ATE322260T1 - Nateglinide zubereitung in tablettenform - Google Patents

Nateglinide zubereitung in tablettenform

Info

Publication number: ATE322260T1
Authority: AT; Austria
Prior art keywords: tablet form; meals; carboxymethyl cellulose; tablet composition; nateglinide preparation
Prior art date: 1996-11-15

Application number

AT97912459T

Other languages

English (en)

Inventor

Akira Yabuki

Kawasaki-Ku

Masato Kaida

Takahiko Ando

Nobutaka Ninomiya

Masanao Ozaki

Original Assignee

Ajinomoto Kk

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1996-11-15

Filing date

1997-11-14

Publication date

2006-04-15

Family has litigation

First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=18100283&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=ATE322260(T1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.

1997-11-14 Application filed by Ajinomoto Kk filed Critical Ajinomoto Kk

2006-04-15 Application granted granted Critical

2006-04-15 Publication of ATE322260T1 publication Critical patent/ATE322260T1/de

Links

OELFLUMRDSZNSF-BRWVUGGUSA-N nateglinide Chemical compound C1C[C@@H](C(C)C)CC[C@@H]1C(=O)N[C@@H](C(O)=O)CC1=CC=CC=C1 OELFLUMRDSZNSF-BRWVUGGUSA-N 0.000 title abstract 2
229960000698 nateglinide Drugs 0.000 title 1
239000001768 carboxy methyl cellulose Substances 0.000 abstract 2
235000012054 meals Nutrition 0.000 abstract 2
239000007916 tablet composition Substances 0.000 abstract 2
OYPRJOBELJOOCE-UHFFFAOYSA-N Calcium Chemical compound [Ca] OYPRJOBELJOOCE-UHFFFAOYSA-N 0.000 abstract 1
229920002134 Carboxymethyl cellulose Polymers 0.000 abstract 1
DPXJVFZANSGRMM-UHFFFAOYSA-N acetic acid;2,3,4,5,6-pentahydroxyhexanal;sodium Chemical compound [Na].CC(O)=O.OCC(O)C(O)C(O)C(O)C=O DPXJVFZANSGRMM-UHFFFAOYSA-N 0.000 abstract 1
239000008280 blood Substances 0.000 abstract 1
210000004369 blood Anatomy 0.000 abstract 1
239000011575 calcium Substances 0.000 abstract 1
229910052791 calcium Inorganic materials 0.000 abstract 1
235000010948 carboxy methyl cellulose Nutrition 0.000 abstract 1
239000008112 carboxymethyl-cellulose Substances 0.000 abstract 1
235000019812 sodium carboxymethyl cellulose Nutrition 0.000 abstract 1
229920001027 sodium carboxymethylcellulose Polymers 0.000 abstract 1
210000002784 stomach Anatomy 0.000 abstract 1

Classifications

- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/185—Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
- A61K31/19—Carboxylic acids, e.g. valproic acid
- A61K31/195—Carboxylic acids, e.g. valproic acid having an amino group
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
- A61K9/2806—Coating materials
- A61K9/2833—Organic macromolecular compounds
- A61K9/2853—Organic macromolecular compounds obtained otherwise than by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyethylene glycol, polyethylene oxide, poloxamers, poly(lactide-co-glycolide)
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/185—Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
- A61K31/19—Carboxylic acids, e.g. valproic acid
- A61K31/195—Carboxylic acids, e.g. valproic acid having an amino group
- A61K31/197—Carboxylic acids, e.g. valproic acid having an amino group the amino and the carboxyl groups being attached to the same acyclic carbon chain, e.g. gamma-aminobutyric acid [GABA], beta-alanine, epsilon-aminocaproic acid or pantothenic acid
- A61K31/198—Alpha-amino acids, e.g. alanine or edetic acid [EDTA]
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2022—Organic macromolecular compounds
- A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
- A61K9/2054—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
- A61K9/2806—Coating materials
- A61K9/2833—Organic macromolecular compounds
- A61K9/286—Polysaccharides, e.g. gums; Cyclodextrin
- A61K9/2866—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Pharmacology & Pharmacy (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Epidemiology (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Diabetes (AREA)
Emergency Medicine (AREA)
Endocrinology (AREA)
Hematology (AREA)
Obesity (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Organic Chemistry (AREA)
Medicinal Preparation (AREA)
Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Medicines Containing Plant Substances (AREA)

AT97912459T 1996-11-15 1997-11-14 Nateglinide zubereitung in tablettenform ATE322260T1 (de)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
JP31854196		1996-11-15

Publications (1)

Publication Number	Publication Date
ATE322260T1 true ATE322260T1 (de)	2006-04-15

Family

ID=18100283

Family Applications (2)

Application Number	Title	Priority Date	Filing Date
AT05014497T ATE503472T1 (de)	1996-11-15	1997-11-14	Nateglinide-tablettenzubereitungen
AT97912459T ATE322260T1 (de)	1996-11-15	1997-11-14	Nateglinide zubereitung in tablettenform

Family Applications Before (1)

Application Number	Title	Priority Date	Filing Date
AT05014497T ATE503472T1 (de)	1996-11-15	1997-11-14	Nateglinide-tablettenzubereitungen

Country Status (14)

Country	Link
US (4)	US6143323A (de)
EP (3)	EP1586314B1 (de)
JP (1)	JP4171091B2 (de)
KR (1)	KR100343062B1 (de)
CN (1)	CN1245158C (de)
AT (2)	ATE503472T1 (de)
AU (1)	AU718350B2 (de)
CA (1)	CA2271865C (de)
DE (2)	DE69740161D1 (de)
DK (1)	DK1586314T3 (de)
ES (2)	ES2364145T3 (de)
PT (2)	PT965339E (de)
TW (1)	TW492878B (de)
WO (1)	WO1998022105A1 (de)

Families Citing this family (34)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
ATE503472T1 (de)	1996-11-15	2011-04-15	Ajinomoto Kk	Nateglinide-tablettenzubereitungen
DE69934505T2 (de)	1998-05-18	2007-10-04	Takeda Pharmaceutical Co. Ltd.	Im munde zerfallende tablette enthaltend ein benzimidazole
TW585786B (en) *	1998-07-28	2004-05-01	Takeda Chemical Industries Ltd	Lansoprazole-containing rapidly disintegrable solid pharmaceutical composition
JP2000119160A (ja) *	1998-10-06	2000-04-25	Kanebo Ltd	皮膚化粧料
US6559188B1 (en)	1999-09-17	2003-05-06	Novartis Ag	Method of treating metabolic disorders especially diabetes, or a disease or condition associated with diabetes
CO5200844A1 (es) *	1999-09-17	2002-09-27	Novartis Ag	Una combinacion que comprende nateglinida y cuando por menos otro compuesto antidiabetico usada para el tratamiento de desordenes metabolicos, especialmente diabetes, o de una enfermedad o condicion asociada con dibetes
US6878749B2 (en)	1999-09-17	2005-04-12	Novartis Ag	Method of treating metabolic disorders, especially diabetes, or a disease or condition associated with diabetes
CA2395993A1 (en)	1999-12-28	2001-07-05	Ajinomoto Co., Inc.	Antidiabetic preparation for oral administration
KR20070104953A (ko) *	2000-03-17	2007-10-29	아지노모토 가부시키가이샤	신경 장애용 약제
ATE368641T1 (de) *	2000-10-18	2007-08-15	Ajinomoto Kk	Verfahren zur herstellung von nateglinidin- kristallen
CN1273442C (zh)	2000-10-18	2006-09-06	味之素株式会社	酰基苯丙氨酸的制备方法
MXPA03003685A (es) *	2000-10-24	2004-01-26	Ajinomoto Kk	Preparaciones que contienen nateglinida.
AU2001296000A1 (en) *	2000-10-24	2002-05-27	Ajinomoto Co., Inc.	Nateglinide-containing hydrophilic drug preparations
RU2275354C2 (ru) *	2000-10-24	2006-04-27	Адзиномото Ко., Инк.	Способы получения кристаллов в-типа натеглинида
US20080058424A1 (en) *	2002-05-23	2008-03-06	Cephalon, Inc.	Novel pharmaceutical formulations of modafinil
JP2003252749A (ja) *	2002-03-04	2003-09-10	Shin Etsu Chem Co Ltd	外用基剤
US6830759B2 (en)	2002-06-28	2004-12-14	Ajinomoto Co., Inc.	Antidiabetic preparation for oral administration
CN1247194C (zh) *	2002-08-27	2006-03-29	石药集团中奇制药技术（石家庄）有限公司	一种那格列奈包合物
US20040116532A1 (en)	2002-09-13	2004-06-17	Craig Heacock	Pharmaceutical formulations of modafinil
US20050065183A1 (en) *	2003-07-31	2005-03-24	Indranil Nandi	Fexofenadine composition and process for preparing
WO2005013964A1 (ja)	2003-08-08	2005-02-17	Ajinomoto Co., Inc.	ナテグリニド含有製剤
WO2005016315A1 (en) *	2003-08-14	2005-02-24	Ranbaxy Laboratories Limited	Pharmaceutical compositions of nateglinide and a high amount of a water-soluble filler
JP5168712B2 (ja) *	2004-04-01	2013-03-27	味の素株式会社	ナテグリニド含有製剤
WO2005117840A1 (en) *	2004-05-31	2005-12-15	Ranbaxy Laboratories Limited	Stable pharmaceutical compositions comprising pulverized granules of nateglinide of form b
EP1776102A1 (de) *	2004-07-28	2007-04-25	Ranbaxy Laboratories Limited	Präparate aus stabilen pharmazeutischen zusammensetzungen aus nateglinid und herstellungsverfahren dafür
BRPI0513089B8 (pt) *	2004-08-04	2021-05-25	Alza Corp	forma de dosagem para liberação controlada de um fármaco de ordem ascendente de zero
AU2005290829B2 (en) *	2004-10-01	2011-06-09	Nippon Zoki Pharmaceutical Co., Ltd.	Solid pharmaceutical preparation
US7276198B2 (en) *	2004-12-28	2007-10-02	The Goodyear Tire & Rubber Company	Method and mold for making tire with tie bar
WO2006080524A1 (ja) *	2005-01-31	2006-08-03	Ajinomoto Co., Inc.	血糖降下剤を含有する、耐糖能異常、境界型糖尿病、インスリン抵抗性及び高インスリン血症の改善ないし治療用医薬組成物
US9034860B2 (en)	2006-12-07	2015-05-19	Daiichi Sankyo Company, Limited	Pharmaceutical composition containing low-substituted hydroxypropyl cellulose
CN101600431B (zh) *	2006-12-07	2011-09-07	第一三共株式会社	具有改进贮存稳定性的药物组合物
CA2672157C (en) *	2006-12-07	2016-07-26	Daiichi Sankyo Company, Limited	Method for producing solid preparation
CA2672134C (en) *	2006-12-07	2015-02-10	Daiichi Sankyo Company, Limited	Solid medicinal preparation containing mannitol or lactose
TWI405574B (zh) *	2007-06-21	2013-08-21	Otsuka Pharma Co Ltd	藥學固體製劑及其製造方法

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
JPS6354321A (ja) *	1985-03-27	1988-03-08	Ajinomoto Co Inc	血糖降下剤
JP3586471B2 (ja) *	1991-06-25	2004-11-10	三菱ウェルファーマ株式会社	トラセミド含有医薬組成物
ES2100291T3 (es)	1991-07-30	1997-06-16	Ajinomoto Kk	Cristales de n-(trans-4-isopropilciclohexilcarbonil)-d-fenilalanina y metodos para prepararlos.
JPH07503236A (ja) *	1991-11-26	1995-04-06	ワーナー−ランバート・コンパニー	制御放出性ジェムフィブロジル剤形の開発のための方法および組成物
ATE503472T1 (de) *	1996-11-15	2011-04-15	Ajinomoto Kk	Nateglinide-tablettenzubereitungen

1997
- 1997-11-14 AT AT05014497T patent/ATE503472T1/de active
- 1997-11-14 PT PT97912459T patent/PT965339E/pt unknown
- 1997-11-14 AT AT97912459T patent/ATE322260T1/de not_active IP Right Cessation
- 1997-11-14 KR KR1019997004308A patent/KR100343062B1/ko not_active Expired - Lifetime
- 1997-11-14 DE DE69740161T patent/DE69740161D1/de not_active Expired - Lifetime
- 1997-11-14 WO PCT/JP1997/004152 patent/WO1998022105A1/ja not_active Ceased
- 1997-11-14 TW TW086117009A patent/TW492878B/zh not_active IP Right Cessation
- 1997-11-14 EP EP05014497A patent/EP1586314B1/de not_active Expired - Lifetime
- 1997-11-14 ES ES05014497T patent/ES2364145T3/es not_active Expired - Lifetime
- 1997-11-14 EP EP97912459A patent/EP0965339B1/de not_active Expired - Lifetime
- 1997-11-14 EP EP10010714A patent/EP2277517A1/de not_active Withdrawn
- 1997-11-14 JP JP32974597A patent/JP4171091B2/ja not_active Expired - Lifetime
- 1997-11-14 DE DE69735644T patent/DE69735644T2/de not_active Expired - Lifetime
- 1997-11-14 AU AU49654/97A patent/AU718350B2/en not_active Ceased
- 1997-11-14 CA CA002271865A patent/CA2271865C/en not_active Expired - Lifetime
- 1997-11-14 DK DK05014497.1T patent/DK1586314T3/da active
- 1997-11-14 ES ES97912459T patent/ES2257772T3/es not_active Expired - Lifetime
- 1997-11-14 PT PT05014497T patent/PT1586314E/pt unknown
- 1997-11-14 CN CNB971811407A patent/CN1245158C/zh not_active Expired - Lifetime
1999
- 1999-05-14 US US09/311,060 patent/US6143323A/en not_active Expired - Lifetime
2000
- 2000-09-29 US US09/672,896 patent/US6296872B1/en not_active Expired - Lifetime
2001
- 2001-08-03 US US09/920,830 patent/US6641841B2/en not_active Expired - Lifetime
2003
- 2003-02-05 US US10/358,324 patent/US6844008B2/en not_active Expired - Lifetime

Also Published As

Publication number	Publication date
KR100343062B1 (ko)	2002-07-02
JPH10194969A (ja)	1998-07-28
DE69735644D1 (de)	2006-05-18
PT965339E (pt)	2006-06-30
US6844008B2 (en)	2005-01-18
DK1586314T3 (da)	2011-06-20
CA2271865A1 (en)	1998-05-28
AU718350B2 (en)	2000-04-13
EP0965339B1 (de)	2006-04-05
CN1245158C (zh)	2006-03-15
EP1586314A1 (de)	2005-10-19
KR20000053312A (ko)	2000-08-25
ES2364145T3 (es)	2011-08-25
EP1586314B1 (de)	2011-03-30
CA2271865C (en)	2003-10-14
ATE503472T1 (de)	2011-04-15
US6143323A (en)	2000-11-07
TW492878B (en)	2002-07-01
JP4171091B2 (ja)	2008-10-22
US6641841B2 (en)	2003-11-04
US20030147951A1 (en)	2003-08-07
EP0965339A4 (de)	2003-04-23
AU4965497A (en)	1998-06-10
US20020028239A1 (en)	2002-03-07
WO1998022105A1 (en)	1998-05-28
DE69740161D1 (de)	2011-05-12
US6296872B1 (en)	2001-10-02
EP0965339A1 (de)	1999-12-22
EP2277517A1 (de)	2011-01-26
PT1586314E (pt)	2011-07-01
DE69735644T2 (de)	2007-05-03
CN1242704A (zh)	2000-01-26
ES2257772T3 (es)	2006-08-01

Legal Events

Date	Code	Title	Description
2006-10-15	RER	Ceased as to paragraph 5 lit. 3 law introducing patent treaties

Publication	Publication Date	Title
ATE322260T1 (de)	2006-04-15	Nateglinide zubereitung in tablettenform
ID24901A (id)	2000-08-31	Metode pengobatan keadaan terkoagulasi tinggi atau defisiensi protein c yang diperoleh
KR880010764A (ko)	1988-10-24	과콜레스테롤혈중 치료용 혼합물
MX9605940A (es)	1998-04-30	Compuestos bioaromaticos que llevan un grupo adamantilo en orto, composiciones farmaceuticas y cosmeticas que los contienen y utilizaciones.
BR0109336A (pt)	2003-06-24	Medicamento para a prevenção, melhora e/ou tratamento de uma complicação diabética, droga medicinal adequada ou utilizável como o mesmo, método para prevenir, melhorar e/ou tratar a complicação diabética, e a neuropatia, e, usos de um agente redutor do açúcar no sangue pós-prandial e pelo menos um agente selecionado de um agente anti-hipertensivo, um agente vasodilatador e um agente anti-hiperlipidêmico
DK420385A (da)	1985-09-17	Antioestrogent laegemiddel til perkutan indgift
MY118164A (en)	2004-09-30	Pharmaceutical composition comprising a combination of metformin and fibrate, and its use for the preparation of medicines intended to reduce hyperglycaemia
ES2123903T3 (es)	1999-01-16	Composicion nutritiva conteniendo fibra.
ES2040232T3 (es)	1993-10-16	Preparaciones medicinales para administracion oral conteniendo una sola dosis de 10 a 240 mg de dihidropiridina.
CO5160272A1 (es)	2002-05-30	Combinacion de cerivastatina y fibratos
NO870772D0 (no)	1987-02-25	Vevplasminogenaktivator for normale humane tykktarmceller.
MX9100246A (es)	1992-02-28	Preparacion farmaceutica en forma de tabletas o grageas que contienen sulcralfato y procedimiento para su preparacion
IS5416A (is)	2000-03-24	Samsetning til að bæla fráhvarfseinkenni og fíkn í áfengi hjá áfengissjúklingum og fyrirbyggja misnotkun áfengis hjá heilbrigðum einstaklingum
BR9912533A (pt)	2002-02-13	Composição farmacêutica tendo sabor melhorado
EP1108429A3 (de)	2002-06-19	Verbesserte Aminosäurenzusammensetzung zum Bereitstellen von Aminosäurenergänzungen oder Eiweissersatz, insbesondere zur Behandlung und/oder Verwaltung von bestimmten Erkrankungen
CN1109357A (zh)	1995-10-04	一种美容保健制品及工艺方法
US6683098B1 (en)	2004-01-27	Use of drug miglitol (Glyset) for treatment of obesity to prevent weight gain for losing weight and for weight control
RU2053782C1 (ru)	1996-02-10	Способ лечения язвенно-некротического стоматита
JPS54148090A (en)	1979-11-19	Peroral cholesterol-depressant
KR970058708A (ko)	1997-08-12	엘-무스콘(l-muscone)의 의약용도
KR910015294A (ko)	1991-09-30	약제 조성물
RU94030887A (ru)	1996-09-20	N-ацетил-дегидрофенилаланил-l-метионин
蕭裕明 et al.	1988	Surgical Correction of Pes Cavus and Equinus Deformity in Two Young Adults
LT2000063A (en)	2002-01-25	Food additive
TH26907A (th)	1997-10-31	องค์ประกอบทางเภสัชภัณฑ์ที่คงตัว