BG61202B2 - Стабилизиран фармацевтичен състав и неговото получаване - Google Patents

Стабилизиран фармацевтичен състав и неговото получаване Download PDF

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Publication number
BG61202B2
BG61202B2 BG098473A BG9847394A BG61202B2 BG 61202 B2 BG61202 B2 BG 61202B2 BG 098473 A BG098473 A BG 098473A BG 9847394 A BG9847394 A BG 9847394A BG 61202 B2 BG61202 B2 BG 61202B2
Authority
BG
Bulgaria
Prior art keywords
pharmaceutical composition
compound
hydrogen
composition according
alkyl
Prior art date
Application number
BG098473A
Other languages
Bulgarian (bg)
English (en)
Inventor
Tadashi Makino
Tetsuro Tabata
Shin-Ichiro Hirai
Original Assignee
Takeda Chemical Industries, Ltd.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=26367776&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=BG61202(B2) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Takeda Chemical Industries, Ltd. filed Critical Takeda Chemical Industries, Ltd.
Publication of BG61202B2 publication Critical patent/BG61202B2/bg

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/02—Inorganic compounds
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • A61K9/1605—Excipients; Inactive ingredients
    • A61K9/1611—Inorganic compounds
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2009—Inorganic compounds
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
    • A61K9/5005—Wall or coating material
    • A61K9/5021—Organic macromolecular compounds
    • A61K9/5026—Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
    • A61K9/5073—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals having two or more different coatings optionally including drug-containing subcoatings
    • A61K9/5078—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals having two or more different coatings optionally including drug-containing subcoatings with drug-free core

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Inorganic Chemistry (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
BG098473A 1986-02-13 1994-02-14 Стабилизиран фармацевтичен състав и неговото получаване BG61202B2 (bg)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP2956786 1986-02-13
JP3805986 1986-02-21

Publications (1)

Publication Number Publication Date
BG61202B2 true BG61202B2 (bg) 1997-02-28

Family

ID=26367776

Family Applications (1)

Application Number Title Priority Date Filing Date
BG098473A BG61202B2 (bg) 1986-02-13 1994-02-14 Стабилизиран фармацевтичен състав и неговото получаване

Country Status (7)

Country Link
US (2) US5045321A (de)
EP (3) EP0237200B1 (de)
BG (1) BG61202B2 (de)
CA (1) CA1327010C (de)
DE (3) DE3751845T2 (de)
HK (2) HK188195A (de)
SG (1) SG50619A1 (de)

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* Cited by examiner, † Cited by third party
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US5045321A (en) 1991-09-03
EP0237200A2 (de) 1987-09-16
DE3751845D1 (de) 1996-07-25
EP0446961A3 (en) 1992-04-01
SG50619A1 (en) 1998-07-20
US5093132A (en) 1992-03-03
CA1327010C (en) 1994-02-15
EP0237200A3 (en) 1988-02-03
EP0446961B1 (de) 1996-06-19
HK188195A (en) 1995-12-22
EP0423748B1 (de) 1994-08-24
DE3750431T2 (de) 1994-12-22
EP0237200B1 (de) 1992-07-01
DE3780045T2 (de) 1992-12-24
DE3750431D1 (de) 1994-09-29
HK1002021A1 (en) 1998-07-24
EP0446961A2 (de) 1991-09-18
DE3780045D1 (de) 1992-08-06
DE3751845T2 (de) 1996-11-28
EP0423748A1 (de) 1991-04-24

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