ATE121101T1 - Aus dalbaheptide hergestellte tetrapeptidantibiotika. - Google Patents

Aus dalbaheptide hergestellte tetrapeptidantibiotika.

Info

Publication number: ATE121101T1
Authority: AT; Austria
Prior art keywords: group; dalbaheptide; carboxyacid; tetrapeptide; aglucodalbaheptides
Prior art date: 1990-12-10

Application number

AT91920590T

Other languages

English (en)

Inventor

Adriano Malabarba

Romeo Ciabatti

Original Assignee

Lepetit Spa

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1990-12-10

Filing date

1991-11-28

Publication date

1995-04-15

1991-11-28 Application filed by Lepetit Spa filed Critical Lepetit Spa

1995-04-15 Application granted granted Critical

1995-04-15 Publication of ATE121101T1 publication Critical patent/ATE121101T1/de

Links

230000003115 biocidal effect Effects 0.000 title abstract 2
239000003242 anti bacterial agent Substances 0.000 abstract 2
150000003839 salts Chemical class 0.000 abstract 2
239000002253 acid Substances 0.000 abstract 1
150000007513 acids Chemical class 0.000 abstract 1
125000003277 amino group Chemical group 0.000 abstract 1
229940088710 antibiotic agent Drugs 0.000 abstract 1
229910052739 hydrogen Inorganic materials 0.000 abstract 1
239000001257 hydrogen Substances 0.000 abstract 1
125000004435 hydrogen atom Chemical group [H]* 0.000 abstract 1
125000002924 primary amino group Chemical group [H]N([H])* 0.000 abstract 1
125000006239 protecting group Chemical group 0.000 abstract 1
DKVBOUDTNWVDEP-NJCHZNEYSA-N teicoplanin aglycone Chemical compound N([C@H](C(N[C@@H](C1=CC(O)=CC(O)=C1C=1C(O)=CC=C2C=1)C(O)=O)=O)[C@H](O)C1=CC=C(C(=C1)Cl)OC=1C=C3C=C(C=1O)OC1=CC=C(C=C1Cl)C[C@H](C(=O)N1)NC([C@H](N)C=4C=C(O5)C(O)=CC=4)=O)C(=O)[C@@H]2NC(=O)[C@@H]3NC(=O)[C@@H]1C1=CC5=CC(O)=C1 DKVBOUDTNWVDEP-NJCHZNEYSA-N 0.000 abstract 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K9/00—Peptides having up to 20 amino acids, containing saccharide radicals and having a fully defined sequence; Derivatives thereof
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K9/00—Peptides having up to 20 amino acids, containing saccharide radicals and having a fully defined sequence; Derivatives thereof
- C07K9/006—Peptides having up to 20 amino acids, containing saccharide radicals and having a fully defined sequence; Derivatives thereof the peptide sequence being part of a ring structure
- C07K9/008—Peptides having up to 20 amino acids, containing saccharide radicals and having a fully defined sequence; Derivatives thereof the peptide sequence being part of a ring structure directly attached to a hetero atom of the saccharide radical, e.g. actaplanin, avoparcin, ristomycin, vancomycin
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/10—Tetrapeptides
- C07K5/1002—Tetrapeptides with the first amino acid being neutral
- C07K5/1016—Tetrapeptides with the first amino acid being neutral and aromatic or cycloaliphatic
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P20/00—Technologies relating to chemical industry
- Y02P20/50—Improvements relating to the production of bulk chemicals
- Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
General Health & Medical Sciences (AREA)
Medicinal Chemistry (AREA)
Life Sciences & Earth Sciences (AREA)
Biophysics (AREA)
Biochemistry (AREA)
Genetics & Genomics (AREA)
Molecular Biology (AREA)
Proteomics, Peptides & Aminoacids (AREA)
Oncology (AREA)
Communicable Diseases (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Pharmacology & Pharmacy (AREA)
Animal Behavior & Ethology (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Peptides Or Proteins (AREA)
Medicines Containing Material From Animals Or Micro-Organisms (AREA)

AT91920590T 1990-12-10 1991-11-28 Aus dalbaheptide hergestellte tetrapeptidantibiotika. ATE121101T1 (de)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
EP90123672		1990-12-10

Publications (1)

Publication Number	Publication Date
ATE121101T1 true ATE121101T1 (de)	1995-04-15

Family

ID=8204819

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
AT91920590T ATE121101T1 (de)	1990-12-10	1991-11-28	Aus dalbaheptide hergestellte tetrapeptidantibiotika.

Country Status (10)

Country	Link
EP (1)	EP0561827B1 (de)
JP (1)	JP3276632B2 (de)
KR (1)	KR100202250B1 (de)
AT (1)	ATE121101T1 (de)
CA (1)	CA2098098C (de)
DE (1)	DE69108930T2 (de)
DK (1)	DK0561827T3 (de)
ES (1)	ES2071346T3 (de)
IE (1)	IE914265A1 (de)
WO (1)	WO1992010517A1 (de)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
AU683881B2 (en) *	1993-05-19	1997-11-27	Vicuron Pharmaceuticals Inc.	Synthetic aglucodalbaheptide antibiotics

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
ES2110401T3 (es) *	1989-07-18	1998-02-16	Biosearch Italia Spa	Antibioticos pentapeptidicos derivados de dalbaheptidos.

1991
- 1991-11-28 DK DK91920590.6T patent/DK0561827T3/da active
- 1991-11-28 JP JP51867691A patent/JP3276632B2/ja not_active Expired - Fee Related
- 1991-11-28 WO PCT/EP1991/002250 patent/WO1992010517A1/en not_active Ceased
- 1991-11-28 EP EP91920590A patent/EP0561827B1/de not_active Expired - Lifetime
- 1991-11-28 CA CA002098098A patent/CA2098098C/en not_active Expired - Fee Related
- 1991-11-28 AT AT91920590T patent/ATE121101T1/de not_active IP Right Cessation
- 1991-11-28 ES ES91920590T patent/ES2071346T3/es not_active Expired - Lifetime
- 1991-11-28 DE DE69108930T patent/DE69108930T2/de not_active Expired - Fee Related
- 1991-11-28 KR KR1019930701721A patent/KR100202250B1/ko not_active Expired - Fee Related
- 1991-12-09 IE IE426591A patent/IE914265A1/en not_active IP Right Cessation

Also Published As

Publication number	Publication date
EP0561827A1 (de)	1993-09-29
JP3276632B2 (ja)	2002-04-22
WO1992010517A1 (en)	1992-06-25
CA2098098C (en)	2003-04-08
JPH06503307A (ja)	1994-04-14
EP0561827B1 (de)	1995-04-12
CA2098098A1 (en)	1992-06-10
KR930703358A (ko)	1993-11-29
DE69108930T2 (de)	1995-08-24
IE914265A1 (en)	1992-06-17
KR100202250B1 (ko)	1999-06-15
DE69108930D1 (de)	1995-05-18
ES2071346T3 (es)	1995-06-16
DK0561827T3 (da)	1995-07-03

Legal Events

Date	Code	Title
1996-03-15	UEP	Publication of translation of european patent specification
2003-12-15	EEIH	Change in the person of patent owner
2005-08-15	REN	Ceased due to non-payment of the annual fee

Publication	Publication Date	Title
ATE302180T1 (de)	2005-09-15	Zwischenprodukte zur herstellung von non-peptiden retroviralproteasehemmenden verbindungen
AU551463B2 (en)	1986-05-01	2-oxoazetidine derivatives
DK0876388T3 (da)	2004-06-07	Tricykliske erythromycinderivater
IT7909592A0 (it)	1979-11-12	Procedimento per la produzione di un derivato n acilato selettivamente protetto di un antibiotico amino glicosidico
CA2021379A1 (en)	1991-01-19	Pentapeptide antibiotics derived from dalbaheptides
FI893842A0 (fi)	1989-08-15	Menetelmä uuden antibiootin, mersasidiinin, valmistamiseksi
DE69108930D1 (de)	1995-05-18	Aus dalbaheptide hergestellte tetrapeptidantibiotika.
ATE159533T1 (de)	1997-11-15	Syntetische aglukodalbaheptid-antibiotika
ES2121293T3 (es)	1998-11-16	Uso de trovafloxacina o derivados de la misma para la fabricacion de un medicamento para el tratamiento de infecciones por h. pylori.
ES2144271T3 (es)	2000-06-01	Sintesis de derivados de acido carboxilico.
GR1001309B (el)	1993-08-31	Μεθοδος παρασκευης παραγωγου ενωσεως της διχλωροανιλινης.
DE69116383D1 (de)	1996-02-22	Hexapeptidderivate von teicoplanin und verfahren zu deren herstellung
ES2191778T3 (es)	2003-09-16	Derivados de 3-desoxi-3-descladinosa de las eritromicinas a y b.
HUP9601528A2 (hu)	1998-10-28	Véralvadásgátló hatású peptidszármazékok és a vegyületeket tartalmazó gyógyszerkészítmények
HUP9601525A2 (hu)	1998-10-28	Trombin- és Xa-faktor-gátló hatású peptidil-arginin-aldehid-származékok és a vegyületeket tartalmazó gyógyszerkészítmények
KR940022256U (ko)	1994-10-19	사출성형기용 셧 오프(Shut Off)식 노즐의 구조