ATE523493T1 - 2-(1-oxo-1h-isochinolin-2-yl) acetamid-derivate - Google Patents
2-(1-oxo-1h-isochinolin-2-yl) acetamid-derivateInfo
- Publication number
- ATE523493T1 ATE523493T1 AT07842137T AT07842137T ATE523493T1 AT E523493 T1 ATE523493 T1 AT E523493T1 AT 07842137 T AT07842137 T AT 07842137T AT 07842137 T AT07842137 T AT 07842137T AT E523493 T1 ATE523493 T1 AT E523493T1
- Authority
- AT
- Austria
- Prior art keywords
- isochinolin
- oxo
- acetamide derivatives
- acetamide
- derivatives
- Prior art date
Links
- DLFVBJFMPXGRIB-UHFFFAOYSA-N Acetamide Chemical class CC(N)=O DLFVBJFMPXGRIB-UHFFFAOYSA-N 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D217/00—Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems
- C07D217/22—Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to carbon atoms of the nitrogen-containing ring
- C07D217/24—Oxygen atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/22—Anxiolytics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Veterinary Medicine (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Public Health (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Psychiatry (AREA)
- Pain & Pain Management (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Other In-Based Heterocyclic Compounds (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US84371306P | 2006-09-11 | 2006-09-11 | |
| PCT/US2007/077999 WO2008033757A2 (en) | 2006-09-11 | 2007-09-10 | 2-(1-oxo-1h-isoquinolin-2-yl) acetamide derivatives |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ATE523493T1 true ATE523493T1 (de) | 2011-09-15 |
Family
ID=39184481
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AT07842137T ATE523493T1 (de) | 2006-09-11 | 2007-09-10 | 2-(1-oxo-1h-isochinolin-2-yl) acetamid-derivate |
Country Status (9)
| Country | Link |
|---|---|
| US (1) | US7906504B2 (de) |
| EP (1) | EP2066640B1 (de) |
| JP (1) | JP5271909B2 (de) |
| CN (1) | CN101528703B (de) |
| AR (1) | AR062734A1 (de) |
| AT (1) | ATE523493T1 (de) |
| CA (1) | CA2663193A1 (de) |
| MX (1) | MX2009002685A (de) |
| WO (1) | WO2008033757A2 (de) |
Families Citing this family (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN101600698B (zh) * | 2006-09-11 | 2012-01-11 | 欧加农股份有限公司;药典有限责任公司 | 喹唑啉酮和异喹啉酮乙酰胺衍生物 |
| ME02169B (me) | 2010-10-01 | 2015-10-20 | Taisho Pharmaceutical Co Ltd | Derivat 1,2,4-triazolona |
| CN103889951B (zh) | 2011-10-27 | 2016-12-14 | 大正制药株式会社 | 唑类衍生物 |
| HK1200829A1 (en) | 2012-03-30 | 2015-08-14 | 大正制药株式会社 | Fused azole derivative |
| ES2821010T3 (es) | 2015-12-09 | 2021-04-23 | Cadent Therapeutics Inc | Moduladores heteroaromáticos del receptor NMDA y usos de los mismos |
| US10500205B2 (en) | 2015-12-09 | 2019-12-10 | Cadent Therapeutics, Inc. | Thienopyrimidinone NMDA receptor modulators and uses thereof |
| CA3047403A1 (en) | 2016-12-22 | 2018-06-28 | Cadent Therapeutics, Inc. | Nmda receptor modulators and uses thereof |
| CA3108519A1 (en) | 2018-08-03 | 2020-04-30 | Cadent Therapeutics, Inc. | Heteroaromatic nmda receptor modulators and uses thereof |
Family Cites Families (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FR2506767A1 (fr) * | 1981-05-26 | 1982-12-03 | Synthelabo | Derives heterocycliques d'amidoximes, leur preparation et leur application en therapeutique |
| JP2004511465A (ja) * | 2000-10-10 | 2004-04-15 | カリックス セラピューティックス インコーポレイテッド | 三環式化合物およびその使用 |
| BR0312232A (pt) * | 2002-06-28 | 2005-05-10 | Vertex Pharma | Inibidores de caspases e seus usos |
| KR20070056060A (ko) * | 2004-07-14 | 2007-05-31 | 리간드 파마슈티칼스 인코포레이티드 | 세포내 수용체 조절화합물 및 방법 |
| TW200643015A (en) * | 2005-03-11 | 2006-12-16 | Akzo Nobel Nv | 2-(4-oxo-4H-quinazolin-3-yl)acetamide derivatives |
| PT1910333E (pt) * | 2005-07-26 | 2013-08-01 | Sanofi Sa | Derivados de isoquinolona substituída com piperidinilo como inibidores da rho-cinase |
| SI1912949T1 (sl) * | 2005-07-26 | 2011-12-30 | Sanofi Sa | Cikloheksilamin izokinolonski derivati kot inhibitorji Rho-kinaze |
-
2007
- 2007-09-10 AT AT07842137T patent/ATE523493T1/de not_active IP Right Cessation
- 2007-09-10 US US11/852,737 patent/US7906504B2/en active Active
- 2007-09-10 CA CA002663193A patent/CA2663193A1/en not_active Abandoned
- 2007-09-10 JP JP2009527606A patent/JP5271909B2/ja not_active Expired - Fee Related
- 2007-09-10 WO PCT/US2007/077999 patent/WO2008033757A2/en not_active Ceased
- 2007-09-10 EP EP07842137A patent/EP2066640B1/de active Active
- 2007-09-10 MX MX2009002685A patent/MX2009002685A/es active IP Right Grant
- 2007-09-10 CN CN2007800395254A patent/CN101528703B/zh not_active Expired - Fee Related
- 2007-09-11 AR ARP070104003A patent/AR062734A1/es not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| US20080064678A1 (en) | 2008-03-13 |
| EP2066640A2 (de) | 2009-06-10 |
| MX2009002685A (es) | 2009-10-13 |
| EP2066640B1 (de) | 2011-09-07 |
| AR062734A1 (es) | 2008-11-26 |
| CN101528703B (zh) | 2011-09-07 |
| WO2008033757A2 (en) | 2008-03-20 |
| JP2010502745A (ja) | 2010-01-28 |
| CN101528703A (zh) | 2009-09-09 |
| US7906504B2 (en) | 2011-03-15 |
| CA2663193A1 (en) | 2008-03-20 |
| WO2008033757A3 (en) | 2008-12-11 |
| JP5271909B2 (ja) | 2013-08-21 |
| EP2066640A4 (de) | 2010-12-22 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| RER | Ceased as to paragraph 5 lit. 3 law introducing patent treaties |