ATE458476T1 - Verfahren für die zubereitung der amorphen form eines medikamentes - Google Patents

Verfahren für die zubereitung der amorphen form eines medikamentes

Info

Publication number
ATE458476T1
ATE458476T1 AT05758626T AT05758626T ATE458476T1 AT E458476 T1 ATE458476 T1 AT E458476T1 AT 05758626 T AT05758626 T AT 05758626T AT 05758626 T AT05758626 T AT 05758626T AT E458476 T1 ATE458476 T1 AT E458476T1
Authority
AT
Austria
Prior art keywords
medication
preparing
amorphic form
amorphic
preparation
Prior art date
Application number
AT05758626T
Other languages
English (en)
Inventor
Szabolcs Szoke
Csaba Szabo
Lorant Gyuricza
Claude Singer
Valerie Niddam-Hildesheim
Greta Sterimbaum
Original Assignee
Teva Gyogyszergyar Zartkoeruen
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Teva Gyogyszergyar Zartkoeruen filed Critical Teva Gyogyszergyar Zartkoeruen
Application granted granted Critical
Publication of ATE458476T1 publication Critical patent/ATE458476T1/de

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/14Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D215/00Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
    • C07D215/02Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
    • C07D215/16Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D215/18Halogen atoms or nitro radicals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/14Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D407/00Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen atoms as the only ring hetero atoms, not provided for by group C07D405/00
    • C07D407/02Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen atoms as the only ring hetero atoms, not provided for by group C07D405/00 containing two hetero rings
    • C07D407/06Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen atoms as the only ring hetero atoms, not provided for by group C07D405/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • FMECHANICAL ENGINEERING; LIGHTING; HEATING; WEAPONS; BLASTING
    • F26DRYING
    • F26BDRYING SOLID MATERIALS OR OBJECTS BY REMOVING LIQUID THEREFROM
    • F26B11/00Machines or apparatus for drying solid materials or objects with movement which is non-progressive
    • F26B11/12Machines or apparatus for drying solid materials or objects with movement which is non-progressive in stationary drums or other mainly-closed receptacles with moving stirring devices
    • FMECHANICAL ENGINEERING; LIGHTING; HEATING; WEAPONS; BLASTING
    • F26DRYING
    • F26BDRYING SOLID MATERIALS OR OBJECTS BY REMOVING LIQUID THEREFROM
    • F26B5/00Drying solid materials or objects by processes not involving the application of heat
    • F26B5/04Drying solid materials or objects by processes not involving the application of heat by evaporation or sublimation of moisture under reduced pressure, e.g. in a vacuum
    • F26B5/041Drying solid materials or objects by processes not involving the application of heat by evaporation or sublimation of moisture under reduced pressure, e.g. in a vacuum for drying flowable materials, e.g. suspensions, bulk goods, in a continuous operation, e.g. with locks or other air tight arrangements for charging/discharging

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Mechanical Engineering (AREA)
  • General Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Molecular Biology (AREA)
  • Epidemiology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Medicinal Preparation (AREA)
  • Steroid Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
AT05758626T 2004-06-01 2005-06-01 Verfahren für die zubereitung der amorphen form eines medikamentes ATE458476T1 (de)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US57621604P 2004-06-01 2004-06-01
US58377804P 2004-06-28 2004-06-28
US59970004P 2004-08-05 2004-08-05
PCT/US2005/019485 WO2005117837A1 (en) 2004-06-01 2005-06-01 Process for preparation of amorphous form of a drug

Publications (1)

Publication Number Publication Date
ATE458476T1 true ATE458476T1 (de) 2010-03-15

Family

ID=35134738

Family Applications (1)

Application Number Title Priority Date Filing Date
AT05758626T ATE458476T1 (de) 2004-06-01 2005-06-01 Verfahren für die zubereitung der amorphen form eines medikamentes

Country Status (11)

Country Link
US (1) US7589128B2 (de)
JP (1) JP2008500405A (de)
KR (1) KR20060123772A (de)
AT (1) ATE458476T1 (de)
CA (1) CA2560984A1 (de)
DE (1) DE602005019509D1 (de)
DK (1) DK1641438T3 (de)
ES (1) ES2339682T3 (de)
IL (1) IL179719A0 (de)
MX (1) MXPA06010084A (de)
WO (1) WO2005117837A1 (de)

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US20060083784A1 (en) * 2002-08-07 2006-04-20 Smithkline Beecham Corporation Amorphous pharmaceutical compositions
MX2007004426A (es) 2004-10-15 2007-06-14 Teva Pharma Procesos para preparar telmisartan.
WO2006050509A2 (en) * 2004-11-03 2006-05-11 Teva Pharmaceutical Industries Ltd. Amorphous and polymorphic forms of telmisartan sodium
CA2584430A1 (en) 2004-12-01 2006-06-08 Teva Gyogyszergyar Zartkoruen Mukodo Reszvenytarsasag Methods for preparing pimecrolimus
CA2594694A1 (en) 2005-01-28 2006-08-03 Pfizer Products Inc. Drying of drug-containing particles
EP1904448B1 (de) 2005-07-05 2011-02-02 Teva Pharmaceutical Industries, Ltd. Reinigung von montelukast
US20070161796A1 (en) * 2005-11-16 2007-07-12 Ilan Kor-Sade Drying methods of montelukast sodium by azeotropic removal of the solvent
GB0613925D0 (en) 2006-07-13 2006-08-23 Unilever Plc Improvements relating to nanodispersions
WO2008012617A1 (en) 2006-07-21 2008-01-31 Pfizer Products Inc. Drying of drug-containing particles
GB2441328A (en) * 2006-08-30 2008-03-05 Alpharma Aps A method for obtaining mupirocin calcium
US20080187684A1 (en) * 2007-02-07 2008-08-07 Imra America, Inc. Method for depositing crystalline titania nanoparticles and films
US20090234125A1 (en) * 2007-11-26 2009-09-17 Eli Lancry Amorphous retapamulin and processes for preparation thereof
GB2457452B (en) * 2008-02-12 2010-05-12 Pliva Lachema As Amorphous form of (OC-6-43)-bis(acetate)(1-tricyclo[3,3,1,13,7]decylamine) amminedichloroplatinum (IV)
EP2366378A1 (de) 2010-03-01 2011-09-21 Dexcel Pharma Technologies Ltd. Donepezilformulierungen mit verzögerter Freisetzung
WO2011121596A2 (en) * 2010-04-01 2011-10-06 Neuland Laboratories Ltd. Crystal modification of moxifloxacin hydrochloride
US8471030B2 (en) 2010-12-06 2013-06-25 Orochem Technologies Inc. Purification of montelukast using simulated moving bed
EP3846792A4 (de) 2018-09-06 2022-10-12 Innopharmascreen Inc. Verfahren und zusammensetzungen zur behandlung von asthma oder morbus parkinson
WO2025146702A1 (en) * 2024-01-03 2025-07-10 Msn Laboratories Private Limited, R&D Center Solid state forms of 1-{(2s,5r)-2-methyl-5-[(7h-pyrrolo[2,3-d]pyrimidin-4-yl)amino] piperidine-1-yl}prop-2-en-1-one 4-methylbenzene-1-sulfonic acid

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CA2584430A1 (en) * 2004-12-01 2006-06-08 Teva Gyogyszergyar Zartkoruen Mukodo Reszvenytarsasag Methods for preparing pimecrolimus

Also Published As

Publication number Publication date
IL179719A0 (en) 2007-05-15
JP2008500405A (ja) 2008-01-10
US7589128B2 (en) 2009-09-15
DK1641438T3 (da) 2010-06-07
US20050272768A1 (en) 2005-12-08
ES2339682T3 (es) 2010-05-24
DE602005019509D1 (de) 2010-04-08
KR20060123772A (ko) 2006-12-04
MXPA06010084A (es) 2007-03-01
WO2005117837A1 (en) 2005-12-15
CA2560984A1 (en) 2005-12-15

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Legal Events

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RER Ceased as to paragraph 5 lit. 3 law introducing patent treaties