SG55239A1 - Process for the preparation of dihaloazpyrimidines - Google Patents
Process for the preparation of dihaloazpyrimidinesInfo
- Publication number
- SG55239A1 SG55239A1 SG1996010896A SG1996010896A SG55239A1 SG 55239 A1 SG55239 A1 SG 55239A1 SG 1996010896 A SG1996010896 A SG 1996010896A SG 1996010896 A SG1996010896 A SG 1996010896A SG 55239 A1 SG55239 A1 SG 55239A1
- Authority
- SG
- Singapore
- Prior art keywords
- dihaloazpyrimidines
- preparation
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US802295P | 1995-10-27 | 1995-10-27 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| SG55239A1 true SG55239A1 (en) | 1998-12-21 |
Family
ID=21729405
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| SG1996010896A SG55239A1 (en) | 1995-10-27 | 1996-10-18 | Process for the preparation of dihaloazpyrimidines |
Country Status (22)
| Country | Link |
|---|---|
| US (1) | US5808066A (de) |
| EP (1) | EP0770615B1 (de) |
| JP (1) | JP4018182B2 (de) |
| KR (1) | KR100443182B1 (de) |
| AR (1) | AR004122A1 (de) |
| AT (1) | ATE243211T1 (de) |
| BR (1) | BR9605258A (de) |
| CA (1) | CA2188905C (de) |
| DE (1) | DE69628712T2 (de) |
| DK (1) | DK0770615T3 (de) |
| ES (1) | ES2202419T3 (de) |
| HU (1) | HU217773B (de) |
| IL (1) | IL119496A (de) |
| MX (1) | MX9604882A (de) |
| PT (1) | PT770615E (de) |
| RU (1) | RU2147584C1 (de) |
| SG (1) | SG55239A1 (de) |
| SI (1) | SI0770615T1 (de) |
| SK (1) | SK284071B6 (de) |
| TR (1) | TR199600792A2 (de) |
| UA (1) | UA48132C2 (de) |
| ZA (1) | ZA968957B (de) |
Families Citing this family (40)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US6117876A (en) | 1997-04-14 | 2000-09-12 | American Cyanamid Company | Fungicidal trifluorophenyl-triazolopyrimidines |
| HUP0100885A3 (en) * | 1998-02-11 | 2002-12-28 | American Cyanamid Company Madi | Fungicidal 7-alkyl-triazolopyrimidines |
| US6117865A (en) * | 1998-09-10 | 2000-09-12 | American Cyanamid Company | Fungicidal trifluorophenyl-triazolopyrimidines |
| US6156925A (en) * | 1998-09-25 | 2000-12-05 | American Cyanamid Company | Process for the preparation of halogenated phenylmaloates |
| US6242451B1 (en) * | 1998-09-25 | 2001-06-05 | Klaus-Juergen Pees | Fungicidal trihalophenyl-triazolopyrimidines |
| US6380202B1 (en) * | 1998-09-25 | 2002-04-30 | Basf Aktiengesellschaft | Fungicidal fluoro-substituted 7-heterocyclyl-triazolopyrimidines |
| US6559151B2 (en) | 2000-05-08 | 2003-05-06 | Basf Aktiengesellschaft | 6-(2-trifluoromethyl-phenyl)-triazolopyrimidines |
| US6756379B2 (en) | 2001-07-26 | 2004-06-29 | Taro Pharmaceutical Industries Ltd. | Non-sedating barbiturate compounds as neuroprotective agents |
| US7683071B2 (en) * | 2000-07-26 | 2010-03-23 | Taro Pharmaceuticals Industries Ltd. | Composition and method for improved bioavailability and enhanced brain delivery of 5,5-diphenyl barbituric acid |
| US6939873B2 (en) * | 2000-07-26 | 2005-09-06 | Taro Pharmaceuticals Industries Limited | Non-sedating barbituric acid derivatives |
| DE10063115A1 (de) * | 2000-12-18 | 2002-06-27 | Bayer Ag | Triazolopyrimidine |
| JP2002249492A (ja) * | 2000-12-22 | 2002-09-06 | Nippon Bayer Agrochem Co Ltd | トリアゾロピリミジン類 |
| DE10121101A1 (de) * | 2001-04-27 | 2002-10-31 | Bayer Ag | Triazolopyrimidine |
| KR100619216B1 (ko) | 2001-07-05 | 2006-09-08 | 바스프 악티엔게젤샤프트 | 살진균성 트리아졸로피리미딘, 이의 제조방법 및 유해진균 방제를 위한 이의 용도 및 상기 화합물을 포함하는조성물 |
| US7038047B2 (en) | 2001-07-18 | 2006-05-02 | Basf Aktiengesellschaft | Substituted 6-(2-methoxyphenyl) triazolopyrimides as fungicides |
| HUP0401488A2 (hu) | 2001-07-26 | 2004-12-28 | Basf Aktiengesellschaft | Fungicid hatású 7-amino-triazolopirimidinek, előállításuk, alkalmazásuk és ilyeneket tartalmazó készítmények |
| ES2287312T3 (es) | 2001-09-04 | 2007-12-16 | Sumitomo Chemical Company, Limited | Imidazo(1,2-a)pirimidinas y composiciones fungicidas que las contienen. |
| CA2479766A1 (en) | 2002-03-21 | 2003-10-02 | Basf Aktiengesellschaft | Fungicidal triazolopyrimidines, methods for producing the same, use thereof for combating harmful fungi and agents containing said substances |
| WO2004052350A2 (en) * | 2002-12-11 | 2004-06-24 | Taro Pharmaceutical Industries Limited | Method of treating movement disorders using barbituric acid derivatives |
| US7419982B2 (en) * | 2003-09-24 | 2008-09-02 | Wyeth Holdings Corporation | Crystalline forms of 5-chloro-6-{2,6-difluoro-4-[3-(methylamino)propoxy]phenyl}-N-[(1S)-2,2,2-trifluoro-1-methylethyl][1,2,4]triazolo[1,5-a]pyrimidin-7-amine salts |
| SI1680425T1 (sl) * | 2003-09-24 | 2007-04-30 | Wyeth Corp | 6-((substituirani)fenil)triazolopirimidini kot sredstva proti raku |
| ES2308256T3 (es) * | 2003-09-24 | 2008-12-01 | Wyeth Holdings Corporation | 6-aril-7-halo-imidazo(1,2-a)pirimidinas como agentes anticancerosos. |
| MY179926A (en) * | 2003-12-08 | 2020-11-19 | Wyeth Corp | Process for the preparation of tubulin inhibitors |
| TW200533670A (en) * | 2003-12-19 | 2005-10-16 | Basf Ag | 6-(aminocarbonylphenyl)triazolopyrimidines, their preparation and their use for controlling harmful fungi, and compositions comprising these compounds |
| DE102004007076A1 (de) * | 2004-02-13 | 2005-08-25 | Bayer Cropscience Ag | Imidazolopyrimidine |
| DE502005009862D1 (de) * | 2004-03-10 | 2010-08-19 | Basf Se | 5,6-dialkyl-7-aminotriazolopyrimidine, verfahren zu ihrer herstellung und ihre verwendung zur bekämpfung von schadpilzen sowie sie enthaltende mittel |
| EP1725560B1 (de) * | 2004-03-10 | 2010-07-07 | Basf Se | 5,6-dialkyl-7-amino-triazolopyrimidine, verfahren zu ihrer herstellung und ihre verwendung zur bekämpfung von schadpilzen sowie sie enthaltende mittel |
| PE20060020A1 (es) * | 2004-03-30 | 2006-03-10 | Basf Ag | 5-6-cicloalquil-7-amino-triazolopirimidinas para combatir hongos fitopatogenos y procedimientos para su obtencion |
| WO2006003651A2 (en) * | 2004-07-02 | 2006-01-12 | Taro Pharmaceutical Industries, Ltd | A process for preparing 1-methoxymethyl-5,5-diphenylbarbituric acid |
| JP2008536806A (ja) * | 2005-03-01 | 2008-09-11 | ビーエーエスエフ ソシエタス・ヨーロピア | ５，６−ジアルキル−７−アミノアゾロピリミジン、それらの製造方法、植物病原性菌類を防除するためのそれらの使用、および該化合物を含む薬剤 |
| JP2008532944A (ja) * | 2005-03-01 | 2008-08-21 | ビーエーエスエフ ソシエタス・ヨーロピア | ５，６−ジアルキル−７−アミノアゾロピリミジン、それらの製造方法、有害な菌類を防除するためのそれらの使用、およびそれらの化合物を含む物質 |
| JP2008531653A (ja) * | 2005-03-01 | 2008-08-14 | ビーエーエスエフ ソシエタス・ヨーロピア | ５，６−ジアルキル−７−アミノアゾロピリミジン類、その調製法および有害菌類を防除するためのその使用、ならびにこれらの化合物を含む組成物 |
| US20080139581A1 (en) * | 2005-03-02 | 2008-06-12 | Basf Aktiengesellschaft | 2-Substituted 7-Aminoazolopyrimidines, Processes For Their Preparation And Their Use For Controlling Harmful Fungi, And Compositions Comprising These Compounds |
| US20080176744A1 (en) * | 2005-03-10 | 2008-07-24 | Basf Aktiengesellschaft | Use of 4-Aminopyrimidines for Controlling Harmful Fungi, Novel 4-Aminopyrimidines, Processes for Their Preparation and Compositions Comprising Them |
| US20080146839A1 (en) * | 2005-03-18 | 2008-06-19 | Basf Aktiengesellschaft | Method for Producing 5-Halo-2,4,6-Trifluoroisophthalic Acid |
| CN101208289A (zh) * | 2005-06-27 | 2008-06-25 | 巴斯福股份公司 | 生产取代的苯基丙二酸酯中间体化合物的方法及其在生产5,7-二羟基-6-(2,4,6-三氟苯基)[1,2,4]三唑并[1,5-a]嘧啶中的用途 |
| CN101208287A (zh) * | 2005-06-27 | 2008-06-25 | 巴斯福股份公司 | 生产取代的苯基丙二酸酯的方法，新的苯基丙二酸酯及其用途 |
| EP2081576A4 (de) * | 2006-11-14 | 2010-06-30 | Taro Pharmaceuticals North Ame | Verfahren zur verbesserung der bioverfügbarkeit für nichtsedierende barbiturate |
| WO2008084082A1 (de) * | 2007-01-11 | 2008-07-17 | Basf Se | Verfahren zur herstellung arylsubstituierter anellierter pyrimidine |
| US8343977B2 (en) * | 2009-12-30 | 2013-01-01 | Arqule, Inc. | Substituted triazolo-pyrimidine compounds |
Family Cites Families (15)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3907799A (en) * | 1971-08-16 | 1975-09-23 | Icn Pharmaceuticals | Xanthine oxidase inhibitors |
| AU557300B2 (en) * | 1982-03-16 | 1986-12-18 | Farmitalia Carlo Erba S.P.A. | Substituted 1h-pyrazolo(1,5-alpha)pyrimidines and processes for their preparation |
| JPS5962593A (ja) * | 1982-09-30 | 1984-04-10 | Ss Pharmaceut Co Ltd | ３―置換―５，７―ジクロルトリアゾロピリミジン誘導体 |
| DE3522463A1 (de) * | 1985-06-22 | 1987-01-02 | Bayer Ag | Herbizide mittel |
| US4910306A (en) * | 1987-11-09 | 1990-03-20 | The Dow Chemical Company | Preparation of substituted 1,2,4-triazolo[1,5-a]pyrimidine-2-sulfonanilides |
| US4892945A (en) * | 1987-12-21 | 1990-01-09 | Ciba-Geigy Corporation | Isoindoline pigments containing at least one triazolopyrimidone radical |
| US5006656A (en) * | 1990-02-26 | 1991-04-09 | Dowelanco | Preparation of 5,7-dihydroxy-1,2,4-triazolo[1,5-a]pyrimidine-2-sulfonanilides |
| KR100191774B1 (ko) * | 1991-04-22 | 1999-06-15 | 오스카 아끼히꼬 | 피라졸로[1,5-알파] 피리미딘 유도체 및 이것을 함유하는 항염증제 |
| US5356897A (en) * | 1991-09-09 | 1994-10-18 | Fujisawa Pharmaceutical Co., Ltd. | 3-(heteroaryl)-pyrazololi[1,5-a]pyrimidines |
| US5177206A (en) * | 1991-10-08 | 1993-01-05 | Dowelanco | Process for the preparation of substituted N-(aryl)-1,2,4-triazolopyrimidine-2-sulfonamides |
| TW224044B (de) * | 1991-12-30 | 1994-05-21 | Shell Internat Res Schappej B V | |
| IL108731A (en) * | 1993-03-04 | 1997-03-18 | Shell Int Research | 6, N-DISUBSTITUTED-£1, 2, 4| TRIAZOLO-£1, 5-a| PYRIMIDINE- 7-AMINE DERIVATIVES, THEIR PREPARATION AND THEIR USE AS FUNGICIDES |
| RU2066295C1 (ru) * | 1993-05-19 | 1996-09-10 | Институт структурной макрокинетики РАН | Способ получения порошкового материала на основе карбида титана |
| EP0628559B1 (de) * | 1993-06-10 | 2002-04-03 | Beiersdorf-Lilly GmbH | Pyrimidinverbindungen und ihre Verwendung als Pharmazeutika |
| DE69429728T2 (de) * | 1993-10-18 | 2002-10-31 | Dow Agrosciences Llc, Indianapolis | Verfahren zur herstellung von n-(2,6-dichloro-3-methylphenyl)-5-7-dihalo[1,2,4]triazolo[1,5a]pyrimidin-2-sulfonamid durch cyclisierung und halo-dehydroxylierung |
-
1996
- 1996-09-30 RU RU96120421A patent/RU2147584C1/ru not_active IP Right Cessation
- 1996-10-03 TR TR96/00792A patent/TR199600792A2/xx unknown
- 1996-10-15 US US08/729,204 patent/US5808066A/en not_active Expired - Lifetime
- 1996-10-16 MX MX9604882A patent/MX9604882A/es not_active IP Right Cessation
- 1996-10-16 DK DK96307528T patent/DK0770615T3/da active
- 1996-10-16 AT AT96307528T patent/ATE243211T1/de not_active IP Right Cessation
- 1996-10-16 DE DE69628712T patent/DE69628712T2/de not_active Expired - Lifetime
- 1996-10-16 SI SI9630630T patent/SI0770615T1/xx unknown
- 1996-10-16 PT PT96307528T patent/PT770615E/pt unknown
- 1996-10-16 ES ES96307528T patent/ES2202419T3/es not_active Expired - Lifetime
- 1996-10-16 EP EP96307528A patent/EP0770615B1/de not_active Expired - Lifetime
- 1996-10-18 SG SG1996010896A patent/SG55239A1/en unknown
- 1996-10-23 UA UA96104029A patent/UA48132C2/uk unknown
- 1996-10-23 JP JP29790396A patent/JP4018182B2/ja not_active Expired - Fee Related
- 1996-10-24 ZA ZA9608957A patent/ZA968957B/xx unknown
- 1996-10-25 SK SK1377-96A patent/SK284071B6/sk unknown
- 1996-10-25 BR BR9605258A patent/BR9605258A/pt not_active IP Right Cessation
- 1996-10-25 CA CA002188905A patent/CA2188905C/en not_active Expired - Fee Related
- 1996-10-25 AR ARP960104928A patent/AR004122A1/es active IP Right Grant
- 1996-10-25 HU HU9602957A patent/HU217773B/hu not_active IP Right Cessation
- 1996-10-26 KR KR1019960048877A patent/KR100443182B1/ko not_active Expired - Fee Related
- 1996-10-27 IL IL11949696A patent/IL119496A/en not_active IP Right Cessation
Also Published As
| Publication number | Publication date |
|---|---|
| JP4018182B2 (ja) | 2007-12-05 |
| SK284071B6 (sk) | 2004-09-08 |
| HUP9602957A3 (en) | 1998-01-28 |
| KR970021081A (ko) | 1997-05-28 |
| ATE243211T1 (de) | 2003-07-15 |
| HU217773B (hu) | 2000-04-28 |
| US5808066A (en) | 1998-09-15 |
| SI0770615T1 (en) | 2003-12-31 |
| EP0770615B1 (de) | 2003-06-18 |
| JPH09124651A (ja) | 1997-05-13 |
| ZA968957B (en) | 1998-04-24 |
| SK137796A3 (en) | 1997-05-07 |
| DK0770615T3 (da) | 2003-07-14 |
| AR004122A1 (es) | 1998-09-30 |
| BR9605258A (pt) | 1998-07-21 |
| IL119496A (en) | 2001-07-24 |
| IL119496A0 (en) | 1997-01-10 |
| CA2188905C (en) | 2005-12-06 |
| TR199600792A2 (tr) | 1997-05-21 |
| EP0770615A1 (de) | 1997-05-02 |
| HU9602957D0 (en) | 1996-12-30 |
| UA48132C2 (uk) | 2002-08-15 |
| DE69628712D1 (de) | 2003-07-24 |
| KR100443182B1 (ko) | 2005-04-19 |
| PT770615E (pt) | 2003-10-31 |
| HUP9602957A2 (en) | 1997-06-30 |
| DE69628712T2 (de) | 2004-04-29 |
| ES2202419T3 (es) | 2004-04-01 |
| RU2147584C1 (ru) | 2000-04-20 |
| CA2188905A1 (en) | 1997-04-28 |
| MX9604882A (es) | 1997-04-30 |
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