ATE443713T1 - Makrozyklische peptide mit wirkung gegen das hepatitis-c-virus - Google Patents

Makrozyklische peptide mit wirkung gegen das hepatitis-c-virus

Info

Publication number: ATE443713T1
Authority: AT; Austria
Prior art keywords: alkyl; virus; active against; against hepatitis; macrocyclic peptides
Prior art date: 2002-10-25

Application number

AT03809217T

Other languages

English (en)

Inventor

Montse Llinas-Brunet

Murray Bailey

Original Assignee

Boehringer Ingelheim Int

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2002-10-25

Filing date

2003-10-20

Publication date

2009-10-15

Family has litigation

First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=32180514&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=ATE443713(T1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.

2003-10-20 Application filed by Boehringer Ingelheim Int filed Critical Boehringer Ingelheim Int

2009-10-15 Application granted granted Critical

2009-10-15 Publication of ATE443713T1 publication Critical patent/ATE443713T1/de

Links

241000711549 Hepacivirus C Species 0.000 title 1
102000004196 processed proteins & peptides Human genes 0.000 title 1
108090000765 processed proteins & peptides Proteins 0.000 title 1
-1 O-(C1-6)alkyl Chemical group 0.000 abstract 2
125000003368 amide group Chemical group 0.000 abstract 2
125000004093 cyano group Chemical group *C#N 0.000 abstract 2
125000000753 cycloalkyl group Chemical group 0.000 abstract 2
125000001475 halogen functional group Chemical group 0.000 abstract 2
125000000449 nitro group Chemical group [O-][N+](*)=O 0.000 abstract 2
125000001997 phenyl group Chemical group [H]C1=C([H])C([H])=C(*)C([H])=C1[H] 0.000 abstract 2
125000002924 primary amino group Chemical group [H]N([H])* 0.000 abstract 2
125000004169 (C1-C6) alkyl group Chemical group 0.000 abstract 1
125000004209 (C1-C8) alkyl group Chemical group 0.000 abstract 1
101800001838 Serine protease/helicase NS3 Proteins 0.000 abstract 1
125000003118 aryl group Chemical group 0.000 abstract 1
150000001875 compounds Chemical class 0.000 abstract 1
239000003112 inhibitor Substances 0.000 abstract 1
150000003839 salts Chemical class 0.000 abstract 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/08—Tripeptides
- C07K5/0802—Tripeptides with the first amino acid being neutral
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
- A61P31/14—Antivirals for RNA viruses
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides

Landscapes

Chemical & Material Sciences (AREA)
Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
Organic Chemistry (AREA)
General Health & Medical Sciences (AREA)
Medicinal Chemistry (AREA)
Molecular Biology (AREA)
Biochemistry (AREA)
Biophysics (AREA)
Genetics & Genomics (AREA)
Proteomics, Peptides & Aminoacids (AREA)
Virology (AREA)
Communicable Diseases (AREA)
Oncology (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Pharmacology & Pharmacy (AREA)
Animal Behavior & Ethology (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Peptides Or Proteins (AREA)

AT03809217T 2002-10-25 2003-10-20 Makrozyklische peptide mit wirkung gegen das hepatitis-c-virus ATE443713T1 (de)

Applications Claiming Priority (4)

Application Number	Priority Date	Filing Date	Title
US42141402P	2002-10-25	2002-10-25
US43382002P	2002-12-16	2002-12-16
US44276803P	2003-01-27	2003-01-27
PCT/CA2003/001604 WO2004037855A1 (en)	2002-10-25	2003-10-20	Macrocyclic peptides active against the hepatitis c virus

Publications (1)

Publication Number	Publication Date
ATE443713T1 true ATE443713T1 (de)	2009-10-15

Family

ID=32180514

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
AT03809217T ATE443713T1 (de)	2002-10-25	2003-10-20	Makrozyklische peptide mit wirkung gegen das hepatitis-c-virus

Country Status (9)

Country	Link
US (2)	US20050075279A1 (de)
EP (1)	EP1558632B1 (de)
JP (1)	JP4398424B2 (de)
AT (1)	ATE443713T1 (de)
AU (1)	AU2003275826A1 (de)
CA (1)	CA2498572C (de)
DE (1)	DE60329408D1 (de)
ES (1)	ES2330932T3 (de)
WO (1)	WO2004037855A1 (de)

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2003
- 2003-10-16 US US10/686,755 patent/US20050075279A1/en not_active Abandoned
- 2003-10-20 ES ES03809217T patent/ES2330932T3/es not_active Expired - Lifetime
- 2003-10-20 AT AT03809217T patent/ATE443713T1/de active
- 2003-10-20 WO PCT/CA2003/001604 patent/WO2004037855A1/en not_active Ceased
- 2003-10-20 DE DE60329408T patent/DE60329408D1/de not_active Expired - Lifetime
- 2003-10-20 JP JP2005501488A patent/JP4398424B2/ja not_active Expired - Fee Related
- 2003-10-20 AU AU2003275826A patent/AU2003275826A1/en not_active Abandoned
- 2003-10-20 EP EP03809217A patent/EP1558632B1/de not_active Expired - Lifetime
- 2003-10-20 CA CA2498572A patent/CA2498572C/en not_active Expired - Fee Related
2005
- 2005-12-10 US US11/298,443 patent/US7504378B2/en not_active Expired - Lifetime

Also Published As

Publication number	Publication date
ES2330932T3 (es)	2009-12-17
CA2498572C (en)	2011-08-23
US7504378B2 (en)	2009-03-17
JP4398424B2 (ja)	2010-01-13
AU2003275826A1 (en)	2004-05-13
WO2004037855A1 (en)	2004-05-06
JP2006517915A (ja)	2006-08-03
EP1558632B1 (de)	2009-09-23
CA2498572A1 (en)	2004-05-06
US20060089300A1 (en)	2006-04-27
DE60329408D1 (de)	2009-11-05
EP1558632A1 (de)	2005-08-03
US20050075279A1 (en)	2005-04-07

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