ATE240300T1 - Verfahren zur herstellung von phenylimidazolin- derivaten - Google Patents

Verfahren zur herstellung von phenylimidazolin- derivaten

Info

Publication number
ATE240300T1
ATE240300T1 AT96938306T AT96938306T ATE240300T1 AT E240300 T1 ATE240300 T1 AT E240300T1 AT 96938306 T AT96938306 T AT 96938306T AT 96938306 T AT96938306 T AT 96938306T AT E240300 T1 ATE240300 T1 AT E240300T1
Authority
AT
Austria
Prior art keywords
phenylimidazoline
derivatives
producing
producing phenylimidazoline
phenylimidazoline derivatives
Prior art date
Application number
AT96938306T
Other languages
English (en)
Inventor
Rapha L Bouchet
Michel Delthil
Daniel Guilmard
Philippe Mackiewicz
Original Assignee
Aventis Pharma Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Aventis Pharma Sa filed Critical Aventis Pharma Sa
Application granted granted Critical
Publication of ATE240300T1 publication Critical patent/ATE240300T1/de

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/66—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D233/72—Two oxygen atoms, e.g. hydantoin
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
    • C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
    • C07D491/10—Spiro-condensed systems
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Solid-Sorbent Or Filter-Aiding Compositions (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
AT96938306T 1995-11-16 1996-11-14 Verfahren zur herstellung von phenylimidazolin- derivaten ATE240300T1 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR9513589A FR2741346B1 (fr) 1995-11-16 1995-11-16 Nouveau procede de preparation de derives phenylimidazolidine
PCT/FR1996/001794 WO1997018197A1 (fr) 1995-11-16 1996-11-14 Nouveau procede de preparation de derives phenylimidazolidine

Publications (1)

Publication Number Publication Date
ATE240300T1 true ATE240300T1 (de) 2003-05-15

Family

ID=9484624

Family Applications (1)

Application Number Title Priority Date Filing Date
AT96938306T ATE240300T1 (de) 1995-11-16 1996-11-14 Verfahren zur herstellung von phenylimidazolin- derivaten

Country Status (29)

Country Link
US (1) US6107488A (de)
EP (1) EP0877738B1 (de)
JP (1) JP2000500150A (de)
KR (1) KR100466991B1 (de)
CN (1) CN1131219C (de)
AR (1) AR004965A1 (de)
AT (1) ATE240300T1 (de)
AU (1) AU718832B2 (de)
BR (1) BR9611573A (de)
CA (1) CA2235335A1 (de)
CU (1) CU22890A3 (de)
CZ (1) CZ144498A3 (de)
DE (1) DE69628203T2 (de)
DK (1) DK0877738T3 (de)
EA (1) EA002658B1 (de)
ES (1) ES2193271T3 (de)
FR (1) FR2741346B1 (de)
HU (1) HUP9904034A3 (de)
IL (1) IL124382A0 (de)
MX (1) MX9803730A (de)
NO (1) NO316514B1 (de)
PL (1) PL189697B1 (de)
PT (1) PT877738E (de)
SI (1) SI0877738T1 (de)
TR (1) TR199800865T2 (de)
TW (1) TW404942B (de)
UA (1) UA67720C2 (de)
WO (1) WO1997018197A1 (de)
ZA (1) ZA969442B (de)

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP1709193B1 (de) * 2003-12-19 2011-03-16 The Regents of The University of California Verfahren und materialien zur beurteilung von prostatakrebstherapien
WO2005099693A2 (en) * 2004-02-24 2005-10-27 The Regents Of The University Of California Methods and materials for assessing prostate cancer therapies and compounds
US7709517B2 (en) 2005-05-13 2010-05-04 The Regents Of The University Of California Diarylhydantoin compounds
ES2689292T3 (es) 2006-03-27 2018-11-13 The Regents Of The University Of California Modulador del receptor de andrógenos para el tratamiento del cáncer de próstata y enfermedades asociadas con el receptor de andrógenos
NZ572374A (en) 2006-03-29 2011-12-22 Univ California Diarylthiohydantoin compounds
EP2220050A2 (de) 2007-10-26 2010-08-25 The Regents Of The University Of California Diarylhydantoinverbindungen als androgenrezeptormodulatoren
JP2013504531A (ja) 2009-09-11 2013-02-07 バイエル・ファルマ・アクチェンゲゼルシャフト 抗癌薬としての置換（ヘテロアリールメチル）チオヒダントイン
US9482944B2 (en) 2009-09-15 2016-11-01 Mylan Group Copolymers, polymeric particles comprising said copolymers and copolymeric binders for radiation-sensitive coating compositions for negative-working radiation-sensitive lithographic printing plates
SG10201907588XA (en) 2010-02-16 2019-09-27 Aragon Pharmaceuticals Inc Androgen Receptor Modulators And Uses Thereof
KR101471310B1 (ko) 2010-09-14 2014-12-09 밀란 그룹 포지티브형 서멀 리소그래픽 인쇄판을 위한 근적외선-감응 코팅 조성물용 코폴리머
CN115737643A (zh) 2012-09-26 2023-03-07 阿拉贡药品公司 用于治疗非转移性去势抵抗性前列腺癌的抗雄激素
DK2945628T3 (da) 2013-01-15 2020-05-04 Aragon Pharmaceuticals Inc Androgen receptormodulator i kombination med abirateronacetat og prednison til behandling af prostatacancer
TWI726969B (zh) 2016-01-11 2021-05-11 比利時商健生藥品公司 用作雄性激素受體拮抗劑之經取代之硫尿囊素衍生物
MX2020003845A (es) 2017-10-16 2020-11-06 Aragon Pharmaceuticals Inc Antiandrógenos para el tratamiento de cáncer de próstata no metastásico resistente a la castración.
CN108218784A (zh) * 2018-01-16 2018-06-29 吴江信凯医药科技有限公司 一种尼鲁米特的制备方法

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS4916937B1 (de) * 1970-01-21 1974-04-25
JPS5136332B1 (de) * 1970-12-09 1976-10-07
CH544491A (de) * 1971-03-16 1973-11-30 Ciba Geigy Ag Herbizides Mittel
MC1220A1 (fr) * 1977-10-28 1979-07-20 Hoffmann La Roche Nouveaux derives d'imidazolidine
JPS57197268A (en) * 1981-05-29 1982-12-03 Sumitomo Chem Co Ltd Substituted phenylhydantoin derivative, its preparation, and herbicide containing the same as active ingredient
JPS62298562A (ja) * 1986-06-17 1987-12-25 Nippon Kayaku Co Ltd ブロモアニリン類の製造法
FR2656302B1 (fr) * 1989-12-22 1992-05-07 Roussel Uclaf Nouveau procede de preparation de l'anandron et derives de l'anandron.
US5411981A (en) * 1991-01-09 1995-05-02 Roussel Uclaf Phenylimidazolidines having antiandrogenic activity
FR2694290B1 (fr) * 1992-07-08 1994-09-02 Roussel Uclaf Nouvelles phénylimidazolidines éventuellement substituées, leur procédé de préparation, leur application comme médicaments et les compositions pharmaceutiques les renfermant.

Also Published As

Publication number Publication date
DK0877738T3 (da) 2003-09-08
EA002658B1 (ru) 2002-08-29
PL326491A1 (en) 1998-09-28
MX9803730A (es) 1998-11-30
PL189697B1 (pl) 2005-09-30
EP0877738A1 (de) 1998-11-18
CU22890A3 (es) 2004-01-23
TR199800865T2 (xx) 1998-08-21
TW404942B (en) 2000-09-11
KR100466991B1 (ko) 2005-04-06
NO982237L (no) 1998-07-10
HUP9904034A2 (hu) 2000-05-28
IL124382A0 (en) 1998-12-06
FR2741346B1 (fr) 1997-12-19
PT877738E (pt) 2003-09-30
DE69628203D1 (de) 2003-06-18
EA199800378A1 (ru) 1998-10-29
KR19990067639A (ko) 1999-08-25
NO316514B1 (no) 2004-02-02
AU718832B2 (en) 2000-04-20
WO1997018197A1 (fr) 1997-05-22
CZ144498A3 (cs) 1998-09-16
EP0877738B1 (de) 2003-05-14
JP2000500150A (ja) 2000-01-11
CN1131219C (zh) 2003-12-17
HUP9904034A3 (en) 2001-08-28
CA2235335A1 (fr) 1997-05-22
AU7577396A (en) 1997-06-05
SI0877738T1 (en) 2003-10-31
ES2193271T3 (es) 2003-11-01
US6107488A (en) 2000-08-22
AR004965A1 (es) 1999-04-07
CN1207732A (zh) 1999-02-10
NO982237D0 (no) 1998-05-15
FR2741346A1 (fr) 1997-05-23
ZA969442B (en) 1997-11-11
BR9611573A (pt) 1999-05-11
DE69628203T2 (de) 2004-02-05
UA67720C2 (en) 2004-07-15

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