UA81111C2 - Use of a microglia inhibitor for the production of a pharmaceutical agent that inhibits immune reactions mediated by interleukin 12 (il 12) and interferon-? (variants) - Google Patents

Use of a microglia inhibitor for the production of a pharmaceutical agent that inhibits immune reactions mediated by interleukin 12 (il 12) and interferon-? (variants) Download PDF

Info

Publication number: UA81111C2
Authority: UA; Ukraine
Prior art keywords: group; ring; atom; residues; alkyl
Prior art date: 2002-02-15

Application number

UA20040907401A

Other languages

English (en)

Ukrainian (uk)

Inventor

Torsten Blume

Wolfgang Halfbrodt

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2002-02-15

Filing date

2003-01-17

Publication date

2007-12-10

2003-01-17 Application filed filed Critical

2007-12-10 Publication of UA81111C2 publication Critical patent/UA81111C2/uk

Links

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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/02—Immunomodulators
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/02—Immunomodulators
- A61P37/06—Immunosuppressants, e.g. drugs for graft rejection
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid

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Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
Pharmacology & Pharmacy (AREA)
Chemical & Material Sciences (AREA)
Veterinary Medicine (AREA)
Public Health (AREA)
Medicinal Chemistry (AREA)
General Health & Medical Sciences (AREA)
Organic Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
General Chemical & Material Sciences (AREA)
Chemical Kinetics & Catalysis (AREA)
Bioinformatics & Cheminformatics (AREA)
Engineering & Computer Science (AREA)
Immunology (AREA)
Pulmonology (AREA)
Diabetes (AREA)
Dermatology (AREA)
Rheumatology (AREA)
Epidemiology (AREA)
Hematology (AREA)
Obesity (AREA)
Transplantation (AREA)
Pain & Pain Management (AREA)
Virology (AREA)
Communicable Diseases (AREA)
Oncology (AREA)
Gastroenterology & Hepatology (AREA)
Endocrinology (AREA)
Orthopedic Medicine & Surgery (AREA)
Physical Education & Sports Medicine (AREA)
Emergency Medicine (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Plural Heterocyclic Compounds (AREA)

UA20040907401A 2002-02-15 2003-01-17 Use of a microglia inhibitor for the production of a pharmaceutical agent that inhibits immune reactions mediated by interleukin 12 (il 12) and interferon-? (variants) UA81111C2 (en)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
DE10207843A DE10207843A1 (de)	2002-02-15	2002-02-15	Mikrolia-Inhibitoren zur Unterbrechung von Interleukin 12 und IFN-gamma vermittelten Immunreaktionen
PCT/EP2003/000467 WO2003068225A1 (de)	2002-02-15	2003-01-17	Mikroglia-inhibitoren zur unterbrechung von interleukin 12 und ifn-gamma vermittelten immunreaktionen

Publications (1)

Publication Number	Publication Date
UA81111C2 true UA81111C2 (en)	2007-12-10

Family

ID=27674912

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
UA20040907401A UA81111C2 (en)	2002-02-15	2003-01-17	Use of a microglia inhibitor for the production of a pharmaceutical agent that inhibits immune reactions mediated by interleukin 12 (il 12) and interferon-? (variants)

Country Status (21)

Country	Link
EP (1)	EP1474138A1 (sr)
JP (1)	JP2005522447A (sr)
KR (1)	KR20040084909A (sr)
CN (1)	CN1756546A (sr)
AR (1)	AR039556A1 (sr)
AU (1)	AU2003245523A1 (sr)
BR (1)	BR0307706A (sr)
CA (1)	CA2475770A1 (sr)
DE (1)	DE10207843A1 (sr)
EC (1)	ECSP045297A (sr)
MX (1)	MXPA04007943A (sr)
NO (1)	NO20043840L (sr)
PE (1)	PE20030906A1 (sr)
PL (1)	PL371327A1 (sr)
RS (1)	RS71304A (sr)
RU (1)	RU2004127677A (sr)
TW (1)	TW200306823A (sr)
UA (1)	UA81111C2 (sr)
UY (1)	UY27662A1 (sr)
WO (1)	WO2003068225A1 (sr)
ZA (1)	ZA200407382B (sr)

Families Citing this family (14)

* Cited by examiner, † Cited by third party
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DE10207844A1 (de) *	2002-02-15	2003-09-04	Schering Ag	1-Phenyl-2-heteroaryl-substituierte Benzimidazolderivate, deren Verwendung zur Herstellung von Arzneimitteln sowie diese Derivate enthaltende pharmazeutische Präparate
US7820637B2 (en) *	2005-03-17	2010-10-26	Proyecto De Biomedicina Cima, S.L.	Use of 5′-methylthioadenosine (MTA) in the prevention and/or treatment of autoimmune diseases and/or transplant rejection
CA2874303C (en) *	2012-06-11	2020-10-13	Ucb Biopharma Sprl	Tnf -alpha modulating benz imidazoles
WO2016130501A1 (en)	2015-02-09	2016-08-18	Incyte Corporation	Aza-heteroaryl compounds as pi3k-gamma inhibitors
TWI744256B (zh)	2015-11-06	2021-11-01	美商英塞特公司	作為ＰＩ３Ｋ-γ抑制劑之雜環化合物
EP3390367B1 (en) *	2015-12-15	2020-09-09	The Board of Trustees of the Leland Stanford Junior University	Method for preventing and/or treating aging-associated cognitive impairment and neuroinflammation
TW201734003A (zh)	2016-01-05	2017-10-01	英塞特公司	作為ＰＩ３Ｋ-γ抑制劑之吡啶及嘧啶化合物
AR108875A1 (es)	2016-06-24	2018-10-03	Incyte Corp	COMPUESTOS HETEROCÍCLICOS COMO INHIBIDORES DE PI3K-g
AU2018350980C1 (en)	2017-10-18	2024-12-12	Incyte Corporation	Condensed imidazole derivatives substituted by tertiary hydroxy groups as pi3k-y gamma inhibitors
CR20250050A (es)	2018-09-05	2025-03-19	Incyte Corp	Formas cristalinas de un inhibidor de fosfoinositida 3–quinasa (pi3k) (divisional 2021-0165)
PT3860998T (pt)	2018-10-05	2024-04-02	Annapurna Bio Inc	Compostos e composições para o tratamento de condições associadas à atividade do recetor apj
CN112341451B (zh) *	2019-08-09	2022-06-17	成都先导药物开发股份有限公司	一种免疫调节剂
CN112341450B (zh) *	2019-08-09	2022-05-17	成都先导药物开发股份有限公司	一种免疫调节剂
CA3165339A1 (en) *	2019-12-19	2021-06-24	The United States Of America, As Represented By The Secretary, Dept. Of Health And Human Services	Cd206 modulators their use and methods for preparation

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
DE4330959A1 (de) *	1993-09-09	1995-03-16	Schering Ag	Neue Benzimidazolderivate, Verfahren zu ihrer Herstellung und ihre pharmazeutische Verwendung
NZ519326A (en) *	2000-01-14	2005-02-25	Schering Ag	1,2-diarylbenzimidazoles for treating diseases that are associated with a microglia activation
DE10134775A1 (de) *	2001-07-06	2003-01-30	Schering Ag	1-Alkyl-2.aryl-benzimidazolderivate, deren Verwendung zur Herstellung von Arzneimitteln sowie diese Derivate enthaltende pharmazeutische Präparate
DE10135050A1 (de) *	2001-07-09	2003-02-06	Schering Ag	1-Ary1-2-N-, S- oder O-substituierte Benzimidazolderivate, deren Verwendung zur Herstellung von Arzneimitteln sowie diese Derivate enthaltende pharmazeutische Präparate

2002
- 2002-02-15 DE DE10207843A patent/DE10207843A1/de not_active Ceased
2003
- 2003-01-17 RS YU71304A patent/RS71304A/sr unknown
- 2003-01-17 PL PL03371327A patent/PL371327A1/xx not_active Application Discontinuation
- 2003-01-17 UA UA20040907401A patent/UA81111C2/uk unknown
- 2003-01-17 JP JP2003567407A patent/JP2005522447A/ja active Pending
- 2003-01-17 RU RU2004127677/15A patent/RU2004127677A/ru unknown
- 2003-01-17 EP EP03739380A patent/EP1474138A1/de not_active Withdrawn
- 2003-01-17 CN CNA038039923A patent/CN1756546A/zh active Pending
- 2003-01-17 MX MXPA04007943A patent/MXPA04007943A/es unknown
- 2003-01-17 CA CA002475770A patent/CA2475770A1/en not_active Abandoned
- 2003-01-17 KR KR10-2004-7012557A patent/KR20040084909A/ko not_active Ceased
- 2003-01-17 BR BR0307706-3A patent/BR0307706A/pt not_active IP Right Cessation
- 2003-01-17 WO PCT/EP2003/000467 patent/WO2003068225A1/de not_active Ceased
- 2003-01-17 AU AU2003245523A patent/AU2003245523A1/en not_active Abandoned
- 2003-02-03 PE PE2003000119A patent/PE20030906A1/es not_active Application Discontinuation
- 2003-02-11 UY UY27662A patent/UY27662A1/es not_active Application Discontinuation
- 2003-02-12 AR ARP030100436A patent/AR039556A1/es unknown
- 2003-02-14 TW TW092103072A patent/TW200306823A/zh unknown
2004
- 2004-09-14 EC EC2004005297A patent/ECSP045297A/es unknown
- 2004-09-14 ZA ZA200407382A patent/ZA200407382B/en unknown
- 2004-09-14 NO NO20043840A patent/NO20043840L/no not_active Application Discontinuation

Also Published As

Publication number	Publication date
TW200306823A (en)	2003-12-01
JP2005522447A (ja)	2005-07-28
BR0307706A (pt)	2005-01-11
PE20030906A1 (es)	2004-01-17
MXPA04007943A (es)	2004-11-26
ZA200407382B (en)	2005-09-14
WO2003068225A1 (de)	2003-08-21
KR20040084909A (ko)	2004-10-06
AU2003245523A1 (en)	2003-09-04
CN1756546A (zh)	2006-04-05
RS71304A (sr)	2006-10-27
NO20043840L (no)	2004-11-12
AR039556A1 (es)	2005-02-23
CA2475770A1 (en)	2003-08-21
DE10207843A1 (de)	2003-09-04
UY27662A1 (es)	2003-09-30
PL371327A1 (en)	2005-06-13
RU2004127677A (ru)	2005-06-10
EP1474138A1 (de)	2004-11-10
ECSP045297A (es)	2004-10-26

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