ZA200605632B - UV-light stable semi-solid transdermal systems that contain a light-sensitive substance and a UV-absorber - Google Patents

UV-light stable semi-solid transdermal systems that contain a light-sensitive substance and a UV-absorber Download PDF

Info

Publication number: ZA200605632B
Authority: ZA; South Africa
Prior art keywords: semisolid; absorber; transdermal therapeutic; therapeutic system; acid
Prior art date: 2003-12-10

Application number

ZA200605632A

Other languages

English (en)

Inventor

Hans-Peter Podhaisky

Stefan Bracht

Original Assignee

Bayer Schering Pharma Ag Nm

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2003-12-10

Filing date

2006-07-07

Publication date

2008-06-25

Family has litigation

First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=34486168&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=ZA200605632(B) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.

2006-07-07 Application filed by Bayer Schering Pharma Ag Nm filed Critical Bayer Schering Pharma Ag Nm

2008-06-25 Publication of ZA200605632B publication Critical patent/ZA200605632B/en

Links

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229920000058 polyacrylate Polymers 0.000 description 1
229920000193 polymethacrylate Polymers 0.000 description 1
229920002451 polyvinyl alcohol Polymers 0.000 description 1
229940068984 polyvinyl alcohol Drugs 0.000 description 1
235000019422 polyvinyl alcohol Nutrition 0.000 description 1
229920000036 polyvinylpyrrolidone Polymers 0.000 description 1
239000001267 polyvinylpyrrolidone Substances 0.000 description 1
235000013855 polyvinylpyrrolidone Nutrition 0.000 description 1
229920001592 potato starch Polymers 0.000 description 1
229940116317 potato starch Drugs 0.000 description 1
230000008569 process Effects 0.000 description 1
239000000047 product Substances 0.000 description 1
238000011321 prophylaxis Methods 0.000 description 1
230000001681 protective effect Effects 0.000 description 1
229940100486 rice starch Drugs 0.000 description 1
150000003839 salts Chemical class 0.000 description 1
FWFUWXVFYKCSQA-UHFFFAOYSA-M sodium;2-methyl-2-(prop-2-enoylamino)propane-1-sulfonate Chemical compound [Na+].[O-]S(=O)(=O)CC(C)(C)NC(=O)C=C FWFUWXVFYKCSQA-UHFFFAOYSA-M 0.000 description 1
230000003595 spectral effect Effects 0.000 description 1
235000019698 starch Nutrition 0.000 description 1
150000003460 sulfonic acids Chemical class 0.000 description 1
239000000725 suspension Substances 0.000 description 1
230000008961 swelling Effects 0.000 description 1
230000001839 systemic circulation Effects 0.000 description 1
229960003604 testosterone Drugs 0.000 description 1
239000000196 tragacanth Substances 0.000 description 1
235000010487 tragacanth Nutrition 0.000 description 1
229940116362 tragacanth Drugs 0.000 description 1
229960000281 trometamol Drugs 0.000 description 1
229940100445 wheat starch Drugs 0.000 description 1

Classifications

- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0014—Skin, i.e. galenical aspects of topical compositions
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/08—Solutions
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
- A61K31/565—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
- A61K31/565—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol
- A61K31/567—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol substituted in position 17 alpha, e.g. mestranol, norethandrolone
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
- A61K47/08—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
- A61K47/10—Alcohols; Phenols; Salts thereof, e.g. glycerol; Polyethylene glycols [PEG]; Poloxamers; PEG/POE alkyl ethers
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
- A61K47/08—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
- A61K47/14—Esters of carboxylic acids, e.g. fatty acid monoglycerides, medium-chain triglycerides, parabens or PEG fatty acid esters
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/30—Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
- A61K47/32—Macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. carbomers, poly(meth)acrylates, or polyvinyl pyrrolidone
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/18—Feminine contraceptives
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
- A61P5/26—Androgens
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
- A61P5/30—Oestrogens
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
- A61P5/34—Gestagens

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Pharmacology & Pharmacy (AREA)
Veterinary Medicine (AREA)
Public Health (AREA)
General Health & Medical Sciences (AREA)
Animal Behavior & Ethology (AREA)
Medicinal Chemistry (AREA)
Life Sciences & Earth Sciences (AREA)
Epidemiology (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Engineering & Computer Science (AREA)
Organic Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Endocrinology (AREA)
Bioinformatics & Cheminformatics (AREA)
Diabetes (AREA)
Oil, Petroleum & Natural Gas (AREA)
Dermatology (AREA)
Reproductive Health (AREA)
Gynecology & Obstetrics (AREA)
Inorganic Chemistry (AREA)
Medicinal Preparation (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Cosmetics (AREA)

ZA200605632A 2003-12-10 2006-07-07 UV-light stable semi-solid transdermal systems that contain a light-sensitive substance and a UV-absorber ZA200605632B (en)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
EP03028353A EP1541136A1 (de)	2003-12-10	2003-12-10	UV-Licht stabile halbfeste transdermale Systeme, die einen lichtempfindlichen Wirkstoff und einen UV-Absorber enthalten

Publications (1)

Publication Number	Publication Date
ZA200605632B true ZA200605632B (en)	2008-06-25

Family

ID=34486168

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
ZA200605632A ZA200605632B (en)	2003-12-10	2006-07-07	UV-light stable semi-solid transdermal systems that contain a light-sensitive substance and a UV-absorber

Country Status (24)

Country	Link
EP (2)	EP1541136A1 (pt)
JP (1)	JP2007534643A (pt)
KR (1)	KR20060096512A (pt)
CN (1)	CN101415402A (pt)
AR (1)	AR047140A1 (pt)
AU (1)	AU2004296539B2 (pt)
BR (1)	BRPI0416979A (pt)
CA (1)	CA2548739C (pt)
CR (1)	CR8461A (pt)
EA (1)	EA010239B1 (pt)
EC (1)	ECSP066689A (pt)
GT (1)	GT200400261A (pt)
HN (1)	HN2004000525A (pt)
IL (1)	IL176208A0 (pt)
MX (1)	MXPA06006534A (pt)
MY (1)	MY141728A (pt)
NO (1)	NO20063208L (pt)
NZ (1)	NZ547733A (pt)
PE (1)	PE20050863A1 (pt)
SV (1)	SV2006001971A (pt)
TW (1)	TW200528136A (pt)
UA (1)	UA85861C2 (pt)
WO (1)	WO2005055975A2 (pt)
ZA (1)	ZA200605632B (pt)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
TWI395806B (zh)	2010-04-14	2013-05-11	Ind Tech Res Inst	封裝材料
SI2613772T1 (sl) *	2010-09-06	2017-03-31	Bayer Intellectual Property Gmbh	Transdermalni obliži z nizkim odmerkom z visoko stopnjo sproščanja zdravila
WO2014152122A2 (en) *	2013-03-15	2014-09-25	Children's Medical Center Corporation	Methods of altering vascular permeability and uses thereof
JP2024000555A (ja) *	2022-06-21	2024-01-09	東ソー株式会社	紫外線抑制下でのエストラジオール測定試薬の製造方法

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
JPS60155111A (ja) *	1983-10-20	1985-08-15	Hisamitsu Pharmaceut Co Inc	安定なケトプロフェン含有外用経皮製剤
JP2981523B2 (ja) *	1990-11-19	1999-11-22	株式会社林原生物化学研究所	皮膚外用剤
AUPN814496A0 (en) *	1996-02-19	1996-03-14	Monash University	Dermal penetration enhancer
CA2301016A1 (en) *	1997-08-21	1999-02-25	Johnson & Johnson Consumer Companies, Inc.	Use of 17-.alpha.-estradiol for the treatment of aged or sundamaged ski n and/or skin atrophy
JP2000292428A (ja) *	1999-04-05	2000-10-20	Umeda Jimusho:Kk	環境化学物質の内分泌攪乱活性の新規測定方法及びその装置
JP2001129566A (ja) *	1999-11-05	2001-05-15	Mitsubishi Heavy Ind Ltd	有害物質処理方法およびその装置
FR2804024B1 (fr) *	2000-01-21	2002-09-13	Menarini France	Nouvelles compositions pharmaceutiques a action anti- inflammatoire et leur procede de preparation
DE10053375C1 (de) *	2000-10-27	2002-01-24	Lohmann Therapie Syst Lts	Transdermale therapeutische Systeme mit lichtempfindlichen Wirkstoffen
FR2834895B1 (fr) *	2002-01-22	2006-06-23	Ellipse Pharmaceuticals	Compositions dermatologiques, resistantes a l'eau, avec filtres solaires, procede de fabrication et utilisations de ces compositions
ITFI20020144A1 (it) *	2002-08-01	2004-02-02	Menarini Farma Ind	Formulazioni topiche stabilizzate contenenti ketoprofene.

2003
- 2003-12-10 EP EP03028353A patent/EP1541136A1/de not_active Withdrawn
2004
- 2004-06-12 UA UAA200607539A patent/UA85861C2/uk unknown
- 2004-12-02 TW TW93137245A patent/TW200528136A/zh unknown
- 2004-12-06 KR KR1020067013775A patent/KR20060096512A/ko not_active Ceased
- 2004-12-06 JP JP2006543451A patent/JP2007534643A/ja active Pending
- 2004-12-06 CN CNA2004800369947A patent/CN101415402A/zh active Pending
- 2004-12-06 EP EP04803546A patent/EP1703892A2/de not_active Withdrawn
- 2004-12-06 CA CA002548739A patent/CA2548739C/en not_active Expired - Fee Related
- 2004-12-06 NZ NZ547733A patent/NZ547733A/en unknown
- 2004-12-06 WO PCT/EP2004/013839 patent/WO2005055975A2/de not_active Ceased
- 2004-12-06 EA EA200601084A patent/EA010239B1/ru not_active IP Right Cessation
- 2004-12-06 BR BRPI0416979-4A patent/BRPI0416979A/pt not_active IP Right Cessation
- 2004-12-06 AU AU2004296539A patent/AU2004296539B2/en not_active Ceased
- 2004-12-10 PE PE2004001228A patent/PE20050863A1/es not_active Application Discontinuation
- 2004-12-10 HN HN2004000525A patent/HN2004000525A/es unknown
- 2004-12-10 MY MYPI20045109A patent/MY141728A/en unknown
- 2004-12-10 AR ARP040104604A patent/AR047140A1/es unknown
- 2004-12-10 SV SV2004001971A patent/SV2006001971A/es not_active Application Discontinuation
- 2004-12-10 GT GT200400261A patent/GT200400261A/es unknown
2006
- 2006-06-08 MX MXPA06006534 patent/MXPA06006534A/es unknown
- 2006-06-08 IL IL176208A patent/IL176208A0/en unknown
- 2006-06-16 CR CR8461A patent/CR8461A/es not_active Application Discontinuation
- 2006-07-07 EC EC2006006689A patent/ECSP066689A/es unknown
- 2006-07-07 ZA ZA200605632A patent/ZA200605632B/en unknown
- 2006-07-10 NO NO20063208A patent/NO20063208L/no not_active Application Discontinuation

Also Published As

Publication number	Publication date
WO2005055975A3 (de)	2009-03-12
CN101415402A (zh)	2009-04-22
GT200400261A (es)	2005-10-31
HN2004000525A (es)	2010-09-17
TW200528136A (en)	2005-09-01
MY141728A (en)	2010-06-15
IL176208A0 (en)	2006-10-05
CA2548739A1 (en)	2005-06-23
NZ547733A (en)	2010-02-26
JP2007534643A (ja)	2007-11-29
EP1541136A1 (de)	2005-06-15
ECSP066689A (es)	2006-10-31
EA010239B1 (ru)	2008-06-30
AR047140A1 (es)	2006-01-11
CA2548739C (en)	2009-08-18
UA85861C2 (uk)	2009-03-10
SV2006001971A (es)	2006-02-15
WO2005055975A2 (de)	2005-06-23
EA200601084A1 (ru)	2006-12-29
AU2004296539A1 (en)	2005-06-23
KR20060096512A (ko)	2006-09-11
MXPA06006534A (es)	2006-08-01
NO20063208L (no)	2006-07-10
AU2004296539B2 (en)	2008-10-09
PE20050863A1 (es)	2005-11-02
CR8461A (es)	2006-12-07
EP1703892A2 (de)	2006-09-27
BRPI0416979A (pt)	2007-02-21

Publication	Publication Date	Title
US20050129756A1 (en)	2005-06-16	UV-stable, liquid or semisolid transdermal pharmaceutical preparation with light sensitive active ingredient
AU676562B2 (en)	1997-03-13	Solubilizing agent and external preparation containing the same
EP0782861B1 (en)	2001-12-12	Drug compounding ingredients comprising n-substituted-o-toluidine derivative and percutaneously absorbable preparation
ES2399900T3 (es)	2013-04-04	Composición farmacéutica que comprende un andrógeno
US20150150827A1 (en)	2015-06-04	Multi-layered transdermal system with triazine uv absorber
HU221598B (hu)	2002-11-28	Glicerin alkalmazása bőrön keresztüli hatóanyag-bevitel szabályozására
EP2138169B1 (en)	2013-11-06	Transdermal delivery system of hormones without penetration enhancers
SK126093A3 (en)	1994-09-07	Lanoline derivatives as a penetration-promoting substances
AU2004296539B2 (en)	2008-10-09	UV-stable, liquid or semi-solid transdermal administration form comprising a photosensitive active ingredient
US20180078493A1 (en)	2018-03-22	Transdermal hormone delivery
AU2004298930B2 (en)	2009-11-26	Transdermal delivery system of hormones without penetration enhancers
JP5075622B2 (ja)	2012-11-21	非ステロイド系消炎鎮痛剤を含有する外用経皮製剤
EP1752164B1 (en)	2014-05-07	Percutaneous pharmaceutical preparation for external use containing nonsteroidal antiinflammatory analgesic
HK1129209A (en)	2009-11-20	Uv-stable, liquid or semi-solid transdermal administration form comprising a photosensitive active ingredient
JP2852816B2 (ja)	1999-02-03	溶解剤および該溶解剤を含有する外用製剤
KR20080003854A (ko)	2008-01-08	Ｕｖ 흡수제를 포함하는 고상 경피 치료 시스템
HK1132682B (en)	2014-07-11	Transdermal delivery system of hormones without penetration enhancers
KR20070015954A (ko)	2007-02-06	비스테로이드계 소염 진통제를 함유하는 외용 경피 제제
HK1074801B (en)	2010-05-20	Transdermal delivery system of gestodene