UA71938C2 - BENZYOXAZOLES AND PHENONES AS a2-ANTAGONISTS - Google Patents
BENZYOXAZOLES AND PHENONES AS a2-ANTAGONISTS Download PDFInfo
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- UA71938C2 UA71938C2 UA2001064352A UA2001064352A UA71938C2 UA 71938 C2 UA71938 C2 UA 71938C2 UA 2001064352 A UA2001064352 A UA 2001064352A UA 2001064352 A UA2001064352 A UA 2001064352A UA 71938 C2 UA71938 C2 UA 71938C2
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- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
- C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
- C07D491/04—Ortho-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
- C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D495/04—Ortho-condensed systems
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- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Medicinal Chemistry (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Biomedical Technology (AREA)
- Diabetes (AREA)
- Psychiatry (AREA)
- Endocrinology (AREA)
- Pain & Pain Management (AREA)
- Gynecology & Obstetrics (AREA)
- Emergency Medicine (AREA)
- Psychology (AREA)
- Hematology (AREA)
- Obesity (AREA)
- Hospice & Palliative Care (AREA)
- Ophthalmology & Optometry (AREA)
- Reproductive Health (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP98204358 | 1998-12-21 | ||
| PCT/EP1999/010054 WO2000037466A1 (en) | 1998-12-21 | 1999-12-14 | BENZISOXAZOLES AND PHENONES AS α2-ANTAGONISTS |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| UA71938C2 true UA71938C2 (en) | 2005-01-17 |
Family
ID=8234508
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| UA2001064352A UA71938C2 (en) | 1998-12-21 | 1999-12-14 | BENZYOXAZOLES AND PHENONES AS a2-ANTAGONISTS |
Country Status (30)
| Country | Link |
|---|---|
| US (1) | US6576640B1 (cs) |
| EP (1) | EP1140934B1 (cs) |
| JP (1) | JP4717216B2 (cs) |
| KR (2) | KR20060093139A (cs) |
| CN (1) | CN1154646C (cs) |
| AR (1) | AR021924A1 (cs) |
| AT (1) | ATE251622T1 (cs) |
| AU (1) | AU765751B2 (cs) |
| BG (1) | BG65162B1 (cs) |
| BR (1) | BR9916427A (cs) |
| CA (1) | CA2355716C (cs) |
| CZ (1) | CZ294532B6 (cs) |
| DE (1) | DE69911995T2 (cs) |
| EA (1) | EA003606B1 (cs) |
| EE (1) | EE200100329A (cs) |
| ES (1) | ES2209553T3 (cs) |
| HK (1) | HK1045686B (cs) |
| HR (1) | HRP20010444A2 (cs) |
| HU (1) | HUP0104812A3 (cs) |
| ID (1) | ID28967A (cs) |
| IL (2) | IL143830A0 (cs) |
| NO (1) | NO317892B1 (cs) |
| NZ (1) | NZ511411A (cs) |
| PL (1) | PL196958B1 (cs) |
| SK (1) | SK285560B6 (cs) |
| TR (1) | TR200101813T2 (cs) |
| TW (1) | TWI229673B (cs) |
| UA (1) | UA71938C2 (cs) |
| WO (1) | WO2000037466A1 (cs) |
| ZA (1) | ZA200105067B (cs) |
Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| RU2407744C2 (ru) * | 2008-12-19 | 2010-12-27 | Андрей Александрович Иващенко | Лиганды альфа-адреноцепторов, допаминовых, гистаминовых, имидазолиновых и серотониновых рецепторов и их применение |
Families Citing this family (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2003004501A2 (en) * | 2001-07-05 | 2003-01-16 | Pharmacia & Upjohn Company | (hetero) aryl substituted benzofurans as 5-ht ligands |
| AU2003219199A1 (en) * | 2002-04-03 | 2003-10-13 | Orion Corporation | Use of an alfa2-adrenoreceptor antagonist for cns-related diseases |
| AU2005233456A1 (en) | 2004-04-12 | 2005-10-27 | Taisho Pharmaceutical Co., Ltd. | Cyclic amine compound |
| JP2009502959A (ja) * | 2005-07-28 | 2009-01-29 | ブリストル−マイヤーズ スクイブ カンパニー | セロトニン受容体アゴニストおよびアンタゴニストとしての置換テトラヒドロ−１ｈ−ピリド［４，３，ｂ］インドール |
| CN117327065A (zh) * | 2022-06-23 | 2024-01-02 | 北京大学 | 作为多巴胺d2/3受体调节剂的咔唑类衍生物 |
Family Cites Families (14)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3419568A (en) * | 1966-12-07 | 1968-12-31 | Abbott Lab | Derivatives of 1,2,3,4-tetrahydro-5h-pyrido[4,3b]indoles |
| US3382250A (en) * | 1966-12-07 | 1968-05-07 | Abbott Lab | Aroylalkyl derivatives of 1, 2, 3, 4-tetrahydro-5h-pyrido[4, 3b]indoles |
| US3718657A (en) * | 1970-12-03 | 1973-02-27 | Abbott Lab | Certain-2-substituted-1,2,3,4-tetrahydro-beta or gamma carbolines |
| JPS4729395U (cs) * | 1971-04-26 | 1972-12-04 | ||
| AR207799A1 (es) * | 1974-04-01 | 1976-10-29 | Pfizer | Procedimiento para preparar azaciclo(3,4-a)-n-fenilindoles-2-substituidos |
| US4001263A (en) * | 1974-04-01 | 1977-01-04 | Pfizer Inc. | 5-Aryl-1,2,3,4-tetrahydro-γ-carbolines |
| US4224329A (en) * | 1979-01-23 | 1980-09-23 | Pfizer Inc. | 2-Substituted-trans-5-aryl-2,3,4,4a,5,9b-hexahydro-1H-pyrido[4,3-b]indoles |
| FR2570701B1 (fr) * | 1984-09-27 | 1987-05-22 | Synthelabo | Derives de furo(3,2-c)pyridines, leur preparation et leur application en therapeutique |
| DE3522959A1 (de) * | 1985-06-27 | 1987-01-08 | Merck Patent Gmbh | Indolderivate |
| EP0339959A3 (en) * | 1988-04-27 | 1991-03-20 | Glaxo Group Limited | Lactam derivatives |
| WO1994008040A1 (en) * | 1992-09-25 | 1994-04-14 | Synaptic Pharmaceutical Corporation | Dna encoding human alpha 1 adrenergic receptors and uses thereof |
| US5508306A (en) * | 1992-11-13 | 1996-04-16 | Synaptic Pharmaceutical Corporation | Aromatic amine derivatives |
| US5403847A (en) | 1992-11-13 | 1995-04-04 | Synaptic Pharmaceutical Corporation | Use of α1C specific compounds to treat benign prostatic hyperlasia |
| UA52681C2 (uk) * | 1997-04-08 | 2003-01-15 | Янссен Фармацевтика Н.В. | Похідні 1,2,3,4-тетрагідро-бензофуро[3,2,-c]піридину, спосіб їх одержання та фармацевтична композиція на їх основі |
-
1999
- 1999-12-14 CZ CZ20012120A patent/CZ294532B6/cs not_active IP Right Cessation
- 1999-12-14 DE DE69911995T patent/DE69911995T2/de not_active Expired - Lifetime
- 1999-12-14 CN CNB998147095A patent/CN1154646C/zh not_active Expired - Fee Related
- 1999-12-14 UA UA2001064352A patent/UA71938C2/uk unknown
- 1999-12-14 JP JP2000589537A patent/JP4717216B2/ja not_active Expired - Fee Related
- 1999-12-14 EP EP99967955A patent/EP1140934B1/en not_active Expired - Lifetime
- 1999-12-14 PL PL348421A patent/PL196958B1/pl unknown
- 1999-12-14 TR TR2001/01813T patent/TR200101813T2/xx unknown
- 1999-12-14 KR KR1020067015507A patent/KR20060093139A/ko not_active Ceased
- 1999-12-14 EE EEP200100329A patent/EE200100329A/xx unknown
- 1999-12-14 EA EA200100709A patent/EA003606B1/ru not_active IP Right Cessation
- 1999-12-14 CA CA2355716A patent/CA2355716C/en not_active Expired - Fee Related
- 1999-12-14 US US09/868,756 patent/US6576640B1/en not_active Expired - Lifetime
- 1999-12-14 ES ES99967955T patent/ES2209553T3/es not_active Expired - Lifetime
- 1999-12-14 ID IDW00200101335A patent/ID28967A/id unknown
- 1999-12-14 AT AT99967955T patent/ATE251622T1/de not_active IP Right Cessation
- 1999-12-14 IL IL14383099A patent/IL143830A0/xx active IP Right Grant
- 1999-12-14 SK SK858-2001A patent/SK285560B6/sk unknown
- 1999-12-14 NZ NZ511411A patent/NZ511411A/xx unknown
- 1999-12-14 HR HR20010444A patent/HRP20010444A2/hr not_active Application Discontinuation
- 1999-12-14 HU HU0104812A patent/HUP0104812A3/hu unknown
- 1999-12-14 KR KR1020017004946A patent/KR100657540B1/ko not_active Expired - Fee Related
- 1999-12-14 HK HK02105098.8A patent/HK1045686B/zh not_active IP Right Cessation
- 1999-12-14 WO PCT/EP1999/010054 patent/WO2000037466A1/en not_active Ceased
- 1999-12-14 AU AU24327/00A patent/AU765751B2/en not_active Ceased
- 1999-12-14 BR BR9916427-2A patent/BR9916427A/pt not_active Application Discontinuation
- 1999-12-16 TW TW088122067A patent/TWI229673B/zh not_active IP Right Cessation
- 1999-12-20 AR ARP990106577A patent/AR021924A1/es active IP Right Grant
-
2001
- 2001-05-18 BG BG105521A patent/BG65162B1/bg unknown
- 2001-06-06 NO NO20012783A patent/NO317892B1/no unknown
- 2001-06-19 IL IL143830A patent/IL143830A/en not_active IP Right Cessation
- 2001-06-20 ZA ZA200105067A patent/ZA200105067B/en unknown
Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| RU2407744C2 (ru) * | 2008-12-19 | 2010-12-27 | Андрей Александрович Иващенко | Лиганды альфа-адреноцепторов, допаминовых, гистаминовых, имидазолиновых и серотониновых рецепторов и их применение |
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