BRPI0618381A2 - processo para a preparação do hemi-sal de cálcio do ácido (3r, 5r) -7-[2-(4-fluorofenil) -5-isopropil-3-fenil-4-[(4-hidroximetilfenilamino) carbonil]-pirrol-1-il] -3, 5-diidroxi heptanóico - Google Patents

processo para a preparação do hemi-sal de cálcio do ácido (3r, 5r) -7-[2-(4-fluorofenil) -5-isopropil-3-fenil-4-[(4-hidroximetilfenilamino) carbonil]-pirrol-1-il] -3, 5-diidroxi heptanóico Download PDF

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BRPI0618381A2
BRPI0618381A2 BRPI0618381-6A BRPI0618381A BRPI0618381A2 BR PI0618381 A2 BRPI0618381 A2 BR PI0618381A2 BR PI0618381 A BRPI0618381 A BR PI0618381A BR PI0618381 A2 BRPI0618381 A2 BR PI0618381A2
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carbonyl
isopropyl
phenyl
preparation
fluorophenyl
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BRPI0618381-6A
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English (en)
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Jitendra Anant Sattigeri
Sachin Sethi
Kaushal Kishore
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Ranbaxy Lab Ltd
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    • C07D207/30—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members
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Abstract

PROCESSO PARA A PREPARAçãO DO HEMI-SAL DE CáLCIO DO áCIDO (3R, 5R) -7- [2- (4-FLUOROFENIL) -5-ISOPROPIL-3-FENIL-4- [(4- HIDROXIMETILFENILAMINO) CARBONIL] -PIRROL-1-IL] -3, 5-DIIDROXI HEPTANóICO. A presente invenção refere-se a processos para a preparação do hemi-sal de cálcio do ácido (3R,5R)-7-[2-(4- fluorofenil) -5-isopropil-3-fenil-4- [ (4-hidroximetilfenil amino) carbonil] -pirrol-l-il] -3, 5-diidroxiheptanóico.
BRPI0618381-6A 2005-11-08 2006-11-08 processo para a preparação do hemi-sal de cálcio do ácido (3r, 5r) -7-[2-(4-fluorofenil) -5-isopropil-3-fenil-4-[(4-hidroximetilfenilamino) carbonil]-pirrol-1-il] -3, 5-diidroxi heptanóico BRPI0618381A2 (pt)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
IN2967DE2005 2005-11-08
IN2964DE2005 2005-11-08
IN3033DE2005 2005-11-14
PCT/IB2006/003153 WO2007054790A1 (en) 2005-11-08 2006-11-08 Process for preparation of (3r, 5r)-7-[2-(4-fluorophenyl)-5-isopropyl-3-phenyl-4-[(4-hydroxy methyl phenyl amino) carbonyl]-pyrrol-1-yl]-3,5-dihydroxy-heptanoic acid hemi calcium salt

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BRPI0618381A2 true BRPI0618381A2 (pt) 2011-08-30

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BRPI0618379-4A BRPI0618379A2 (pt) 2005-11-08 2006-11-07 processo para preparação do hemi-sal de cálcio do ácido (3r,5r) -7-[2-(4-fluorofenil)-5-isopropil-3-fenil-4-[(4-hidroxime tilfenilamino) carbonil]-pirrol-1-il] -3, 5-diidroxi heptanóico
BRPI0618381-6A BRPI0618381A2 (pt) 2005-11-08 2006-11-08 processo para a preparação do hemi-sal de cálcio do ácido (3r, 5r) -7-[2-(4-fluorofenil) -5-isopropil-3-fenil-4-[(4-hidroximetilfenilamino) carbonil]-pirrol-1-il] -3, 5-diidroxi heptanóico
BRPI0618380-8A BRPI0618380A2 (pt) 2005-11-08 2006-11-08 combinação farmacêutica e seu uso

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BRPI0618379-4A BRPI0618379A2 (pt) 2005-11-08 2006-11-07 processo para preparação do hemi-sal de cálcio do ácido (3r,5r) -7-[2-(4-fluorofenil)-5-isopropil-3-fenil-4-[(4-hidroxime tilfenilamino) carbonil]-pirrol-1-il] -3, 5-diidroxi heptanóico

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BRPI0618380-8A BRPI0618380A2 (pt) 2005-11-08 2006-11-08 combinação farmacêutica e seu uso

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US (5) US8026377B2 (pt)
EP (3) EP1948599A1 (pt)
JP (3) JP2009514851A (pt)
KR (3) KR101329112B1 (pt)
CN (1) CN102526029A (pt)
AU (3) AU2006313430B2 (pt)
BR (3) BRPI0618379A2 (pt)
CA (3) CA2627599A1 (pt)
IL (1) IL191203A0 (pt)
MY (1) MY147450A (pt)
NZ (1) NZ567738A (pt)
SG (1) SG166829A1 (pt)
WO (3) WO2007054896A1 (pt)

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US20080287690A1 (en) 2008-11-20
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