PT95519A - Processo para a preparacao de derivados de 1,4-di-hidro-4-oxo-3-quinolina uteiscomo agentes antibacterianos selectivos em mamiferos - Google Patents

Processo para a preparacao de derivados de 1,4-di-hidro-4-oxo-3-quinolina uteiscomo agentes antibacterianos selectivos em mamiferos

Info

Publication number
PT95519A
PT95519A PT95519A PT9551990A PT95519A PT 95519 A PT95519 A PT 95519A PT 95519 A PT95519 A PT 95519A PT 9551990 A PT9551990 A PT 9551990A PT 95519 A PT95519 A PT 95519A
Authority
PT
Portugal
Prior art keywords
antibacterial agents
kinoline
dihydro
mammals
oxo
Prior art date
Application number
PT95519A
Other languages
English (en)
Other versions
PT95519B (pt
Inventor
Paul R Mcguirk
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of PT95519A publication Critical patent/PT95519A/pt
Publication of PT95519B publication Critical patent/PT95519B/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/08Bridged systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
PT95519A 1989-10-06 1990-10-04 Processo para a preparacao de derivados de 1,4-di-hidro-4-oxo-3-quinolina uteiscomo agentes antibacterianos selectivos em mamiferos PT95519B (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
PCT/US1989/004438 WO1991004972A1 (en) 1989-10-06 1989-10-06 1,4-dihydro-4-oxo-3-quinoline derivatives as selectively toxic mammalian antibacterial agents

Publications (2)

Publication Number Publication Date
PT95519A true PT95519A (pt) 1991-08-14
PT95519B PT95519B (pt) 1997-07-31

Family

ID=22215279

Family Applications (1)

Application Number Title Priority Date Filing Date
PT95519A PT95519B (pt) 1989-10-06 1990-10-04 Processo para a preparacao de derivados de 1,4-di-hidro-4-oxo-3-quinolina uteiscomo agentes antibacterianos selectivos em mamiferos

Country Status (12)

Country Link
EP (1) EP0421668B1 (pt)
JP (1) JPH03130286A (pt)
AT (1) ATE116649T1 (pt)
CA (1) CA2026972A1 (pt)
DE (1) DE69015756T2 (pt)
DK (1) DK0421668T3 (pt)
ES (1) ES2066147T3 (pt)
FI (1) FI921475A7 (pt)
GR (1) GR3015002T3 (pt)
IE (1) IE64194B1 (pt)
PT (1) PT95519B (pt)
WO (1) WO1991004972A1 (pt)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20080139574A1 (en) 2006-11-30 2008-06-12 Cadila Healthcare Limited Novel quinoline derivatives
US7902227B2 (en) * 2007-07-27 2011-03-08 Janssen Pharmaceutica Nv. C-7 isoxazolinyl quinolone / naphthyridine derivatives useful as antibacterial agents

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4571396A (en) * 1984-04-16 1986-02-18 Warner-Lambert Company Antibacterial agents
IN166416B (pt) * 1985-09-18 1990-05-05 Pfizer
DE3601567A1 (de) * 1986-01-21 1987-07-23 Bayer Ag 7-(azabicycloalkyl)-chinoloncarbonsaeure- und -naphthyridon-carbonsaeure-derivate
JPH089597B2 (ja) * 1986-01-21 1996-01-31 杏林製薬株式会社 選択毒性に優れた8‐アルコキシキノロンカルボン酸およびその塩並びにその製造方法
JPS63198664A (ja) * 1986-03-31 1988-08-17 Sankyo Co Ltd キノロンカルボン酸誘導体
DK164287A (da) * 1986-03-31 1987-10-01 Sankyo Co Quinolin-3-carboxylsyrederivater og fremgangsmaade til fremstilling deraf og deres anvendelse
DE3641312A1 (de) * 1986-12-03 1988-06-09 Bayer Ag Verfahren zur herstellung von chinolincarbonsaeuren
DE3711193A1 (de) * 1987-04-02 1988-10-13 Bayer Ag 5-substituierte chinolon- und naphthyridoncarbonsaeure-derivate
DE3713672A1 (de) * 1987-04-24 1988-11-17 Bayer Ag Verfahren zur herstellung von parenteral verabreichbaren chinoloncarbonsaeuren
US4851418A (en) * 1987-08-21 1989-07-25 Warner-Lambert Company Naphthyridine antibacterial agents containing an α-amino acid in the side chain of the 7-substituent

Also Published As

Publication number Publication date
IE903566A1 (en) 1991-04-10
GR3015002T3 (en) 1995-05-31
DK0421668T3 (da) 1995-03-20
FI921475A0 (fi) 1992-04-03
PT95519B (pt) 1997-07-31
ES2066147T3 (es) 1995-03-01
EP0421668A2 (en) 1991-04-10
IE64194B1 (en) 1995-07-12
FI921475L (fi) 1992-04-03
WO1991004972A1 (en) 1991-04-18
CA2026972A1 (en) 1991-04-07
JPH03130286A (ja) 1991-06-04
FI921475A7 (fi) 1992-04-03
EP0421668A3 (en) 1991-08-07
ATE116649T1 (de) 1995-01-15
EP0421668B1 (en) 1995-01-04
DE69015756T2 (de) 1995-05-11
DE69015756D1 (de) 1995-02-16

Similar Documents

Publication Publication Date Title
DK0423714T3 (da) Hårrevitaliseringsmiddel
PT94085A (pt) Processo para a preparacao de derivados de amino-fenol anti-inflamatorios
NO954080D0 (no) Amino(tio)eterderivater
FI943142A0 (fi) Amidi- ja ureajohdannaiset, joilla on veren korkeita kolesteroliarvoja vastustava vaikutus, niiden valmistus ja terapeuttiset käytöt
IT1209953B (it) Derivati di 1,4-diidro-4-ossonaftiridina e relativi sali, procedimento per la loro produzione e agenti antibatterici che comprendono i medesimi
BR9503536A (pt) Composto processo para sua preparação seu uso e composição farmacêutica
PT85668A (en) Benzo-fused cycloalkane and oxa-and thai-, cycloalkane trans-1,2-daimine derivatives
ES2051479T3 (es) Uso de imidazoles substituidos en 4 para disminuir la presion intraocular.
PT90022A (pt) Processo para a preparacao de derivados cefem e dos intermediarios correspondentes
SE8600017D0 (sv) New compound
BR9713159A (pt) Composição substancialmente sólida, composto, composição de sal substancialmente sólida, mistura, e, processo para preparar um composto
ATE156486T1 (de) Fungizide 3,4-diaryl-(5h)-furan-2-onederivate
PT92540A (pt) Processo para a preparacao de derivados de anfotericina b
PT95519A (pt) Processo para a preparacao de derivados de 1,4-di-hidro-4-oxo-3-quinolina uteiscomo agentes antibacterianos selectivos em mamiferos
ATE90685T1 (de) Disaccharidderivate.
ES548196A0 (es) Un procedimiento para la preparacion de nuevos derivados de 1,5-benzotiazepina
PT89935A (pt) Processo para a preparacao de novos compostos cefem
ES532836A0 (es) Metodo para preparar derivados de acidos b-carbolin-3-barboxilicos
IT1239950B (it) Processo per la preparazione di composti con attivita' analgesica centrale
ES2038185T3 (es) Procedimiento para preparar inhibidores de dopamina-beta-hidroxilasa.
IT1204960B (it) Composti dotati di attivita' antiallergica
ES2045335T3 (es) Un procedimiento para la preparacion de nuevas s-difluorometilhomocisteinas.
IT1204959B (it) Composti dotati di attivita' antiallergica
BR9501713A (pt) Derivado de imidazopiridina processo para preparar um derivado de imidazopiridina composição farmacêutica e método para a profilaxia ou tratamento de hipertensão em um animal de sangue quente

Legal Events

Date Code Title Description
BB1A Laying open of patent application

Effective date: 19910306

FG3A Patent granted, date of granting

Effective date: 19970430

MM3A Annulment or lapse

Effective date: 20041102