011209A1 (en) | 1990-09-04 |
| AU633304B2 (en) | 1993-01-28 |
| KR900014412A (ko) | 1990-10-23 |
| NZ232692A (en) | 1992-06-25 |
| IL93598A0 (en) | 1990-12-23 |
| HUT53111A (en) | 1990-09-28 |
| FI93122C (fi) | 1995-02-27 |
| ATE121409T1 (de) | 1995-05-15 |
| JPH0341027A (ja) | 1991-02-21 |
| HU204057B (en) | 1991-11-28 |
| EP0395849B1 (de) | 1995-04-19 |
| AU5059690A (en) | 1990-09-06 |
| HU901280D0 (en) | 1990-05-28 |
| DE3906952A1 (de) | 1990-09-06 |
| NO901008D0 (no) | 1990-03-02 |
| FI93122B (fi) | 1994-11-15 |
| ZA901601B (en) | 1990-12-28 |
| PT93324B (pt) | 1996-02-29 |
| IE900743L (en) | 1990-09-04 |
| FI901096A0 (fi) | 1990-03-02 |
| EP0395849A1 (de) | 1990-11-07 |
| RU2035466C1 (ru) | 1995-05-20 |
| MX19722A (es) | 1993-11-01 |
| DD292259A5 (de) | 1991-07-25 |
| DE59008915D1 (de) | 1995-05-24 |
| US5543402A (en) | 1996-08-06 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FG3A | Patent granted, date of granting |
Effective date: 19951123 |
|
| MM3A | Annulment or lapse |
Free format text: LAPSE DUE TO NON-PAYMENT OF FEES Effective date: 19970531 |