ATE10741T1 - Dibenzo(b,f)(1,4)oxazepin-derivate, verfahren zu ihrer herstellung und diese enthaltende pharmazeutische zusammensetzungen. - Google Patents

Dibenzo(b,f)(1,4)oxazepin-derivate, verfahren zu ihrer herstellung und diese enthaltende pharmazeutische zusammensetzungen.

Info

Publication number
ATE10741T1
ATE10741T1 AT81110655T AT81110655T ATE10741T1 AT E10741 T1 ATE10741 T1 AT E10741T1 AT 81110655 T AT81110655 T AT 81110655T AT 81110655 T AT81110655 T AT 81110655T AT E10741 T1 ATE10741 T1 AT E10741T1
Authority
AT
Austria
Prior art keywords
group
pharmaceutical compositions
derivatives
lower alkyl
alkyl group
Prior art date
Application number
AT81110655T
Other languages
English (en)
Inventor
Kiyohiko Ito
Masuo Koizumi
Yasushi Murakami
Mitchitaka Akima
Jinichiro Aono
Yasuhiro Ohba
Tamotsu Yamazaki
Kazushige Sakai
Shun-Ichi Hata
Shigeru Takanashi
Original Assignee
Chugai Seiyaku Kabushiki Kaisha
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Chugai Seiyaku Kabushiki Kaisha filed Critical Chugai Seiyaku Kabushiki Kaisha
Application granted granted Critical
Publication of ATE10741T1 publication Critical patent/ATE10741T1/de

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D267/00—Heterocyclic compounds containing rings of more than six members having one nitrogen atom and one oxygen atom as the only ring hetero atoms
    • C07D267/02—Seven-membered rings
    • C07D267/08—Seven-membered rings having the hetero atoms in positions 1 and 4
    • C07D267/12—Seven-membered rings having the hetero atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
    • C07D267/16—Seven-membered rings having the hetero atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems condensed with two six-membered rings
    • C07D267/20—[b, f]-condensed
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/08—Vasodilators for multiple indications
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Cardiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Urology & Nephrology (AREA)
  • Vascular Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
AT81110655T 1980-12-24 1981-12-21 Dibenzo(b,f)(1,4)oxazepin-derivate, verfahren zu ihrer herstellung und diese enthaltende pharmazeutische zusammensetzungen. ATE10741T1 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP55181831A JPS57106673A (en) 1980-12-24 1980-12-24 Dibenzo(b,f)(1,4)oxazepin derivative
EP81110655A EP0054951B1 (de) 1980-12-24 1981-12-21 Dibenzo(b,f)(1,4)oxazepin-Derivate, Verfahren zu ihrer Herstellung und diese enthaltende pharmazeutische Zusammensetzungen

Publications (1)

Publication Number Publication Date
ATE10741T1 true ATE10741T1 (de) 1984-12-15

Family

ID=16107575

Family Applications (1)

Application Number Title Priority Date Filing Date
AT81110655T ATE10741T1 (de) 1980-12-24 1981-12-21 Dibenzo(b,f)(1,4)oxazepin-derivate, verfahren zu ihrer herstellung und diese enthaltende pharmazeutische zusammensetzungen.

Country Status (6)

Country Link
US (1) US4379150A (de)
EP (1) EP0054951B1 (de)
JP (1) JPS57106673A (de)
AT (1) ATE10741T1 (de)
CA (1) CA1169059A (de)
DE (2) DE54951T1 (de)

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US5395932A (en) * 1993-04-30 1995-03-07 G. D. Searle & Co. 2,3-,4-,5-,6-,7-,8-,9- and/or 10-substituted dibenzoxazepine compounds, pharmaceutical compositions and methods of use
US5354746A (en) * 1993-06-01 1994-10-11 G. D. Searle & Co. Squaric acid derivatives of substituted dibenzoxazepine compounds, pharmaceutical compositions and methods of use
US5461047A (en) * 1993-06-16 1995-10-24 G. D. Searle & Co. 2-,3-,4-,5-,6-,7-,8-,9- and/or 10-substituted dibenzoxazepine and dibenzthiazepine compounds, pharmaceutical compositions and methods of use
US5354747A (en) * 1993-06-16 1994-10-11 G. D. Searle & Co. 2-, 3-, 4-, 5-, 6-, 7-, 8-, 9- and/or 10-substituted dibenzoxazepine and dibenzthiazepine compounds, pharmaceutical compositions and methods of use
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Publication number Priority date Publication date Assignee Title
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CH484179A (de) * 1965-06-23 1970-01-15 Ciba Geigy Verfahren zur Herstellung von Oxazaheterocyclen
FR4500M (de) * 1965-07-15 1966-10-10
DE1670414A1 (de) * 1966-12-17 1970-10-29 Ciba Geigy Oxyzaheterocyclen

Also Published As

Publication number Publication date
US4379150A (en) 1983-04-05
JPS57106673A (en) 1982-07-02
DE54951T1 (de) 1983-04-28
EP0054951B1 (de) 1984-12-12
EP0054951A1 (de) 1982-06-30
DE3167757D1 (en) 1985-01-24
CA1169059A (en) 1984-06-12

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