BRPI0512168A - processo para preparar tiazol por aminometilação - Google Patents
processo para preparar tiazol por aminometilaçãoInfo
- Publication number
- BRPI0512168A BRPI0512168A BRPI0512168-0A BRPI0512168A BRPI0512168A BR PI0512168 A BRPI0512168 A BR PI0512168A BR PI0512168 A BRPI0512168 A BR PI0512168A BR PI0512168 A BRPI0512168 A BR PI0512168A
- Authority
- BR
- Brazil
- Prior art keywords
- formula
- compound
- aminomethylation
- preparing
- thiazole
- Prior art date
Links
- 238000004519 manufacturing process Methods 0.000 title abstract 3
- FZWLAAWBMGSTSO-UHFFFAOYSA-N Thiazole Chemical compound C1=CSC=N1 FZWLAAWBMGSTSO-UHFFFAOYSA-N 0.000 title abstract 2
- 238000005902 aminomethylation reaction Methods 0.000 title 1
- WSFSSNUMVMOOMR-UHFFFAOYSA-N Formaldehyde Chemical compound O=C WSFSSNUMVMOOMR-UHFFFAOYSA-N 0.000 abstract 3
- QGZKDVFQNNGYKY-UHFFFAOYSA-N Ammonia Chemical compound N QGZKDVFQNNGYKY-UHFFFAOYSA-N 0.000 abstract 2
- 150000001875 compounds Chemical class 0.000 abstract 2
- 125000005843 halogen group Chemical group 0.000 abstract 2
- -1 thiazole compound Chemical class 0.000 abstract 2
- 229910021529 ammonia Inorganic materials 0.000 abstract 1
- 125000004435 hydrogen atom Chemical group [H]* 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
- C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D277/22—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
- C07D277/28—Radicals substituted by nitrogen atoms
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Thiazole And Isothizaole Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Abstract
PROCESSO PARA PREPARAR TIAZOL POR AMINOMETILAçãO. A presente invenção refere-se a um processo para preparar um composto de tiazol da fórmula (3): em que X¬ 1¬ representa um átomo de hidrogênio ou um átomo de halogênio compreendendo reagir um composto da fórmula (1):em que X¬ 1¬ é como definido acima, e X¬ 2¬ representa um átomo de halogênio, com amónia e formaldeído para obter um composto de hexaidrotriazina da fórmula (2):em que X¬ 1¬ é como definido acima, e hidrolizar o composto da fórmula (2).
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2004179472 | 2004-06-17 | ||
| JP2005110701 | 2005-04-07 | ||
| PCT/JP2005/011095 WO2005123704A1 (en) | 2004-06-17 | 2005-06-10 | Compound for preparing thiazole by aminomethylation |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| BRPI0512168A true BRPI0512168A (pt) | 2008-02-12 |
| BRPI0512168B1 BRPI0512168B1 (pt) | 2013-12-31 |
Family
ID=34970323
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BRPI0512168-0B1A BRPI0512168B1 (pt) | 2004-06-17 | 2005-06-10 | Processo para preparar tiazol por aminometilação |
Country Status (14)
| Country | Link |
|---|---|
| US (1) | US7439357B2 (pt) |
| EP (1) | EP1756075B1 (pt) |
| JP (1) | JP4788201B2 (pt) |
| KR (1) | KR101214414B1 (pt) |
| CN (1) | CN1968938B (pt) |
| AR (1) | AR049695A1 (pt) |
| AU (1) | AU2005254863B2 (pt) |
| BR (1) | BRPI0512168B1 (pt) |
| DK (1) | DK1756075T3 (pt) |
| ES (1) | ES2425477T3 (pt) |
| IL (1) | IL179701A (pt) |
| RU (1) | RU2372340C2 (pt) |
| TW (1) | TWI344958B (pt) |
| WO (1) | WO2005123704A1 (pt) |
Families Citing this family (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP4839660B2 (ja) * | 2005-04-07 | 2011-12-21 | 住友化学株式会社 | チアゾール化合物の製造法 |
| WO2007069685A1 (ja) * | 2005-12-15 | 2007-06-21 | Sumitomo Chemical Company, Limited | 選択的一級アミン化合物の製造方法 |
| JP5130706B2 (ja) * | 2005-12-15 | 2013-01-30 | 住友化学株式会社 | 選択的一級アミン化合物の製造方法 |
| JP4848762B2 (ja) * | 2005-12-26 | 2011-12-28 | 住友化学株式会社 | 一級アミン化合物の製造方法 |
| KR101682339B1 (ko) * | 2007-04-24 | 2016-12-02 | 닛뽕소다 가부시키가이샤 | 치환 메틸아민 화합물의 제조방법 및 트리아진 유도체 |
| CN104755476B (zh) * | 2012-11-02 | 2017-12-05 | 住友化学株式会社 | 化合物的制造方法 |
| EP3484857B1 (de) * | 2016-07-18 | 2021-03-03 | Sika Technology AG | Katalysator für härtbare zusammensetzungen enthaltend hexahydrotriazin-struktureinheiten |
Family Cites Families (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| SU407905A1 (ru) * | 1972-01-07 | 1973-12-10 | Ордена Трудового Красного Знамени институт органического синтеза Латвийской ССР | Способ получения 4-аминометилтиазол-2-олов |
| SU798102A1 (ru) | 1977-08-25 | 1981-01-23 | Предприятие П/Я В-2287 | Способ совместного получени , , -ТРибЕНзилгЕКСАгидРО-ТРиАзиНА-1,3,5 и -МЕТилбЕНзил-АМиНО- -бЕНзилиМиНОМЕТилЕНА |
| IL100688A (en) | 1987-08-01 | 1995-08-31 | Takeda Chemical Industries Ltd | Intermediates for the production of unsaturated amines in position A and the process for their preparation |
| US5180833A (en) * | 1990-03-16 | 1993-01-19 | Takeda Chemical Industries, Ltd. | Process for the preparation of chlorothiazole derivatives |
| JPH0421674A (ja) | 1990-05-15 | 1992-01-24 | Nippon Soda Co Ltd | 2―クロロ―5―(アミノメチル)チアゾールの製造方法 |
| JPH05286936A (ja) | 1992-04-06 | 1993-11-02 | Takeda Chem Ind Ltd | ホルムアミド誘導体の製造法及び新規ホルムアミド誘導体 |
| TW541294B (en) | 1998-10-12 | 2003-07-11 | Ihara Chemical Ind Co | Process for producing aminomethyl-heterocyclic derivative |
| JP4276720B2 (ja) | 1998-11-05 | 2009-06-10 | 住友化学株式会社 | 5−アミノメチル−2−クロロチアゾールまたはその塩の製造方法 |
| DE10061083A1 (de) | 2000-12-08 | 2002-06-13 | Bayer Ag | Bis-(2-chlor-thiazolyl-5-methyl)-amin und seine Salze sowie Verfahren zur Aufarbeitung von 5-Aminomethyl-2-chlor-thiazol und Bis-(2-chlor-thiazol-5-methyl)-amin enthaltenden Reaktionsgemischen |
| JP4839660B2 (ja) * | 2005-04-07 | 2011-12-21 | 住友化学株式会社 | チアゾール化合物の製造法 |
-
2005
- 2005-05-30 TW TW094117685A patent/TWI344958B/zh not_active IP Right Cessation
- 2005-06-02 JP JP2005162231A patent/JP4788201B2/ja not_active Expired - Fee Related
- 2005-06-10 AU AU2005254863A patent/AU2005254863B2/en not_active Ceased
- 2005-06-10 RU RU2007101508/04A patent/RU2372340C2/ru not_active IP Right Cessation
- 2005-06-10 US US11/629,754 patent/US7439357B2/en not_active Expired - Lifetime
- 2005-06-10 CN CN200580019523XA patent/CN1968938B/zh not_active Expired - Lifetime
- 2005-06-10 BR BRPI0512168-0B1A patent/BRPI0512168B1/pt not_active IP Right Cessation
- 2005-06-10 EP EP05751282.4A patent/EP1756075B1/en not_active Expired - Lifetime
- 2005-06-10 WO PCT/JP2005/011095 patent/WO2005123704A1/en not_active Ceased
- 2005-06-10 DK DK05751282.4T patent/DK1756075T3/da active
- 2005-06-10 ES ES05751282T patent/ES2425477T3/es not_active Expired - Lifetime
- 2005-06-13 AR ARP050102393A patent/AR049695A1/es unknown
-
2006
- 2006-11-29 IL IL179701A patent/IL179701A/en not_active IP Right Cessation
- 2006-12-15 KR KR1020067026415A patent/KR101214414B1/ko not_active Expired - Fee Related
Also Published As
| Publication number | Publication date |
|---|---|
| US20070197803A1 (en) | 2007-08-23 |
| WO2005123704A1 (en) | 2005-12-29 |
| JP2006312617A (ja) | 2006-11-16 |
| ES2425477T3 (es) | 2013-10-15 |
| IL179701A (en) | 2012-03-29 |
| TWI344958B (en) | 2011-07-11 |
| EP1756075A1 (en) | 2007-02-28 |
| US7439357B2 (en) | 2008-10-21 |
| IL179701A0 (en) | 2007-05-15 |
| BRPI0512168B1 (pt) | 2013-12-31 |
| AR049695A1 (es) | 2006-08-30 |
| RU2007101508A (ru) | 2008-07-27 |
| RU2372340C2 (ru) | 2009-11-10 |
| CN1968938A (zh) | 2007-05-23 |
| KR20070026597A (ko) | 2007-03-08 |
| JP4788201B2 (ja) | 2011-10-05 |
| KR101214414B1 (ko) | 2012-12-21 |
| CN1968938B (zh) | 2010-05-05 |
| AU2005254863B2 (en) | 2010-12-23 |
| AU2005254863A1 (en) | 2005-12-29 |
| DK1756075T3 (da) | 2013-08-26 |
| TW200602331A (en) | 2006-01-16 |
| EP1756075B1 (en) | 2013-08-07 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| B06F | Objections, documents and/or translations needed after an examination request according [chapter 6.6 patent gazette] | ||
| B09A | Decision: intention to grant [chapter 9.1 patent gazette] | ||
| B16A | Patent or certificate of addition of invention granted [chapter 16.1 patent gazette] |
Free format text: PRAZO DE VALIDADE: 20 (VINTE) ANOS CONTADOS A PARTIR DE 10/06/2005, OBSERVADAS AS CONDICOES LEGAIS. |
|
| B21F | Lapse acc. art. 78, item iv - on non-payment of the annual fees in time |
Free format text: REFERENTE A 11A ANUIDADE. |
|
| B24J | Lapse because of non-payment of annual fees (definitively: art 78 iv lpi, resolution 113/2013 art. 12) |
Free format text: EM VIRTUDE DA EXTINCAO PUBLICADA NA RPI 2385 DE 20-09-2016 E CONSIDERANDO AUSENCIA DE MANIFESTACAO DENTRO DOS PRAZOS LEGAIS, INFORMO QUE CABE SER MANTIDA A EXTINCAO DA PATENTE E SEUS CERTIFICADOS, CONFORME O DISPOSTO NO ARTIGO 12, DA RESOLUCAO 113/2013. |