ATE546446T1 - 5-aminocyclylmethyl-oxazolidin-2-eins-derivativ - Google Patents

5-aminocyclylmethyl-oxazolidin-2-eins-derivativ

Info

Publication number
ATE546446T1
ATE546446T1 AT08861657T AT08861657T ATE546446T1 AT E546446 T1 ATE546446 T1 AT E546446T1 AT 08861657 T AT08861657 T AT 08861657T AT 08861657 T AT08861657 T AT 08861657T AT E546446 T1 ATE546446 T1 AT E546446T1
Authority
AT
Austria
Prior art keywords
aminocyclylmethyl
oxazolidine
derivative
Prior art date
Application number
AT08861657T
Other languages
English (en)
Inventor
Christian Hubschwerlen
Georg Rueedi
Jean-Philippe Surivet
Acklin Cornelia Zumbrunn
Original Assignee
Actelion Pharmaceuticals Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=40471513&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=ATE546446(T1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Actelion Pharmaceuticals Ltd filed Critical Actelion Pharmaceuticals Ltd
Application granted granted Critical
Publication of ATE546446T1 publication Critical patent/ATE546446T1/de

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A61P31/06—Antibacterial agents for tuberculosis
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Veterinary Medicine (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Oncology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Pulmonology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
AT08861657T 2007-12-18 2008-12-17 5-aminocyclylmethyl-oxazolidin-2-eins-derivativ ATE546446T1 (de)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
IB2007055194 2007-12-18
IB2008054170 2008-10-10
PCT/IB2008/055374 WO2009077989A1 (en) 2007-12-18 2008-12-17 5-aminocyclylmethyl-oxazolidin-2-one derivatives

Publications (1)

Publication Number Publication Date
ATE546446T1 true ATE546446T1 (de) 2012-03-15

Family

ID=40471513

Family Applications (1)

Application Number Title Priority Date Filing Date
AT08861657T ATE546446T1 (de) 2007-12-18 2008-12-17 5-aminocyclylmethyl-oxazolidin-2-eins-derivativ

Country Status (16)

Country Link
US (1) US9505750B2 (de)
EP (1) EP2245028B1 (de)
JP (1) JP5323088B2 (de)
KR (1) KR101578234B1 (de)
CN (1) CN101903380B (de)
AR (1) AR069800A1 (de)
AT (1) ATE546446T1 (de)
AU (1) AU2008337096B2 (de)
BR (1) BRPI0820985A2 (de)
CA (1) CA2706837C (de)
ES (1) ES2380398T3 (de)
MX (1) MX2010006111A (de)
PL (1) PL2245028T3 (de)
RU (1) RU2492169C2 (de)
TW (1) TWI441636B (de)
WO (1) WO2009077989A1 (de)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2411930T3 (es) 2008-02-20 2013-07-09 Actelion Pharmaceuticals Ltd. Compuestos antibióticos azatricíclicos
KR101294962B1 (ko) 2008-10-07 2013-08-12 액테리온 파마슈티칼 리미티드 트리사이클 옥사졸리디논 항생제 화합물
CA2738775A1 (en) * 2008-10-10 2010-04-15 Actelion Pharmaceuticals Ltd 2-benzothiophenyl-and 2-naphthyl-0xaz0lidin0nes and their azaisostere analogues as antibacterial agents
MX2011003188A (es) 2008-10-10 2011-04-27 Actelion Pharmaceuticals Ltd Antibioticos de oxazolidinilo.
US8952010B2 (en) 2011-02-07 2015-02-10 Daiichi Sankyo Company, Limited Amino group-containing pyrrolidinone derivative
JP6030146B2 (ja) * 2011-11-08 2016-11-24 アクテリオン ファーマシューティカルズ リミテッドＡｃｔｅｌｉｏｎ Ｐｈａｒｍａｃｅｕｔｉｃａｌｓ Ｌｔｄ ２−オキソ−オキサゾリジン−３，５−ジイル抗生物質誘導体
WO2014024056A1 (en) 2012-08-06 2014-02-13 Daiichi Sankyo Company, Limited Pyrrolidine derivatives with antibacterial properties
AR102256A1 (es) 2014-10-15 2017-02-15 Actelion Pharmaceuticals Ltd Derivados biaromáticos básicos antibacterianos con sustitución de aminoalcoxi
TW201833120A (zh) 2017-02-17 2018-09-16 瑞士商愛杜西亞製藥有限公司 芳基噁唑啶酮抗生素化合物

Family Cites Families (22)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE19707628A1 (de) * 1997-02-26 1998-08-27 Merck Patent Gmbh Oxazolidinone
IT1297874B1 (it) 1997-06-19 1999-12-20 Ezio Pellegrinotti Cerniera elastica per occhiali.
DE60011570T2 (de) 1999-01-07 2004-11-25 Wyeth Arylpiperazinyl-cyclohexyl indolderivate zur behandlung von depressionen
MY137020A (en) 2000-04-27 2008-12-31 Abbott Lab Diazabicyclic central nervous system active agents
GB0031086D0 (en) * 2000-12-20 2001-01-31 Smithkline Beecham Plc Medicaments
JP2004535411A (ja) 2001-05-25 2004-11-25 ブリストルーマイヤーズ スクイブ カンパニー マトリックスメタロプロテナーゼ及び／またはＴＮＦ−α転換酵素（ＴＡＣＥ）の阻害剤としてのヒダントイン及び関連複素環化合物
GB0112834D0 (en) 2001-05-25 2001-07-18 Smithkline Beecham Plc Medicaments
GB0112836D0 (en) * 2001-05-25 2001-07-18 Smithkline Beecham Plc Medicaments
TW200409637A (en) 2002-06-26 2004-06-16 Glaxo Group Ltd Compounds
WO2004032856A2 (en) 2002-10-07 2004-04-22 Smithkline Beecham Corporation Compounds
ATE411312T1 (de) * 2002-12-04 2008-10-15 Glaxo Group Ltd Chinoline und stickstoffhaltige derivatedavon und deren verwendung als antibakterielle mittel
DE10316081A1 (de) 2003-04-08 2004-10-21 Morphochem AG Aktiengesellschaft für kombinatorische Chemie Neue Verbindungen mit antibakterieller Aktivität
US7160888B2 (en) 2003-08-22 2007-01-09 Warner Lambert Company Llc [1,8]naphthyridin-2-ones and related compounds for the treatment of schizophrenia
EP1771456A2 (de) * 2004-07-30 2007-04-11 Palumed SA Hybride qa-moleküle, in denen q ein aminochinolin und a ein antibiotikarückstand ist, ihre synthese und ihre verwendung als antibakterielles mittel
DE102004041163A1 (de) 2004-08-25 2006-03-02 Morphochem Aktiengesellschaft für kombinatorische Chemie Neue Verbindungen mit antibakterieller Aktivität
JP4887297B2 (ja) 2004-09-24 2012-02-29 アクテリオン ファーマシューティカルズ リミテッド 新規二環式抗生物質
WO2006046552A1 (ja) 2004-10-27 2006-05-04 Toyama Chemical Co., Ltd. 新規な含窒素複素環化合物およびその塩
WO2007012210A2 (de) 2005-07-23 2007-02-01 Schlittler & Co. Ag Reiniger mit einweg-wischtasche
EP1996579A2 (de) 2006-03-10 2008-12-03 Actelion Pharmaceuticals Ltd. Antibiotische verbindungen
ATE469649T1 (de) 2006-03-23 2010-06-15 Actelion Pharmaceuticals Ltd Antibiotische cyclohexyl- oder piperidinylcarboxamid-derivate
CL2008001002A1 (es) * 2007-04-11 2008-10-17 Actelion Pharmaceuticals Ltd Compuestos derivados de oxazolidinona; composicion farmaceutica que comprende a dichos compuestos; y su uso para preparar un medicamento para tratar una infeccion bacteriana.
CL2008001003A1 (es) 2007-04-11 2008-10-17 Actelion Pharmaceuticals Ltd Compuestos derivados de oxazolidinona; composicion farmaceutica que comprende a dichos compuestos; y su uso para preparar un medicamento para tratar una infeccion bacteriana.

Also Published As

Publication number Publication date
US20110003789A1 (en) 2011-01-06
KR101578234B1 (ko) 2015-12-16
WO2009077989A1 (en) 2009-06-25
CN101903380A (zh) 2010-12-01
ES2380398T3 (es) 2012-05-11
TW200932230A (en) 2009-08-01
CN101903380B (zh) 2013-04-17
EP2245028B1 (de) 2012-02-22
JP2011506593A (ja) 2011-03-03
TWI441636B (zh) 2014-06-21
RU2492169C2 (ru) 2013-09-10
AR069800A1 (es) 2010-02-17
US9505750B2 (en) 2016-11-29
AU2008337096B2 (en) 2013-10-17
RU2010129113A (ru) 2012-01-27
EP2245028A1 (de) 2010-11-03
BRPI0820985A2 (pt) 2015-06-16
KR20100092965A (ko) 2010-08-23
MX2010006111A (es) 2010-06-25
AU2008337096A1 (en) 2009-06-25
CA2706837C (en) 2016-05-03
JP5323088B2 (ja) 2013-10-23
PL2245028T3 (pl) 2012-07-31
CA2706837A1 (en) 2009-06-25

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