SV2002000320A - Proceso para la simple preparacion de (3-cloro-4- fluorofenilo)-[7-(3-morfolina-4ilo-propoxi)-6-nitroquinazolina-4ilo]-amina o (3-cloro-4-fluorofenilo-[7-(3-morfolina-4-il-propoxi)-6-aminoquinazolina-4-ilo]-amina ref.b.12187/rm/shh - Google Patents

Proceso para la simple preparacion de (3-cloro-4- fluorofenilo)-[7-(3-morfolina-4ilo-propoxi)-6-nitroquinazolina-4ilo]-amina o (3-cloro-4-fluorofenilo-[7-(3-morfolina-4-il-propoxi)-6-aminoquinazolina-4-ilo]-amina ref.b.12187/rm/shh

Info

Publication number
SV2002000320A
SV2002000320A SV2001000320A SV2001000320A SV2002000320A SV 2002000320 A SV2002000320 A SV 2002000320A SV 2001000320 A SV2001000320 A SV 2001000320A SV 2001000320 A SV2001000320 A SV 2001000320A SV 2002000320 A SV2002000320 A SV 2002000320A
Authority
SV
El Salvador
Prior art keywords
propoxi
amina
4ilo
ilo
morfolina
Prior art date
Application number
SV2001000320A
Other languages
English (en)
Inventor
Hubert Barth
Simon Schneider
Klaus Steiner
Original Assignee
Godecke Gmbh
Sanofi Aventis Deutschland
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Godecke Gmbh, Sanofi Aventis Deutschland filed Critical Godecke Gmbh
Publication of SV2002000320A publication Critical patent/SV2002000320A/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/70Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
    • C07D239/72Quinazolines; Hydrogenated quinazolines
    • C07D239/86Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in position 4
    • C07D239/94Nitrogen atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)

Abstract

ESTA INVENCION SE REFIERE A UNA REACCION GLOBAL PARA LA PREPARACION DE (3-CLORO-4-FLUOROFENILO)-[7-(3-MORFOLINA-4-ILO-PROPOXI)-6-NITROQUINAZOLINA-4-ILO]-AMINA(I)VER FORMULAS O DE (3-CLORO-4-FLUOROFENILO)-[7-(3-MORFOLINA-4-ILO-PROPOXI)-6-AMINOQUINAZOLINA-4-ILO]-AMINA(VII), VER FORMULA.
SV2001000320A 2000-02-26 2001-02-23 Proceso para la simple preparacion de (3-cloro-4- fluorofenilo)-[7-(3-morfolina-4ilo-propoxi)-6-nitroquinazolina-4ilo]-amina o (3-cloro-4-fluorofenilo-[7-(3-morfolina-4-il-propoxi)-6-aminoquinazolina-4-ilo]-amina ref.b.12187/rm/shh SV2002000320A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE10009267A DE10009267A1 (de) 2000-02-26 2000-02-26 Verfahren zur einfachen Herstellung von (3-Chlor-4-fluor-phenyl)-[7-(3-morpholin-4-yl-propoxy)-6-nitro-quinazolin-4-yl]-amin bzw. (3-Chlor-4-fluor-phenyl)-[7-(3-morpholin-4-yl-propoxy)-6-amino-quinazolin-4-yl]-amin

Publications (1)

Publication Number Publication Date
SV2002000320A true SV2002000320A (es) 2002-06-07

Family

ID=7632648

Family Applications (1)

Application Number Title Priority Date Filing Date
SV2001000320A SV2002000320A (es) 2000-02-26 2001-02-23 Proceso para la simple preparacion de (3-cloro-4- fluorofenilo)-[7-(3-morfolina-4ilo-propoxi)-6-nitroquinazolina-4ilo]-amina o (3-cloro-4-fluorofenilo-[7-(3-morfolina-4-il-propoxi)-6-aminoquinazolina-4-ilo]-amina ref.b.12187/rm/shh

Country Status (32)

Country Link
US (1) US20030050313A1 (es)
EP (1) EP1265874B1 (es)
JP (1) JP2003524006A (es)
KR (1) KR20030011773A (es)
CN (1) CN1171877C (es)
AR (1) AR027377A1 (es)
AT (1) ATE296810T1 (es)
AU (1) AU2001228478A1 (es)
BR (1) BR0108695A (es)
CA (1) CA2401171A1 (es)
CO (1) CO5280058A1 (es)
DE (2) DE10009267A1 (es)
EA (1) EA005213B1 (es)
EG (1) EG23221A (es)
ES (1) ES2240483T3 (es)
GT (1) GT200100025A (es)
HK (1) HK1054551B (es)
HU (1) HUP0204510A3 (es)
IL (1) IL151206A0 (es)
MX (1) MXPA02008301A (es)
MY (1) MY133846A (es)
PA (1) PA8512701A1 (es)
PE (1) PE20011073A1 (es)
PL (1) PL357774A1 (es)
PT (1) PT1265874E (es)
PY (1) PY0102711A (es)
SV (1) SV2002000320A (es)
TN (1) TNSN01031A1 (es)
UY (1) UY26594A1 (es)
WO (1) WO2001062743A2 (es)
YU (1) YU62502A (es)
ZA (1) ZA200206107B (es)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PE20040945A1 (es) * 2003-02-05 2004-12-14 Warner Lambert Co Preparacion de quinazolinas substituidas
WO2006081741A1 (en) * 2005-02-05 2006-08-10 Piaoyang Sun Quinazoline compounds or their medical salts and preparation and medical usage thereof
JP5250901B2 (ja) * 2007-02-23 2013-07-31 学校法人慶應義塾 アニリノキナゾリン系化合物及びその用途
US7829574B2 (en) 2008-05-09 2010-11-09 Hutchison Medipharma Enterprises Limited Substituted quinazoline compounds and their use in treating angiogenesis-related diseases
CN105399688A (zh) * 2015-12-02 2016-03-16 西南科技大学 一种吉非替尼的制备方法

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
HU228446B1 (en) * 1996-04-12 2013-03-28 Warner Lambert Co Kinazoline derivatives as irreversible inhibitors of protein-kinase, pharmaceutical compositions containing these compounds and use thereof

Also Published As

Publication number Publication date
AU2001228478A1 (en) 2001-09-03
JP2003524006A (ja) 2003-08-12
HK1054551B (zh) 2005-06-03
WO2001062743A3 (de) 2002-03-14
GT200100025A (es) 2003-09-22
BR0108695A (pt) 2002-12-10
DE50106391D1 (de) 2005-07-07
ES2240483T3 (es) 2005-10-16
EA005213B1 (ru) 2004-12-30
PY0102711A (es) 2003-10-01
CN1171877C (zh) 2004-10-20
ATE296810T1 (de) 2005-06-15
MXPA02008301A (es) 2004-05-14
HUP0204510A2 (en) 2003-05-28
CO5280058A1 (es) 2003-05-30
DE10009267A1 (de) 2001-08-30
EA200200885A1 (ru) 2003-02-27
EP1265874A2 (de) 2002-12-18
TNSN01031A1 (en) 2005-11-10
YU62502A (sh) 2005-03-15
WO2001062743A2 (de) 2001-08-30
AR027377A1 (es) 2003-03-26
ZA200206107B (en) 2003-07-31
UY26594A1 (es) 2001-09-28
CA2401171A1 (en) 2001-08-30
IL151206A0 (en) 2003-04-10
KR20030011773A (ko) 2003-02-11
US20030050313A1 (en) 2003-03-13
EP1265874B1 (de) 2005-06-01
CN1406232A (zh) 2003-03-26
PT1265874E (pt) 2005-08-31
HUP0204510A3 (en) 2003-07-28
MY133846A (en) 2007-11-30
PA8512701A1 (es) 2002-02-21
EG23221A (en) 2004-08-31
PE20011073A1 (es) 2001-12-16
PL357774A1 (pl) 2004-07-26
HK1054551A1 (en) 2003-12-05

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