YU63482A - Process for obtaining new antagonists of the antidiuretic and/or vasopressoric activity of the arginine vasopressin - Google Patents

Process for obtaining new antagonists of the antidiuretic and/or vasopressoric activity of the arginine vasopressin

Info

Publication number: YU63482A
Authority: YU; Yugoslavia
Prior art keywords: vasopressoric; antidiuretic; activity; obtaining new; arginine vasopressin
Prior art date: 1981-03-24

Application number

YU00634/82A

Other languages

English (en)

Inventor

M Manning

W Sawyer

Original Assignee

Ohio Med College

Univ Columbia

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1981-03-24

Filing date

1982-03-24

Publication date

1985-10-31

1981-03-24 Priority claimed from US06/247,008 external-priority patent/US4367225A/en

1982-03-24 Application filed by Ohio Med College, Univ Columbia filed Critical Ohio Med College

1985-10-31 Publication of YU63482A publication Critical patent/YU63482A/xx

Links

101800001144 Arg-vasopressin Proteins 0.000 title 1
102100026383 Vasopressin-neurophysin 2-copeptin Human genes 0.000 title 1
239000005557 antagonist Substances 0.000 title 1
230000002686 anti-diuretic effect Effects 0.000 title 1
229940124538 antidiuretic agent Drugs 0.000 title 1
239000003160 antidiuretic agent Substances 0.000 title 1
KBZOIRJILGZLEJ-LGYYRGKSSA-N argipressin Chemical compound C([C@H]1C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CSSC[C@@H](C(N[C@@H](CC=2C=CC(O)=CC=2)C(=O)N1)=O)N)C(=O)N1[C@@H](CCC1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)NCC(N)=O)C1=CC=CC=C1 KBZOIRJILGZLEJ-LGYYRGKSSA-N 0.000 title 1
230000000694 effects Effects 0.000 title 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K7/00—Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
- C07K7/04—Linear peptides containing only normal peptide links
- C07K7/16—Oxytocins; Vasopressins; Related peptides
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y10—TECHNICAL SUBJECTS COVERED BY FORMER USPC
- Y10S—TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y10S930/00—Peptide or protein sequence
- Y10S930/01—Peptide or protein sequence
- Y10S930/15—Oxytocin or vasopressin; related peptides

Landscapes

Chemical & Material Sciences (AREA)
Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
Organic Chemistry (AREA)
General Health & Medical Sciences (AREA)
Medicinal Chemistry (AREA)
Proteomics, Peptides & Aminoacids (AREA)
Biophysics (AREA)
Genetics & Genomics (AREA)
Molecular Biology (AREA)
Biochemistry (AREA)
Immunology (AREA)
Bioinformatics & Cheminformatics (AREA)
Engineering & Computer Science (AREA)
Pharmacology & Pharmacy (AREA)
Epidemiology (AREA)
Animal Behavior & Ethology (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Peptides Or Proteins (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)

YU00634/82A 1981-03-24 1982-03-24 Process for obtaining new antagonists of the antidiuretic and/or vasopressoric activity of the arginine vasopressin YU63482A (en)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
US06/247,008 US4367225A (en)	1981-03-24	1981-03-24	Novel antagonists of the antidiuretic and/or vasopressor action of arginine vasopressin
US06/322,071 US4399125A (en)	1981-03-24	1981-11-16	Novel antagonists of the antidiuretic action of arginine vasopressin

Publications (1)

Publication Number	Publication Date
YU63482A true YU63482A (en)	1985-10-31

Family

ID=26938391

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
YU00634/82A YU63482A (en)	1981-03-24	1982-03-24	Process for obtaining new antagonists of the antidiuretic and/or vasopressoric activity of the arginine vasopressin

Country Status (21)

Country	Link
US (1)	US4399125A (fr)
EP (1)	EP0061356B1 (fr)
KR (1)	KR880000758B1 (fr)
AU (1)	AU546865B2 (fr)
BG (1)	BG38487A3 (fr)
CA (1)	CA1185235A (fr)
DD (2)	DD202695A5 (fr)
DE (1)	DE3264734D1 (fr)
DK (1)	DK130182A (fr)
ES (2)	ES8604264A1 (fr)
FI (1)	FI77047C (fr)
HU (1)	HU189127B (fr)
IE (1)	IE52624B1 (fr)
IL (1)	IL65211A (fr)
NO (1)	NO162024C (fr)
NZ (1)	NZ199908A (fr)
PH (1)	PH19237A (fr)
PT (1)	PT74615B (fr)
RO (1)	RO84361B (fr)
YU (1)	YU63482A (fr)
ZW (1)	ZW4882A1 (fr)

Families Citing this family (26)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US4491577A (en) *	1981-11-16	1985-01-01	The Medical College Of Ohio	Antagonists of the antidiuretic action of arginine vasopressin
DK153883A (da) *	1982-04-20	1983-10-21	Ceskoslovenska Akademie Ved	Vasopressin-analoge
US4469679A (en) *	1983-02-16	1984-09-04	Smithkline Beckman Corporation	Octapeptide vasopressin antagonists
US4587045A (en) *	1983-02-16	1986-05-06	Smithkline Beckman Corporation	Intermediates for preparing octapeptide vasopressin antagonists
US4483794A (en) *	1983-05-10	1984-11-20	Ceskoslovenska Akademie Ved	Analogs of neurohypophysial hormones
CA1238314A (fr) *	1983-09-22	1988-06-21	James F. Callahan	Procede de preparation d'heptapeptides inhibiteurs de la vasopressine
US4551445A (en) *	1983-10-14	1985-11-05	The Medical College Of Ohio	Derivatives of arginine vasopressin antagonists
US4649130A (en) *	1984-01-26	1987-03-10	Medical College Of Ohio	Novel derivatives of arginine vasopressin antagonists
US4714696A (en) *	1984-01-26	1987-12-22	Medical College Of Ohio	Novel derivatives of arginine vasopressin antagonists
US4481194A (en) *	1984-03-07	1984-11-06	Smithkline Beckman Corporation	Des-proline-des-glycine vasopressin antagonists
US4481193A (en) *	1984-03-07	1984-11-06	Smithkline Beckman Corporation	Des-proline vasopressin antagonists
CA1249397A (fr) *	1984-03-07	1989-01-24	Fadia E. Ali	Procede de preparation de la des-proline inhibitrice de la vasopressine
US4684716A (en) *	1984-12-14	1987-08-04	Smithkline Beckman Corporation	Polypeptide intermediates
US4597901A (en) *	1984-12-14	1986-07-01	Smithkline Beckman Corporation	β-indolylalanyl or β-indolylglycinyl vasopressin antagonists
US4719199A (en) *	1984-12-14	1988-01-12	Smithkline Beckman Corporation	Diuretic compositions and methods of producing diuresis
US4624943A (en) *	1985-03-20	1986-11-25	Smithkline Beckman Corporation	Aromatic basic-tailed vasopressin antagonists
EP0247033A1 (fr) *	1985-10-25	1987-12-02	Gibson-Stephens Neuropharmaceuticals, Inc.	Antagonistes de l'oxytocine a conformation limitee presentant des activites biologiques prolongees
PT84342B (pt) *	1986-02-25	1989-09-14	Smithkline Beecham Corp	Processo de preparacao de compostos de vasopressina
US4762820A (en) *	1986-03-03	1988-08-09	Trustees Of Boston University	Therapeutic treatment for congestive heart failure
EP0300036A4 (fr) *	1987-01-30	1989-06-14	Biomed Res Consultants Ltd	Compositions pharmaceutiques a base de vasopressine.
US5055448A (en) *	1987-06-25	1991-10-08	Medical College Of Ohio	Linear derivatives of arginine vasopressin antagonists
AT398766B (de) *	1988-05-26	1995-01-25	Gebro Broschek Gmbh	Verfahren zur intramolekularen oxidation von zwei -sh gruppen in einer peptidverbindung zu einer disulfidbrücke
US5070187A (en) *	1989-11-03	1991-12-03	Trustees Of Boston University	Pharmacologically effective antagonists of arginine-vasopressin
US5051400A (en) *	1990-06-28	1991-09-24	Smithkline Beecham Corporation	Method of treating nausea and emesis related to motion sickness with vasopressin antagonists
RU2342949C1 (ru) *	2007-03-26	2009-01-10	Юрий Георгиевич Жуковский	Применение [дезамино-1, изолейцин-3, аргинин-8]вазопрессина в качестве средства для увеличения выведения почкой солей натрия и усиления обратного избирательного всасывания из почечных канальцев в кровь воды-растворителя
CN111253569B (zh) *	2020-02-26	2021-06-01	山东大学	一种聚合物、其制剂及其制备方法和应用

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
DE1193509B (de) *	1960-06-02	1965-05-26	Hoechst Ag	Verfahren zur Herstellung eines neuen Oktapeptids mit vasopressorischer Wirksamkeit
CH426861A (de) *	1963-06-06	1966-12-31	Sandoz Ag	Verfahren zur Herstellung eines bisher unbekannten Polypeptids
CH442342A (de) *	1964-07-17	1967-08-31	Sandoz Ag	Verfahren zur Herstellung eines neuen Polypeptids
CH460039A (de) *	1965-04-15	1968-07-31	Sandoz Ag	Verfahren zur Herstellung eines neuen Polypeptids
CH495957A (de) *	1966-09-15	1970-09-15	Ceskoslovenska Akademie Ved	Verfahren zur Herstellung eines antidiuretisch wirksamen Polypeptids
US4148787A (en) *	1976-05-24	1979-04-10	Ferring Ab	Antidiuretically effective polypeptide and a process for preparing the same

1981
- 1981-11-16 US US06/322,071 patent/US4399125A/en not_active Expired - Fee Related
1982
- 1982-03-02 IE IE465/82A patent/IE52624B1/en unknown
- 1982-03-03 CA CA000397464A patent/CA1185235A/fr not_active Expired
- 1982-03-04 NZ NZ199908A patent/NZ199908A/xx unknown
- 1982-03-09 IL IL65211A patent/IL65211A/xx unknown
- 1982-03-10 PH PH26975A patent/PH19237A/en unknown
- 1982-03-16 ZW ZW48/82A patent/ZW4882A1/xx unknown
- 1982-03-17 AU AU81617/82A patent/AU546865B2/en not_active Ceased
- 1982-03-18 ES ES510579A patent/ES8604264A1/es not_active Expired
- 1982-03-19 PT PT74615A patent/PT74615B/pt unknown
- 1982-03-23 RO RO107007A patent/RO84361B/ro unknown
- 1982-03-23 FI FI821019A patent/FI77047C/fi not_active IP Right Cessation
- 1982-03-23 KR KR8201234A patent/KR880000758B1/ko not_active Expired
- 1982-03-23 NO NO820967A patent/NO162024C/no unknown
- 1982-03-23 BG BG055925A patent/BG38487A3/xx unknown
- 1982-03-23 DK DK130182A patent/DK130182A/da not_active Application Discontinuation
- 1982-03-23 HU HU82880A patent/HU189127B/hu unknown
- 1982-03-24 DE DE8282301555T patent/DE3264734D1/de not_active Expired
- 1982-03-24 YU YU00634/82A patent/YU63482A/xx unknown
- 1982-03-24 DD DD82238409A patent/DD202695A5/de not_active IP Right Cessation
- 1982-03-24 EP EP82301555A patent/EP0061356B1/fr not_active Expired
- 1982-03-24 DD DD82255304A patent/DD212735A5/de not_active IP Right Cessation
1985
- 1985-08-14 ES ES546137A patent/ES8703489A1/es not_active Expired

Also Published As

Publication number	Publication date
ES8604264A1 (es)	1986-01-16
IL65211A (en)	1986-02-28
IL65211A0 (en)	1982-05-31
NO162024B (no)	1989-07-17
ZW4882A1 (en)	1983-02-23
RO84361B (ro)	1984-07-30
AU8161782A (en)	1982-09-30
BG38487A3 (en)	1985-12-16
NZ199908A (en)	1985-09-13
KR830008683A (ko)	1983-12-14
DK130182A (da)	1982-09-25
ES510579A0 (es)	1986-01-16
NO162024C (no)	1989-10-25
ES546137A0 (es)	1987-03-01
NO820967L (no)	1982-09-27
HU189127B (en)	1986-06-30
FI77047C (fi)	1989-01-10
FI821019L (fi)	1982-09-25
IE52624B1 (en)	1988-01-06
IE820465L (en)	1982-09-24
PT74615B (en)	1983-10-20
FI821019A0 (fi)	1982-03-23
EP0061356A3 (en)	1982-12-29
FI77047B (fi)	1988-09-30
DD202695A5 (de)	1983-09-28
DE3264734D1 (en)	1985-08-22
ES8703489A1 (es)	1987-03-01
RO84361A (fr)	1984-05-23
CA1185235A (fr)	1985-04-09
KR880000758B1 (ko)	1988-05-06
EP0061356A2 (fr)	1982-09-29
US4399125A (en)	1983-08-16
PT74615A (en)	1982-04-01
AU546865B2 (en)	1985-09-26
EP0061356B1 (fr)	1985-07-17
DD212735A5 (de)	1984-08-22
PH19237A (en)	1986-02-14

Publication	Publication Date	Title
YU63482A (en)	1985-10-31	Process for obtaining new antagonists of the antidiuretic and/or vasopressoric activity of the arginine vasopressin
DE3263071D1 (en)	1985-05-23	Snap-fit button
GB2094613B (en)	1984-04-18	Snap-fit button
PT80149B (en)	1987-03-23	Process for the preparation of new cyclosporines
ZA821422B (en)	1983-04-27	Novel antagonists of the antidiuretic and/or vasopressor action of arginine vasopressin
PT79059A (en)	1984-09-01	Phono-and electrocardiograph background of the invention
JPS57141488A (en)	1982-09-01	Manufacture of carbon article precurcor substance
PT80783A (en)	1985-08-01	Process for the preparation of benzimidazols bezoxazols and benzothiazols
DE3274017D1 (en)	1986-12-04	Assay and use
NZ200599A (en)	1985-04-30	Process for the production of dimethylether and catalyst therefor
GB2107705B (en)	1985-09-04	Process for the preparation of urea
GB2109771B (en)	1986-04-03	Bags and the manufacture of bags
DE3664464D1 (en)	1989-08-24	Process for the manufacture of gamma-butyrolactames
JPS57158782A (en)	1982-09-30	1,4,5,6,7,8-hexahydro-2-alkyl-4-aryl-5-oxo- 1,7-naphthyridine-3-carboxylic acid esters and use
DE3266101D1 (en)	1985-10-17	Process for the preparation of n substituted di and/or polyurethanes
HUT35480A (en)	1985-07-29	Herbicide preparations containing pyrazolile- and isoxazolile-sulfonyl-urea-derivatives and process for the production of the agents
ZW20982A1 (en)	1983-04-27	Aminooxazolyl compounds processes for their manufacture pharmaceutical preparations containing these compounds and the use of the latter
HUT36343A (en)	1985-09-30	Herbicides containing sulfonil-guanidine-derivatives as agent and process for the production of the agents
GB2098318B (en)	1984-12-05	Measuring the area of flat workpieces
HUT41589A (en)	1987-05-28	Artropodicids and process for production of the active substances
PT83528A (en)	1986-11-01	Process for the preparation of cardiotonic aroylthiazolones
YU29282A (en)	1985-03-20	Process for the manufacture of tetrahydronaphthaline and indiane
GB2145722B (en)	1987-07-08	Process for the preparation of 6-demethyl-6-deoxy-6-methylene-5-oxytetracyclin and the 11a-chloro-derivative thereof
IL67332A0 (en)	1983-03-31	Inter-m-phenylene-prostacycline analogues and process for the preparation thereof
JPS57135149A (en)	1982-08-20	Duster mat and its manufacture