BRPI0607765A2 - pirazolopirimidinas - Google Patents

pirazolopirimidinas

Info

Publication number
BRPI0607765A2
BRPI0607765A2 BRPI0607765-0A BRPI0607765A BRPI0607765A2 BR PI0607765 A2 BRPI0607765 A2 BR PI0607765A2 BR PI0607765 A BRPI0607765 A BR PI0607765A BR PI0607765 A2 BRPI0607765 A2 BR PI0607765A2
Authority
BR
Brazil
Prior art keywords
pyrazolopyrimidines
pirazolopyrimidines
formula
preparation
description
Prior art date
Application number
BRPI0607765-0A
Other languages
English (en)
Inventor
Stefan Herrmann
Olaf Gebauer
Herbert Gayer
Stefan Hillebrand
Ulrich Heinemann
Oliver Guth
Kerstin Ilg
Ronald Ebbert
Ulrike Wachendorff-Neumann
Karl-Heinz Kuck
Thomas Seitz
Peter Dahmen
Horst-Peter Antonicek
Original Assignee
Bayer Cropscience Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Cropscience Ag filed Critical Bayer Cropscience Ag
Publication of BRPI0607765A2 publication Critical patent/BRPI0607765A2/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/90—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system

Landscapes

  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Dentistry (AREA)
  • Pest Control & Pesticides (AREA)
  • Plant Pathology (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Agronomy & Crop Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)

Abstract

PIRAZOLOPIRIMIDINAS. A presente invenção refere-se a pirazolopirimidinas da fórmula (I) na qual R^ 1^, R^ 2^, R^ 3^, R^ 4^, R^ 5^ e X têm os significados indicados na descrição, processo para sua preparação e seu emprego para o controle de microor- ganismos indesejados.
BRPI0607765-0A 2005-02-17 2006-02-07 pirazolopirimidinas BRPI0607765A2 (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE102005007534A DE102005007534A1 (de) 2005-02-17 2005-02-17 Pyrazolopyrimidine
PCT/EP2006/001064 WO2006087120A2 (de) 2005-02-17 2006-02-07 Pyrazolopyrimidine

Publications (1)

Publication Number Publication Date
BRPI0607765A2 true BRPI0607765A2 (pt) 2009-10-06

Family

ID=36793966

Family Applications (1)

Application Number Title Priority Date Filing Date
BRPI0607765-0A BRPI0607765A2 (pt) 2005-02-17 2006-02-07 pirazolopirimidinas

Country Status (16)

Country Link
US (1) US7781439B2 (pt)
EP (1) EP1853607A2 (pt)
JP (1) JP2008530155A (pt)
KR (1) KR20070103473A (pt)
CN (1) CN101120000B (pt)
AR (1) AR052913A1 (pt)
AU (1) AU2006215858A1 (pt)
BR (1) BRPI0607765A2 (pt)
CA (1) CA2597833A1 (pt)
DE (1) DE102005007534A1 (pt)
EA (1) EA200701707A1 (pt)
IL (1) IL185092A0 (pt)
MX (1) MX2007010045A (pt)
TW (1) TW200640926A (pt)
WO (1) WO2006087120A2 (pt)
ZA (1) ZA200706734B (pt)

Families Citing this family (23)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE102006039255A1 (de) * 2006-08-17 2008-02-21 Bayer Cropscience Ag Insektizide heterocyclische Carbonsäurederivate
EP2014661A1 (de) * 2007-06-13 2009-01-14 Bayer CropScience AG Heterocyclisch substituierte Heterocyclyl-carbonsäurederivate
GB0712653D0 (en) 2007-06-28 2007-08-08 Syngenta Ltd Novel herbicides
GB0717082D0 (en) 2007-09-03 2007-10-10 Syngenta Ltd Novel herbicides
WO2010045615A2 (en) 2008-10-16 2010-04-22 Cenomed Biosciences, Llc Treatment of organophosphate exposure with ocinaplon
EP2649075B1 (en) * 2010-12-08 2018-04-25 The U.S.A. As Represented By The Secretary, Department Of Health And Human Services Substituted pyrazolopyrimidines as glucocerebrosidase activators
US9309250B2 (en) 2011-06-22 2016-04-12 Vertex Pharmaceuticals Incorporated Substituted pyrrolo[2,3-b]pyrazines as ATR kinase inhibitors
WO2014089379A1 (en) 2012-12-07 2014-06-12 Vertex Pharmaceuticals Incorporated Compounds useful as inhibitors of atr kinase
US9663519B2 (en) 2013-03-15 2017-05-30 Vertex Pharmaceuticals Incorporated Compounds useful as inhibitors of ATR kinase
EP2970288A1 (en) 2013-03-15 2016-01-20 Vertex Pharmaceuticals Incorporated Compounds useful as inhibitors of atr kinase
EP2970289A1 (en) 2013-03-15 2016-01-20 Vertex Pharmaceuticals Inc. Compounds useful as inhibitors of atr kinase
WO2015085132A1 (en) 2013-12-06 2015-06-11 Vertex Pharmaceuticals Incorporated 2-amino-6-fluoro-n-[5-fluoro-pyridin-3-yl]pyrazolo[1,5-a]pyrimidin-3-carboxamide compound useful as atr kinase inhibitor, its preparation, different solid forms and radiolabelled derivatives thereof
HRP20200186T1 (hr) 2014-06-05 2020-05-29 Vertex Pharmaceuticals Inc. Radioaktivno obilježeni derivati 2-amino-6-fluoro-n-[5-fluoro-piridin-3-il]-pirazolo[1,5-a]pirimidin-3-karboksamid spojeva koji se koriste kao inhibitori atr kinaze, priprava navedenih spojeva i njihovi različiti čvrsti oblici
JP6936007B2 (ja) 2014-06-17 2021-09-15 バーテックス ファーマシューティカルズ インコーポレイテッドＶｅｒｔｅｘ Ｐｈａｒｍａｃｅｕｔｉｃａｌｓ Ｉｎｃｏｒｐｏｒａｔｅｄ Ｃｈｋ１阻害剤とａｔｒ阻害剤との組み合わせを使用してがんを処置する方法
HRP20240644T1 (hr) 2014-11-06 2024-08-02 Bial-R&D Investments, S.A. Supstituirani pirazolo(1,5-a)pirimidini i njihova uporaba u liječenju medicinskih poremećaja
EP3355926B1 (en) 2015-09-30 2025-12-24 Vertex Pharmaceuticals Inc. Combination of dna damaging agents and atr inhibitors for use in a method for treating cancer using
SG11201808830YA (en) * 2016-04-06 2018-11-29 Lysosomal Therapeutics Inc Pyrazolo[1,5-a]pyrimidinyl carboxamide compounds and their use in the treatment of medical disorders
JP7046827B2 (ja) 2016-04-06 2022-04-04 リソソーマル・セラピューティクス・インコーポレイテッド イミダゾ［１，５－ａ］ピリミジニルカルボキサミド化合物および医学的障害の処置におけるその使用
US11124516B2 (en) 2016-04-06 2021-09-21 BIAL-BioTech Investments, Inc. Pyrrolo[1,2-A]pyrimidinyl carboxamide compounds and their use in the treatment of medical disorders
JP7164774B2 (ja) 2016-05-05 2022-11-02 ビアル－アール・アンド・ディ・インベストメンツ・ソシエダーデ・アノニマ 置換イミダゾ［１，２－ｂ］ピリダジン、置換イミダゾ［１，５－ｂ］ピリダジン、関連化合物、および医学的障害の治療におけるその使用
JP7216705B2 (ja) * 2017-07-28 2023-02-02 ニンバス ラクシュミ， インコーポレイテッド Ｔｙｋ２阻害剤およびその使用方法
MY210039A (en) 2018-10-30 2025-08-22 Kronos Bio Inc Compounds, compositions, and methods for modulating cdk9 activity
CN113287620B (zh) * 2021-06-18 2021-11-19 浙江大学 1H-吡唑并[3,4-d]嘧啶类化合物在制备禾谷镰刀菌杀菌剂中的应用

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US2444606A (en) * 1945-12-15 1948-07-06 Gen Aniline & Film Corp Stabilizers for photographic emulsions
US3515715A (en) * 1967-01-23 1970-06-02 Eastman Kodak Co Quaternized pyrazolylazo dyes
US3634391A (en) * 1969-07-25 1972-01-11 Eastman Kodak Co Pyrazolyl-azo-indole dyestuffs
US4838925A (en) * 1986-04-25 1989-06-13 E. I. Du Pont De Nemours And Company Heterocyclic acyl sulfonamides
DE3825043A1 (de) 1988-07-20 1990-02-15 Schering Ag 3-methylsulfonyl-pyrazolo(1,5-a)pyrimidin-sulfonsaeureamide, verfahren zu ihrer herstellung und ihre verwendung als mittel mit herbizider, pflanzenwuchsregulierender und fungizider wirkung
US6156925A (en) * 1998-09-25 2000-12-05 American Cyanamid Company Process for the preparation of halogenated phenylmaloates
IL131912A (en) 1998-09-25 2005-12-18 American Cyanamid Co Process for preparing halogenated phenylmalonates
EP1343787B1 (en) 2000-12-11 2004-11-10 Basf Aktiengesellschaft 6-phenyl-pyrazolopyrimidines
NZ531169A (en) 2001-07-26 2005-09-30 Basf Ag 7-amino triazolopyrimidines for controlling harmful fungi
NZ518658A (en) * 2002-04-30 2004-10-29 Lionel Evans Method of water treatment
DE10223917A1 (de) 2002-05-29 2003-12-11 Bayer Cropscience Ag Pyrazolopyrimidine
FR2841982B1 (fr) 2002-07-03 2005-03-25 Inst Francais Du Petrole Capteur de pression a fibre optique compense en temperature
EP1536786A1 (en) 2002-07-17 2005-06-08 Warner-Lambert Company Llc Combination of an allosteric inhibitor of matrix metalloproteinase-13 with celecoxib or valdecoxib
EP1599482A4 (en) * 2003-02-28 2008-10-01 Teijin Pharma Ltd PYRAZOLO1,5-A PYRIMIDINE DERIVATIVES
CA2527136A1 (en) 2003-06-03 2004-12-09 Basf Aktiengesellschaft Substituted pyrazolopyrimidines, methods for the production thereof, use of the same for controlling pathogenic fungi, and agents containing said compounds
CA2530378A1 (en) 2003-06-27 2005-01-06 Bayer Cropscience Ag Pyrazolopyrimidines
DE10357567A1 (de) 2003-12-10 2005-07-07 Bayer Cropscience Ag Pyrazolopyrimidine
DE10357565A1 (de) * 2003-12-10 2005-07-07 Bayer Cropscience Ag Pyrazolopyrimidine
DE10357568A1 (de) 2003-12-10 2005-07-07 Bayer Cropscience Ag Pyrazolopyrimidine
DE10357569A1 (de) * 2003-12-10 2005-07-07 Bayer Cropscience Ag Pyrazolopyrimidine
DE102004008807A1 (de) 2004-02-20 2005-09-08 Bayer Cropscience Ag Pyrazolopyrimidine

Also Published As

Publication number Publication date
JP2008530155A (ja) 2008-08-07
WO2006087120A2 (de) 2006-08-24
TW200640926A (en) 2006-12-01
US7781439B2 (en) 2010-08-24
AR052913A1 (es) 2007-04-11
IL185092A0 (en) 2007-12-03
CN101120000A (zh) 2008-02-06
MX2007010045A (es) 2007-10-02
KR20070103473A (ko) 2007-10-23
EA200701707A1 (ru) 2008-02-28
DE102005007534A1 (de) 2006-08-31
EP1853607A2 (de) 2007-11-14
CN101120000B (zh) 2011-05-18
ZA200706734B (en) 2009-01-28
CA2597833A1 (en) 2006-08-24
WO2006087120A3 (de) 2006-12-14
US20080287463A1 (en) 2008-11-20
WO2006087120A8 (de) 2007-08-30
AU2006215858A1 (en) 2006-08-24

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Legal Events

Date Code Title Description
B08F Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette]

Free format text: REFERENTE A 6A ANUIDADE.

B08K Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette]

Free format text: REFERENTE AO DESPACHO 8.6 PUBLICADO NA RPI 2161 DE 05/06/2012.