ATE546446T1 - 5-aminocyclylmethyl-oxazolidin-2-eins-derivativ - Google Patents

5-aminocyclylmethyl-oxazolidin-2-eins-derivativ

Info

Publication number
ATE546446T1
ATE546446T1 AT08861657T AT08861657T ATE546446T1 AT E546446 T1 ATE546446 T1 AT E546446T1 AT 08861657 T AT08861657 T AT 08861657T AT 08861657 T AT08861657 T AT 08861657T AT E546446 T1 ATE546446 T1 AT E546446T1
Authority
AT
Austria
Prior art keywords
aminocyclylmethyl
oxazolidine
derivative
Prior art date
Application number
AT08861657T
Other languages
English (en)
Inventor
Christian Hubschwerlen
Georg Rueedi
Jean-Philippe Surivet
Acklin Cornelia Zumbrunn
Original Assignee
Actelion Pharmaceuticals Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=40471513&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=ATE546446(T1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Actelion Pharmaceuticals Ltd filed Critical Actelion Pharmaceuticals Ltd
Application granted granted Critical
Publication of ATE546446T1 publication Critical patent/ATE546446T1/de

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • A61P31/06Antibacterial agents for tuberculosis
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D413/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/14Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/14Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Oncology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Communicable Diseases (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pulmonology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
AT08861657T 2007-12-18 2008-12-17 5-aminocyclylmethyl-oxazolidin-2-eins-derivativ ATE546446T1 (de)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
IB2007055194 2007-12-18
IB2008054170 2008-10-10
PCT/IB2008/055374 WO2009077989A1 (en) 2007-12-18 2008-12-17 5-aminocyclylmethyl-oxazolidin-2-one derivatives

Publications (1)

Publication Number Publication Date
ATE546446T1 true ATE546446T1 (de) 2012-03-15

Family

ID=40471513

Family Applications (1)

Application Number Title Priority Date Filing Date
AT08861657T ATE546446T1 (de) 2007-12-18 2008-12-17 5-aminocyclylmethyl-oxazolidin-2-eins-derivativ

Country Status (16)

Country Link
US (1) US9505750B2 (de)
EP (1) EP2245028B1 (de)
JP (1) JP5323088B2 (de)
KR (1) KR101578234B1 (de)
CN (1) CN101903380B (de)
AR (1) AR069800A1 (de)
AT (1) ATE546446T1 (de)
AU (1) AU2008337096B2 (de)
BR (1) BRPI0820985A2 (de)
CA (1) CA2706837C (de)
ES (1) ES2380398T3 (de)
MX (1) MX2010006111A (de)
PL (1) PL2245028T3 (de)
RU (1) RU2492169C2 (de)
TW (1) TWI441636B (de)
WO (1) WO2009077989A1 (de)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2411930T3 (es) 2008-02-20 2013-07-09 Actelion Pharmaceuticals Ltd. Compuestos antibióticos azatricíclicos
DK2344495T3 (en) 2008-10-07 2015-02-02 Actelion Pharmaceuticals Ltd TRICYCLIC OXAZOLIDINON ANTIBIOTIC COMPOUNDS
ES2395491T3 (es) * 2008-10-10 2013-02-13 Actelion Pharmaceuticals Ltd. 2-Benzotiofenil y 2-naftil-oxazolidinonas y sus análogos azaisósteros como agentes antibacterianos
RU2516701C2 (ru) * 2008-10-10 2014-05-20 Актелион Фармасьютиклз Лтд Оксазолидиниловые антибиотики
EP2674430A4 (de) 2011-02-07 2014-07-02 Daiichi Sankyo Co Ltd Aminogruppenhaltige pyrrolidinonderivate
SG11201401710PA (en) * 2011-11-08 2014-09-26 Actelion Pharmaceuticals Ltd 2-oxo-oxazolidin-3,5-diyl antibiotic derivatives
WO2014024056A1 (en) 2012-08-06 2014-02-13 Daiichi Sankyo Company, Limited Pyrrolidine derivatives with antibacterial properties
AR102256A1 (es) 2014-10-15 2017-02-15 Actelion Pharmaceuticals Ltd Derivados biaromáticos básicos antibacterianos con sustitución de aminoalcoxi
TW201833120A (zh) 2017-02-17 2018-09-16 瑞士商愛杜西亞製藥有限公司 芳基噁唑啶酮抗生素化合物

Family Cites Families (22)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE19707628A1 (de) * 1997-02-26 1998-08-27 Merck Patent Gmbh Oxazolidinone
IT1297874B1 (it) 1997-06-19 1999-12-20 Ezio Pellegrinotti Cerniera elastica per occhiali.
ES2219302T3 (es) 1999-01-07 2004-12-01 Wyeth Derivados de arilpiperazinil-ciclohexilindol para el tratamiento de la depresion.
MY145722A (en) 2000-04-27 2012-03-30 Abbott Lab Diazabicyclic central nervous system active agents
GB0031086D0 (en) 2000-12-20 2001-01-31 Smithkline Beecham Plc Medicaments
CA2447475A1 (en) 2001-05-25 2002-12-05 Chu-Biao Xue Hydantion derivatives as inhibitors of matrix metalloproteinases
GB0112836D0 (en) 2001-05-25 2001-07-18 Smithkline Beecham Plc Medicaments
GB0112834D0 (en) 2001-05-25 2001-07-18 Smithkline Beecham Plc Medicaments
AR040336A1 (es) 2002-06-26 2005-03-30 Glaxo Group Ltd Compuesto de piperidina, uso del mismo para la fabricacion de un medicamento, composicion farmaceutica que lo comprende y procedimiento para preparar dicho compuesto
WO2004032856A2 (en) 2002-10-07 2004-04-22 Smithkline Beecham Corporation Compounds
WO2004050036A2 (en) 2002-12-04 2004-06-17 Glaxo Group Limited Quinolines and nitrogenated derivatives thereof and their use as antibacterial agents
DE10316081A1 (de) * 2003-04-08 2004-10-21 Morphochem AG Aktiengesellschaft für kombinatorische Chemie Neue Verbindungen mit antibakterieller Aktivität
US7160888B2 (en) 2003-08-22 2007-01-09 Warner Lambert Company Llc [1,8]naphthyridin-2-ones and related compounds for the treatment of schizophrenia
BRPI0514381A (pt) 2004-07-30 2008-06-10 Palumed Sa compostos hìbridos de aminoquinolina-antibiótico, composições farmacêuticas, método de preparação e uso destes
DE102004041163A1 (de) 2004-08-25 2006-03-02 Morphochem Aktiengesellschaft für kombinatorische Chemie Neue Verbindungen mit antibakterieller Aktivität
JP4887297B2 (ja) 2004-09-24 2012-02-29 アクテリオン ファーマシューティカルズ リミテッド 新規二環式抗生物質
JP5314244B2 (ja) 2004-10-27 2013-10-16 富山化学工業株式会社 新規な含窒素複素環化合物およびその塩
WO2007012210A2 (de) 2005-07-23 2007-02-01 Schlittler & Co. Ag Reiniger mit einweg-wischtasche
CA2643962A1 (en) 2006-03-10 2007-09-20 Actelion Pharmaceuticals Ltd Antibiotic compounds
EP2001478B1 (de) 2006-03-23 2010-06-02 Actelion Pharmaceuticals Ltd. Antibiotische cyclohexyl- oder piperidinylcarboxamid-derivate
CL2008001002A1 (es) * 2007-04-11 2008-10-17 Actelion Pharmaceuticals Ltd Compuestos derivados de oxazolidinona; composicion farmaceutica que comprende a dichos compuestos; y su uso para preparar un medicamento para tratar una infeccion bacteriana.
CL2008001003A1 (es) 2007-04-11 2008-10-17 Actelion Pharmaceuticals Ltd Compuestos derivados de oxazolidinona; composicion farmaceutica que comprende a dichos compuestos; y su uso para preparar un medicamento para tratar una infeccion bacteriana.

Also Published As

Publication number Publication date
CA2706837C (en) 2016-05-03
CN101903380A (zh) 2010-12-01
EP2245028A1 (de) 2010-11-03
CN101903380B (zh) 2013-04-17
WO2009077989A1 (en) 2009-06-25
CA2706837A1 (en) 2009-06-25
AU2008337096A1 (en) 2009-06-25
EP2245028B1 (de) 2012-02-22
KR101578234B1 (ko) 2015-12-16
PL2245028T3 (pl) 2012-07-31
TW200932230A (en) 2009-08-01
AU2008337096B2 (en) 2013-10-17
JP2011506593A (ja) 2011-03-03
ES2380398T3 (es) 2012-05-11
KR20100092965A (ko) 2010-08-23
JP5323088B2 (ja) 2013-10-23
RU2492169C2 (ru) 2013-09-10
MX2010006111A (es) 2010-06-25
BRPI0820985A2 (pt) 2015-06-16
TWI441636B (zh) 2014-06-21
AR069800A1 (es) 2010-02-17
RU2010129113A (ru) 2012-01-27
US20110003789A1 (en) 2011-01-06
US9505750B2 (en) 2016-11-29

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