AP2009004880A0 - Spiroketone acetyl-COA carboxylase inhibitors - Google Patents

Spiroketone acetyl-COA carboxylase inhibitors

Info

Publication number
AP2009004880A0
AP2009004880A0 AP2009004880A AP2009004880A AP2009004880A0 AP 2009004880 A0 AP2009004880 A0 AP 2009004880A0 AP 2009004880 A AP2009004880 A AP 2009004880A AP 2009004880 A AP2009004880 A AP 2009004880A AP 2009004880 A0 AP2009004880 A0 AP 2009004880A0
Authority
AP
ARIPO
Prior art keywords
spiroketone
acetyl
coa carboxylase
carboxylase inhibitors
inhibitors
Prior art date
Application number
AP2009004880A
Other languages
English (en)
Inventor
Richard Louis Elliot
Jeffrey Wayne Corbett
Andrew Simon Bell
Original Assignee
Pfizer Prod Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Prod Inc filed Critical Pfizer Prod Inc
Publication of AP2009004880A0 publication Critical patent/AP2009004880A0/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
    • C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
    • C07D491/10—Spiro-condensed systems
    • C07D491/107—Spiro-condensed systems with only one oxygen atom as ring hetero atom in the oxygen-containing ring
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/38—Heterocyclic compounds having sulfur as a ring hetero atom
    • A61K31/39—Heterocyclic compounds having sulfur as a ring hetero atom having oxygen in the same ring
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/06—Antihyperlipidemics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/04—Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
    • C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
    • C07D491/10—Spiro-condensed systems

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Diabetes (AREA)
  • Cardiology (AREA)
  • Obesity (AREA)
  • Hematology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Endocrinology (AREA)
  • Urology & Nephrology (AREA)
  • Emergency Medicine (AREA)
  • Hospice & Palliative Care (AREA)
  • Vascular Medicine (AREA)
  • Child & Adolescent Psychology (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Plural Heterocyclic Compounds (AREA)
AP2009004880A 2006-11-29 2007-11-16 Spiroketone acetyl-COA carboxylase inhibitors AP2009004880A0 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US86177906P 2006-11-29 2006-11-29
PCT/IB2007/003639 WO2008065508A1 (en) 2006-11-29 2007-11-16 Spiroketone acetyl-coa carboxylase inhibitors

Publications (1)

Publication Number Publication Date
AP2009004880A0 true AP2009004880A0 (en) 2009-06-30

Family

ID=39126209

Family Applications (1)

Application Number Title Priority Date Filing Date
AP2009004880A AP2009004880A0 (en) 2006-11-29 2007-11-16 Spiroketone acetyl-COA carboxylase inhibitors

Country Status (23)

Country Link
US (1) US20090270435A1 (pt)
EP (1) EP2097420B1 (pt)
JP (1) JP2010511035A (pt)
KR (1) KR20090083956A (pt)
CN (1) CN101541809A (pt)
AP (1) AP2009004880A0 (pt)
AT (1) ATE552262T1 (pt)
AU (1) AU2007326950B2 (pt)
BR (1) BRPI0721053A2 (pt)
CA (1) CA2670422C (pt)
CO (1) CO6180424A2 (pt)
CR (1) CR10831A (pt)
EA (1) EA200900613A1 (pt)
EC (1) ECSP099371A (pt)
IL (1) IL198779A0 (pt)
MA (1) MA30932B1 (pt)
MX (1) MX2009005604A (pt)
NO (1) NO20091889L (pt)
RS (1) RS20090249A (pt)
SV (1) SV2009003281A (pt)
TN (1) TN2009000204A1 (pt)
WO (1) WO2008065508A1 (pt)
ZA (1) ZA200903268B (pt)

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DE102008038222A1 (de) 2008-08-18 2010-02-25 Merck Patent Gmbh Indazol-5-carbonsäurehydrazid-derivate
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Also Published As

Publication number Publication date
US20090270435A1 (en) 2009-10-29
CO6180424A2 (es) 2010-07-19
EP2097420A1 (en) 2009-09-09
EA200900613A1 (ru) 2009-10-30
TN2009000204A1 (fr) 2010-10-18
AU2007326950B2 (en) 2010-10-14
NO20091889L (no) 2009-06-17
MA30932B1 (fr) 2009-11-02
EP2097420B1 (en) 2012-04-04
CA2670422C (en) 2011-09-06
CN101541809A (zh) 2009-09-23
SV2009003281A (es) 2010-08-17
WO2008065508A1 (en) 2008-06-05
RS20090249A (sr) 2010-06-30
MX2009005604A (es) 2009-06-08
JP2010511035A (ja) 2010-04-08
IL198779A0 (en) 2010-02-17
ATE552262T1 (de) 2012-04-15
BRPI0721053A2 (pt) 2014-07-29
ZA200903268B (en) 2010-07-28
KR20090083956A (ko) 2009-08-04
CR10831A (es) 2009-06-18
CA2670422A1 (en) 2008-06-05
AU2007326950A1 (en) 2008-06-05
ECSP099371A (es) 2009-06-30

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GB2452595B8 (en) An insert
IL197981A0 (en) Kinase inhibitors
GB0605795D0 (en) Spirit level
GB0619177D0 (en) Level
ZA200806993B (en) Hydantoin based kinase inhibitors
GB0714941D0 (en) Inhibitors
PL2126486T3 (pl) Lodówka
GB0610713D0 (en) Flexi-garden-design
GB0708255D0 (en) Cysteine prtease inhibitors
GB0613519D0 (en) Insert
GB0713152D0 (en) Phosphodlesterase inhibitors