UA75828C2 - Tetrahydropyranyl cyclopentyl tetrahydropyridopyridine modulators of chemokine receptor activity, pharmaceutical composition based thereon and method for treatment of disorder or disease (variants) - Google Patents

Tetrahydropyranyl cyclopentyl tetrahydropyridopyridine modulators of chemokine receptor activity, pharmaceutical composition based thereon and method for treatment of disorder or disease (variants) Download PDF

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Publication number: UA75828C2
Authority: UA; Ukraine
Prior art keywords: compound; compound according; solution; compounds; stage
Prior art date: 2002-04-29

Application number

UA20041109704A

Other languages

English (en)

Ukrainian (uk)

Original Assignee

Merck & Co Inc

Merck Sharp & Dohme

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2002-04-29

Filing date

2003-04-25

Publication date

2006-05-15

2003-04-25 Application filed by Merck & Co Inc, Merck Sharp & Dohme filed Critical Merck & Co Inc

2006-05-15 Publication of UA75828C2 publication Critical patent/UA75828C2/uk

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Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/02—Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/02—Immunomodulators
- A61P37/04—Immunostimulants

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Chemical & Material Sciences (AREA)
Health & Medical Sciences (AREA)
Organic Chemistry (AREA)
Immunology (AREA)
Pharmacology & Pharmacy (AREA)
Public Health (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Chemical Kinetics & Catalysis (AREA)
Veterinary Medicine (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Bioinformatics & Cheminformatics (AREA)
Engineering & Computer Science (AREA)
Rheumatology (AREA)
Pain & Pain Management (AREA)
Orthopedic Medicine & Surgery (AREA)
Physical Education & Sports Medicine (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)
Plural Heterocyclic Compounds (AREA)

UA20041109704A 2002-04-29 2003-04-25 Tetrahydropyranyl cyclopentyl tetrahydropyridopyridine modulators of chemokine receptor activity, pharmaceutical composition based thereon and method for treatment of disorder or disease (variants) UA75828C2 (en)

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US37629102P	2002-04-29	2002-04-29
PCT/US2003/013042 WO2003093266A1 (en)	2002-04-29	2003-04-25	Tetrahydropyranyl cyclopentyl tetrahydropyridopyridine modulators of chemokine receptor activity

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UA75828C2 true UA75828C2 (en)	2006-05-15

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US (1)	US7786305B2 (pl)
KR (1)	KR100754760B1 (pl)
CN (1)	CN1310917C (pl)
AR (1)	AR039489A1 (pl)
AU (1)	AU2003234251A1 (pl)
BR (1)	BR0309650A (pl)
DO (1)	DOP2003000638A (pl)
EC (1)	ECSP045392A (pl)
HR (1)	HRP20041023A2 (pl)
IL (1)	IL164909A (pl)
IS (1)	IS7512A (pl)
JO (1)	JO2479B1 (pl)
MA (1)	MA27119A1 (pl)
MX (1)	MXPA04010702A (pl)
MY (1)	MY129850A (pl)
NO (1)	NO20045235L (pl)
PE (1)	PE20040598A1 (pl)
PL (1)	PL373401A1 (pl)
RU (1)	RU2285004C2 (pl)
TW (1)	TWI262077B (pl)
UA (1)	UA75828C2 (pl)
WO (1)	WO2003093266A1 (pl)

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2003
- 2003-04-22 JO JO200343A patent/JO2479B1/en active
- 2003-04-22 MY MYPI20031503A patent/MY129850A/en unknown
- 2003-04-22 TW TW092109364A patent/TWI262077B/zh not_active IP Right Cessation
- 2003-04-25 RU RU2004134604/04A patent/RU2285004C2/ru not_active IP Right Cessation
- 2003-04-25 AU AU2003234251A patent/AU2003234251A1/en not_active Abandoned
- 2003-04-25 KR KR1020047017373A patent/KR100754760B1/ko not_active Expired - Fee Related
- 2003-04-25 UA UA20041109704A patent/UA75828C2/uk unknown
- 2003-04-25 BR BR0309650-5A patent/BR0309650A/pt not_active Application Discontinuation
- 2003-04-25 HR HR20041023A patent/HRP20041023A2/hr not_active Application Discontinuation
- 2003-04-25 MX MXPA04010702A patent/MXPA04010702A/es active IP Right Grant
- 2003-04-25 PE PE2003000418A patent/PE20040598A1/es not_active Application Discontinuation
- 2003-04-25 CN CNB038150417A patent/CN1310917C/zh not_active Expired - Fee Related
- 2003-04-25 WO PCT/US2003/013042 patent/WO2003093266A1/en not_active Ceased
- 2003-04-25 PL PL03373401A patent/PL373401A1/pl not_active Application Discontinuation
- 2003-04-29 AR ARP030101487A patent/AR039489A1/es unknown
- 2003-04-29 DO DO2003000638A patent/DOP2003000638A/es unknown
2004
- 2004-05-28 US US10/856,012 patent/US7786305B2/en active Active
- 2004-10-18 IS IS7512A patent/IS7512A/is unknown
- 2004-10-27 EC EC2004005392A patent/ECSP045392A/es unknown
- 2004-10-28 IL IL164909A patent/IL164909A/en not_active IP Right Cessation
- 2004-11-17 MA MA27955A patent/MA27119A1/fr unknown
- 2004-11-29 NO NO20045235A patent/NO20045235L/no not_active Application Discontinuation

Also Published As

Publication number	Publication date
PE20040598A1 (es)	2004-10-05
JO2479B1 (en)	2009-01-20
HRP20041023A2 (en)	2005-02-28
AU2003234251A8 (en)	2003-11-17
WO2003093266A1 (en)	2003-11-13
MXPA04010702A (es)	2005-02-17
US7786305B2 (en)	2010-08-31
CN1662532A (zh)	2005-08-31
US20050101628A1 (en)	2005-05-12
RU2004134604A (ru)	2005-05-27
AR039489A1 (es)	2005-02-23
TW200307543A (en)	2003-12-16
TWI262077B (en)	2006-09-21
ECSP045392A (es)	2005-01-03
KR20050000413A (ko)	2005-01-03
IL164909A0 (en)	2005-12-18
IL164909A (en)	2010-04-15
RU2285004C2 (ru)	2006-10-10
PL373401A1 (pl)	2005-08-22
CN1310917C (zh)	2007-04-18
AU2003234251A1 (en)	2003-11-17
MY129850A (en)	2007-05-31
NO20045235L (no)	2004-11-29
BR0309650A (pt)	2005-04-26
KR100754760B1 (ko)	2007-09-04
MA27119A1 (fr)	2004-12-20
DOP2003000638A (es)	2003-11-30
HK1081967A1 (en)	2006-05-26
IS7512A (is)	2004-10-18

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