UA85097C2 - Бициклические гетеросоединения как ингибиторы вич-интегразы - Google Patents
Бициклические гетеросоединения как ингибиторы вич-интегразыInfo
- Publication number
- UA85097C2 UA85097C2 UAA200613941A UAA200613941A UA85097C2 UA 85097 C2 UA85097 C2 UA 85097C2 UA A200613941 A UAA200613941 A UA A200613941A UA A200613941 A UAA200613941 A UA A200613941A UA 85097 C2 UA85097 C2 UA 85097C2
- Authority
- UA
- Ukraine
- Prior art keywords
- hiv integrase
- integrase inhibitors
- bicyclic heterocycles
- hiv
- treating
- Prior art date
Links
- 229940099797 HIV integrase inhibitor Drugs 0.000 title 1
- 125000002618 bicyclic heterocycle group Chemical group 0.000 title 1
- 239000003084 hiv integrase inhibitor Substances 0.000 title 1
- 208000030507 AIDS Diseases 0.000 abstract 1
- 108010002459 HIV Integrase Proteins 0.000 abstract 1
- 150000001875 compounds Chemical class 0.000 abstract 1
- -1 cyclic bicyclic pyrimidinone compounds Chemical class 0.000 abstract 1
- 208000015181 infectious disease Diseases 0.000 abstract 1
- 230000010354 integration Effects 0.000 abstract 1
- 239000008194 pharmaceutical composition Substances 0.000 abstract 1
- 230000003612 virological effect Effects 0.000 abstract 1
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
Изобретением охватывается ряд бициклческих пиримидиноновых соединений в соответствии с формулой І, которые ингибируют ВИЧ-интегразу и предотвращают интегрирование вирусов в ДНК человека. Эта способность предложенных соединений делает их полезными в леченииВИЧ-инфекции и СПИДА.Изобретением охватываются также фармацевтические составы и процессы для лечения ВИЧ-инфицированных пациентов.I
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US57551304P | 2004-05-28 | 2004-05-28 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| UA85097C2 true UA85097C2 (ru) | 2008-12-25 |
Family
ID=38185422
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| UAA200613941A UA85097C2 (ru) | 2004-05-28 | 2005-05-12 | Бициклические гетеросоединения как ингибиторы вич-интегразы |
Country Status (3)
| Country | Link |
|---|---|
| CN (1) | CN1989141B (ru) |
| UA (1) | UA85097C2 (ru) |
| ZA (1) | ZA200609935B (ru) |
Families Citing this family (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN112028816B (zh) * | 2020-09-11 | 2022-10-14 | 江阴迈康升华医药科技有限公司 | 一种取代异吲哚啉的合成方法 |
-
2005
- 2005-05-12 UA UAA200613941A patent/UA85097C2/ru unknown
- 2005-05-12 CN CN2005800253288A patent/CN1989141B/zh not_active Expired - Fee Related
-
2006
- 2006-11-28 ZA ZA200609935A patent/ZA200609935B/xx unknown
Also Published As
| Publication number | Publication date |
|---|---|
| CN1989141B (zh) | 2010-06-16 |
| CN1989141A (zh) | 2007-06-27 |
| ZA200609935B (en) | 2008-06-25 |
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