SE7708592L - Forfarande for framstellning av fosfonsyraderivat - Google Patents

Forfarande for framstellning av fosfonsyraderivat

Info

Publication number: SE7708592L
Authority: SE; Sweden
Prior art keywords: acid derivatives; procedure; preparation; phosphonic acid; hydroxyamino
Prior art date: 1976-07-27

Application number

SE7708592A

Other languages

English (en)

Other versions

SE441360B (sv

Inventor

Y Kuroda

M Okuhara

E Iguchi

H Aoki

H Imanaka

T Kamiya

M Hashimoto

K Hemmi

H Takeno

Original Assignee

Fujisawa Pharmaceutical Co

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1976-07-27

Filing date

1977-07-26

Publication date

1978-01-28

1977-07-26 Application filed by Fujisawa Pharmaceutical Co filed Critical Fujisawa Pharmaceutical Co

1978-01-28 Publication of SE7708592L publication Critical patent/SE7708592L/sv

1985-09-30 Publication of SE441360B publication Critical patent/SE441360B/sv

Links

229940042400 direct acting antivirals phosphonic acid derivative Drugs 0.000 title 1
150000003007 phosphonic acid derivatives Chemical class 0.000 title 1
PKMNDDZSIHLLLI-UHFFFAOYSA-N FR900098 Natural products CC(=O)N(O)CCCP(O)(O)=O PKMNDDZSIHLLLI-UHFFFAOYSA-N 0.000 abstract 2
125000002252 acyl group Chemical group 0.000 abstract 2
125000000217 alkyl group Chemical group 0.000 abstract 2
125000002947 alkylene group Chemical group 0.000 abstract 2
229910052739 hydrogen Inorganic materials 0.000 abstract 2
239000001257 hydrogen Substances 0.000 abstract 2
125000004435 hydrogen atom Chemical group [H]* 0.000 abstract 2
150000003839 salts Chemical class 0.000 abstract 2
SMXUDUOWTDBXDT-UHFFFAOYSA-N [3-[acetyl(hydroxy)amino]-2-hydroxypropyl]phosphonic acid Chemical compound CC(=O)N(O)CC(O)CP(O)(O)=O SMXUDUOWTDBXDT-UHFFFAOYSA-N 0.000 abstract 1
239000002253 acid Substances 0.000 abstract 1
125000004450 alkenylene group Chemical group 0.000 abstract 1
230000000845 anti-microbial effect Effects 0.000 abstract 1
150000001875 compounds Chemical class 0.000 abstract 1
150000002148 esters Chemical class 0.000 abstract 1
125000002887 hydroxy group Chemical group [H]O* 0.000 abstract 1
244000052769 pathogen Species 0.000 abstract 1
125000001476 phosphono group Chemical group [H]OP(*)(=O)O[H] 0.000 abstract 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
- C07F9/02—Phosphorus compounds
- C07F9/28—Phosphorus compounds with one or more P—C bonds
- C07F9/38—Phosphonic acids [RP(=O)(OH)2]; Thiophosphonic acids ; [RP(=X1)(X2H)2(X1, X2 are each independently O, S or Se)]
- C07F9/40—Esters thereof
- C07F9/4003—Esters thereof the acid moiety containing a substituent or a structure which is considered as characteristic
- C07F9/4006—Esters of acyclic acids which can have further substituents on alkyl
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
- C07F9/02—Phosphorus compounds
- C07F9/28—Phosphorus compounds with one or more P—C bonds
- C07F9/38—Phosphonic acids [RP(=O)(OH)2]; Thiophosphonic acids ; [RP(=X1)(X2H)2(X1, X2 are each independently O, S or Se)]
- C07F9/3804—Phosphonic acids [RP(=O)(OH)2]; Thiophosphonic acids ; [RP(=X1)(X2H)2(X1, X2 are each independently O, S or Se)] not used, see subgroups
- C07F9/3808—Acyclic saturated acids which can have further substituents on alkyl
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
- C07F9/02—Phosphorus compounds
- C07F9/28—Phosphorus compounds with one or more P—C bonds
- C07F9/38—Phosphonic acids [RP(=O)(OH)2]; Thiophosphonic acids ; [RP(=X1)(X2H)2(X1, X2 are each independently O, S or Se)]
- C07F9/3804—Phosphonic acids [RP(=O)(OH)2]; Thiophosphonic acids ; [RP(=X1)(X2H)2(X1, X2 are each independently O, S or Se)] not used, see subgroups
- C07F9/3826—Acyclic unsaturated acids

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
General Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
Biochemistry (AREA)
Molecular Biology (AREA)
Oncology (AREA)
Veterinary Medicine (AREA)
Pharmacology & Pharmacy (AREA)
Chemical Kinetics & Catalysis (AREA)
Animal Behavior & Ethology (AREA)
Medicinal Chemistry (AREA)
Public Health (AREA)
General Chemical & Material Sciences (AREA)
Communicable Diseases (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Preparation Of Compounds By Using Micro-Organisms (AREA)
Cephalosporin Compounds (AREA)
Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

SE7708592A 1976-07-27 1977-07-26 Forfarande for framstellning av fosfonsyraderivat SE441360B (sv)

Applications Claiming Priority (3)

Application Number	Priority Date	Filing Date	Title
GB3133976		1976-07-27
GB4222276		1976-10-11
GB31339/76A GB1580899A (en)	1976-07-27	1977-06-20	Hydroxyaminohydrocarbonphosphonic acid derivatives and production and use thereof

Publications (2)

Publication Number	Publication Date
SE7708592L true SE7708592L (sv)	1978-01-28
SE441360B SE441360B (sv)	1985-09-30

Family

ID=27258468

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
SE7708592A SE441360B (sv)	1976-07-27	1977-07-26	Forfarande for framstellning av fosfonsyraderivat

Country Status (21)

Country	Link
US (1)	US4182758A (sv)
JP (1)	JPS5340720A (sv)
AR (1)	AR226522A1 (sv)
AT (2)	AT367064B (sv)
CA (1)	CA1091241A (sv)
CH (5)	CH640862A5 (sv)
DE (2)	DE2733658A1 (sv)
DK (1)	DK149609C (sv)
ES (3)	ES461084A1 (sv)
FI (1)	FI64377C (sv)
FR (1)	FR2474505A1 (sv)
GB (1)	GB1580899A (sv)
GR (1)	GR61140B (sv)
HU (1)	HU182023B (sv)
IE (1)	IE45536B1 (sv)
NL (1)	NL7708325A (sv)
NO (1)	NO157504C (sv)
OA (1)	OA05725A (sv)
PH (1)	PH14401A (sv)
PT (1)	PT66854B (sv)
SE (1)	SE441360B (sv)

Families Citing this family (23)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US4084953A (en) *	1977-03-09	1978-04-18	Monsanto Company	N-hydroxy-N-phosphonomethylglycines and the herbicidal use thereof
US4210635A (en) *	1978-02-15	1980-07-01	Fujisawa Pharmaceutical Co., Ltd.	Antibacterial composition
US4268503A (en) *	1978-09-14	1981-05-19	Fujisawa Pharmaceutical Co., Ltd.	Antibacterial composition
US4693742A (en) *	1983-12-20	1987-09-15	Rohm And Hass Company	Herbicidal hydroxyamino phosphonic acids and derivatives
US5189030A (en) *	1985-06-11	1993-02-23	Ciba-Geigy Corporation	1-amino-2-phenylethanephosphonic acids as microbiocides
JPH0340299U (sv) *	1989-08-31	1991-04-18
DE19843223A1 (de) *	1998-09-22	2000-03-30	Hassan Jomaa	Phosphororganische Verbindungen und ihre Verwendung
BR9909668A (pt)	1998-04-14	2000-12-19	Jomaa Hassan	Uso de compostos de organofósforo para o tratamento terapêutico e profilático de infecções
DE19825585A1 (de) *	1998-04-14	1999-10-21	Hassan Jomaa	Verwendung von Aminohydrocarbylphosphonsäurederivaten zur therapeutischen und prophylaktischen Behandlung von Infektionen, die durch Parasiten, Pilze oder Viren hervorgerufen werden
CN1309659A (zh)	1998-07-15	2001-08-22	哈桑·朱马	有机磷化合物及其用途
US6753324B2 (en)	1998-07-15	2004-06-22	Hassan Jomaa	Phosphorous organic compounds and their use
AU5034899A (en) *	1998-07-15	2000-02-07	Jomaa Hassan	Drugs containing phosphoric acid derivatives as active ingredient and their use
DE19854403A1 (de)	1998-11-25	2000-05-31	Hassan Jomaa	Phosphororganische Verbindungen und ihre Verwendung
WO2001060829A1 (de) *	2000-02-18	2001-08-23	Jomaa Pharmaka Gmbh	Phosphororganische verbindungen und ihre verwendung
DE10035189A1 (de) *	2000-07-20	2002-02-21	Hassan Jomaa	Arzneimittel zur oralen Applikation mit einem Gehalt an 3-N-Formylhydroxylaminopropylphosphonsäureestern oder 3-N-Acetylhydroxylaminopropylphosphonsäureestern als Wirkstoff
JP2009511449A (ja) *	2005-10-06	2009-03-19	イナート・ファルマ	有機塩基のリン酸化抗原塩およびその結晶化方法
JP5198877B2 (ja) *	2006-01-31	2013-05-15	株式会社エーピーアイコーポレーション	ベンゾアゼピノン類の製造方法
CA2733390A1 (en)	2008-08-01	2010-02-04	Bioxiness Pharmaceuticals, Inc.	Methionine analogs and methods of using same
EP2404601A1 (en)	2010-07-06	2012-01-11	BioAgency AG	New drug combinations for the treatment of Malaria
EP2725029A1 (en)	2012-10-29	2014-04-30	Laboratoire Biodim	New antibacterial compounds and biological applications thereof
WO2019246119A1 (en) *	2018-06-18	2019-12-26	The George Washington University a Congressionally Chartered Not-for-Profit Corporation	Antibiotics for veterinary staphylococcal infections
EP4045056A1 (de)	2019-10-19	2022-08-24	DMG Deutsche Malaria GmbH	Kombinationspräparate von 3-n-formylhydroxylaminopropylphosphonsäurederivaten oder 3-n-acetylhydroxylaminopropylphosphonsäurederivaten mit clindamycin und artesunat
EP3960176A1 (en)	2020-08-26	2022-03-02	DMG Deutsche Malaria GmbH	Piperaquine and related drug combinations for use in the treatment of covid-19

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
NL6905272A (sv)	1968-05-15	1969-11-18
US3764677A (en) *	1971-06-25	1973-10-09	Gates Rubber Co	Diethyl betaaminoethylphosphonate as an antimicrobial agent

1977
- 1977-06-20 GB GB31339/76A patent/GB1580899A/en not_active Expired
- 1977-07-25 HU HU77FU356A patent/HU182023B/hu not_active IP Right Cessation
- 1977-07-25 PH PH20031A patent/PH14401A/en unknown
- 1977-07-26 SE SE7708592A patent/SE441360B/sv not_active IP Right Cessation
- 1977-07-26 DK DK337877A patent/DK149609C/da not_active IP Right Cessation
- 1977-07-26 NO NO772652A patent/NO157504C/no unknown
- 1977-07-26 CA CA283,566A patent/CA1091241A/en not_active Expired
- 1977-07-26 DE DE19772733658 patent/DE2733658A1/de active Granted
- 1977-07-26 FI FI772280A patent/FI64377C/fi not_active IP Right Cessation
- 1977-07-26 DE DE2760320A patent/DE2760320C2/de not_active Expired
- 1977-07-26 GR GR54041A patent/GR61140B/el unknown
- 1977-07-26 IE IE1555/77A patent/IE45536B1/en unknown
- 1977-07-27 US US05/819,554 patent/US4182758A/en not_active Expired - Lifetime
- 1977-07-27 PT PT66854A patent/PT66854B/pt unknown
- 1977-07-27 OA OA56240A patent/OA05725A/xx unknown
- 1977-07-27 AR AR268576A patent/AR226522A1/es active
- 1977-07-27 ES ES461084A patent/ES461084A1/es not_active Expired
- 1977-07-27 NL NL7708325A patent/NL7708325A/xx not_active Application Discontinuation
- 1977-07-27 AT AT0550977A patent/AT367064B/de not_active IP Right Cessation
- 1977-07-27 CH CH930777A patent/CH640862A5/de not_active IP Right Cessation
- 1977-07-27 JP JP9081077A patent/JPS5340720A/ja active Granted
- 1977-07-27 FR FR7723128A patent/FR2474505A1/fr active Granted
1978
- 1978-07-17 ES ES471822A patent/ES471822A1/es not_active Expired
1979
- 1979-04-02 ES ES479211A patent/ES479211A1/es not_active Expired
- 1979-08-22 AT AT0564879A patent/AT367430B/de not_active IP Right Cessation
1984
- 1984-01-31 CH CH427/84A patent/CH647807A5/de not_active IP Right Cessation
- 1984-01-31 CH CH42484A patent/CH646978A5/de not_active IP Right Cessation
- 1984-01-31 CH CH42584A patent/CH646979A5/de not_active IP Right Cessation
- 1984-01-31 CH CH42684A patent/CH646980A5/de not_active IP Right Cessation

Also Published As

Publication number	Publication date
US4182758A (en)	1980-01-08
PT66854B (en)	1978-12-28
FR2474505B1 (sv)	1984-01-27
NO772652L (no)	1978-01-30
JPS613799B2 (sv)	1986-02-04
ES461084A1 (es)	1978-12-01
CH646978A5 (de)	1984-12-28
FR2474505A1 (fr)	1981-07-31
HU182023B (en)	1983-12-28
CH647807A5 (de)	1985-02-15
ES471822A1 (es)	1979-10-16
PH14401A (en)	1981-06-25
CH646979A5 (de)	1984-12-28
CH640862A5 (de)	1984-01-31
IE45536B1 (en)	1982-09-22
PT66854A (en)	1977-08-01
AT367430B (de)	1982-07-12
ATA550977A (de)	1981-10-15
DE2760320C2 (sv)	1988-11-03
DE2733658C2 (sv)	1987-06-25
SE441360B (sv)	1985-09-30
ES479211A1 (es)	1979-12-16
DK149609C (da)	1987-02-09
IE45536L (en)	1978-01-27
GR61140B (en)	1978-09-23
NL7708325A (nl)	1978-01-31
JPS5340720A (en)	1978-04-13
NO157504C (no)	1988-03-30
DK149609B (da)	1986-08-11
FI64377C (fi)	1983-11-10
FI772280A7 (sv)	1978-01-28
AR226522A1 (es)	1982-07-30
FI64377B (fi)	1983-07-29
DK337877A (da)	1978-01-28
CH646980A5 (de)	1984-12-28
AT367064B (de)	1982-05-25
NO157504B (no)	1987-12-21
GB1580899A (en)	1980-12-10
ATA564879A (de)	1981-11-15
OA05725A (fr)	1981-05-31
CA1091241A (en)	1980-12-09
DE2733658A1 (de)	1978-02-09

Legal Events

Date

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Title

Description

1995-01-31

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Patent has lapsed

Ref document number: 7708592-6

Effective date: 19950210

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1995-04-03

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