ATE69446T1 - 5-lipoxygenase-inhibitoren. - Google Patents

5-lipoxygenase-inhibitoren.

Info

Publication number: ATE69446T1
Authority: AT; Austria
Prior art keywords: substituted; lipoxygenase inhibitors; tetrazol; benzothiazine; dioxides
Prior art date: 1985-04-16

Application number

AT86302746T

Other languages

English (en)

Inventor

Isao Nagakura

Susumu Nakanishi

Original Assignee

Pfizer

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1985-04-16

Filing date

1986-04-14

Publication date

1991-11-15

1986-04-14 Application filed by Pfizer filed Critical Pfizer

1991-11-15 Application granted granted Critical

1991-11-15 Publication of ATE69446T1 publication Critical patent/ATE69446T1/de

Links

239000000867 Lipoxygenase Inhibitor Substances 0.000 title 1
-1 2-substituted-1,3,4-oxadiazol-5-yl Chemical group 0.000 abstract 3
UJVBZCCNLAAMOV-UHFFFAOYSA-N 2h-1,2-benzothiazine Chemical compound C1=CC=C2C=CNSC2=C1 UJVBZCCNLAAMOV-UHFFFAOYSA-N 0.000 abstract 1
102000001381 Arachidonate 5-Lipoxygenase Human genes 0.000 abstract 1
108010093579 Arachidonate 5-lipoxygenase Proteins 0.000 abstract 1
239000003112 inhibitor Substances 0.000 abstract 1
230000037361 pathway Effects 0.000 abstract 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Veterinary Medicine (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Bioinformatics & Cheminformatics (AREA)
Pharmacology & Pharmacy (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Engineering & Computer Science (AREA)
Immunology (AREA)
Pulmonology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Plural Heterocyclic Compounds (AREA)
Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Medicines Containing Material From Animals Or Micro-Organisms (AREA)
Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Food Preservation Except Freezing, Refrigeration, And Drying (AREA)
Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
Agricultural Chemicals And Associated Chemicals (AREA)
Preparation Of Compounds By Using Micro-Organisms (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Saccharide Compounds (AREA)

AT86302746T 1985-04-16 1986-04-14 5-lipoxygenase-inhibitoren. ATE69446T1 (de)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
JP60080666A JPS61238785A (ja)	1985-04-16	1985-04-16	１、２―ベンゾチアジン類
EP86302746A EP0200408B1 (de)	1985-04-16	1986-04-14	5-Lipoxygenase-Inhibitoren

Publications (1)

Publication Number	Publication Date
ATE69446T1 true ATE69446T1 (de)	1991-11-15

Family

ID=13724685

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
AT86302746T ATE69446T1 (de)	1985-04-16	1986-04-14	5-lipoxygenase-inhibitoren.

Country Status (21)

Country	Link
US (1)	US4694080A (de)
EP (1)	EP0200408B1 (de)
JP (1)	JPS61238785A (de)
AT (1)	ATE69446T1 (de)
AU (1)	AU562532B2 (de)
CA (1)	CA1277318C (de)
DD (4)	DD258010A5 (de)
DE (1)	DE3682424D1 (de)
DK (1)	DK170086A (de)
ES (2)	ES8800218A1 (de)
FI (1)	FI87353C (de)
GR (1)	GR860977B (de)
HU (1)	HU207862B (de)
IE (1)	IE59041B1 (de)
IL (1)	IL78501A (de)
NZ (1)	NZ215821A (de)
PH (1)	PH22452A (de)
PL (2)	PL149169B1 (de)
PT (1)	PT82385B (de)
YU (2)	YU45012B (de)
ZA (1)	ZA862790B (de)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
CN122404318A (zh) *	2026-06-22	2026-07-17	齐鲁医药学院	1,2-苯并噻嗪双噁二唑衍生物及其制备方法

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US3303189A (en) *	1965-03-11	1967-02-07	Smith Kline French Lab	2, 1-benzothiazine-2, 2-dioxides
US3957772A (en) *	1975-05-21	1976-05-18	Warner-Lambert Company	Process for the preparation of 4-hydroxy-3-(5-methyl-3-isoxazolylcarbamoyl)-2-methyl-2h-1,2-benzothiazine 1,1-dioxide
US3987038A (en) *	1975-05-21	1976-10-19	Warner-Lambert Company	Process for the preparation of {1-[5-(4-hydroxy-2H-1,2-benzothiazin-3-yl)-1,2,4-oxadiazol-3-yl]methyl}ethanone S,S-dioxide

1985
- 1985-04-16 JP JP60080666A patent/JPS61238785A/ja active Granted
1986
- 1986-03-19 US US06/841,509 patent/US4694080A/en not_active Expired - Fee Related
- 1986-04-14 NZ NZ215821A patent/NZ215821A/xx unknown
- 1986-04-14 EP EP86302746A patent/EP0200408B1/de not_active Expired - Lifetime
- 1986-04-14 PT PT82385A patent/PT82385B/pt not_active IP Right Cessation
- 1986-04-14 DE DE8686302746T patent/DE3682424D1/de not_active Expired - Lifetime
- 1986-04-14 CA CA000506537A patent/CA1277318C/en not_active Expired - Lifetime
- 1986-04-14 GR GR860977A patent/GR860977B/el unknown
- 1986-04-14 AT AT86302746T patent/ATE69446T1/de not_active IP Right Cessation
- 1986-04-15 HU HU861575A patent/HU207862B/hu not_active IP Right Cessation
- 1986-04-15 YU YU608/86A patent/YU45012B/xx unknown
- 1986-04-15 IE IE97986A patent/IE59041B1/en not_active IP Right Cessation
- 1986-04-15 AU AU56100/86A patent/AU562532B2/en not_active Ceased
- 1986-04-15 ZA ZA862790A patent/ZA862790B/xx unknown
- 1986-04-15 DK DK170086A patent/DK170086A/da not_active Application Discontinuation
- 1986-04-15 FI FI861587A patent/FI87353C/fi not_active IP Right Cessation
- 1986-04-15 IL IL78501A patent/IL78501A/xx not_active IP Right Cessation
- 1986-04-15 ES ES554005A patent/ES8800218A1/es not_active Expired
- 1986-04-16 PH PH33663A patent/PH22452A/en unknown
- 1986-04-16 PL PL1986258986A patent/PL149169B1/pl unknown
- 1986-04-16 DD DD86289231A patent/DD258010A5/de not_active IP Right Cessation
- 1986-04-16 DD DD86314100A patent/DD269385A5/de not_active IP Right Cessation
- 1986-04-16 DD DD86314101A patent/DD269386A5/de not_active IP Right Cessation
- 1986-04-16 PL PL1986268860A patent/PL149788B1/pl unknown
- 1986-04-16 DD DD86314099A patent/DD273257A5/de not_active IP Right Cessation
1987
- 1987-05-16 ES ES557555A patent/ES8802519A1/es not_active Expired
- 1987-06-15 YU YU1110/87A patent/YU44631B/xx unknown

Also Published As

Publication number	Publication date
IE59041B1 (en)	1993-12-15
DK170086D0 (da)	1986-04-15
DD258010A5 (de)	1988-07-06
FI87353C (fi)	1992-12-28
YU44631B (en)	1990-10-31
DK170086A (da)	1986-10-17
DD269386A5 (de)	1989-06-28
JPH058711B2 (de)	1993-02-02
ES557555A0 (es)	1988-07-16
CA1277318C (en)	1990-12-04
EP0200408B1 (de)	1991-11-13
FI861587A0 (fi)	1986-04-15
IL78501A0 (en)	1986-08-31
PL149169B1 (en)	1990-01-31
PT82385B (pt)	1988-10-14
ES8802519A1 (es)	1988-07-16
PT82385A (en)	1986-05-01
JPS61238785A (ja)	1986-10-24
DD273257A5 (de)	1989-11-08
EP0200408A1 (de)	1986-11-05
DD269385A5 (de)	1989-06-28
PL149788B1 (en)	1990-03-31
NZ215821A (en)	1988-09-29
US4694080A (en)	1987-09-15
ZA862790B (en)	1987-11-25
ES554005A0 (es)	1987-10-16
AU562532B2 (en)	1987-06-11
YU45012B (en)	1991-06-30
IL78501A (en)	1991-03-10
PH22452A (en)	1988-09-12
HUT42086A (en)	1987-06-29
FI87353B (fi)	1992-09-15
PL268860A1 (en)	1988-07-07
HU207862B (en)	1993-06-28
YU111087A (en)	1988-06-30
IE860979L (en)	1986-10-16
YU60886A (en)	1988-02-29
GR860977B (en)	1986-08-06
AU5610086A (en)	1986-10-23
DE3682424D1 (de)	1991-12-19
ES8800218A1 (es)	1987-10-16
FI861587L (fi)	1986-10-17

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Legal Events

Date	Code	Title	Description
1992-07-15	UEP	Publication of translation of european patent specification
1998-01-15	REN	Ceased due to non-payment of the annual fee