ZA968957B - Process for the preparation of dihaloazolopyrimidines. - Google Patents

Process for the preparation of dihaloazolopyrimidines.

Info

Publication number
ZA968957B
ZA968957B ZA9608957A ZA968957A ZA968957B ZA 968957 B ZA968957 B ZA 968957B ZA 9608957 A ZA9608957 A ZA 9608957A ZA 968957 A ZA968957 A ZA 968957A ZA 968957 B ZA968957 B ZA 968957B
Authority
ZA
South Africa
Prior art keywords
dihaloazolopyrimidines
preparation
Prior art date
Application number
ZA9608957A
Other languages
English (en)
Inventor
Guenter Krummel
Karl-Otto Stumm
Klaus-Juergen Pees
Peter Heinz Rudi Liers
Original Assignee
American Cyanamid Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by American Cyanamid Co filed Critical American Cyanamid Co
Publication of ZA968957B publication Critical patent/ZA968957B/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
ZA9608957A 1995-10-27 1996-10-24 Process for the preparation of dihaloazolopyrimidines. ZA968957B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US802295P 1995-10-27 1995-10-27

Publications (1)

Publication Number Publication Date
ZA968957B true ZA968957B (en) 1998-04-24

Family

ID=21729405

Family Applications (1)

Application Number Title Priority Date Filing Date
ZA9608957A ZA968957B (en) 1995-10-27 1996-10-24 Process for the preparation of dihaloazolopyrimidines.

Country Status (22)

Country Link
US (1) US5808066A (de)
EP (1) EP0770615B1 (de)
JP (1) JP4018182B2 (de)
KR (1) KR100443182B1 (de)
AR (1) AR004122A1 (de)
AT (1) ATE243211T1 (de)
BR (1) BR9605258A (de)
CA (1) CA2188905C (de)
DE (1) DE69628712T2 (de)
DK (1) DK0770615T3 (de)
ES (1) ES2202419T3 (de)
HU (1) HU217773B (de)
IL (1) IL119496A (de)
MX (1) MX9604882A (de)
PT (1) PT770615E (de)
RU (1) RU2147584C1 (de)
SG (1) SG55239A1 (de)
SI (1) SI0770615T1 (de)
SK (1) SK284071B6 (de)
TR (1) TR199600792A2 (de)
UA (1) UA48132C2 (de)
ZA (1) ZA968957B (de)

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NZ506247A (en) * 1998-02-11 2003-03-28 American Cyanamid Co Fungicidal 7-(alkyl, alkenyl, alkadienyl, cycloalkyl, cycloalkenyl or aryl)-[1,2,4]triazolo[1,5-a]pyrimidines
US6117865A (en) * 1998-09-10 2000-09-12 American Cyanamid Company Fungicidal trifluorophenyl-triazolopyrimidines
US6380202B1 (en) * 1998-09-25 2002-04-30 Basf Aktiengesellschaft Fungicidal fluoro-substituted 7-heterocyclyl-triazolopyrimidines
US6242451B1 (en) * 1998-09-25 2001-06-05 Klaus-Juergen Pees Fungicidal trihalophenyl-triazolopyrimidines
US6156925A (en) * 1998-09-25 2000-12-05 American Cyanamid Company Process for the preparation of halogenated phenylmaloates
US6559151B2 (en) 2000-05-08 2003-05-06 Basf Aktiengesellschaft 6-(2-trifluoromethyl-phenyl)-triazolopyrimidines
US6756379B2 (en) 2001-07-26 2004-06-29 Taro Pharmaceutical Industries Ltd. Non-sedating barbiturate compounds as neuroprotective agents
US7683071B2 (en) * 2000-07-26 2010-03-23 Taro Pharmaceuticals Industries Ltd. Composition and method for improved bioavailability and enhanced brain delivery of 5,5-diphenyl barbituric acid
US6939873B2 (en) * 2000-07-26 2005-09-06 Taro Pharmaceuticals Industries Limited Non-sedating barbituric acid derivatives
DE10063115A1 (de) * 2000-12-18 2002-06-27 Bayer Ag Triazolopyrimidine
JP2002249492A (ja) * 2000-12-22 2002-09-06 Nippon Bayer Agrochem Co Ltd トリアゾロピリミジン類
DE10121101A1 (de) * 2001-04-27 2002-10-31 Bayer Ag Triazolopyrimidine
US7300908B2 (en) 2001-07-05 2007-11-27 Basf Aktiengesellschaft Fungicidal triazolopyrimidines, method for the production thereof and use thereof in controlling noxious fungi and agents containing said compounds
JP2005504743A (ja) 2001-07-18 2005-02-17 ビーエーエスエフ アクチェンゲゼルシャフト 殺菌薬としての置換された６−（２−メトキシ−フェニル）−トリアゾロピリミジン
UA76486C2 (en) 2001-07-26 2006-08-15 Basf Ag 7-amino triazolopyrimidines, a process of praparation, a fungicidal preparations based thereon and a method to control phytopathogenic fungi
US7211545B2 (en) 2001-09-04 2007-05-01 Sumitomo Chemical Company, Limited Imidazo[1,2-a]pyrimidine and fungicidal compositions containing thereof
WO2003080615A1 (de) 2002-03-21 2003-10-02 Basf Aktiengesellschaft Fungizide triazolopyrimidine, verfahren zu ihrer herstellung und ihre verwendung zur bekämpfung von schadpilzen sowie sie enthaltende mittel
CL2003002588A1 (es) * 2002-12-11 2005-01-07 Taro Pharmaceuticals Ireland L Uso de una composicion farmaceutica que comprende acido n,n-dimetoximetildifenil barbiturico, acido n-metoximetildifenil barbiturico o acido difenil barbiturico o una sal farmaceuticamente aceptable del mismo para preparar un medicamento util en el t
US7419982B2 (en) * 2003-09-24 2008-09-02 Wyeth Holdings Corporation Crystalline forms of 5-chloro-6-{2,6-difluoro-4-[3-(methylamino)propoxy]phenyl}-N-[(1S)-2,2,2-trifluoro-1-methylethyl][1,2,4]triazolo[1,5-a]pyrimidin-7-amine salts
MXPA06003206A (es) * 2003-09-24 2006-06-23 Wyeth Corp 6-[(sustituido)fenil]triazolopirimidinas como agentes anticancer.
JP4695595B2 (ja) * 2003-09-24 2011-06-08 ワイス・ホールディングズ・コーポレイション 抗癌剤としての６−アリール−７−ハロ−イミダゾ［１，２−ａ］ピリミジン類
MY179926A (en) * 2003-12-08 2020-11-19 Wyeth Corp Process for the preparation of tubulin inhibitors
TW200533670A (en) * 2003-12-19 2005-10-16 Basf Ag 6-(aminocarbonylphenyl)triazolopyrimidines, their preparation and their use for controlling harmful fungi, and compositions comprising these compounds
DE102004007076A1 (de) * 2004-02-13 2005-08-25 Bayer Cropscience Ag Imidazolopyrimidine
DE502005009861D1 (de) * 2004-03-10 2010-08-19 Basf Se 5,6-dialkyl-7-amino-triazolopyrimidine, verfahren zu ihrer herstellung und ihre verwendung zur bekämpfung von schadpilzen sowie sie enthaltende mittel
US9487519B2 (en) * 2004-03-10 2016-11-08 Basf Se 5,6-Dialkyl-7-aminotriazolopyrimidines, their preparation and their use for controlling harmful fungi, and compositions comprising these compounds
PE20060020A1 (es) * 2004-03-30 2006-03-10 Basf Ag 5-6-cicloalquil-7-amino-triazolopirimidinas para combatir hongos fitopatogenos y procedimientos para su obtencion
EP1781624A4 (de) * 2004-07-02 2010-06-23 Taro Pharma Ind Verfahren zur herstellung von 1-methoxymethyl-5,5-diphenylbarbitursäure
EP1856118A1 (de) * 2005-03-01 2007-11-21 Basf Aktiengesellschaft 5,6-dialkyl-7-amino-azolopyrimidine, verfahren zu ihrer herstellung und ihre verwendung zur bekämpfung von schadpilzen sowie sie enthaltende mittel
US20080125445A1 (en) * 2005-03-01 2008-05-29 Basf Aktiengesellschaft 5,6-Dialkyl-7-Amino-Azolopyrimidines, Method For Their Production, Their Use For Controlling Pathogenic Fungi and Agents Containing Said Compounds
US20080188493A1 (en) * 2005-03-01 2008-08-07 Basf Aktiengesellschaft 5,6-Dialkyl-7-Aminoazolopyrimidines, Their Preparation and Their Use For Controlling Harmful Fungi, and Compositions Comprising These Compounds
EP1856122A2 (de) * 2005-03-02 2007-11-21 Basf Aktiengesellschaft 2-substituierte 7-amino-azolopyrimidine, verfahren zu ihrer herstellung und ihre verwendung zur bekämpfung von schadpilzen sowie sie enthaltende mittel
BRPI0608411A2 (pt) * 2005-03-10 2009-12-29 Basf Ag uso de um composto, composto, processo para preparar compostos, agente, semente, e, processo para combater fungos nocivos fitopatogênicos
BRPI0608712A2 (pt) * 2005-03-18 2010-12-07 Basf Ag processo para a preparação de composto, e, uso do composto
US20090131708A1 (en) * 2005-06-27 2009-05-21 Basf Aktiengesellschaft Method For Production of Substituted Phenylmalonate Esters, Intermediate Compounds and The Use Thereof for production of 5, 7-dihydroxy-6-(2,4,5-trifluorophenyl)-(1,2,4)triazolo(1,5-A)pyrimidines
US20080200675A1 (en) * 2005-06-27 2008-08-21 Basf Aktiengesellschaft Method for Production of Substituted Phenylmalonate Esters, Novel Phenylmalonate Esters and Use Thereof
WO2008066704A2 (en) * 2006-11-14 2008-06-05 Taro Pharmaceuticals North America, Inc. Method of improving bioavailability for non-sedating barbiturates
CN101583613A (zh) * 2007-01-11 2009-11-18 巴斯夫欧洲公司 生产芳基取代的稠合嘧啶的方法
WO2011082271A2 (en) * 2009-12-30 2011-07-07 Arqule, Inc. Substituted triazolo-pyrimidine compounds

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US3907799A (en) * 1971-08-16 1975-09-23 Icn Pharmaceuticals Xanthine oxidase inhibitors
AU557300B2 (en) * 1982-03-16 1986-12-18 Farmitalia Carlo Erba S.P.A. Substituted 1h-pyrazolo(1,5-alpha)pyrimidines and processes for their preparation
JPS5962593A (ja) * 1982-09-30 1984-04-10 Ss Pharmaceut Co Ltd ３―置換―５，７―ジクロルトリアゾロピリミジン誘導体
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US4910306A (en) * 1987-11-09 1990-03-20 The Dow Chemical Company Preparation of substituted 1,2,4-triazolo[1,5-a]pyrimidine-2-sulfonanilides
US4892945A (en) * 1987-12-21 1990-01-09 Ciba-Geigy Corporation Isoindoline pigments containing at least one triazolopyrimidone radical
US5006656A (en) * 1990-02-26 1991-04-09 Dowelanco Preparation of 5,7-dihydroxy-1,2,4-triazolo[1,5-a]pyrimidine-2-sulfonanilides
WO1992018504A1 (en) * 1991-04-22 1992-10-29 Otsuka Pharmaceutical Factory, Inc. PYRAZOLO[1,5-a]PYRIMIDINE DERIVATIVE AND ANTI-INFLAMMATORY CONTAINING THE SAME
US5356897A (en) * 1991-09-09 1994-10-18 Fujisawa Pharmaceutical Co., Ltd. 3-(heteroaryl)-pyrazololi[1,5-a]pyrimidines
US5177206A (en) * 1991-10-08 1993-01-05 Dowelanco Process for the preparation of substituted N-(aryl)-1,2,4-triazolopyrimidine-2-sulfonamides
TW224044B (de) * 1991-12-30 1994-05-21 Shell Internat Res Schappej B V
IL108731A (en) * 1993-03-04 1997-03-18 Shell Int Research 6, N-DISUBSTITUTED-£1, 2, 4| TRIAZOLO-£1, 5-a| PYRIMIDINE- 7-AMINE DERIVATIVES, THEIR PREPARATION AND THEIR USE AS FUNGICIDES
RU2066295C1 (ru) * 1993-05-19 1996-09-10 Институт структурной макрокинетики РАН Способ получения порошкового материала на основе карбида титана
EP0628559B1 (de) * 1993-06-10 2002-04-03 Beiersdorf-Lilly GmbH Pyrimidinverbindungen und ihre Verwendung als Pharmazeutika
CA2171003C (en) * 1993-10-18 2005-12-13 James W. Ringer Process for preparing n-(2,6-dichloro-3-methylphenyl)-5-7-dihalo[1,2,4]triazolo[1,5a]pyrimidine-2-sulfonamide by cyclization and halo-dehydroxylation

Also Published As

Publication number Publication date
EP0770615B1 (de) 2003-06-18
SG55239A1 (en) 1998-12-21
HUP9602957A2 (en) 1997-06-30
SI0770615T1 (en) 2003-12-31
DE69628712T2 (de) 2004-04-29
MX9604882A (es) 1997-04-30
HU217773B (hu) 2000-04-28
UA48132C2 (uk) 2002-08-15
SK137796A3 (en) 1997-05-07
TR199600792A2 (tr) 1997-05-21
IL119496A0 (en) 1997-01-10
PT770615E (pt) 2003-10-31
JPH09124651A (ja) 1997-05-13
SK284071B6 (sk) 2004-09-08
CA2188905A1 (en) 1997-04-28
EP0770615A1 (de) 1997-05-02
ES2202419T3 (es) 2004-04-01
KR970021081A (ko) 1997-05-28
IL119496A (en) 2001-07-24
ATE243211T1 (de) 2003-07-15
HUP9602957A3 (en) 1998-01-28
BR9605258A (pt) 1998-07-21
DK0770615T3 (da) 2003-07-14
KR100443182B1 (ko) 2005-04-19
US5808066A (en) 1998-09-15
HU9602957D0 (en) 1996-12-30
AR004122A1 (es) 1998-09-30
RU2147584C1 (ru) 2000-04-20
JP4018182B2 (ja) 2007-12-05
CA2188905C (en) 2005-12-06
DE69628712D1 (de) 2003-07-24

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