BRPI0410888A - uso de derivados de difenilmetano como inibidores de tirosinase - Google Patents

uso de derivados de difenilmetano como inibidores de tirosinase

Info

Publication number
BRPI0410888A
BRPI0410888A BRPI0410888-4A BRPI0410888A BRPI0410888A BR PI0410888 A BRPI0410888 A BR PI0410888A BR PI0410888 A BRPI0410888 A BR PI0410888A BR PI0410888 A BRPI0410888 A BR PI0410888A
Authority
BR
Brazil
Prior art keywords
tyrosinase inhibitors
compounds
diphenylmethane derivatives
formula
browning
Prior art date
Application number
BRPI0410888-4A
Other languages
English (en)
Inventor
Gerhard Schmaus
Martina Herrmann
Holger Joppe
Gabriele Vielhaber
Original Assignee
Symrise Gmbh & Co Kg
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=33441495&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=BRPI0410888(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Symrise Gmbh & Co Kg filed Critical Symrise Gmbh & Co Kg
Publication of BRPI0410888A publication Critical patent/BRPI0410888A/pt

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K8/00—Cosmetics or similar toiletry preparations
    • A61K8/18—Cosmetics or similar toiletry preparations characterised by the composition
    • A61K8/30—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds
    • A61K8/33—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing oxygen
    • A61K8/34—Alcohols
    • A61K8/347—Phenols
    • A—HUMAN NECESSITIES
    • A23—FOODS OR FOODSTUFFS; TREATMENT THEREOF, NOT COVERED BY OTHER CLASSES
    • A23L—FOODS, FOODSTUFFS OR NON-ALCOHOLIC BEVERAGES, NOT OTHERWISE PROVIDED FOR; PREPARATION OR TREATMENT THEREOF
    • A23L5/00—Preparation or treatment of foods or foodstuffs, in general; Food or foodstuffs obtained thereby; Materials therefor
    • A23L5/40—Colouring or decolouring of foods
    • A23L5/41—Retaining or modifying natural colour by use of additives, e.g. optical brighteners
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K8/00—Cosmetics or similar toiletry preparations
    • A61K8/18—Cosmetics or similar toiletry preparations characterised by the composition
    • A61K8/30—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds
    • A61K8/33—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing oxygen
    • A61K8/34—Alcohols
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61Q—SPECIFIC USE OF COSMETICS OR SIMILAR TOILETRY PREPARATIONS
    • A61Q19/00—Preparations for care of the skin
    • A61Q19/02—Preparations for care of the skin for chemically bleaching or whitening the skin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61Q—SPECIFIC USE OF COSMETICS OR SIMILAR TOILETRY PREPARATIONS
    • A61Q19/00—Preparations for care of the skin
    • A61Q19/08—Anti-ageing preparations
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61Q—SPECIFIC USE OF COSMETICS OR SIMILAR TOILETRY PREPARATIONS
    • A61Q5/00—Preparations for care of the hair
    • A61Q5/08—Preparations for bleaching the hair
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K2800/00—Properties of cosmetic compositions or active ingredients thereof or formulation aids used therein and process related aspects
    • A61K2800/74—Biological properties of particular ingredients
    • A61K2800/78—Enzyme modulators, e.g. Enzyme agonists
    • A61K2800/782—Enzyme inhibitors; Enzyme antagonists

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical & Material Sciences (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Dermatology (AREA)
  • Birds (AREA)
  • Emergency Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Food Science & Technology (AREA)
  • Polymers & Plastics (AREA)
  • Nutrition Science (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Gerontology & Geriatric Medicine (AREA)
  • Cosmetics (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Food Preservation Except Freezing, Refrigeration, And Drying (AREA)

Abstract

"USO DE DERIVADOS DE DIFENILMETANO COMO INIBIDORES DE TIROSINASE". A presente invenção refere-se ao uso de compostos da fórmula 1 ou misturas de substâncias que contêm um ou mais compostos da fórmula 1. Os referidos compostos são adequados como agentes contra a formação de cor marrom na pele e cabelos, para o combate de manchas pela idade e para a inibição da formação de cor marrom indesejada de alimentos.
BRPI0410888-4A 2003-05-30 2004-05-24 uso de derivados de difenilmetano como inibidores de tirosinase BRPI0410888A (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE10324566A DE10324566A1 (de) 2003-05-30 2003-05-30 Verwendung von Diphenylmethan-Derivaten als Tyrosinase-Inhibitoren
PCT/EP2004/050896 WO2004105736A1 (de) 2003-05-30 2004-05-24 Verwendung von diphenylmethan-derivaten als tyrosinase-inhibitoren

Publications (1)

Publication Number Publication Date
BRPI0410888A true BRPI0410888A (pt) 2006-07-04

Family

ID=33441495

Family Applications (1)

Application Number Title Priority Date Filing Date
BRPI0410888-4A BRPI0410888A (pt) 2003-05-30 2004-05-24 uso de derivados de difenilmetano como inibidores de tirosinase

Country Status (11)

Country Link
US (1) US9655824B2 (pt)
EP (1) EP1633206B1 (pt)
JP (1) JP4733018B2 (pt)
KR (1) KR101118139B1 (pt)
CN (1) CN100441174C (pt)
AT (1) ATE369755T1 (pt)
BR (1) BRPI0410888A (pt)
DE (2) DE10324566A1 (pt)
ES (1) ES2289532T3 (pt)
WO (1) WO2004105736A1 (pt)
ZA (1) ZA200510114B (pt)

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FR2949330B1 (fr) 2009-08-28 2012-08-10 Oreal Composition cosmetique comprenant un derive diphenyl-methane hydroxyle
US8906432B2 (en) 2009-10-02 2014-12-09 Johnson & Johnson Consumer Companies, Inc. Compositions comprising an NFκB-inhibitor and a non-retinoid collagen promoter
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US8084504B2 (en) 2009-10-02 2011-12-27 Johnson & Johnson Consumer Companies, Inc. High-clarity aqueous concentrates of 4-hexylresorcinol
FR2954140A1 (fr) 2009-12-17 2011-06-24 Oreal Compositions cosmetiques ou dermatologiques a base de bacteriocines et de prebiotiques
FR2956582B1 (fr) 2010-02-19 2012-08-24 Oreal Composition sous forme de poudre comprenant au moins une charge, au moins une huile essentielle et au moins un ester hydroxyle de polyol et d'acide(s) carboxylique(s) en c4 a c16
EP2389922A1 (en) 2010-05-25 2011-11-30 Symrise AG Cyclohexyl carbamate compounds as anti-ageing actives
FR2968569B1 (fr) 2010-12-13 2013-01-04 Oreal Procede de traitement de la peau grasse non acneique.
WO2012105060A1 (en) 2011-02-04 2012-08-09 L'oreal Composite pigment and method for preparation thereof
FR2971249B1 (fr) 2011-02-07 2013-10-18 Fabre Pierre Dermo Cosmetique Derives heterocycliques du resorcinol, leur preparation et leurs utilisations cosmetiques
AU2012231008B2 (en) 2011-03-24 2017-05-11 Unigen, Inc. Compounds and methods for preparation of diarylpropanes
WO2013010590A1 (en) 2011-07-21 2013-01-24 L'oreal Cosmetic and/or dermatological composition containing a merocyanine derivative comprising specific polar groups consisting of hydroxyl- and ether-functionalities
MX2014008225A (es) * 2012-01-05 2014-10-06 Merz North America Inc Composiciones para aclarar la piel.
ITBS20120092A1 (it) * 2012-06-04 2013-12-05 Paoli Ambrosi Gianfranco De Miscela per l'inibizione della biosintesi della melanina
JP6096898B2 (ja) 2012-07-13 2017-03-15 ロレアル 化粧料組成物
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US20140086859A1 (en) 2012-09-24 2014-03-27 Johnson & Johnson Consumer Companies, Inc. Low oil compositions comprising a 4-substituted resorcinol and a high carbon chain ester
EP2789369B1 (en) 2013-04-14 2018-06-06 Symrise AG A composition for lightening skin and hair
EP2853254B1 (en) 2013-09-26 2017-11-08 Symrise AG A composition for lightening skin and/or hair
CN103536454A (zh) * 2013-10-30 2014-01-29 东南大学 苯乙基间苯二酚羟丙基-β-环糊精包合物及其制备方法
FR3012328B1 (fr) * 2013-10-30 2016-12-30 Oreal Methode de peeling cosmetique
JP6510177B2 (ja) 2014-04-01 2019-05-08 ロレアル ナノ又はマイクロエマルションの形態の組成物
JP6537788B2 (ja) * 2014-06-25 2019-07-03 ロレアル ナノエマルション若しくはマイクロエマルションの形態の又はラメラ構造を有する組成物
WO2016090551A1 (en) * 2014-12-09 2016-06-16 L'oreal Composition comprising visible beads
KR102348045B1 (ko) * 2015-02-27 2022-01-11 (주)아모레퍼시픽 미백성분의 부작용을 예측하는 방법
ES2933563T3 (es) 2015-04-16 2023-02-10 Symrise Ag Uso de una composición de liposoma
CN108697600B (zh) * 2015-10-30 2021-08-13 欧莱雅 含羟基化二苯基甲烷衍生物的无水组合物
EP3373895B1 (en) * 2015-11-15 2020-08-19 Symrise AG Reduction of stinging sensation on skin
WO2017096583A1 (en) 2015-12-10 2017-06-15 L'oreal Composition comprising hydroxylated diphenylmethane derivatives
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Also Published As

Publication number Publication date
WO2004105736A8 (de) 2006-10-05
KR101118139B1 (ko) 2012-06-20
EP1633206A1 (de) 2006-03-15
JP2006526005A (ja) 2006-11-16
DE502004004659D1 (de) 2007-09-27
JP4733018B2 (ja) 2011-07-27
KR20060014402A (ko) 2006-02-15
ES2289532T3 (es) 2008-02-01
CN1798550A (zh) 2006-07-05
EP1633206B1 (de) 2007-08-15
US20070098655A1 (en) 2007-05-03
ZA200510114B (en) 2006-12-27
WO2004105736A1 (de) 2004-12-09
DE10324566A1 (de) 2004-12-16
HK1086169A1 (en) 2006-09-15
CN100441174C (zh) 2008-12-10
US9655824B2 (en) 2017-05-23
ATE369755T1 (de) 2007-09-15

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Legal Events

Date Code Title Description
B25A Requested transfer of rights approved

Owner name: SYMRISE AG (DE)

Free format text: TRANSFERIDO POR INCORPORACAO DE: SYMRISE GMBH AND CO. KG

B06F Objections, documents and/or translations needed after an examination request according [chapter 6.6 patent gazette]
B15K Others concerning applications: alteration of classification

Free format text: AS CLASSIFICACOES ANTERIORES ERAM: A61K 8/34 , A23L 1/272

Ipc: A61K 8/34 (2006.01), A61Q 5/08 (2006.01), A61Q 19/

B07A Application suspended after technical examination (opinion) [chapter 7.1 patent gazette]
B09B Patent application refused [chapter 9.2 patent gazette]

Free format text: INDEFIRO O PEDIDO DE ACORDO COM O ART. 8O C/C ART. 13 E ART. 25 DA LPI.

B12B Appeal against refusal [chapter 12.2 patent gazette]
B15K Others concerning applications: alteration of classification

Ipc: A61K 8/34 (2006.01), A23L 5/41 (2016.01), A61Q 5/0