BRPI0607765A2 - pirazolopirimidinas - Google Patents

pirazolopirimidinas

Info

Publication number
BRPI0607765A2
BRPI0607765A2 BRPI0607765-0A BRPI0607765A BRPI0607765A2 BR PI0607765 A2 BRPI0607765 A2 BR PI0607765A2 BR PI0607765 A BRPI0607765 A BR PI0607765A BR PI0607765 A2 BRPI0607765 A2 BR PI0607765A2
Authority
BR
Brazil
Prior art keywords
pyrazolopyrimidines
pirazolopyrimidines
formula
preparation
description
Prior art date
Application number
BRPI0607765-0A
Other languages
English (en)
Inventor
Stefan Herrmann
Olaf Gebauer
Herbert Gayer
Stefan Hillebrand
Ulrich Heinemann
Oliver Guth
Kerstin Ilg
Ronald Ebbert
Ulrike Wachendorff-Neumann
Karl-Heinz Kuck
Thomas Seitz
Peter Dahmen
Horst-Peter Antonicek
Original Assignee
Bayer Cropscience Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Cropscience Ag filed Critical Bayer Cropscience Ag
Publication of BRPI0607765A2 publication Critical patent/BRPI0607765A2/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/90—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system

Landscapes

  • Life Sciences & Earth Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Plant Pathology (AREA)
  • Engineering & Computer Science (AREA)
  • Dentistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Pest Control & Pesticides (AREA)
  • Agronomy & Crop Science (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)

Abstract

PIRAZOLOPIRIMIDINAS. A presente invenção refere-se a pirazolopirimidinas da fórmula (I) na qual R^ 1^, R^ 2^, R^ 3^, R^ 4^, R^ 5^ e X têm os significados indicados na descrição, processo para sua preparação e seu emprego para o controle de microor- ganismos indesejados.
BRPI0607765-0A 2005-02-17 2006-02-07 pirazolopirimidinas BRPI0607765A2 (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE102005007534A DE102005007534A1 (de) 2005-02-17 2005-02-17 Pyrazolopyrimidine
PCT/EP2006/001064 WO2006087120A2 (de) 2005-02-17 2006-02-07 Pyrazolopyrimidine

Publications (1)

Publication Number Publication Date
BRPI0607765A2 true BRPI0607765A2 (pt) 2009-10-06

Family

ID=36793966

Family Applications (1)

Application Number Title Priority Date Filing Date
BRPI0607765-0A BRPI0607765A2 (pt) 2005-02-17 2006-02-07 pirazolopirimidinas

Country Status (16)

Country Link
US (1) US7781439B2 (pt)
EP (1) EP1853607A2 (pt)
JP (1) JP2008530155A (pt)
KR (1) KR20070103473A (pt)
CN (1) CN101120000B (pt)
AR (1) AR052913A1 (pt)
AU (1) AU2006215858A1 (pt)
BR (1) BRPI0607765A2 (pt)
CA (1) CA2597833A1 (pt)
DE (1) DE102005007534A1 (pt)
EA (1) EA200701707A1 (pt)
IL (1) IL185092A0 (pt)
MX (1) MX2007010045A (pt)
TW (1) TW200640926A (pt)
WO (1) WO2006087120A2 (pt)
ZA (1) ZA200706734B (pt)

Families Citing this family (23)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE102006039255A1 (de) * 2006-08-17 2008-02-21 Bayer Cropscience Ag Insektizide heterocyclische Carbonsäurederivate
EP2014661A1 (de) * 2007-06-13 2009-01-14 Bayer CropScience AG Heterocyclisch substituierte Heterocyclyl-carbonsäurederivate
GB0712653D0 (en) 2007-06-28 2007-08-08 Syngenta Ltd Novel herbicides
GB0717082D0 (en) 2007-09-03 2007-10-10 Syngenta Ltd Novel herbicides
WO2010045615A2 (en) 2008-10-16 2010-04-22 Cenomed Biosciences, Llc Treatment of organophosphate exposure with ocinaplon
EP3366688B1 (en) * 2010-12-08 2022-02-09 The U.S.A. as represented by the Secretary, Department of Health and Human Services Substituted pyrazolopyrimidines as glucocerebrosidase activators
US9309250B2 (en) 2011-06-22 2016-04-12 Vertex Pharmaceuticals Incorporated Substituted pyrrolo[2,3-b]pyrazines as ATR kinase inhibitors
SI2941432T1 (en) 2012-12-07 2018-07-31 Vertex Pharmaceuticals Incorporated 2-AMINO-6-FLUORO-N- (5-FLUORO-4- (4- (4- (OXETHAN-3-YL) PIPERAZIN-1-CARBONYL) PIPERIDIN-1-YLIPRIDIN-3-YL) 1,5 ALFA) PYRIMIDINE-3-CARBOXAMIDE AS ATR KINAZE INHIBITOR
US8957078B2 (en) 2013-03-15 2015-02-17 Vertex Pharmaceuticals Incorporated Compounds useful as inhibitors of ATR kinase
WO2014143240A1 (en) 2013-03-15 2014-09-18 Vertex Pharmaceuticals Incorporated Fused pyrazolopyrimidine derivatives useful as inhibitors of atr kinase
EP2970288A1 (en) 2013-03-15 2016-01-20 Vertex Pharmaceuticals Incorporated Compounds useful as inhibitors of atr kinase
PT3077397T (pt) 2013-12-06 2020-01-22 Vertex Pharma Composto de 2-amino-6-fluoro-n-[5-fluoro-piridin-3-il]pirazolo[1,5-a]pirimidin-3-carboxamida útil como inibidor da atr quinase, a sua preparação, diferentes formas sólidas e derivados radiomarcados do mesmo
MX373102B (es) 2014-06-05 2020-04-17 Vertex Pharma Derivados radiomarcados de un compuesto de 2-amino-6-fluoro-n-[5-fluoro-piridin-3-il]-pirazolo[1,5-a]pirimidin-3-carboxamida útil como inhibidor de ataxia telangiectasia mutada y rad3 relacionado (atr) cinasa, preparación de tal compuesto y diferentes formas sólidas del mismo.
SG11201610500WA (en) 2014-06-17 2017-01-27 Vertex Pharma Method for treating cancer using a combination of chk1 and atr inhibitors
EP4406616A3 (en) 2014-11-06 2024-11-06 Bial-R&D Investments, S.A. Substituted pyrazolo(1,5-a)pyrimidines and their use in the treatment of medical disorders
AU2016331955B2 (en) 2015-09-30 2022-07-21 Vertex Pharmaceuticals Incorporated Method for treating cancer using a combination of DNA damaging agents and ATR inhibitors
CA3020305A1 (en) 2016-04-06 2017-10-12 Lysosomal Therapeutics Inc. Imidazo [1,5-a]pyrimidinyl carboxamide compounds and their use in the treatment of medical disorders
AU2017246455B2 (en) * 2016-04-06 2021-09-30 Bial - R&D Investments, S.A. Pyrazolo[1,5-a]pyrimidinyl carboxamide compounds and their use in the treatment of medical disorders
EP3440081A4 (en) 2016-04-06 2019-09-18 Lysosomal Therapeutics Inc. PYRROLO [1,2-A] PYRIMIDINYL-CARBOXAMIDE COMPOUNDS AND THEIR USE IN THE TREATMENT OF MEDICAL DISORDER
KR102530515B1 (ko) 2016-05-05 2023-05-09 비알 - 알&디 인베스트먼츠, 에스.에이. 치환된 이미다조[1,2-b]피리다진, 치환된 이미다조[1,5-b]피리다진, 관련 화합물, 및 의학적 장애의 치료에서의 그의 용도
SI3658557T1 (sl) * 2017-07-28 2024-10-30 Takeda Pharmaceutical Company Limited Zaviralci TYK2 in njihova uporaba
US11155560B2 (en) 2018-10-30 2021-10-26 Kronos Bio, Inc. Substituted pyrazolo[1,5-a]pyrimidines for modulating CDK9 activity
CN113287620B (zh) * 2021-06-18 2021-11-19 浙江大学 1H-吡唑并[3,4-d]嘧啶类化合物在制备禾谷镰刀菌杀菌剂中的应用

Family Cites Families (21)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2444606A (en) * 1945-12-15 1948-07-06 Gen Aniline & Film Corp Stabilizers for photographic emulsions
US3515715A (en) * 1967-01-23 1970-06-02 Eastman Kodak Co Quaternized pyrazolylazo dyes
US3634391A (en) * 1969-07-25 1972-01-11 Eastman Kodak Co Pyrazolyl-azo-indole dyestuffs
US4838925A (en) * 1986-04-25 1989-06-13 E. I. Du Pont De Nemours And Company Heterocyclic acyl sulfonamides
DE3825043A1 (de) 1988-07-20 1990-02-15 Schering Ag 3-methylsulfonyl-pyrazolo(1,5-a)pyrimidin-sulfonsaeureamide, verfahren zu ihrer herstellung und ihre verwendung als mittel mit herbizider, pflanzenwuchsregulierender und fungizider wirkung
US6156925A (en) * 1998-09-25 2000-12-05 American Cyanamid Company Process for the preparation of halogenated phenylmaloates
IL131912A (en) 1998-09-25 2005-12-18 American Cyanamid Co Process for preparing halogenated phenylmalonates
WO2002048151A1 (en) 2000-12-11 2002-06-20 Basf Aktiengesellschaft 6-phenyl-pyrazolopyrimidines
DK1414302T3 (da) 2001-07-26 2007-06-18 Basf Ag 7-aminotriazolopyrimidiner til bekæmpelse af skadelige svampe
NZ518658A (en) * 2002-04-30 2004-10-29 Lionel Evans Method of water treatment
DE10223917A1 (de) 2002-05-29 2003-12-11 Bayer Cropscience Ag Pyrazolopyrimidine
FR2841982B1 (fr) 2002-07-03 2005-03-25 Inst Francais Du Petrole Capteur de pression a fibre optique compense en temperature
WO2004006913A1 (en) 2002-07-17 2004-01-22 Warner-Lambert Company Llc Combination of an allosteric inhibitor of matrix metalloproteinase-13 with celecoxib or valdecoxib
US7557110B2 (en) * 2003-02-28 2009-07-07 Teijin Pharma Limited Pyrazolo[1,5-A] pyrimidine derivatives
BRPI0410610A (pt) 2003-06-03 2006-07-04 Basf Ag compostos, processos para a produção dos mesmos e para o combate de fungos nocivos fitopatogênicos, produtos intermediários, e, agente adequado para o combate de fungos nocivos
ATE388138T1 (de) * 2003-06-27 2008-03-15 Bayer Cropscience Ag Pyrazolopyrimidine
DE10357568A1 (de) 2003-12-10 2005-07-07 Bayer Cropscience Ag Pyrazolopyrimidine
DE10357565A1 (de) * 2003-12-10 2005-07-07 Bayer Cropscience Ag Pyrazolopyrimidine
DE10357569A1 (de) 2003-12-10 2005-07-07 Bayer Cropscience Ag Pyrazolopyrimidine
DE10357567A1 (de) * 2003-12-10 2005-07-07 Bayer Cropscience Ag Pyrazolopyrimidine
DE102004008807A1 (de) 2004-02-20 2005-09-08 Bayer Cropscience Ag Pyrazolopyrimidine

Also Published As

Publication number Publication date
IL185092A0 (en) 2007-12-03
WO2006087120A8 (de) 2007-08-30
DE102005007534A1 (de) 2006-08-31
CN101120000B (zh) 2011-05-18
KR20070103473A (ko) 2007-10-23
US20080287463A1 (en) 2008-11-20
JP2008530155A (ja) 2008-08-07
MX2007010045A (es) 2007-10-02
EA200701707A1 (ru) 2008-02-28
WO2006087120A2 (de) 2006-08-24
US7781439B2 (en) 2010-08-24
CN101120000A (zh) 2008-02-06
EP1853607A2 (de) 2007-11-14
CA2597833A1 (en) 2006-08-24
AR052913A1 (es) 2007-04-11
WO2006087120A3 (de) 2006-12-14
TW200640926A (en) 2006-12-01
AU2006215858A1 (en) 2006-08-24
ZA200706734B (en) 2009-01-28

Similar Documents

Publication Publication Date Title
BRPI0607765A2 (pt) pirazolopirimidinas
BRPI0507894A (pt) pirazolopirimidinas
BR0309242A (pt) Derivados de acil-4-carboxifenil-uréia, processo para a sua preparação e sua aplicação
BRPI0407284A (pt) Bactérias e processo para produção de compostos quìmicos pelas bactérias i
BRPI0514361A (pt) processo para a produção de dihidropteridinonas
BRPI0610088A2 (pt) mÉtodo para o controle de doenÇa na soja mon89788
BRPI0411713B8 (pt) compostos, processo para a sua manufatura, composições farmacêuticas que compreendem os mesmos, método para tratamento e/ou profilaxia de enfermidades que estão associadas com dpp-iv e sua utilização
BR0215493A (pt) Processo para preparação de ésteres escopìnicos
BRPI0618451A2 (pt) derivados de piridopirazina, seu uso, composição farmacêutica e estojo
BRPI0410494A (pt) iodopirazolilcarboxanilidas
BRPI0510412A (pt) compostos orgánicos
BR0312379A (pt) Produtos de poliadição contendo grupos uretodiona
BRPI0512335A (pt) compostos, processo para a sua manufatura, composições farmacêuticas que os compreendem, método para o tratamento e/ou prevenção de enfermidades e sua utilização
BRPI0519316B8 (pt) composição aquosa herbicida, e, processo para a preparação de uma composição
BRPI0410238A (pt) compostos orgánicos
BRPI0719367B8 (pt) processo para a preparação de nebivolol, seus intermediários e usos
BRPI0712889A8 (pt) composto, processo para a preparação de um composto, composto intermediário, e, composição farmacêutica.
BRPI0406596A (pt) Métodos para tratar a dor articular e melhorar o sono utilizando um agonista/antagonista de estrogênio
BRPI0514439A (pt) bifeniltiazolcarboxamidas
BR0309568A (pt) Triazolopirimidinas
BRPI0415454A (pt) 1,3-dimetilbutilcarboxanilidas para controle de microorganismos indesejáveis
BR0112927A (pt) Pirazolilbifenilcarboxamidas e sua aplicação para combater microorganismos indesejados
BRPI0416571A (pt) nicotinoilcarbamatos substituìdos como pesticidas
BRPI0410906A (pt) triazolopirimidinas
BRPI0514678A (pt) bifeniltiazolcarboxamida

Legal Events

Date Code Title Description
B08F Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette]

Free format text: REFERENTE A 6A ANUIDADE.

B08K Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette]

Free format text: REFERENTE AO DESPACHO 8.6 PUBLICADO NA RPI 2161 DE 05/06/2012.