SK16552002A3 - Stála, biologicky zlúčiteľná, dobre znášateľná mikroemulzia voda v oleji a jej použitie - Google Patents

Stála, biologicky zlúčiteľná, dobre znášateľná mikroemulzia voda v oleji a jej použitie Download PDF

Info

Publication number: SK16552002A3
Authority: SK; Slovakia
Prior art keywords: microemulsion; biologically active; surfactant; active compound; days
Prior art date: 2000-05-26

Application number

SK1655-2002A

Other languages

English (en)

Slovak (sk)

Inventor

Francesco Autuori

Carlo Bianchini

Giuseppe Bottoni

Flavio Leoni

Paolo Mascagni

Valmen Monzani

Oreste Piccolo

Original Assignee

Italfarmaco S. P. A.

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2000-05-26

Filing date

2001-05-23

Publication date

2003-05-02

2001-05-23 Application filed by Italfarmaco S. P. A. filed Critical Italfarmaco S. P. A.

2003-05-02 Publication of SK16552002A3 publication Critical patent/SK16552002A3/sk

Links

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RUGAHXUZHWYHNG-NLGNTGLNSA-N acetic acid;(4r,7s,10s,13r,16s,19r)-10-(4-aminobutyl)-n-[(2s,3r)-1-amino-3-hydroxy-1-oxobutan-2-yl]-19-[[(2r)-2-amino-3-naphthalen-2-ylpropanoyl]amino]-16-[(4-hydroxyphenyl)methyl]-13-(1h-indol-3-ylmethyl)-6,9,12,15,18-pentaoxo-7-propan-2-yl-1,2-dithia-5, Chemical compound CC(O)=O.CC(O)=O.CC(O)=O.CC(O)=O.CC(O)=O.C([C@H]1C(=O)N[C@H](CC=2C3=CC=CC=C3NC=2)C(=O)N[C@@H](CCCCN)C(=O)N[C@H](C(N[C@@H](CSSC[C@@H](C(=O)N1)NC(=O)[C@H](N)CC=1C=C2C=CC=CC2=CC=1)C(=O)N[C@@H]([C@@H](C)O)C(N)=O)=O)C(C)C)C1=CC=C(O)C=C1.C([C@H]1C(=O)N[C@H](CC=2C3=CC=CC=C3NC=2)C(=O)N[C@@H](CCCCN)C(=O)N[C@H](C(N[C@@H](CSSC[C@@H](C(=O)N1)NC(=O)[C@H](N)CC=1C=C2C=CC=CC2=CC=1)C(=O)N[C@@H]([C@@H](C)O)C(N)=O)=O)C(C)C)C1=CC=C(O)C=C1 RUGAHXUZHWYHNG-NLGNTGLNSA-N 0.000 description 1
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WQZGKKKJIJFFOK-PHYPRBDBSA-N alpha-D-galactose Chemical compound OC[C@H]1O[C@H](O)[C@H](O)[C@@H](O)[C@H]1O WQZGKKKJIJFFOK-PHYPRBDBSA-N 0.000 description 1
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GONOPSZTUGRENK-UHFFFAOYSA-N benzyl(trichloro)silane Chemical compound Cl[Si](Cl)(Cl)CC1=CC=CC=C1 GONOPSZTUGRENK-UHFFFAOYSA-N 0.000 description 1
WQZGKKKJIJFFOK-VFUOTHLCSA-N beta-D-glucose Chemical compound OC[C@H]1O[C@@H](O)[C@H](O)[C@@H](O)[C@@H]1O WQZGKKKJIJFFOK-VFUOTHLCSA-N 0.000 description 1
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ACCCMOQWYVYDOT-UHFFFAOYSA-N hexane-1,1-diol Chemical compound CCCCCC(O)O ACCCMOQWYVYDOT-UHFFFAOYSA-N 0.000 description 1
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RGLRXNKKBLIBQS-XNHQSDQCSA-N leuprolide acetate Chemical compound CC(O)=O.CCNC(=O)[C@@H]1CCCN1C(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](CC(C)C)NC(=O)[C@@H](NC(=O)[C@H](CO)NC(=O)[C@H](CC=1C2=CC=CC=C2NC=1)NC(=O)[C@H](CC=1N=CNC=1)NC(=O)[C@H]1NC(=O)CC1)CC1=CC=C(O)C=C1 RGLRXNKKBLIBQS-XNHQSDQCSA-N 0.000 description 1
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Classifications

- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/10—Dispersions; Emulsions
- A61K9/107—Emulsions ; Emulsion preconcentrates; Micelles
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/10—Dispersions; Emulsions
- A61K9/107—Emulsions ; Emulsion preconcentrates; Micelles
- A61K9/1075—Microemulsions or submicron emulsions; Preconcentrates or solids thereof; Micelles, e.g. made of phospholipids or block copolymers
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/02—Drugs for disorders of the endocrine system of the hypothalamic hormones, e.g. TRH, GnRH, CRH, GRH, somatostatin
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/06—Drugs for disorders of the endocrine system of the anterior pituitary hormones, e.g. TSH, ACTH, FSH, LH, PRL, GH
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
- A61P5/26—Androgens

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Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
Veterinary Medicine (AREA)
Public Health (AREA)
Medicinal Chemistry (AREA)
General Health & Medical Sciences (AREA)
Pharmacology & Pharmacy (AREA)
Organic Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
General Chemical & Material Sciences (AREA)
Chemical Kinetics & Catalysis (AREA)
Endocrinology (AREA)
Bioinformatics & Cheminformatics (AREA)
Diabetes (AREA)
Engineering & Computer Science (AREA)
Dispersion Chemistry (AREA)
Epidemiology (AREA)
Biophysics (AREA)
Molecular Biology (AREA)
Medicinal Preparation (AREA)
Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

SK1655-2002A 2000-05-26 2001-05-23 Stála, biologicky zlúčiteľná, dobre znášateľná mikroemulzia voda v oleji a jej použitie SK16552002A3 (sk)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
IT2000MI001173A IT1318539B1 (it)	2000-05-26	2000-05-26	Composizioni farmaceutiche a rilascio prolungato per lasomministrazione parenterale di sostanze idrofile biologicamente
PCT/EP2001/005949 WO2001089479A2 (en)	2000-05-26	2001-05-23	Sustained release pharmaceutical compositions for parenteral administration of hydrophilic compounds

Publications (1)

Publication Number	Publication Date
SK16552002A3 true SK16552002A3 (sk)	2003-05-02

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Country Status (28)

Country	Link
US (1)	US7157099B2 (pt)
EP (1)	EP1283700B1 (pt)
JP (1)	JP4954423B2 (pt)
KR (1)	KR100802625B1 (pt)
CN (1)	CN100479856C (pt)
AT (1)	ATE321533T1 (pt)
AU (2)	AU8178601A (pt)
BR (1)	BRPI0111016B8 (pt)
CA (1)	CA2409854C (pt)
CY (1)	CY1105262T1 (pt)
CZ (1)	CZ302059B6 (pt)
DE (1)	DE60118395T2 (pt)
DK (1)	DK1283700T3 (pt)
ES (1)	ES2257428T3 (pt)
HR (1)	HRP20020929A2 (pt)
HU (1)	HU228926B1 (pt)
IL (1)	IL153011A0 (pt)
IT (1)	IT1318539B1 (pt)
MX (1)	MXPA02011539A (pt)
NO (1)	NO334880B1 (pt)
PL (1)	PL203354B1 (pt)
PT (1)	PT1283700E (pt)
RU (1)	RU2272615C2 (pt)
SI (1)	SI1283700T1 (pt)
SK (1)	SK16552002A3 (pt)
WO (1)	WO2001089479A2 (pt)
YU (1)	YU88202A (pt)
ZA (1)	ZA200209520B (pt)

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2000
- 2000-05-26 IT IT2000MI001173A patent/IT1318539B1/it active
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- 2001-05-23 CN CNB018099254A patent/CN100479856C/zh not_active Expired - Lifetime
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Also Published As

Publication number	Publication date
AU8178601A (en)	2001-12-03
BR0111016A (pt)	2003-04-15
CN1430502A (zh)	2003-07-16
HUP0301921A2 (hu)	2003-09-29
IL153011A0 (en)	2003-06-24
PT1283700E (pt)	2006-07-31
RU2272615C2 (ru)	2006-03-27
KR100802625B1 (ko)	2008-02-13
NO20025621L (no)	2003-01-27
DE60118395T2 (de)	2006-12-07
DE60118395D1 (de)	2006-05-18
JP4954423B2 (ja)	2012-06-13
CZ20023772A3 (cs)	2003-02-12
CA2409854C (en)	2011-02-08
CY1105262T1 (el)	2010-03-03
US7157099B2 (en)	2007-01-02
EP1283700B1 (en)	2006-03-29
ATE321533T1 (de)	2006-04-15
JP2003534265A (ja)	2003-11-18
BRPI0111016B1 (pt)	2017-11-21
YU88202A (sh)	2006-01-16
WO2001089479A3 (en)	2002-03-28
EP1283700A2 (en)	2003-02-19
DK1283700T3 (da)	2006-07-24
CN100479856C (zh)	2009-04-22
BRPI0111016B8 (pt)	2021-05-25
AU2001281786B8 (en)	2005-11-17
SI1283700T1 (sl)	2006-08-31
HRP20020929A2 (en)	2004-02-29
CZ302059B6 (cs)	2010-09-22
ES2257428T3 (es)	2006-08-01
NO334880B1 (no)	2014-06-30
CA2409854A1 (en)	2001-11-29
PL359601A1 (en)	2004-08-23
PL203354B1 (pl)	2009-09-30
WO2001089479A2 (en)	2001-11-29
KR20030011856A (ko)	2003-02-11
IT1318539B1 (it)	2003-08-27
HU228926B1 (en)	2013-06-28
ITMI20001173A1 (it)	2001-11-26
ITMI20001173A0 (it)	2000-05-26
NO20025621D0 (no)	2002-11-22
ZA200209520B (en)	2003-11-24
AU2001281786B2 (en)	2005-07-21
MXPA02011539A (es)	2004-08-12
HUP0301921A3 (en)	2005-11-28
US20030171299A1 (en)	2003-09-11

Publication	Publication Date	Title
US7157099B2 (en)	2007-01-02	Sustained release pharmaceutical compositions for the parenteral administration of hydrophilic compounds
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AU672441B2 (en)	1996-10-03	Injectable lecithin gel
KR100401119B1 (ko)	2004-03-19	택산계열유도체-기본약학조성물
EA035495B1 (ru)	2020-06-25	Состав-предшественник, содержащий агонист рецепторов соматостатина, способ лечения путем его введения, его применение, предварительно заполненное устройство, содержащее его, и набор, содержащий указанное устройство
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