YU6196A - Transdermalna flasterska formulacija - Google Patents

Transdermalna flasterska formulacija

Info

Publication number
YU6196A
YU6196A YU6196A YU6196A YU6196A YU 6196 A YU6196 A YU 6196A YU 6196 A YU6196 A YU 6196A YU 6196 A YU6196 A YU 6196A YU 6196 A YU6196 A YU 6196A
Authority
YU
Yugoslavia
Prior art keywords
transdermal
formulation
present
provides
butylthio
Prior art date
Application number
YU6196A
Other languages
English (en)
Inventor
Franklin Bymaster
Harlan Shannon
Lisa Shipley
Kirti Valia
Original Assignee
Eli Lilly And Company
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Eli Lilly And Company filed Critical Eli Lilly And Company
Publication of YU6196A publication Critical patent/YU6196A/sh

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/70—Web, sheet or filament bases ; Films; Fibres of the matrix type containing drug
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/70—Web, sheet or filament bases ; Films; Fibres of the matrix type containing drug
    • A61K9/7023—Transdermal patches and similar drug-containing composite devices, e.g. cataplasms
    • A61K9/703—Transdermal patches and similar drug-containing composite devices, e.g. cataplasms characterised by shape or structure; Details concerning release liner or backing; Refillable patches; User-activated patches
    • A61K9/7038—Transdermal patches of the drug-in-adhesive type, i.e. comprising drug in the skin-adhesive layer
    • A61K9/7046—Transdermal patches of the drug-in-adhesive type, i.e. comprising drug in the skin-adhesive layer the adhesive comprising macromolecular compounds
    • A61K9/7053—Transdermal patches of the drug-in-adhesive type, i.e. comprising drug in the skin-adhesive layer the adhesive comprising macromolecular compounds obtained by reactions only involving carbon to carbon unsaturated bonds, e.g. polyvinyl, polyisobutylene, polystyrene
    • A61K9/7061—Polyacrylates
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61F—FILTERS IMPLANTABLE INTO BLOOD VESSELS; PROSTHESES; DEVICES PROVIDING PATENCY TO, OR PREVENTING COLLAPSING OF, TUBULAR STRUCTURES OF THE BODY, e.g. STENTS; ORTHOPAEDIC, NURSING OR CONTRACEPTIVE DEVICES; FOMENTATION; TREATMENT OR PROTECTION OF EYES OR EARS; BANDAGES, DRESSINGS OR ABSORBENT PADS; FIRST-AID KITS
    • A61F13/00—Bandages or dressings; Absorbent pads
    • A61F13/02—Adhesive bandages or dressings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/439—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom the ring forming part of a bridged ring system, e.g. quinuclidine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/70—Web, sheet or filament bases ; Films; Fibres of the matrix type containing drug
    • A61K9/7023—Transdermal patches and similar drug-containing composite devices, e.g. cataplasms
    • A61K9/703—Transdermal patches and similar drug-containing composite devices, e.g. cataplasms characterised by shape or structure; Details concerning release liner or backing; Refillable patches; User-activated patches
    • A61K9/7084—Transdermal patches having a drug layer or reservoir, and one or more separate drug-free skin-adhesive layers, e.g. between drug reservoir and skin, or surrounding the drug reservoir; Liquid-filled reservoir patches
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia

Landscapes

  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Dermatology (AREA)
  • Epidemiology (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pain & Pain Management (AREA)
  • Hospice & Palliative Care (AREA)
  • Psychiatry (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Vascular Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)

Abstract

TRANSDERMALNA FLASTERSKA FORMULACIJA - Ovaj pronalazak obezbedjuje nove transdermalne formulacije koje sadrže farmaceutski aktivno jedinjenje 3-/4-(butiltio)-1,2,5-tiadiazol-3-il/-1-azabiciklo/2.2.2/oktana koje ima muskarinsku aktivnost koja je indikativna za lečenje Alzhajmerove bolesti, stanja sa jakim bolovima i glaukoma. Sadašnji pronalazak obezbedjuje metod za lečenje Alzhajmerove bolesti i, stanja sa jakim bolovima sa malo nuz efekata koji su obično povezani sa muskarinskim antagonistima kao što je 3-/4-(butiltio)-1,2,5-tiadiazol-3-il/-1-azabiciklo/2.2.2/oktan. Transdermalna formulacija ovoga pronalaska obezbedjuje konzistentnu dozu aktivnog sastojka, postiže održavanje plazmatične koncentracije farmaceutski aktivnog agensa, i povećava pokornost pacijenta.
YU6196A 1995-02-17 1996-02-01 Transdermalna flasterska formulacija YU6196A (sh)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US39044595A 1995-02-17 1995-02-17
US48101695A 1995-06-07 1995-06-07

Publications (1)

Publication Number Publication Date
YU6196A true YU6196A (sh) 1998-09-18

Family

ID=27013141

Family Applications (1)

Application Number Title Priority Date Filing Date
YU6196A YU6196A (sh) 1995-02-17 1996-02-01 Transdermalna flasterska formulacija

Country Status (22)

Country Link
US (1) US5858393A (sh)
EP (1) EP0727208B1 (sh)
JP (1) JPH11505513A (sh)
KR (1) KR19980702239A (sh)
CN (1) CN1181007A (sh)
AR (1) AR002027A1 (sh)
AU (1) AU700023B2 (sh)
BR (1) BR9607722A (sh)
CA (1) CA2212874A1 (sh)
CO (1) CO4700408A1 (sh)
CZ (1) CZ255097A3 (sh)
DE (1) DE69614419T2 (sh)
ES (1) ES2159683T3 (sh)
FI (1) FI973362A7 (sh)
HU (1) HUP9802070A3 (sh)
IL (1) IL116997A0 (sh)
NO (1) NO973715D0 (sh)
NZ (1) NZ302147A (sh)
PE (1) PE17897A1 (sh)
TR (1) TR199700799T1 (sh)
WO (1) WO1996025154A1 (sh)
YU (1) YU6196A (sh)

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6528529B1 (en) 1998-03-31 2003-03-04 Acadia Pharmaceuticals Inc. Compounds with activity on muscarinic receptors
US6417227B1 (en) 1999-04-28 2002-07-09 Cg And Associates Methods of delivery of cetyl myristoleate
AU1753301A (en) * 1999-10-28 2001-05-08 3M Innovative Properties Company Transdermal drug delivery devices
EP2258357A3 (en) 2005-08-26 2011-04-06 Braincells, Inc. Neurogenesis with acetylcholinesterase inhibitor
EP2275096A3 (en) 2005-08-26 2011-07-13 Braincells, Inc. Neurogenesis via modulation of the muscarinic receptors
US20070264130A1 (en) * 2006-01-27 2007-11-15 Phluid, Inc. Infusion Pumps and Methods for Use
US8986253B2 (en) * 2008-01-25 2015-03-24 Tandem Diabetes Care, Inc. Two chamber pumps and related methods
EP2276525A4 (en) * 2008-05-19 2012-04-04 Tandem Diabetes Care Inc REMOVABLE PUMP CONTAINER AND RELATED METHOD
US7943187B2 (en) * 2008-05-23 2011-05-17 Bakr Rabie Paeoniflorin preparations and uses thereof for fat reduction
EP2363116A1 (en) 2008-06-25 2011-09-07 US Worldmeds LLC Sustained-release formulations comprising lofexidine for oral delivery
US8408421B2 (en) 2008-09-16 2013-04-02 Tandem Diabetes Care, Inc. Flow regulating stopcocks and related methods
EP2334234A4 (en) * 2008-09-19 2013-03-20 Tandem Diabetes Care Inc DEVICE FOR MEASURING THE CONCENTRATION OF A SOLVED SUBSTANCE AND CORRESPONDING METHOD
US8758323B2 (en) * 2009-07-30 2014-06-24 Tandem Diabetes Care, Inc. Infusion pump system with disposable cartridge having pressure venting and pressure feedback
US9180242B2 (en) 2012-05-17 2015-11-10 Tandem Diabetes Care, Inc. Methods and devices for multiple fluid transfer
US9173998B2 (en) 2013-03-14 2015-11-03 Tandem Diabetes Care, Inc. System and method for detecting occlusions in an infusion pump
EP4415785A4 (en) 2021-10-12 2025-09-03 Tandem Diabetes Care Inc SYSTEMS AND METHODS FOR DELAYED MEAL BOLUSE IN AUTOMATED INSULIN DELIVERY

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4316893A (en) * 1975-06-19 1982-02-23 Nelson Research & Development Co. Vehicle composition containing 1-substituted azacycloalkan-2-ones
IT1233860B (it) * 1988-02-08 1992-04-21 Isf Spa Derivati del peridroazacicloalca (1,2-a) imidazolo ad attivita' nootropa
DK198590D0 (da) * 1990-08-21 1990-08-21 Novo Nordisk As Heterocykliske forbindelser, deres fremstilling og anvendelse
US5238933A (en) * 1991-10-28 1993-08-24 Sri International Skin permeation enhancer compositions
FI960748L (fi) * 1993-08-19 1996-04-18 Novo Nordisk As Antipsykoottinen menetelmä

Also Published As

Publication number Publication date
BR9607722A (pt) 1998-07-14
HUP9802070A2 (hu) 1999-02-01
AR002027A1 (es) 1998-01-07
FI973362L (fi) 1997-08-15
PE17897A1 (es) 1997-06-12
TR199700799T1 (xx) 1998-02-21
NO973715L (no) 1997-08-12
NO973715D0 (no) 1997-08-12
MX9706143A (es) 1997-11-29
IL116997A0 (en) 1996-06-18
JPH11505513A (ja) 1999-05-21
CN1181007A (zh) 1998-05-06
ES2159683T3 (es) 2001-10-16
DE69614419T2 (de) 2002-05-23
DE69614419D1 (de) 2001-09-20
NZ302147A (en) 1998-10-28
EP0727208A1 (en) 1996-08-21
FI973362A0 (fi) 1997-08-15
KR19980702239A (ko) 1998-07-15
CO4700408A1 (es) 1998-12-29
HUP9802070A3 (en) 2000-09-28
EP0727208B1 (en) 2001-08-16
WO1996025154A1 (en) 1996-08-22
CZ255097A3 (en) 1997-12-17
CA2212874A1 (en) 1996-08-22
AU4774296A (en) 1996-09-04
FI973362A7 (fi) 1997-08-15
AU700023B2 (en) 1998-12-17
US5858393A (en) 1999-01-12

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