UA57089C2 - Поліморфна форма 2-(r)-(1(r)-(3,5-біс(трифторметил)феніл)етокси)-3-(s)-(4-фтор)феніл-4-(3-(5-оксо-1h,4h-1,2,4-триазоло)метил)морфоліну як антагоніст рецептора тахікініну - Google Patents

Поліморфна форма 2-(r)-(1(r)-(3,5-біс(трифторметил)феніл)етокси)-3-(s)-(4-фтор)феніл-4-(3-(5-оксо-1h,4h-1,2,4-триазоло)метил)морфоліну як антагоніст рецептора тахікініну Download PDF

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Publication number
UA57089C2
UA57089C2 UA99127240A UA99127240A UA57089C2 UA 57089 C2 UA57089 C2 UA 57089C2 UA 99127240 A UA99127240 A UA 99127240A UA 99127240 A UA99127240 A UA 99127240A UA 57089 C2 UA57089 C2 UA 57089C2
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UA
Ukraine
Prior art keywords
phenyl
trifluoromethyl
bis
fluoro
compound
Prior art date
Application number
UA99127240A
Other languages
English (en)
Russian (ru)
Ukrainian (uk)
Inventor
Луіс Крокер
Джеймс МакКолі
Original Assignee
Мерк Енд Ко., Інк.
Мерк Энд Ко., Инк.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Мерк Енд Ко., Інк., Мерк Энд Ко., Инк. filed Critical Мерк Енд Ко., Інк.
Priority claimed from PCT/US1998/013766 external-priority patent/WO1999001444A1/en
Publication of UA57089C2 publication Critical patent/UA57089C2/uk

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  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
UA99127240A 1997-07-02 1998-01-07 Поліморфна форма 2-(r)-(1(r)-(3,5-біс(трифторметил)феніл)етокси)-3-(s)-(4-фтор)феніл-4-(3-(5-оксо-1h,4h-1,2,4-триазоло)метил)морфоліну як антагоніст рецептора тахікініну UA57089C2 (uk)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US5160097P 1997-07-02 1997-07-02
GBGB9800216.5A GB9800216D0 (en) 1998-01-07 1998-01-07 Polymorphic form of a tachykinin receptor antagonist
PCT/US1998/013766 WO1999001444A1 (en) 1997-07-02 1998-07-01 Polymorphic form of the tachykinin receptor antagonist 2-(r)-(1-(r) -(3,5-bis(trifluoromethyl) phenyl)ethoxy)-3-(s)-(4-fluoro) phenyl-4-(3-5 (-oxo-1h,4h-1,2,4,-triazolo) methylmorpholine

Publications (1)

Publication Number Publication Date
UA57089C2 true UA57089C2 (uk) 2003-06-16

Family

ID=10824888

Family Applications (1)

Application Number Title Priority Date Filing Date
UA99127240A UA57089C2 (uk) 1997-07-02 1998-01-07 Поліморфна форма 2-(r)-(1(r)-(3,5-біс(трифторметил)феніл)етокси)-3-(s)-(4-фтор)феніл-4-(3-(5-оксо-1h,4h-1,2,4-триазоло)метил)морфоліну як антагоніст рецептора тахікініну

Country Status (6)

Country Link
AR (1) AR013160A1 (sr)
CO (1) CO4940431A1 (sr)
GB (1) GB9800216D0 (sr)
MY (1) MY126509A (sr)
RS (1) RS49980B (sr)
UA (1) UA57089C2 (sr)

Also Published As

Publication number Publication date
RS49980B (sr) 2008-09-29
GB9800216D0 (en) 1998-03-04
AR013160A1 (es) 2000-12-13
MY126509A (en) 2006-10-31
CO4940431A1 (es) 2000-07-24

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