BRPI0608011A2 - uso de uma formulação para o tratamento da queratose actìnica e uso de 2-metil-1-(2-metilpropil)-1h-imidazo[4,5-c][1,5] naftiridin-4-amina - Google Patents

uso de uma formulação para o tratamento da queratose actìnica e uso de 2-metil-1-(2-metilpropil)-1h-imidazo[4,5-c][1,5] naftiridin-4-amina

Info

Publication number
BRPI0608011A2
BRPI0608011A2 BRPI0608011-1A BRPI0608011A BRPI0608011A2 BR PI0608011 A2 BRPI0608011 A2 BR PI0608011A2 BR PI0608011 A BRPI0608011 A BR PI0608011A BR PI0608011 A2 BRPI0608011 A2 BR PI0608011A2
Authority
BR
Brazil
Prior art keywords
imidazo
methyl
formulation
naphthyridin
methylpropyl
Prior art date
Application number
BRPI0608011-1A
Other languages
English (en)
Inventor
James H Lee
Terrance L Fox
Original Assignee
Graceway Pharmaceuticals Llc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Graceway Pharmaceuticals Llc filed Critical Graceway Pharmaceuticals Llc
Publication of BRPI0608011A2 publication Critical patent/BRPI0608011A2/pt

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47—Quinolines; Isoquinolines
    • A61K31/4738—Quinolines; Isoquinolines ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/4745—Quinolines; Isoquinolines ortho- or peri-condensed with heterocyclic ring systems condensed with ring systems having nitrogen as a ring hetero atom, e.g. phenantrolines
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/0014—Skin, i.e. galenical aspects of topical compositions
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/06—Ointments; Bases therefor; Other semi-solid forms, e.g. creams, sticks, gels

Landscapes

  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Epidemiology (AREA)
  • Dermatology (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Medicinal Preparation (AREA)

Abstract

USO DE UMA FORMULAçAO PALRA O TRATAMENTO DA QUERATOSE ACTìNICA E USO DE 2-METIL-l-(2-METILPROPIL)-lH-IMIDAZO[4,5-C] [1,5]NAFTIRIDIN-4-ANINA. Trata-se de um método de tratamento da queratose actínica, o qual inclui a aplicação tópica a uma lesão de queratose actínica, duas vezes por semana, por uma duração de oito semanas, de uma formulação que compreende 2-metil-l- (2-metilpropil) -lH-imidazo[4,5-c] [1,5] naftiridin-4-amina.
BRPI0608011-1A 2005-03-14 2006-03-14 uso de uma formulação para o tratamento da queratose actìnica e uso de 2-metil-1-(2-metilpropil)-1h-imidazo[4,5-c][1,5] naftiridin-4-amina BRPI0608011A2 (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US66166105P 2005-03-14 2005-03-14
PCT/US2006/008868 WO2006099275A2 (en) 2005-03-14 2006-03-14 Method of treating actinic keratosis

Publications (1)

Publication Number Publication Date
BRPI0608011A2 true BRPI0608011A2 (pt) 2009-11-03

Family

ID=36992327

Family Applications (1)

Application Number Title Priority Date Filing Date
BRPI0608011-1A BRPI0608011A2 (pt) 2005-03-14 2006-03-14 uso de uma formulação para o tratamento da queratose actìnica e uso de 2-metil-1-(2-metilpropil)-1h-imidazo[4,5-c][1,5] naftiridin-4-amina

Country Status (15)

Country Link
US (1) US8354424B2 (pt)
EP (1) EP1865957A4 (pt)
JP (1) JP2008533148A (pt)
CN (1) CN101175493A (pt)
AU (1) AU2006223148A1 (pt)
BR (1) BRPI0608011A2 (pt)
CA (1) CA2602098A1 (pt)
CR (1) CR9382A (pt)
EC (1) ECSP077736A (pt)
IL (1) IL185581A0 (pt)
MX (1) MX2007011112A (pt)
NI (1) NI200700239A (pt)
NO (1) NO20075278L (pt)
RU (1) RU2007137960A (pt)
WO (1) WO2006099275A2 (pt)

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Also Published As

Publication number Publication date
ECSP077736A (es) 2008-01-23
NI200700239A (es) 2008-06-10
RU2007137960A (ru) 2009-04-20
NO20075278L (no) 2007-12-10
CA2602098A1 (en) 2006-09-21
US8354424B2 (en) 2013-01-15
MX2007011112A (es) 2007-11-07
CR9382A (es) 2008-08-26
WO2006099275A3 (en) 2007-10-25
EP1865957A4 (en) 2009-05-06
IL185581A0 (en) 2008-08-07
WO2006099275A2 (en) 2006-09-21
US20080262022A1 (en) 2008-10-23
AU2006223148A1 (en) 2006-09-21
EP1865957A2 (en) 2007-12-19
CN101175493A (zh) 2008-05-07
JP2008533148A (ja) 2008-08-21

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