UA81111C2 - Use of a microglia inhibitor for the production of a pharmaceutical agent that inhibits immune reactions mediated by interleukin 12 (il 12) and interferon-? (variants) - Google Patents

Use of a microglia inhibitor for the production of a pharmaceutical agent that inhibits immune reactions mediated by interleukin 12 (il 12) and interferon-? (variants) Download PDF

Info

Publication number: UA81111C2
Authority: UA; Ukraine
Prior art keywords: group; ring; atom; residues; alkyl
Prior art date: 2002-02-15

Application number

UA20040907401A

Other languages

English (en)

Ukrainian (uk)

Inventor

Torsten Blume

Wolfgang Halfbrodt

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2002-02-15

Filing date

2003-01-17

Publication date

2007-12-10

2003-01-17 Application filed filed Critical

2007-12-10 Publication of UA81111C2 publication Critical patent/UA81111C2/uk

Links

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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/02—Immunomodulators
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/02—Immunomodulators
- A61P37/06—Immunosuppressants, e.g. drugs for graft rejection
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid

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Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
Pharmacology & Pharmacy (AREA)
General Health & Medical Sciences (AREA)
Animal Behavior & Ethology (AREA)
Veterinary Medicine (AREA)
Chemical & Material Sciences (AREA)
Public Health (AREA)
Medicinal Chemistry (AREA)
Chemical Kinetics & Catalysis (AREA)
Organic Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
General Chemical & Material Sciences (AREA)
Bioinformatics & Cheminformatics (AREA)
Engineering & Computer Science (AREA)
Immunology (AREA)
Pulmonology (AREA)
Diabetes (AREA)
Dermatology (AREA)
Hematology (AREA)
Epidemiology (AREA)
Rheumatology (AREA)
Pain & Pain Management (AREA)
Gastroenterology & Hepatology (AREA)
Endocrinology (AREA)
Obesity (AREA)
Oncology (AREA)
Communicable Diseases (AREA)
Virology (AREA)
Emergency Medicine (AREA)
Orthopedic Medicine & Surgery (AREA)
Physical Education & Sports Medicine (AREA)
Transplantation (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Plural Heterocyclic Compounds (AREA)

UA20040907401A 2002-02-15 2003-01-17 Use of a microglia inhibitor for the production of a pharmaceutical agent that inhibits immune reactions mediated by interleukin 12 (il 12) and interferon-? (variants) UA81111C2 (en)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
DE10207843A DE10207843A1 (de)	2002-02-15	2002-02-15	Mikrolia-Inhibitoren zur Unterbrechung von Interleukin 12 und IFN-gamma vermittelten Immunreaktionen
PCT/EP2003/000467 WO2003068225A1 (de)	2002-02-15	2003-01-17	Mikroglia-inhibitoren zur unterbrechung von interleukin 12 und ifn-gamma vermittelten immunreaktionen

Publications (1)

Publication Number	Publication Date
UA81111C2 true UA81111C2 (en)	2007-12-10

Family

ID=27674912

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
UA20040907401A UA81111C2 (en)	2002-02-15	2003-01-17	Use of a microglia inhibitor for the production of a pharmaceutical agent that inhibits immune reactions mediated by interleukin 12 (il 12) and interferon-? (variants)

Country Status (21)

Country	Link
EP (1)	EP1474138A1 (sr)
JP (1)	JP2005522447A (sr)
KR (1)	KR20040084909A (sr)
CN (1)	CN1756546A (sr)
AR (1)	AR039556A1 (sr)
AU (1)	AU2003245523A1 (sr)
BR (1)	BR0307706A (sr)
CA (1)	CA2475770A1 (sr)
DE (1)	DE10207843A1 (sr)
EC (1)	ECSP045297A (sr)
MX (1)	MXPA04007943A (sr)
NO (1)	NO20043840L (sr)
PE (1)	PE20030906A1 (sr)
PL (1)	PL371327A1 (sr)
RS (1)	RS71304A (sr)
RU (1)	RU2004127677A (sr)
TW (1)	TW200306823A (sr)
UA (1)	UA81111C2 (sr)
UY (1)	UY27662A1 (sr)
WO (1)	WO2003068225A1 (sr)
ZA (1)	ZA200407382B (sr)

Families Citing this family (14)

* Cited by examiner, † Cited by third party
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DE10207844A1 (de) *	2002-02-15	2003-09-04	Schering Ag	1-Phenyl-2-heteroaryl-substituierte Benzimidazolderivate, deren Verwendung zur Herstellung von Arzneimitteln sowie diese Derivate enthaltende pharmazeutische Präparate
HRP20090646T1 (hr) *	2005-03-17	2010-01-31	Proyecto De Biomedicina Cima	Uporaba 5'-metiltioadenozina (mta) kod prevencije i/ili liječenja autoimunih bolesti i/ili odbacivanje transplantata
CA2874303C (en) *	2012-06-11	2020-10-13	Ucb Biopharma Sprl	Tnf -alpha modulating benz imidazoles
WO2016130501A1 (en)	2015-02-09	2016-08-18	Incyte Corporation	Aza-heteroaryl compounds as pi3k-gamma inhibitors
RS63359B1 (sr)	2015-11-06	2022-07-29	Incyte Corp	Heterociklična jedinjenja kao inhibitori pi3k-gama
ES2830447T3 (es) *	2015-12-15	2021-06-03	Univ Leland Stanford Junior	Método para la prevención y/o el tratamiento del deterioro cognitivo asociado al envejecimiento y la neuroinflamación
ES2995198T3 (en)	2016-01-05	2025-02-07	Incyte Corp	Pyridine compounds as pi3k-gamma inhibitors
TW201803871A (zh)	2016-06-24	2018-02-01	英塞特公司	作為ＰＩ３Ｋ-γ抑制劑之雜環化合物
KR102717072B1 (ko)	2017-10-18	2024-10-15	인사이트 코포레이션	Pi3k-감마 저해제로서의 3차 하이드록시기로 치환된 축합된 이미다졸 유도체
CR20250050A (es)	2018-09-05	2025-03-19	Incyte Corp	Formas cristalinas de un inhibidor de fosfoinositida 3–quinasa (pi3k) (divisional 2021-0165)
LT3860998T (lt)	2018-10-05	2024-06-25	Annapurna Bio Inc.	Junginiai ir kompozicijos, skirti gydyti būkles, susijusias su apj receptoriaus aktyvumu
CN112341450B (zh) *	2019-08-09	2022-05-17	成都先导药物开发股份有限公司	一种免疫调节剂
CN112341451B (zh) *	2019-08-09	2022-06-17	成都先导药物开发股份有限公司	一种免疫调节剂
US20230056497A1 (en) *	2019-12-19	2023-02-23	The United States Of America, As Represented By The Secretary, Dept. Of Health And Human Services	CD206 Modulators Their Use and Methods for Preparation

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
DE4330959A1 (de) *	1993-09-09	1995-03-16	Schering Ag	Neue Benzimidazolderivate, Verfahren zu ihrer Herstellung und ihre pharmazeutische Verwendung
IL150150A0 (en) *	2000-01-14	2002-12-01	Schering Ag	1,2-diaryl benzimidazoles for treating illnesses associated with a microglia activation
DE10134775A1 (de) *	2001-07-06	2003-01-30	Schering Ag	1-Alkyl-2.aryl-benzimidazolderivate, deren Verwendung zur Herstellung von Arzneimitteln sowie diese Derivate enthaltende pharmazeutische Präparate
DE10135050A1 (de) *	2001-07-09	2003-02-06	Schering Ag	1-Ary1-2-N-, S- oder O-substituierte Benzimidazolderivate, deren Verwendung zur Herstellung von Arzneimitteln sowie diese Derivate enthaltende pharmazeutische Präparate

2002
- 2002-02-15 DE DE10207843A patent/DE10207843A1/de not_active Ceased
2003
- 2003-01-17 RU RU2004127677/15A patent/RU2004127677A/ru unknown
- 2003-01-17 JP JP2003567407A patent/JP2005522447A/ja active Pending
- 2003-01-17 WO PCT/EP2003/000467 patent/WO2003068225A1/de not_active Ceased
- 2003-01-17 AU AU2003245523A patent/AU2003245523A1/en not_active Abandoned
- 2003-01-17 PL PL03371327A patent/PL371327A1/xx not_active Application Discontinuation
- 2003-01-17 KR KR10-2004-7012557A patent/KR20040084909A/ko not_active Ceased
- 2003-01-17 RS YU71304A patent/RS71304A/sr unknown
- 2003-01-17 EP EP03739380A patent/EP1474138A1/de not_active Withdrawn
- 2003-01-17 CN CNA038039923A patent/CN1756546A/zh active Pending
- 2003-01-17 BR BR0307706-3A patent/BR0307706A/pt not_active IP Right Cessation
- 2003-01-17 UA UA20040907401A patent/UA81111C2/uk unknown
- 2003-01-17 CA CA002475770A patent/CA2475770A1/en not_active Abandoned
- 2003-01-17 MX MXPA04007943A patent/MXPA04007943A/es unknown
- 2003-02-03 PE PE2003000119A patent/PE20030906A1/es not_active Application Discontinuation
- 2003-02-11 UY UY27662A patent/UY27662A1/es not_active Application Discontinuation
- 2003-02-12 AR ARP030100436A patent/AR039556A1/es unknown
- 2003-02-14 TW TW092103072A patent/TW200306823A/zh unknown
2004
- 2004-09-14 NO NO20043840A patent/NO20043840L/no not_active Application Discontinuation
- 2004-09-14 ZA ZA200407382A patent/ZA200407382B/en unknown
- 2004-09-14 EC EC2004005297A patent/ECSP045297A/es unknown

Also Published As

Publication number	Publication date
ECSP045297A (es)	2004-10-26
AR039556A1 (es)	2005-02-23
UY27662A1 (es)	2003-09-30
JP2005522447A (ja)	2005-07-28
AU2003245523A1 (en)	2003-09-04
ZA200407382B (en)	2005-09-14
CN1756546A (zh)	2006-04-05
NO20043840L (no)	2004-11-12
RU2004127677A (ru)	2005-06-10
PL371327A1 (en)	2005-06-13
BR0307706A (pt)	2005-01-11
EP1474138A1 (de)	2004-11-10
KR20040084909A (ko)	2004-10-06
PE20030906A1 (es)	2004-01-17
TW200306823A (en)	2003-12-01
DE10207843A1 (de)	2003-09-04
WO2003068225A1 (de)	2003-08-21
MXPA04007943A (es)	2004-11-26
CA2475770A1 (en)	2003-08-21
RS71304A (sr)	2006-10-27

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