ZA200406332B - ACC inhibitors. - Google Patents

ACC inhibitors. Download PDF

Info

Publication number: ZA200406332B
Authority: ZA; South Africa
Prior art keywords: insulin; moiety; human; patient; conjugate
Prior art date: 2002-02-27

Application number

ZA200406332A

Other languages

English (en)

Inventor

David Austen Perry

Harwood Harold James Jr

Original Assignee

Pfizer Prod Inc

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2002-02-27

Filing date

2004-08-10

Publication date

2005-09-28

2004-08-10 Application filed by Pfizer Prod Inc filed Critical Pfizer Prod Inc

2005-09-28 Publication of ZA200406332B publication Critical patent/ZA200406332B/en

Links

229940121373 acetyl-coa carboxylase inhibitor Drugs 0.000 title 1
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Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D407/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen atoms as the only ring hetero atoms, not provided for by group C07D405/00
- C07D407/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen atoms as the only ring hetero atoms, not provided for by group C07D405/00 containing three or more hetero rings
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings

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Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Diabetes (AREA)
Hematology (AREA)
Obesity (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Pharmacology & Pharmacy (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)
Transition And Organic Metals Composition Catalysts For Addition Polymerization (AREA)
Inorganic Insulating Materials (AREA)
Magnetic Heads (AREA)
Polishing Bodies And Polishing Tools (AREA)
Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)

ZA200406332A 2002-02-27 2004-08-10 ACC inhibitors. ZA200406332B (en)

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US (1)	US6979741B2 (fr)
EP (1)	EP1478437B1 (fr)
KR (1)	KR20040095239A (fr)
CN (1)	CN1642599A (fr)
AT (1)	ATE303178T1 (fr)
AU (1)	AU2003248354A1 (fr)
CO (1)	CO5601002A2 (fr)
DE (1)	DE60301491T2 (fr)
EA (1)	EA200400980A1 (fr)
ES (1)	ES2246481T3 (fr)
HR (1)	HRP20040716A2 (fr)
IL (1)	IL163659A0 (fr)
IS (1)	IS7391A (fr)
MA (1)	MA27178A1 (fr)
NO (1)	NO20044034L (fr)
NZ (1)	NZ534582A (fr)
PL (1)	PL372887A1 (fr)
TN (1)	TNSN04164A1 (fr)
WO (1)	WO2003072197A1 (fr)
ZA (1)	ZA200406332B (fr)

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PL373586A1 (en) *	2002-01-11	2005-09-05	Abbott Laboratories	Histamine-3 receptor ligands for diabetic conditions
WO2004063715A2 (fr) *	2003-01-10	2004-07-29	The Trustees Of Columbia University In The City Of New York	Procedes pour utiliser la structure cristalline du domaine de carboxyltransferase de l'acetyl-coa carboxylase, modulateurs de celle-ci et procedes informatiques
JP2006519229A (ja)	2003-02-13	2006-08-24	アルバート・アインシュタイン・カレッジ・オヴ・メディシン・オヴ・イェシヴァ・ユニヴァーシティ	視床下部内の長鎖脂肪アシルＣｏＡレベルの変調による摂食量およびグルコース産生量の調節
CA2518465A1 (fr)	2003-03-25	2004-10-14	Takeda San Diego, Inc.	Inhibiteurs de dipeptidyle peptidase
US7638638B2 (en)	2003-05-14	2009-12-29	Takeda San Diego, Inc.	Dipeptidyl peptidase inhibitors
US7169926B1 (en)	2003-08-13	2007-01-30	Takeda Pharmaceutical Company Limited	Dipeptidyl peptidase inhibitors
KR20060041309A (ko)	2003-08-13	2006-05-11	다케다 야쿠힌 고교 가부시키가이샤	４-피리미돈 유도체 및 펩티딜 펩티다제 저해제로서의 그의용도
JP2007505121A (ja)	2003-09-08	2007-03-08	武田薬品工業株式会社	ジペプチジルぺプチダーゼ阻害剤
US7371759B2 (en)	2003-09-25	2008-05-13	Bristol-Myers Squibb Company	HMG-CoA reductase inhibitors and method
DE602004008959T2 (de) *	2003-11-07	2008-06-19	F. Hoffmann-La Roche Ag	Benzoäbüä1,4üdioxepinderivate
GB0326029D0 (en) *	2003-11-07	2003-12-10	Astrazeneca Ab	Chemical compounds
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- 2003-02-17 PL PL03372887A patent/PL372887A1/xx not_active Application Discontinuation
- 2003-02-17 ES ES03742882T patent/ES2246481T3/es not_active Expired - Lifetime
- 2003-02-17 WO PCT/IB2003/000573 patent/WO2003072197A1/fr not_active Ceased
- 2003-02-17 KR KR10-2004-7013482A patent/KR20040095239A/ko not_active Ceased
- 2003-02-17 AU AU2003248354A patent/AU2003248354A1/en not_active Abandoned
- 2003-02-17 CN CNA038069903A patent/CN1642599A/zh active Pending
- 2003-02-17 DE DE60301491T patent/DE60301491T2/de not_active Expired - Fee Related
- 2003-02-17 AT AT03742882T patent/ATE303178T1/de not_active IP Right Cessation
- 2003-02-17 IL IL16365903A patent/IL163659A0/xx unknown
- 2003-02-17 EP EP03742882A patent/EP1478437B1/fr not_active Expired - Lifetime
- 2003-02-20 US US10/370,844 patent/US6979741B2/en not_active Expired - Fee Related
2004
- 2004-08-09 IS IS7391A patent/IS7391A/is unknown
- 2004-08-10 ZA ZA200406332A patent/ZA200406332B/en unknown
- 2004-08-18 MA MA27830A patent/MA27178A1/fr unknown
- 2004-08-25 TN TNP2004000164A patent/TNSN04164A1/fr unknown
- 2004-08-26 CO CO04083409A patent/CO5601002A2/es not_active Application Discontinuation
- 2004-09-24 NO NO20044034A patent/NO20044034L/no not_active Application Discontinuation

Also Published As

Publication number	Publication date
EP1478437B1 (fr)	2005-08-31
KR20040095239A (ko)	2004-11-12
ATE303178T1 (de)	2005-09-15
US20030187254A1 (en)	2003-10-02
PL372887A1 (en)	2005-08-08
HRP20040716A2 (en)	2005-02-28
CN1642599A (zh)	2005-07-20
DE60301491D1 (en)	2005-10-06
TNSN04164A1 (fr)	2007-03-12
NZ534582A (en)	2006-03-31
DE60301491T2 (de)	2006-05-18
MA27178A1 (fr)	2005-01-03
IL163659A0 (en)	2005-12-18
AU2003248354A1 (en)	2003-09-09
CO5601002A2 (es)	2006-01-31
US6979741B2 (en)	2005-12-27
EA200400980A1 (ru)	2005-02-24
WO2003072197A1 (fr)	2003-09-04
EP1478437A1 (fr)	2004-11-24
ES2246481T3 (es)	2006-02-16
IS7391A (is)	2004-08-09
NO20044034L (no)	2004-11-24

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