TR200100410T2 - 2-(purin-9-il)-tetrahidrofuran-3,4-diol türevleri. - Google Patents

2-(purin-9-il)-tetrahidrofuran-3,4-diol türevleri.

Info

Publication number
TR200100410T2
TR200100410T2 TR2001/00410T TR200100410T TR200100410T2 TR 200100410 T2 TR200100410 T2 TR 200100410T2 TR 2001/00410 T TR2001/00410 T TR 2001/00410T TR 200100410 T TR200100410 T TR 200100410T TR 200100410 T2 TR200100410 T2 TR 200100410T2
Authority
TR
Turkey
Prior art keywords
purin
tetrahydrofuran
diol derivatives
diol
derivatives
Prior art date
Application number
TR2001/00410T
Other languages
English (en)
Inventor
George Allen David
Chan Chuen
Peter Charles Cousins Richard
Cox Brian
Victoria Geden Joanna
Hobbs Heather
Elaine Keeling Suzanne
Judith Redgrave Alison
Thomas Davis Roper, Iv
Xie Shiping
Original Assignee
Glaxo Group Limited
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GBGB9813538.7A external-priority patent/GB9813538D0/en
Priority claimed from GBGB9909482.3A external-priority patent/GB9909482D0/en
Application filed by Glaxo Group Limited filed Critical Glaxo Group Limited
Publication of TR200100410T2 publication Critical patent/TR200100410T2/tr

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/02—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
    • C07H19/04—Heterocyclic radicals containing only nitrogen atoms as ring hetero atom
    • C07H19/16—Purine radicals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/70—Carbohydrates; Sugars; Derivatives thereof
    • A61K31/7042—Compounds having saccharide radicals and heterocyclic rings
    • A61K31/7052—Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides
    • A61K31/706—Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides containing six-membered rings with nitrogen as a ring hetero atom
    • A61K31/7064—Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides containing six-membered rings with nitrogen as a ring hetero atom containing condensed or non-condensed pyrimidines
    • A61K31/7076—Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides containing six-membered rings with nitrogen as a ring hetero atom containing condensed or non-condensed pyrimidines containing purines, e.g. adenosine, adenylic acid
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/06—Antiasthmatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators
    • A61P37/06—Immunosuppressants, e.g. drugs for graft rejection
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H1/00—Processes for the preparation of sugar derivatives
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H7/00—Compounds containing non-saccharide radicals linked to saccharide radicals by a carbon-to-carbon bond
    • C07H7/06—Heterocyclic radicals

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Molecular Biology (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Biotechnology (AREA)
  • Genetics & Genomics (AREA)
  • Biochemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Immunology (AREA)
  • Epidemiology (AREA)
  • Pulmonology (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Transplantation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)

Abstract

Bulusa göre, yeni formül (I) bilesikleri saglanmaktadir ki burada R1, R2 ve R3 tarifnamede tanimlandigi gibi olup, ayrica bunlarin hazirlanmasi için islemler, bunlari içeren formülasyonlar ve bunlarin enflamatuar hastaliklarin tedavisi için kullanimi saglanmaktadir.
TR2001/00410T 1998-06-23 1999-06-23 2-(purin-9-il)-tetrahidrofuran-3,4-diol türevleri. TR200100410T2 (tr)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GBGB9813538.7A GB9813538D0 (en) 1998-06-23 1998-06-23 Chemical compounds
GBGB9909482.3A GB9909482D0 (en) 1999-04-23 1999-04-23 2-(Purin-9-yl)-tetahydrofuran-3,4-diol derivatives

Publications (1)

Publication Number Publication Date
TR200100410T2 true TR200100410T2 (tr) 2001-06-21

Family

ID=26313917

Family Applications (1)

Application Number Title Priority Date Filing Date
TR2001/00410T TR200100410T2 (tr) 1998-06-23 1999-06-23 2-(purin-9-il)-tetrahidrofuran-3,4-diol türevleri.

Country Status (27)

Country Link
US (1) US6495528B1 (tr)
EP (1) EP1090022B1 (tr)
JP (1) JP3933870B2 (tr)
KR (1) KR20010071591A (tr)
CN (1) CN1313861A (tr)
AP (1) AP2000002016A0 (tr)
AT (1) ATE246701T1 (tr)
AU (1) AU750462B2 (tr)
BR (1) BR9911482A (tr)
CA (1) CA2335809A1 (tr)
CZ (1) CZ20004868A3 (tr)
DE (1) DE69910213T2 (tr)
EA (1) EA200001224A1 (tr)
EE (1) EE200000768A (tr)
ES (1) ES2204139T3 (tr)
HR (1) HRP20000894A2 (tr)
HU (1) HUP0103025A3 (tr)
ID (1) ID29609A (tr)
IL (1) IL140396A0 (tr)
IS (1) IS5779A (tr)
NO (1) NO20006548L (tr)
NZ (1) NZ509030A (tr)
PL (1) PL345062A1 (tr)
SK (1) SK19542000A3 (tr)
TR (1) TR200100410T2 (tr)
WO (1) WO1999067265A1 (tr)
YU (1) YU81100A (tr)

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GB0523845D0 (en) * 2005-11-23 2006-01-04 Glaxo Group Ltd Novel salts
GB0601951D0 (en) 2006-01-31 2006-03-15 Novartis Ag Organic compounds
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GB0607950D0 (en) 2006-04-21 2006-05-31 Novartis Ag Organic compounds
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Also Published As

Publication number Publication date
YU81100A (sh) 2003-10-31
JP2002518512A (ja) 2002-06-25
EP1090022B1 (en) 2003-08-06
HUP0103025A3 (en) 2002-04-29
SK19542000A3 (sk) 2001-09-11
EP1090022A1 (en) 2001-04-11
KR20010071591A (ko) 2001-07-28
BR9911482A (pt) 2002-01-22
JP3933870B2 (ja) 2007-06-20
ES2204139T3 (es) 2004-04-16
AU750462B2 (en) 2002-07-18
NO20006548D0 (no) 2000-12-21
ATE246701T1 (de) 2003-08-15
IS5779A (is) 2000-12-19
DE69910213D1 (de) 2003-09-11
DE69910213T2 (de) 2004-07-01
CZ20004868A3 (cs) 2001-08-15
ID29609A (id) 2001-09-06
IL140396A0 (en) 2002-02-10
HUP0103025A2 (hu) 2001-12-28
CN1313861A (zh) 2001-09-19
AU4774499A (en) 2000-01-10
EA200001224A1 (ru) 2001-08-27
WO1999067265A1 (en) 1999-12-29
PL345062A1 (en) 2001-11-19
CA2335809A1 (en) 1999-12-29
NO20006548L (no) 2001-02-22
HRP20000894A2 (en) 2001-12-31
EE200000768A (et) 2002-04-15
AP2000002016A0 (en) 2000-12-31
NZ509030A (en) 2003-07-25
US6495528B1 (en) 2002-12-17

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