ATE398121T1 - Neue synthese von irbesartan - Google Patents

Neue synthese von irbesartan

Info

Publication number: ATE398121T1
Authority: AT; Austria
Prior art keywords: irbesartan; new synthesis; synthesis; new; provides
Prior art date: 2003-01-16

Application number

AT04702955T

Other languages

English (en)

Inventor

Gennady Nisnevich

Igor Rukhman

Boris Pertsikov

Julia Kaftanov

Ben-Zion Dolitzky

Original Assignee

Teva Pharma

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2003-01-16

Filing date

2004-01-16

Publication date

2008-07-15

2004-01-16 Application filed by Teva Pharma filed Critical Teva Pharma

2008-07-15 Application granted granted Critical

2008-07-15 Publication of ATE398121T1 publication Critical patent/ATE398121T1/de

Links

239000002947 C09CA04 - Irbesartan Substances 0.000 title abstract 2
YCPOHTHPUREGFM-UHFFFAOYSA-N irbesartan Chemical compound O=C1N(CC=2C=CC(=CC=2)C=2C(=CC=CC=2)C=2[N]N=NN=2)C(CCCC)=NC21CCCC2 YCPOHTHPUREGFM-UHFFFAOYSA-N 0.000 title abstract 2
229960002198 irbesartan Drugs 0.000 title abstract 2
230000015572 biosynthetic process Effects 0.000 title 1
238000003786 synthesis reaction Methods 0.000 title 1
238000004519 manufacturing process Methods 0.000 abstract 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D235/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
- C07D235/02—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
- C07D403/10—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a carbon chain containing aromatic rings

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
Plural Heterocyclic Compounds (AREA)
Steroid Compounds (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)
Catalysts (AREA)
Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)

AT04702955T 2003-01-16 2004-01-16 Neue synthese von irbesartan ATE398121T1 (de)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
US44099703P	2003-01-16	2003-01-16

Publications (1)

Publication Number	Publication Date
ATE398121T1 true ATE398121T1 (de)	2008-07-15

Family

ID=32771889

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
AT04702955T ATE398121T1 (de)	2003-01-16	2004-01-16	Neue synthese von irbesartan

Country Status (10)

Country	Link
US (6)	US7019148B2 (de)
EP (3)	EP1509517B1 (de)
CN (2)	CN1759113A (de)
AT (1)	ATE398121T1 (de)
CA (1)	CA2513373A1 (de)
DE (1)	DE602004014321D1 (de)
ES (1)	ES2281312T3 (de)
PT (1)	PT1509517E (de)
SI (1)	SI1509517T1 (de)
WO (1)	WO2004065383A2 (de)

Families Citing this family (22)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US7941149B2 (en)	2002-05-13	2011-05-10	Misonimo Chi Acquistion L.L.C.	Multi-hop ultra wide band wireless network communication
US8780770B2 (en) *	2002-05-13	2014-07-15	Misonimo Chi Acquisition L.L.C.	Systems and methods for voice and video communication over a wireless network
US7957356B2 (en)	2002-05-13	2011-06-07	Misomino Chi Acquisitions L.L.C.	Scalable media access control for multi-hop high bandwidth communications
WO2004065383A2 (en) *	2003-01-16	2004-08-05	Teva Pharmaceutical Industries Ltd.	Novel synthesis of irbesartan
DE602004015071D1 (de)	2003-02-05	2008-08-28	Teva Pharma	Synthese von 2-butyl-3-(2'-(1-trityl-1h-tetrazol-5-yl)biphenyl-4-yl)-1,3-diazaspiro-4,4 -nonen-4-on
EP1751123A4 (de) *	2004-05-20	2010-06-30	Reddys Lab Ltd Dr	Verfahren zur herstellung von irbesartan
TWI346108B (en) *	2004-08-23	2011-08-01	Bristol Myers Squibb Co	A method for preparing irbesartan and intermediates thereof
DE102004060699A1 (de) *	2004-12-16	2006-06-22	Ratiopharm Gmbh	Verfahren zur Herstellung von Candesartan
EP1833801B9 (de) *	2004-12-22	2009-02-25	Algry Quimica, S.L	Zwischenprodukte für die herstellung von antagonisten des angiotensin-ii-rezeptors
SI21965A (sl) *	2005-01-05	2006-08-31	Krka, Tovarna Zdravil, D.D., Novo Mesto	Priprava tetrazolskega derivata
ES2259909B1 (es) *	2005-02-28	2007-06-16	Inke, S.A.	Procedimiento para la obtencion de un compuesto farmaceuticamente activo y de su intermedio de sintesis.
WO2006125592A2 (en) *	2005-05-24	2006-11-30	Lek Pharmaceuticals D.D.	Process for the preparation of 2-alkyl-1-((2'-substituted-biphenyl-4-yl)methyl)-imidazole, dihydroimidazole or benzimidazole derivatives
EP1749828A1 (de)	2005-08-04	2007-02-07	Farmaprojects S.L.	Verfahren zur Herstellung eines Angiotensin-II-Antagonisten
EP1764365A1 (de)	2005-09-20	2007-03-21	KRKA, D.D., Novo Mesto	Verfahren zur Herstellung Sartanderivate und Zwischenprodukte für dieses Verfahren
CA2604404A1 (en) *	2005-10-28	2007-05-03	Alembic Limited	An improved process for preparation of irbesartan
ES2300175B1 (es) *	2006-02-14	2009-06-08	Inke, S.A.	Procedimiento para la obtencion de intermedios utiles en la obtencion de un compuesto farmaceuticamente activo.
US8212051B2 (en)	2006-04-07	2012-07-03	Lek Pharmaceuticals, D.D.	Process for the preparation of pure irbesartan
US8175613B2 (en)	2006-08-04	2012-05-08	Misonimo Chi Acquisitions L.L.C.	Systems and methods for determining location of devices within a wireless network
ES2302671T1 (es) *	2006-08-29	2008-08-01	Teva Pharmaceutical Industries Ltd.	Procedimientos para la sintesis de 5-fenil-1-tritil-1h-tetrazol.
KR101102719B1 (ko) *	2006-12-07	2012-01-05	미소니모 카이 액퀴지션 엘엘씨	타임슬롯 및 채널 할당을 위한 시스템 및 방법
ES2527686T3 (es)	2009-04-28	2015-01-28	Daiichi Sankyo Company, Limited	Procedimiento de producción de olmesartán medoxomil
CN106608886A (zh) *	2015-11-22	2017-05-03	宁夏际华环境安全科技有限公司	一种苯基硼酸生产工艺

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US531929A (en) *		1895-01-01		harden
GB8910547D0 (en) *	1989-05-08	1989-06-21	Ici America Inc	Substituted ketones
US5270317A (en)	1990-03-20	1993-12-14	Elf Sanofi	N-substituted heterocyclic derivatives, their preparation and the pharmaceutical compositions in which they are present
US5164403A (en)	1991-04-05	1992-11-17	G. D. Searle & Co.	N-arylheteroarylalkyl imidazol-2-one compounds for treatment of circulatory disorders
JPH06510763A (ja)	1991-08-19	1994-12-01	イー・アイ・デュポン・ドゥ・ヌムール・アンド・カンパニー	アンジオテンシン２受容体遮断イミダゾリノン誘導体
US5310929A (en) *	1992-08-06	1994-05-10	E. I. Du Pont De Nemours And Company	Prodrugs of imidazole carboxylic acids as angiotensin II receptor antagonists
CA2147503A1 (en)	1992-11-06	1994-05-26	Judith M. Pisano	Substituted dipeptide analogs promote release of growth hormone
US5541209A (en) *	1994-08-22	1996-07-30	Bristol-Myers Squibb Company	Method of treating or preventing cardiac arrhythmia employing an N-substituted heterocyclic derivative
EP0782996B1 (de)	1994-09-20	1999-02-17	Wakunaga Seiyaku Kabushiki Kaisha	Verfahren zur herstellung von n-biphenylmethylthiadiazolin derivaten oder deren salzen sowie dafür benötigte zwischen verbindungen
FR2725987B1 (fr) *	1994-10-19	1997-01-10	Sanofi Sa	Procede pour la preparation d'un derive de tetrazole sous deux formes cristallines et nouvelle forme cristalline de ce derive
US5541204A (en) *	1994-12-02	1996-07-30	Bristol-Myers Squibb Company	Aryloxypropanolamine β 3 adrenergic agonists
IT1292437B1 (it) *	1997-06-30	1999-02-08	Zambon Spa	Processo di orto-metallazione utile per la sintesi di 1 - tetrazol- 5-il) benzeni 2-sostituiti
FR2780403B3 (fr)	1998-06-24	2000-07-21	Sanofi Sa	Nouvelle forme de l'irbesartan, procedes pour obtenir ladite forme et compositions pharmaceutiques en contenant
DE60308708T2 (de)	2002-07-16	2007-08-23	Teva Pharmaceutical Industries Ltd.	Neue synthese von irbesartan
WO2004065383A2 (en) *	2003-01-16	2004-08-05	Teva Pharmaceutical Industries Ltd.	Novel synthesis of irbesartan

2004
- 2004-01-16 WO PCT/US2004/001135 patent/WO2004065383A2/en not_active Ceased
- 2004-01-16 US US10/759,906 patent/US7019148B2/en not_active Expired - Fee Related
- 2004-01-16 EP EP04702955A patent/EP1509517B1/de not_active Expired - Lifetime
- 2004-01-16 SI SI200430833T patent/SI1509517T1/sl unknown
- 2004-01-16 PT PT04702955T patent/PT1509517E/pt unknown
- 2004-01-16 CN CNA2004800067788A patent/CN1759113A/zh active Pending
- 2004-01-16 CA CA002513373A patent/CA2513373A1/en not_active Abandoned
- 2004-01-16 DE DE602004014321T patent/DE602004014321D1/de not_active Expired - Fee Related
- 2004-01-16 CN CNA2007101866764A patent/CN101165062A/zh active Pending
- 2004-01-16 AT AT04702955T patent/ATE398121T1/de not_active IP Right Cessation
- 2004-01-16 EP EP09180682A patent/EP2189457A1/de not_active Withdrawn
- 2004-01-16 ES ES04702955T patent/ES2281312T3/es not_active Expired - Lifetime
- 2004-01-16 EP EP08010340A patent/EP2039693A3/de not_active Withdrawn
2006
- 2006-02-06 US US11/348,945 patent/US7217825B2/en not_active Expired - Fee Related
- 2006-02-06 US US11/348,944 patent/US7301035B2/en not_active Expired - Fee Related
- 2006-02-06 US US11/349,360 patent/US7227026B2/en not_active Expired - Fee Related
2007
- 2007-05-04 US US11/800,332 patent/US7838683B2/en not_active Expired - Fee Related
2008
- 2008-12-18 US US12/317,216 patent/US20090216026A1/en not_active Abandoned

Also Published As

Publication number	Publication date
US7301035B2 (en)	2007-11-27
US20060135780A1 (en)	2006-06-22
US7019148B2 (en)	2006-03-28
WO2004065383A3 (en)	2004-12-16
EP1509517A2 (de)	2005-03-02
DE602004014321D1 (de)	2008-07-24
US20070213539A1 (en)	2007-09-13
US20040192713A1 (en)	2004-09-30
ES2281312T3 (es)	2008-08-01
EP2039693A3 (de)	2009-06-17
EP2039693A2 (de)	2009-03-25
US20060135544A1 (en)	2006-06-22
US20060128968A1 (en)	2006-06-15
CN101165062A (zh)	2008-04-23
US7217825B2 (en)	2007-05-15
EP1509517B1 (de)	2008-06-11
SI1509517T1 (sl)	2008-10-31
US7227026B2 (en)	2007-06-05
WO2004065383A2 (en)	2004-08-05
CN1759113A (zh)	2006-04-12
PT1509517E (pt)	2008-08-05
ES2281312T1 (es)	2007-10-01
EP2189457A1 (de)	2010-05-26
US7838683B2 (en)	2010-11-23
CA2513373A1 (en)	2004-08-05
US20090216026A1 (en)	2009-08-27

Legal Events

Date	Code	Title	Description
2008-12-15	RER	Ceased as to paragraph 5 lit. 3 law introducing patent treaties

Publication	Publication Date	Title
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