AR036407A1 - Tieno[2,3-d]pirimidinas con actividad agonista de lh y fsh para el uso en el control de la fertilidad - Google Patents

Tieno[2,3-d]pirimidinas con actividad agonista de lh y fsh para el uso en el control de la fertilidad

Info

Publication number
AR036407A1
AR036407A1 ARP020103309A ARP020103309A AR036407A1 AR 036407 A1 AR036407 A1 AR 036407A1 AR P020103309 A ARP020103309 A AR P020103309A AR P020103309 A ARP020103309 A AR P020103309A AR 036407 A1 AR036407 A1 AR 036407A1
Authority
AR
Argentina
Prior art keywords
fsh
fertility
pyrimidins
control
agonist activity
Prior art date
Application number
ARP020103309A
Other languages
English (en)
Spanish (es)
Inventor
Robert Gerard Jules Marie Hanssen
Cornelis Marius Timmers
Original Assignee
Akzo Nobel Nv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Akzo Nobel Nv filed Critical Akzo Nobel Nv
Publication of AR036407A1 publication Critical patent/AR036407A1/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A61P15/08—Drugs for genital or sexual disorders; Contraceptives for gonadal disorders or for enhancing fertility, e.g. inducers of ovulation or of spermatogenesis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/06—Drugs for disorders of the endocrine system of the anterior pituitary hormones, e.g. TSH, ACTH, FSH, LH, PRL, GH
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/06—Drugs for disorders of the endocrine system of the anterior pituitary hormones, e.g. TSH, ACTH, FSH, LH, PRL, GH
    • A61P5/08—Drugs for disorders of the endocrine system of the anterior pituitary hormones, e.g. TSH, ACTH, FSH, LH, PRL, GH for decreasing, blocking or antagonising the activity of the anterior pituitary hormones

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Endocrinology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Reproductive Health (AREA)
  • Diabetes (AREA)
  • Gynecology & Obstetrics (AREA)
  • Pregnancy & Childbirth (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
ARP020103309A 2001-09-04 2002-09-02 Tieno[2,3-d]pirimidinas con actividad agonista de lh y fsh para el uso en el control de la fertilidad AR036407A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP01203327 2001-09-04

Publications (1)

Publication Number Publication Date
AR036407A1 true AR036407A1 (es) 2004-09-08

Family

ID=8180876

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP020103309A AR036407A1 (es) 2001-09-04 2002-09-02 Tieno[2,3-d]pirimidinas con actividad agonista de lh y fsh para el uso en el control de la fertilidad

Country Status (28)

Country Link
US (1) US7317006B2 (pl)
EP (1) EP1427733B1 (pl)
JP (1) JP4262092B2 (pl)
KR (1) KR100900018B1 (pl)
CN (1) CN1246324C (pl)
AR (1) AR036407A1 (pl)
AT (1) ATE345345T1 (pl)
AU (1) AU2002337035B2 (pl)
BR (1) BR0211938A (pl)
CA (1) CA2456901C (pl)
CY (1) CY1106012T1 (pl)
DE (1) DE60216128T2 (pl)
DK (1) DK1427733T3 (pl)
ES (1) ES2275005T3 (pl)
HR (1) HRP20040202A2 (pl)
HU (1) HUP0401444A3 (pl)
IL (1) IL160084A0 (pl)
IS (1) IS2424B (pl)
MX (1) MXPA04002045A (pl)
NO (1) NO20040927L (pl)
NZ (1) NZ531340A (pl)
PE (1) PE20030439A1 (pl)
PL (1) PL368502A1 (pl)
PT (1) PT1427733E (pl)
RU (1) RU2298011C2 (pl)
TW (1) TWI228508B (pl)
WO (1) WO2003020726A1 (pl)
ZA (1) ZA200401455B (pl)

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6890923B2 (en) * 2002-12-16 2005-05-10 Astrazeneca Ab Compounds
GB0315950D0 (en) * 2003-06-11 2003-08-13 Xention Discovery Ltd Compounds
GB0525164D0 (en) * 2005-12-09 2006-01-18 Xention Discovery Ltd Compounds
CN100430403C (zh) * 2006-10-13 2008-11-05 中国科学院上海有机化学研究所 3-芳基-5,6-取代噻吩并嘧啶-4-羰基-2-巯基乙腈、合成方法和用途
US20090118276A1 (en) * 2007-11-02 2009-05-07 Wyeth Thienopyrimidines, thienopyridines, and pyrrolopyrimidines as b-raf inhibitors
TWI389913B (zh) * 2008-09-08 2013-03-21 Lg Life Sciences Ltd 并合雜環化合物
WO2010047674A1 (en) 2008-10-20 2010-04-29 The Government Of The United States Of America As Represented By The Secretary Of The Department Of Health And Human Services Low molecular weight thyroid stimulating hormone receptor (tshr) agonists
GB0905525D0 (en) 2009-03-31 2009-05-13 Univ Leiden Compounds and uses
CN102811617A (zh) 2010-01-22 2012-12-05 拜耳知识产权有限责任公司 杀螨和/或杀虫活性物质结合物
WO2011127388A2 (en) 2010-04-08 2011-10-13 The United States Of America, As Represented By The Secretary, Department Of Health And Human Services Inverse agonists and neutral antagonists for the tsh receptor
WO2016029372A1 (en) 2014-08-27 2016-03-03 The Procter & Gamble Company Wearable article having elastic belt
WO2016029375A1 (en) 2014-08-27 2016-03-03 The Procter & Gamble Company Wearable article having elastic belt
RU2619091C2 (ru) * 2015-10-13 2017-05-11 Министерство Промышленности И Торговли Рф Цилиндрический термоэмиссионный катод
CN108883011B (zh) 2016-04-08 2021-05-07 宝洁公司 具有艺术作品的可穿着制品
JP2025524365A (ja) * 2022-06-08 2025-07-30 アイカーン スクール オブ メディスン アット マウント サイナイ 黄体形成ホルモン受容体作動薬を用いた肥満の治療方法

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2054784T3 (es) 1987-08-08 1994-08-16 Akzo Nv Un metodo para la fabricacion de un implante.
TW564247B (en) * 1999-04-08 2003-12-01 Akzo Nobel Nv Bicyclic heteraromatic compound

Also Published As

Publication number Publication date
IS2424B (is) 2008-10-15
RU2298011C2 (ru) 2007-04-27
HUP0401444A2 (hu) 2004-11-29
IL160084A0 (en) 2004-06-20
US20040180873A1 (en) 2004-09-16
PE20030439A1 (es) 2003-05-17
ZA200401455B (en) 2004-11-19
US7317006B2 (en) 2008-01-08
PT1427733E (pt) 2007-02-28
CY1106012T1 (el) 2011-04-06
TWI228508B (en) 2005-03-01
JP2005505555A (ja) 2005-02-24
HRP20040202A2 (en) 2004-08-31
CN1246324C (zh) 2006-03-22
BR0211938A (pt) 2004-09-21
NO20040927L (no) 2004-03-03
AU2002337035B2 (en) 2008-04-24
KR20040029134A (ko) 2004-04-03
CN1551884A (zh) 2004-12-01
CA2456901A1 (en) 2003-03-13
DK1427733T3 (da) 2007-03-19
PL368502A1 (pl) 2005-04-04
HUP0401444A3 (en) 2008-05-28
DE60216128D1 (de) 2006-12-28
CA2456901C (en) 2011-01-04
ES2275005T3 (es) 2007-06-01
EP1427733B1 (en) 2006-11-15
MXPA04002045A (es) 2004-07-08
DE60216128T2 (de) 2007-09-27
KR100900018B1 (ko) 2009-06-01
ATE345345T1 (de) 2006-12-15
IS7130A (is) 2004-01-29
WO2003020726A1 (en) 2003-03-13
NZ531340A (en) 2005-08-26
JP4262092B2 (ja) 2009-05-13
EP1427733A1 (en) 2004-06-16
RU2004110042A (ru) 2005-08-20

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