SE454698B - 6-karboxamidoderivat av 5-oxo-5h-1,3,4-tiadiazolo/3,2-a/pyrimidiner, forfarande for deras framstellning samt farmaceutiska kompositioner innehallande desamma - Google Patents

6-karboxamidoderivat av 5-oxo-5h-1,3,4-tiadiazolo/3,2-a/pyrimidiner, forfarande for deras framstellning samt farmaceutiska kompositioner innehallande desamma

Info

Publication number: SE454698B
Authority: SE; Sweden
Prior art keywords: pyridyl; thiadiazolo; oxo; pyrimidine; carboxamide
Prior art date: 1982-12-23

Application number

SE8307133A

Other languages

English (en)

Swedish (sv)

Other versions

SE8307133D0 (sv

SE8307133L (sv

Inventor

G Doria

C Passarotti

A Buttinoni

Original Assignee

Erba Farmitalia

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1982-12-23

Filing date

1983-12-22

Publication date

1988-05-24

1983-11-08 Priority claimed from GB838329746A external-priority patent/GB8329746D0/en

1983-12-22 Application filed by Erba Farmitalia filed Critical Erba Farmitalia

1983-12-22 Publication of SE8307133D0 publication Critical patent/SE8307133D0/xx

1984-06-24 Publication of SE8307133L publication Critical patent/SE8307133L/xx

1988-05-24 Publication of SE454698B publication Critical patent/SE454698B/sv

Links

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D285/00—Heterocyclic compounds containing rings having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by groups C07D275/00 - C07D283/00
- C07D285/01—Five-membered rings
- C07D285/02—Thiadiazoles; Hydrogenated thiadiazoles
- C07D285/04—Thiadiazoles; Hydrogenated thiadiazoles not condensed with other rings
- C07D285/12—1,3,4-Thiadiazoles; Hydrogenated 1,3,4-thiadiazoles
- C07D285/125—1,3,4-Thiadiazoles; Hydrogenated 1,3,4-thiadiazoles with oxygen, sulfur or nitrogen atoms, directly attached to ring carbon atoms, the nitrogen atoms not forming part of a nitro radical
- C07D285/135—Nitrogen atoms
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
- C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
- C07D513/04—Ortho-condensed systems

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Chemical Kinetics & Catalysis (AREA)
Life Sciences & Earth Sciences (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Pain & Pain Management (AREA)
Pharmacology & Pharmacy (AREA)
Rheumatology (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

SE8307133A 1982-12-23 1983-12-22 6-karboxamidoderivat av 5-oxo-5h-1,3,4-tiadiazolo/3,2-a/pyrimidiner, forfarande for deras framstellning samt farmaceutiska kompositioner innehallande desamma SE454698B (sv)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
GB8236642		1982-12-23
GB838329746A GB8329746D0 (en)	1983-11-08	1983-11-08	Carboxamido-derivatives

Publications (3)

Publication Number	Publication Date
SE8307133D0 SE8307133D0 (sv)	1983-12-22
SE8307133L SE8307133L (sv)	1984-06-24
SE454698B true SE454698B (sv)	1988-05-24

Family

ID=26284768

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
SE8307133A SE454698B (sv)	1982-12-23	1983-12-22	6-karboxamidoderivat av 5-oxo-5h-1,3,4-tiadiazolo/3,2-a/pyrimidiner, forfarande for deras framstellning samt farmaceutiska kompositioner innehallande desamma

Country Status (15)

Country	Link
US (1)	US4522944A (de)
AT (1)	AT385036B (de)
AU (1)	AU558600B2 (de)
CA (1)	CA1211440A (de)
CH (1)	CH657136A5 (de)
DE (1)	DE3346223A1 (de)
DK (1)	DK593983A (de)
FI (1)	FI834698A7 (de)
FR (1)	FR2538392B1 (de)
GR (1)	GR79479B (de)
IL (1)	IL70522A (de)
IT (1)	IT1194521B (de)
NL (1)	NL8304340A (de)
SE (1)	SE454698B (de)
SU (1)	SU1297731A3 (de)

Families Citing this family (27)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
DE3702758A1 (de) *	1987-01-30	1988-09-29	Hoechst Ag	Substituierte 3-phenyl-7h-thiazolo (3,2-b) (1,2,4) triazin-7-one, verfahren zu ihrer herstellung, die sie enthaltenden arzneimittel und ihre verwendung, sowie einige bei der herstellung der genannten verbindungen gebildete zwischenprodukte
KR102107954B1 (ko) *	2007-03-12	2020-05-07	인트라-셀룰라 써래피스, 인코퍼레이티드.	치환된 헤테로환 융합 감마-카르볼린 합성
KR20140146192A (ko)	2012-04-14	2014-12-24	인트라-셀룰라 써래피스, 인코퍼레이티드.	유기 화합물
US9708322B2 (en)	2013-03-15	2017-07-18	Intra-Cellular Therapies, Inc.	Substituted pyrido[3',4':4,5]pyrrolo[1,2,3-de]quinoxalines for inhibiting serotonin reuptake transporter activity
KR102373288B1 (ko)	2013-12-03	2022-03-10	인트라-셀룰라 써래피스, 인코퍼레이티드.	신규한 방법
US10077267B2 (en)	2014-04-04	2018-09-18	Intra-Cellular Therapies, Inc.	Organic compounds
CA2944755A1 (en)	2014-04-04	2015-10-08	Intra-Cellular Therapies, Inc.	Organic compounds
PL3838274T3 (pl)	2016-01-26	2024-04-02	Intra-Cellular Therapies, Inc.	Pochodna pirydo[3',4':4,5]pirolo[1,2,3-DE]chinoksaliny do zastosowania w leczeniu zaburzeń OUN
US10682354B2 (en)	2016-03-28	2020-06-16	Intra-Cellular Therapies, Inc.	Compositions and methods
US11014925B2 (en)	2016-03-28	2021-05-25	Intra-Cellular Therapies, Inc.	Co-crystals of 1-(4-fluoro-phenyl)-4-((6bR,1OaS)-3-methyl-2,3,6b,9,10,10a-hexahydro-1H,7H- pyrido[3′,4′:4,51_pyrrolo [1,2,3-delqcuinoxalin-8-yl)-butan-1-one with nicotinamide or isonicotinamide
EP3436455A4 (de)	2016-03-28	2019-09-04	Intra-Cellular Therapies, Inc.	Neuartige salze und kristalle
EP3525763B1 (de)	2016-10-12	2025-03-05	Intra-Cellular Therapies, Inc.	Amorphe feste dispersionen
WO2018126140A1 (en)	2016-12-29	2018-07-05	Intra-Cellular Therapies, Inc.	Organic compounds
EP3562484B1 (de)	2016-12-29	2021-08-25	Intra-Cellular Therapies, Inc.	Pyrido[3',4':4,5]pyrrolo[1,2,3-de]quinoxalinderivate zur behandlung von erkrankungen des zns
RU2767410C2 (ru)	2017-03-24	2022-03-17	Интра-Селлулар Терапиз, Инк.	Новые композиции и способы
EP3658144B1 (de)	2017-07-26	2022-01-26	Intra-Cellular Therapies, Inc.	Pyridopyrroloquinoxalinverbindungen, deren zusammensetzungen und verwendungen in therapie
WO2019023062A1 (en)	2017-07-26	2019-01-31	Intra-Cellular Therapies, Inc.	ORGANIC COMPOUNDS
CN112040940A (zh)	2018-03-23	2020-12-04	细胞内治疗公司	有机化合物
AU2019280850C1 (en)	2018-06-06	2025-02-13	Intra-Cellular Therapies, Inc.	Novel salts and crystals
EP3801527B1 (de)	2018-06-08	2025-02-19	Intra-Cellular Therapies, Inc.	Anellierte gamma-carboline zur akutbehandlung von angst oder depression
CA3240552A1 (en)	2018-06-11	2019-12-19	Intra-Cellular Therapies, Inc.	Substituted heterocycle fused gamma-carbolines synthesis
US12144808B2 (en)	2018-08-29	2024-11-19	Intra-Cellular Therapies, Inc.	Compositions and methods
WO2020047408A1 (en)	2018-08-31	2020-03-05	Intra-Cellular Therapies, Inc.	Novel methods
BR112021003655A2 (pt)	2018-08-31	2021-05-18	Intra-Cellular Therapies, Inc.	métodos novos
WO2021007245A1 (en)	2019-07-07	2021-01-14	Intra-Cellular Therapies, Inc.	Novel methods
EP4072554A4 (de)	2019-12-11	2023-12-20	Intra-Cellular Therapies, Inc.	Organische verbindung
US12414948B2 (en)	2022-05-18	2025-09-16	Intra-Cellular Therapies, Inc.	Methods

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
JPS5129981B2 (de) *	1973-07-17	1976-08-28
GB1568962A (en) *	1975-10-31	1980-06-11	Beecham Group Ltd	Reparation and compositions containing them (heterocyclic-carbonylamino)pencillins methods for their p
JPS55115889A (en) *	1979-02-28	1980-09-06	Teijin Ltd	6-carbamoylthiazolo 3,2-a pyrimidine derivative and its preparation
JPS57142989A (en) *	1981-02-27	1982-09-03	Dai Ichi Seiyaku Co Ltd	Thiazolopyrimidine derivative

1983
- 1983-12-08 US US06/559,322 patent/US4522944A/en not_active Expired - Fee Related
- 1983-12-15 GR GR73259A patent/GR79479B/el unknown
- 1983-12-15 AT AT0438383A patent/AT385036B/de not_active IP Right Cessation
- 1983-12-16 IT IT24207/83A patent/IT1194521B/it active
- 1983-12-16 NL NL8304340A patent/NL8304340A/nl not_active Application Discontinuation
- 1983-12-19 AU AU22525/83A patent/AU558600B2/en not_active Ceased
- 1983-12-20 FI FI834698A patent/FI834698A7/fi not_active Application Discontinuation
- 1983-12-20 CH CH6783/83A patent/CH657136A5/de not_active IP Right Cessation
- 1983-12-21 DE DE19833346223 patent/DE3346223A1/de not_active Withdrawn
- 1983-12-22 SE SE8307133A patent/SE454698B/sv not_active IP Right Cessation
- 1983-12-22 DK DK593983A patent/DK593983A/da not_active Application Discontinuation
- 1983-12-22 CA CA000444151A patent/CA1211440A/en not_active Expired
- 1983-12-22 SU SU833682101A patent/SU1297731A3/ru active
- 1983-12-22 IL IL70522A patent/IL70522A/xx not_active IP Right Cessation
- 1983-12-23 FR FR8320704A patent/FR2538392B1/fr not_active Expired

Also Published As

Publication number	Publication date
SU1297731A3 (ru)	1987-03-15
ATA438383A (de)	1987-07-15
DK593983A (da)	1984-06-24
AT385036B (de)	1988-02-10
CH657136A5 (de)	1986-08-15
FR2538392A1 (fr)	1984-06-29
CA1211440A (en)	1986-09-16
AU558600B2 (en)	1987-02-05
US4522944A (en)	1985-06-11
IL70522A (en)	1986-02-28
SE8307133D0 (sv)	1983-12-22
NL8304340A (nl)	1984-07-16
FI834698A0 (fi)	1983-12-20
SE8307133L (sv)	1984-06-24
GR79479B (de)	1984-10-30
IT8324207A0 (it)	1983-12-16
FI834698A7 (fi)	1984-06-24
DE3346223A1 (de)	1984-06-28
AU2252583A (en)	1984-06-28
FR2538392B1 (fr)	1987-01-16
DK593983D0 (da)	1983-12-22
IL70522A0 (en)	1984-03-30
IT1194521B (it)	1988-09-22

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Legal Events

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1995-01-31

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