ATE370954T1 - Kristallform von asenapinmaleat - Google Patents

Kristallform von asenapinmaleat

Info

Publication number
ATE370954T1
ATE370954T1 AT06112332T AT06112332T ATE370954T1 AT E370954 T1 ATE370954 T1 AT E370954T1 AT 06112332 T AT06112332 T AT 06112332T AT 06112332 T AT06112332 T AT 06112332T AT E370954 T1 ATE370954 T1 AT E370954T1
Authority
AT
Austria
Prior art keywords
crystal form
asenapine maleate
asenapine
maleate
crystal
Prior art date
Application number
AT06112332T
Other languages
English (en)
Inventor
Gerhardus Heeres
Original Assignee
Organon Nv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=36617328&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=ATE370954(T1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Organon Nv filed Critical Organon Nv
Application granted granted Critical
Publication of ATE370954T1 publication Critical patent/ATE370954T1/de

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
    • C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
    • C07D491/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A61K31/407—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with other heterocyclic ring systems, e.g. ketorolac, physostigmine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • General Chemical & Material Sciences (AREA)
  • Epidemiology (AREA)
  • Biomedical Technology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Psychiatry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Hydrogenated Pyridines (AREA)
  • Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
AT06112332T 2005-04-07 2006-04-06 Kristallform von asenapinmaleat ATE370954T1 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP05102742 2005-04-07
EP05102969 2005-04-14

Publications (1)

Publication Number Publication Date
ATE370954T1 true ATE370954T1 (de) 2007-09-15

Family

ID=36617328

Family Applications (2)

Application Number Title Priority Date Filing Date
AT06725622T ATE418556T1 (de) 2005-04-07 2006-04-06 Kristallform von asenapinmaleat
AT06112332T ATE370954T1 (de) 2005-04-07 2006-04-06 Kristallform von asenapinmaleat

Family Applications Before (1)

Application Number Title Priority Date Filing Date
AT06725622T ATE418556T1 (de) 2005-04-07 2006-04-06 Kristallform von asenapinmaleat

Country Status (31)

Country Link
EP (2) EP1710245B1 (de)
JP (1) JP5058151B2 (de)
KR (1) KR101422843B1 (de)
AR (1) AR056306A1 (de)
AT (2) ATE418556T1 (de)
AU (1) AU2006231617B2 (de)
BR (1) BRPI0609741A8 (de)
CA (1) CA2603509C (de)
CY (2) CY1106902T1 (de)
DE (2) DE602006000080T2 (de)
DK (2) DK1917267T3 (de)
DO (1) DOP2006000082A (de)
ES (2) ES2318742T3 (de)
GT (1) GT200600135A (de)
HN (1) HN2006014095A (de)
HR (1) HRP20070429T3 (de)
IL (1) IL186355A (de)
MX (1) MX2007012445A (de)
MY (1) MY137969A (de)
NO (1) NO340520B1 (de)
NZ (1) NZ562124A (de)
PE (1) PE20061311A1 (de)
PL (2) PL1917267T3 (de)
PT (2) PT1917267E (de)
RS (1) RS50532B (de)
RU (1) RU2405786C2 (de)
SI (2) SI1710245T1 (de)
SV (1) SV2006002473A (de)
TW (1) TWI364423B (de)
UY (1) UY29459A1 (de)
WO (1) WO2006106135A1 (de)

Families Citing this family (24)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PE20081457A1 (es) * 2006-10-06 2008-10-18 Organon Nv Asenapina amorfa, procesos para prepararlas y su uso para tratar trastornos del sistema nervioso central
CN102596172A (zh) * 2009-06-24 2012-07-18 Msd欧斯股份有限公司 含有阿塞那平的注射剂和使用其的治疗方法
EP2582704A4 (de) * 2010-06-18 2014-04-02 Reddys Lab Ltd Dr Asenapin-maleat
WO2012066565A2 (en) * 2010-11-16 2012-05-24 Cadila Healthcare Limited Asenapine maleate amorphous and crystalline form and process for preparation thereof
EP2468750A1 (de) 2010-12-13 2012-06-27 Chemo Ibérica, S.A. Polymorphe Formen von Asenapinmaleat und Verfahren zur ihrer Herstellung
WO2012123325A1 (en) 2011-03-11 2012-09-20 Medichem S.A. NEW CRYSTAL FORMS OF THE SALT OF TRANS-5-CHLORO-2-METHYL-2,3,3A,12b-TETRAHYDRO-1H-DIBENZO[2,3:6,7]OXEPINO[4,5-c]PYRROLE WITH MALEIC ACID
ITMI20110734A1 (it) * 2011-05-02 2012-11-03 Olon Spa Sali cristallini di asenapina
EP2524920A1 (de) 2011-05-17 2012-11-21 Sandoz AG Neue kristalline Formen von Asenapin-Hydrochloridsalz
EP2524921A1 (de) 2011-05-17 2012-11-21 Sandoz AG Neue kristalline Salze von Asenapin
EP2524919A1 (de) 2011-05-17 2012-11-21 Sandoz AG Neue kristalline Salze von Asenapin mit organischen Di-Säuren und Tri-Säuren
US9533994B2 (en) 2011-05-18 2017-01-03 Laboratorios Lesvi S.L. Monoclinic crystalline form of asenapine maleate with a specific particle size distribution
EP2709616B1 (de) * 2011-05-18 2018-01-24 Laboratorios Lesvi, S.L. Synthese von einer stabilen mikronisierten monoklinen form des asenapinmaleates
EP2572703A1 (de) 2011-09-21 2013-03-27 Hexal AG Komprimierte orale Dosierform für Asenapinmaleat
WO2013041604A1 (en) 2011-09-21 2013-03-28 Sandoz Ag Crystal form of asenapine maleate
JP6005741B2 (ja) * 2012-07-26 2016-10-12 久光製薬株式会社 貼付剤及びその製造方法
ITMI20121810A1 (it) 2012-10-24 2014-04-25 Chemo Iberica Sa Poliformi di maleato di asenapina e processo per la loro preparazione
WO2014090386A1 (en) 2012-12-11 2014-06-19 Alfred E. Tiefenbacher (Gmbh & Co. Kg) Orally disintegrating tablet containing asenapine
WO2014127786A1 (en) 2013-02-22 2014-08-28 Zentiva, K.S. Orally disintegrating pharmaceutical composition comprising asenapine
WO2017037718A1 (en) 2015-09-02 2017-03-09 Eloxx Pharmaceuticals Ltd. Aminoglycoside derivatives and uses thereof in treating genetic disorders
KR102614709B1 (ko) 2016-12-20 2023-12-18 에르테에스 로만 테라피-시스테메 아게 아세나핀 및 폴리실록산 또는 폴리이소부틸렌을 함유하는 경피흡수 치료 시스템
CN115813888A (zh) 2016-12-20 2023-03-21 罗曼治疗系统股份公司 包含阿塞那平的透皮治疗系统
JP2020525545A (ja) 2017-06-26 2020-08-27 エルテーエス ローマン テラピー−ジステーメ アーゲー アセナピンおよびシリコーンアクリルハイブリッドポリマーを含有する経皮治療システム
PL3810100T3 (pl) 2018-06-20 2025-05-12 Lts Lohmann Therapie-Systeme Ag Transdermalny system terapeutyczny zawierający asenapinę
US12329862B2 (en) 2018-06-20 2025-06-17 Lts Lohmann Therapie-Systeme Ag Transdermal therapeutic system containing asenapine

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NL7605526A (nl) * 1976-05-24 1977-11-28 Akzo Nv Nieuwe tetracyclische derivaten.
RU2139051C1 (ru) * 1994-03-02 1999-10-10 Акцо Нобель Н.В. Сублингвальная или трансбуккальная фармацевтическая композиция
WO1999032108A1 (en) * 1997-12-19 1999-07-01 Akzo Nobel N.V. Org-5222 in the treatment of depression
TWI327915B (en) * 2003-06-12 2010-08-01 Organon Nv Pharmaceutical composition comprising antipsychotic agent and use of the antipsychotic agent for treating patients with overweight

Also Published As

Publication number Publication date
SI1917267T1 (sl) 2009-04-30
DOP2006000082A (es) 2006-11-30
UY29459A1 (es) 2006-11-30
NO20075142L (no) 2007-11-05
EP1917267B1 (de) 2008-12-24
DE602006000080D1 (de) 2007-10-04
WO2006106135A1 (en) 2006-10-12
RS50532B (sr) 2010-05-07
EP1710245B1 (de) 2007-08-22
ES2293626T3 (es) 2008-03-16
PL1710245T3 (pl) 2008-01-31
NZ562124A (en) 2010-07-30
DE602006004463D1 (de) 2009-02-05
GT200600135A (es) 2006-11-07
IL186355A (en) 2016-05-31
ATE418556T1 (de) 2009-01-15
JP2008534656A (ja) 2008-08-28
CA2603509C (en) 2013-12-03
PE20061311A1 (es) 2007-02-09
HRP20070429T3 (en) 2007-11-30
EP1917267A1 (de) 2008-05-07
RU2405786C2 (ru) 2010-12-10
KR20080005253A (ko) 2008-01-10
IL186355A0 (en) 2008-01-20
NO340520B1 (no) 2017-05-02
AU2006231617B2 (en) 2010-06-03
MY137969A (en) 2009-04-30
RU2007141198A (ru) 2009-05-20
MX2007012445A (es) 2007-11-07
ES2318742T3 (es) 2009-05-01
EP1710245A1 (de) 2006-10-11
PT1710245E (pt) 2007-10-03
JP5058151B2 (ja) 2012-10-24
KR101422843B1 (ko) 2014-07-24
CY1108742T1 (el) 2014-04-09
DK1710245T3 (da) 2007-12-03
HN2006014095A (es) 2010-08-19
PT1917267E (pt) 2009-02-04
DK1917267T3 (da) 2009-04-14
AU2006231617A1 (en) 2006-10-12
PL1917267T3 (pl) 2009-06-30
TW200722428A (en) 2007-06-16
DE602006000080T2 (de) 2008-05-15
SI1710245T1 (sl) 2007-12-31
BRPI0609741A2 (pt) 2010-04-27
CA2603509A1 (en) 2006-10-12
AR056306A1 (es) 2007-10-03
SV2006002473A (es) 2009-11-24
BRPI0609741A8 (pt) 2018-03-13
CY1106902T1 (el) 2012-09-26
TWI364423B (en) 2012-05-21

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