BR9607182A - Antagonistas de vasopressina de benzazepina tricíclicos - Google Patents
Antagonistas de vasopressina de benzazepina tricíclicosInfo
- Publication number
- BR9607182A BR9607182A BR9607182A BR9607182A BR9607182A BR 9607182 A BR9607182 A BR 9607182A BR 9607182 A BR9607182 A BR 9607182A BR 9607182 A BR9607182 A BR 9607182A BR 9607182 A BR9607182 A BR 9607182A
- Authority
- BR
- Brazil
- Prior art keywords
- vasopressin antagonists
- tricyclic benzazepine
- benzazepine vasopressin
- tricyclic
- antagonists
- Prior art date
Links
- DQFQCHIDRBIESA-UHFFFAOYSA-N 1-benzazepine Chemical compound N1C=CC=CC2=CC=CC=C12 DQFQCHIDRBIESA-UHFFFAOYSA-N 0.000 title 1
- 229940116211 Vasopressin antagonist Drugs 0.000 title 1
- 239000003038 vasopressin antagonist Substances 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/12—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains three hetero rings
- C07D471/14—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/16—Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/12—Drugs for disorders of the urinary system of the kidneys
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/12—Drugs for disorders of the metabolism for electrolyte homeostasis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/08—Plasma substitutes; Perfusion solutions; Dialytics or haemodialytics; Drugs for electrolytic or acid-base disorders, e.g. hypovolemic shock
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/02—Non-specific cardiovascular stimulants, e.g. drugs for syncope, antihypotensives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/04—Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/08—Vasodilators for multiple indications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/12—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains three hetero rings
- C07D487/14—Ortho-condensed systems
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Veterinary Medicine (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Public Health (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Hematology (AREA)
- Diabetes (AREA)
- Urology & Nephrology (AREA)
- Neurology (AREA)
- Hospice & Palliative Care (AREA)
- Neurosurgery (AREA)
- Biomedical Technology (AREA)
- Psychiatry (AREA)
- Obesity (AREA)
- Vascular Medicine (AREA)
- Pulmonology (AREA)
- Gastroenterology & Hepatology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US08/373,132 US5536718A (en) | 1995-01-17 | 1995-01-17 | Tricyclic benzazepine vasopressin antagonists |
| PCT/US1996/001076 WO1996022293A1 (en) | 1995-01-17 | 1996-01-16 | Tricyclic benzazepine vasopressin antagonists |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| BR9607182A true BR9607182A (pt) | 1997-11-11 |
Family
ID=23471110
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BR9607182A BR9607182A (pt) | 1995-01-17 | 1996-01-16 | Antagonistas de vasopressina de benzazepina tricíclicos |
Country Status (23)
| Country | Link |
|---|---|
| US (3) | US5536718A (pt) |
| EP (1) | EP0804438B1 (pt) |
| JP (2) | JP4163252B2 (pt) |
| KR (1) | KR100443438B1 (pt) |
| CN (1) | CN1065244C (pt) |
| AR (1) | AR002022A1 (pt) |
| AT (1) | ATE320429T1 (pt) |
| AU (1) | AU707982B2 (pt) |
| BR (1) | BR9607182A (pt) |
| CZ (1) | CZ297797B6 (pt) |
| DE (1) | DE69635922T2 (pt) |
| DK (1) | DK0804438T3 (pt) |
| EA (1) | EA001143B1 (pt) |
| ES (1) | ES2258267T3 (pt) |
| HU (1) | HUP9800646A3 (pt) |
| IL (1) | IL116775A (pt) |
| MX (1) | MX9705313A (pt) |
| NZ (1) | NZ302111A (pt) |
| PT (1) | PT804438E (pt) |
| TW (1) | TW403752B (pt) |
| UA (1) | UA54383C2 (pt) |
| WO (1) | WO1996022293A1 (pt) |
| ZA (1) | ZA96297B (pt) |
Families Citing this family (61)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5736540A (en) * | 1993-07-29 | 1998-04-07 | American Cyanamid Company | Tricyclic diazepine vasopressin antagonists and oxytocin antagonists |
| US7071133B2 (en) * | 1993-11-16 | 2006-07-04 | Ppg Industries Ohio, Inc. | Colored glass compositions and-automotive vision panels with-reduced transmitted-color shift |
| CN1174975C (zh) * | 1994-06-10 | 2004-11-10 | 史密丝克莱恩比彻姆有限公司 | 苯并吡喃类化合物和它们作为治疗剂的用途 |
| PL319406A1 (en) * | 1994-09-30 | 1997-08-04 | Basf Ag | Novel heterocyclically substituted imidazoqunoxalinones, their production and application |
| US5700796A (en) * | 1995-01-17 | 1997-12-23 | American Cyanamid Company | Tricyclic benzazepine vasopressin antagonists |
| US5753648A (en) * | 1995-01-17 | 1998-05-19 | American Cyanamid Company | Tricyclic benzazepine vasopressin antagonists |
| US5880122A (en) * | 1996-11-01 | 1999-03-09 | American Home Products Corporation | 3-Carboxamide derivatives of 5H-pyrrolo 2,1-c! 1,4!-benzodiazepines |
| US7096692B2 (en) * | 1997-03-14 | 2006-08-29 | Ppg Industries Ohio, Inc. | Visible-light-responsive photoactive coating, coated article, and method of making same |
| US20030039843A1 (en) * | 1997-03-14 | 2003-02-27 | Christopher Johnson | Photoactive coating, coated article, and method of making same |
| US20020155299A1 (en) | 1997-03-14 | 2002-10-24 | Harris Caroline S. | Photo-induced hydrophilic article and method of making same |
| WO1998043976A1 (en) * | 1997-03-31 | 1998-10-08 | Wakamoto Pharmaceutical Co., Ltd. | Biphenyl derivatives and medicinal compositions |
| US20030022889A1 (en) * | 1997-04-15 | 2003-01-30 | Bymaster Franklin P. | Method for providing neuro-protective effects |
| WO1998046596A1 (en) * | 1997-04-15 | 1998-10-22 | Eli Lilly And Company | Method for providing neuro-protective effects |
| US6511974B1 (en) | 1997-07-30 | 2003-01-28 | Wyeth | Tricyclic vasopressin agonists |
| US6194407B1 (en) | 1997-07-30 | 2001-02-27 | American Home Products Corporation | Tricyclic pyrido vasopressin agonists |
| US7138393B2 (en) * | 1998-07-24 | 2006-11-21 | Wyeth | Biologically active vasopressin agonist metabolites |
| US6090803A (en) * | 1998-07-24 | 2000-07-18 | American Home Products Corporation | Tricyclic vasopressin agonists |
| US6235900B1 (en) | 1999-02-04 | 2001-05-22 | American Home Products Corporation | Tricyclic pyridine N-oxides vasopressin agonists |
| US6297234B1 (en) | 1999-02-04 | 2001-10-02 | American Home Products Corporation | Arylthiophene vasopressin agonists |
| JP2003510280A (ja) * | 1999-09-27 | 2003-03-18 | アメリカン・サイアナミド・カンパニー | バソプレッシンアゴニスト処方および製法 |
| EP1317266A2 (en) * | 2000-08-08 | 2003-06-11 | Ortho-McNeil Pharmaceutical, Inc. | Neuroprotective 2-pyridinamine compositions and related methods |
| US20050203092A1 (en) * | 2000-08-08 | 2005-09-15 | Benjamin Elfrida R. | 4-Pyrimidinamine derivatives, pharmaceutical compositions and related methods |
| US6677063B2 (en) | 2000-08-31 | 2004-01-13 | Ppg Industries Ohio, Inc. | Methods of obtaining photoactive coatings and/or anatase crystalline phase of titanium oxides and articles made thereby |
| US7323249B2 (en) * | 2000-08-31 | 2008-01-29 | Ppg Industries Ohio, Inc. | Methods of obtaining photoactive coatings and/or anatase crystalline phase of titanium oxides and articles made thereby |
| US6977254B2 (en) * | 2001-04-12 | 2005-12-20 | Wyeth | Hydroxy cyclohexenyl phenyl carboxamides tocolytic oxytocin receptor antagonists |
| US7326700B2 (en) * | 2001-04-12 | 2008-02-05 | Wyeth | Cyclohexenyl phenyl carboxamides tocolytic oxytocin receptor antagonists |
| US7202239B2 (en) * | 2001-04-12 | 2007-04-10 | Wyeth | Cyclohexylphenyl carboxamides tocolytic oxytocin receptor antagonists |
| US6900200B2 (en) | 2001-04-12 | 2005-05-31 | Wyeth | Tricyclic hydroxy carboxamides and derivatives thereof tocolytic oxytocin receptor antagonists |
| US7064120B2 (en) * | 2001-04-12 | 2006-06-20 | Wyeth | Tricyclic pyridyl carboxamides and derivatives thereof tocolytic oxytocin receptor antagonists |
| US7022699B2 (en) | 2001-04-12 | 2006-04-04 | Wyeth | Cyclohexenyl phenyl diazepines vasopressin and oxytocin receptor modulators |
| US7109193B2 (en) | 2001-04-12 | 2006-09-19 | Wyeth | Tricyclic diazepines tocolytic oxytocin receptor antagonists |
| CN1294134C (zh) * | 2001-04-12 | 2007-01-10 | 惠氏公司 | 环己基苯基血管升压素激动剂 |
| EP1381370B1 (en) | 2001-04-12 | 2007-03-07 | Wyeth | N-biphenylcarbonyl- and n-phenylpyridylcarbonyl substituted bi- and tricyclic azepines and diazepines as vasopressing agonists |
| SE0102299D0 (sv) | 2001-06-26 | 2001-06-26 | Astrazeneca Ab | Compounds |
| SE0102764D0 (sv) | 2001-08-17 | 2001-08-17 | Astrazeneca Ab | Compounds |
| US7232615B2 (en) * | 2001-10-22 | 2007-06-19 | Ppg Industries Ohio, Inc. | Coating stack comprising a layer of barrier coating |
| US20040010010A1 (en) * | 2002-04-30 | 2004-01-15 | Ebetino Frank Hallock | Melanocortin receptor ligands |
| EP1603858A2 (en) * | 2003-03-11 | 2005-12-14 | NeuroSearch A/S | Kcnq channel modulating compounds and their pharmaceutical use |
| US20060029754A1 (en) * | 2004-08-05 | 2006-02-09 | Medwick Paul A | Coated substrate with improved solar control properties |
| EP1632494A1 (en) * | 2004-08-24 | 2006-03-08 | Ferring B.V. | Vasopressin v1a antagonists |
| US20060046089A1 (en) * | 2004-09-01 | 2006-03-02 | O'shaughnessy Dennis J | Metal based coating composition and related coated substrates |
| US7947373B2 (en) * | 2004-10-14 | 2011-05-24 | Pittsburgh Glass Works, Llc | High luminance coated glass |
| US7563793B2 (en) * | 2004-12-20 | 2009-07-21 | Wyeth | Pyrrolo[1,2-a]quinoxalin-5-(4H)-yl)sulfonyls and carbonyls and their use as estrogenic agents |
| US7473471B2 (en) * | 2005-03-21 | 2009-01-06 | Ppg Industries Ohio, Inc. | Coating composition with solar properties |
| KR101346902B1 (ko) | 2005-07-09 | 2014-01-02 | 아스트라제네카 아베 | 당뇨병 치료에 있어 glk 활성화제로서 사용하기 위한헤테로아릴 벤즈아미드 유도체 |
| UY30117A1 (es) * | 2006-01-31 | 2007-06-29 | Tanabe Seiyaku Co | Compuesto amina trisustituido |
| US20100124642A1 (en) * | 2008-11-19 | 2010-05-20 | Ppg Industries Ohio, Inc. | Undercoating layers providing improved conductive topcoat functionality |
| JP5343133B2 (ja) | 2008-11-19 | 2013-11-13 | ピーピージー・インダストリーズ・オハイオ・インコーポレイテッド | トップコートの機能を向上させるアンダーコーティング層 |
| US8133599B2 (en) * | 2008-11-19 | 2012-03-13 | Ppg Industries Ohio, Inc | Undercoating layers providing improved photoactive topcoat functionality |
| US7998586B2 (en) | 2008-11-19 | 2011-08-16 | Ppg Industries Ohio, Inc. | Undercoating layers providing improved topcoat functionality |
| AR076221A1 (es) | 2009-04-09 | 2011-05-26 | Astrazeneca Ab | Derivado de pirazol [4,5-e] pirimidina y su uso para tratar diabetes y obesidad |
| US20110146768A1 (en) | 2009-12-21 | 2011-06-23 | Ppg Industries Ohio, Inc. | Silicon thin film solar cell having improved underlayer coating |
| US9224892B2 (en) | 2009-12-21 | 2015-12-29 | Ppg Industries Ohio, Inc. | Silicon thin film solar cell having improved haze and methods of making the same |
| RU2518102C1 (ru) * | 2012-11-01 | 2014-06-10 | Федеральное государственное бюджетное образовательное учреждение высшего профессионального образования "Кубанский государственный технологический университет" (ФГБОУ ВПО "КубГТУ") | Способ получения производных 2-диалкиламинопирроло[1,2-альфа][1,4]бензодиазепина |
| CA3046809A1 (en) * | 2016-12-12 | 2018-06-21 | The University Of Sydney | Non-peptide oxytocin receptor agonists |
| US10961242B2 (en) | 2017-05-17 | 2021-03-30 | Legochem Biosciences, Inc. | Compounds as autotaxin inhibitors and pharmaceutical compositions comprising the same |
| KR101798840B1 (ko) | 2017-05-17 | 2017-11-17 | 주식회사 레고켐 바이오사이언스 | 신규 오토탁신 저해 화합물 및 이를 함유하는 약제학적 조성물 |
| AU2018300150A1 (en) | 2017-07-11 | 2020-01-30 | Vertex Pharmaceuticals Incorporated | Carboxamides as modulators of sodium channels |
| US12440481B2 (en) | 2019-01-10 | 2025-10-14 | Vertex Pharmaceuticals Incorporated | Esters and carbamates as modulators of sodium channels |
| WO2020146682A1 (en) | 2019-01-10 | 2020-07-16 | Vertex Pharmaceuticals Incorporated | Carboxamides as modulators of sodium channels |
| US20240287074A1 (en) * | 2020-09-07 | 2024-08-29 | Kinoxis Therapeutics Pty Ltd | Salts and crystals |
Family Cites Families (20)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4766108A (en) * | 1986-12-04 | 1988-08-23 | Smith Kline Beckman Corporation | Tyr-Arg-vasopressin antagonists |
| US5055448A (en) * | 1987-06-25 | 1991-10-08 | Medical College Of Ohio | Linear derivatives of arginine vasopressin antagonists |
| EP0382185B1 (en) * | 1989-02-10 | 1994-06-15 | Otsuka Pharmaceutical Co., Ltd. | Carbostyril derivatives |
| DK0450097T3 (da) * | 1989-10-20 | 1996-05-20 | Otsuka Pharma Co Ltd | Benzoheterocykliske forbindelser |
| US5258510A (en) * | 1989-10-20 | 1993-11-02 | Otsuka Pharma Co Ltd | Benzoheterocyclic compounds |
| US5070187A (en) * | 1989-11-03 | 1991-12-03 | Trustees Of Boston University | Pharmacologically effective antagonists of arginine-vasopressin |
| TW199153B (pt) * | 1990-08-07 | 1993-02-01 | Dtsuka Seiyaku Kk | |
| JPH04163252A (ja) * | 1990-10-25 | 1992-06-08 | Teijin Ltd | エアーバッグ |
| TW198715B (pt) * | 1991-04-19 | 1993-01-21 | Dtsuka Seiyaku Kk | |
| KR100207360B1 (ko) * | 1991-06-14 | 1999-07-15 | 돈 더블유. 슈미츠 | 이미다조[1,5,-a]퀸옥살린 |
| EP0533242A3 (en) * | 1991-09-16 | 1993-09-15 | Merck & Co. Inc. | Substituted derivatives of piperazinylcamphorsulfonyl oxytocin antagonists |
| EP0533243B1 (en) * | 1991-09-16 | 1997-12-17 | Merck & Co. Inc. | Hydantoin and succinimide-substituted spiroindanylcamphorsulfonyl derivatives |
| EP0533240A3 (en) * | 1991-09-16 | 1993-09-29 | Merck & Co. Inc. | Substituted amine derivatives of piperazinylcamphorsulfonyl oxytocin antagonists |
| US5204349A (en) * | 1991-09-16 | 1993-04-20 | Merck & Co., Inc. | Amide-substituted derivatives of spiroindanylcamphorsulfonyl oxytocin antagonists |
| AU657431B2 (en) * | 1992-08-20 | 1995-03-09 | Otsuka Pharmaceutical Co., Ltd. | Benzoheterocyclic compounds as oxytocin and vasopressin antagonists |
| WO1994012476A1 (fr) * | 1992-11-25 | 1994-06-09 | Yamanouchi Pharmaceutical Co., Ltd. | Derive de benzanilide |
| AU5692094A (en) * | 1992-12-21 | 1994-07-19 | Yamanouchi Pharmaceutical Co., Ltd. | Novel n-(pyridylcarbonyl)benzazepine derivative and intermediate therefor |
| WO1994020473A1 (fr) * | 1993-03-11 | 1994-09-15 | Yamanouchi Pharmaceutical Co., Ltd. | Compose avec action antagoniste de la vasopressine |
| GB9307527D0 (en) * | 1993-04-13 | 1993-06-02 | Fujisawa Pharmaceutical Co | New venzamide derivatives,processes for the preparation thereof and pharmaceutical composition comprising the same |
| US5516774A (en) * | 1993-07-29 | 1996-05-14 | American Cyanamid Company | Tricyclic diazepine vasopressin antagonists and oxytocin antagonists |
-
1995
- 1995-01-17 US US08/373,132 patent/US5536718A/en not_active Expired - Lifetime
- 1995-06-02 US US08/460,346 patent/US5612334A/en not_active Expired - Lifetime
- 1995-06-02 US US08/458,210 patent/US5610156A/en not_active Expired - Lifetime
-
1996
- 1996-01-15 ZA ZA96297A patent/ZA96297B/xx unknown
- 1996-01-15 AR ARP960101025A patent/AR002022A1/es active IP Right Grant
- 1996-01-16 EA EA199700117A patent/EA001143B1/ru not_active IP Right Cessation
- 1996-01-16 UA UA97084258A patent/UA54383C2/uk unknown
- 1996-01-16 CN CN96192641A patent/CN1065244C/zh not_active Expired - Fee Related
- 1996-01-16 AU AU47698/96A patent/AU707982B2/en not_active Ceased
- 1996-01-16 CZ CZ0224997A patent/CZ297797B6/cs not_active IP Right Cessation
- 1996-01-16 DE DE69635922T patent/DE69635922T2/de not_active Expired - Lifetime
- 1996-01-16 KR KR1019970704833A patent/KR100443438B1/ko not_active Expired - Fee Related
- 1996-01-16 PT PT96903698T patent/PT804438E/pt unknown
- 1996-01-16 DK DK96903698T patent/DK0804438T3/da active
- 1996-01-16 HU HU9800646A patent/HUP9800646A3/hu unknown
- 1996-01-16 WO PCT/US1996/001076 patent/WO1996022293A1/en not_active Ceased
- 1996-01-16 TW TW085100461A patent/TW403752B/zh not_active IP Right Cessation
- 1996-01-16 ES ES96903698T patent/ES2258267T3/es not_active Expired - Lifetime
- 1996-01-16 BR BR9607182A patent/BR9607182A/pt not_active IP Right Cessation
- 1996-01-16 JP JP52245296A patent/JP4163252B2/ja not_active Expired - Fee Related
- 1996-01-16 AT AT96903698T patent/ATE320429T1/de not_active IP Right Cessation
- 1996-01-16 EP EP96903698A patent/EP0804438B1/en not_active Expired - Lifetime
- 1996-01-16 NZ NZ302111A patent/NZ302111A/en unknown
- 1996-01-16 IL IL11677596A patent/IL116775A/xx not_active IP Right Cessation
-
1997
- 1997-07-14 MX MX9705313A patent/MX9705313A/es unknown
-
2007
- 2007-11-21 JP JP2007301830A patent/JP2008101012A/ja active Pending
Also Published As
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| BR9607182A (pt) | Antagonistas de vasopressina de benzazepina tricíclicos | |
| BR9606977A (pt) | Antagonistas de vasopressina de benzazepina triciclica | |
| BR9607186A (pt) | Antagonistas de vasopressina de benzazepina triciclica | |
| BR9710087A (pt) | Antagonistas de vasopressina de benzazepina tricíclicos | |
| DE69621225D1 (de) | Tricyclische vasopressin antagonisten | |
| ZA96300B (en) | Tricyclic benzazepine vasopressin antagonists | |
| FI943542L (fi) | Trisyklisiä bentsatsepiineja, jotka ovat vasopressiiniantagonisteja | |
| DE69826487D1 (de) | Trizyclische vasopressin agoniste | |
| ATE264845T1 (de) | Benzazepine mit vasopressin-antagonistischer wirkung | |
| ZA96298B (en) | Tricyclic benzazepine vasopressin antagonists | |
| DE69203955D1 (de) | Benzazepinderivate als Vasopressin-Antagonisten. | |
| ATE249465T1 (de) | Tricyclische benzodiazepine als vasopressin antagonisten | |
| FI960836A7 (fi) | Bentsodiatsepiiniyhdisteet, jotka ovat käyttökelpoisia CCK- tai gastriiniantagonisteina | |
| AU3641497A (en) | Tricyclic benzazepine vasopressin antagonists | |
| AU3296597A (en) | Tricyclic benzazepine vasopressin antagonists | |
| AU3296497A (en) | Tricyclic benzazepine vasopressin antagonists | |
| SI0804438T1 (sl) | Triciklicni benzazepinski antagonisti vazopresina | |
| HK1003892A (en) | Tricyclic benzazepine vasopressin antagonists | |
| HK1002959A (en) | Tricyclic benzazepine vasopressin antagonists | |
| HK1019448A (en) | Tricyclic benzazepine vasopressin antagonists | |
| HK1003264A (en) | Bicyclic benzazepine derivatives as vasopressin antagonists | |
| ZA961293B (en) | Muscarinic antagonists |
Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| B06A | Patent application procedure suspended [chapter 6.1 patent gazette] | ||
| B25D | Requested change of name of applicant approved |
Owner name: WYETH HOLDINGS CORPORATION (US) Free format text: ALTERADO DE: AMERICAN CYANAMID COMPANY |
|
| B09B | Patent application refused [chapter 9.2 patent gazette] |
Free format text: INDEFERIMENTO DO PRESENTE PEDIDO, UMA VEZ QUE O RELATORIO DESCRITIVO NAO DESCREVE CLARA E SUFICIENTE O OBJETO, DE MODO A POSSIBILITAR SUA REALIZACAO POR TECNICI NO ASSUNTO ( ART. 24 DA LPI ) |
|
| B12B | Appeal against refusal [chapter 12.2 patent gazette] | ||
| B07E | Notification of approval relating to section 229 industrial property law [chapter 7.5 patent gazette] | ||
| B08L | Patent application lapsed because of non payment of annual fee [chapter 8.12 patent gazette] |
Free format text: ARQUIVAMENTO DEFINITIVO |
|
| B08I | Publication cancelled [chapter 8.9 patent gazette] |
Free format text: ANULADA A PUBLICACAO CODIGO 8.12 NA RPI NO 2256 DE 01/04/2014 POR TER SIDO INDEVIDA. |
|
| B08F | Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette] |
Free format text: REFERENTE A 15A,16A,17A,18A,19A,20A,21A,22A,23A,24A E 25A ANUIDADES |
|
| B08K | Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette] |
Free format text: REFERENTE AO DESPACHO 8.6 PUBLICADO NA RPI 2611 DE 19/01/2021. |