BRPI0715199A2 - derivados de n-(amino-hetero aril)-1h-indol-2-carboxamida, o respectivo preparo e a respectiva aplicaÇço em terapÊutica - Google Patents

derivados de n-(amino-hetero aril)-1h-indol-2-carboxamida, o respectivo preparo e a respectiva aplicaÇço em terapÊutica

Info

Publication number: BRPI0715199A2
Authority: BR; Brazil
Prior art keywords: aminoheteroaryl; indole; preparation; therapeutic application; carboxamide derivatives
Prior art date: 2006-07-31

Application number

BRPI0715199-3A2A

Other languages

English (en)

Inventor

Laurent Dubois

Yannick Evanno

Andre Malanda

David Machnik

Catherine Gille

Original Assignee

Sanofi Aventis

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2006-07-31

Filing date

2007-07-30

Publication date

2013-10-01

2007-07-30 Application filed by Sanofi Aventis filed Critical Sanofi Aventis

2013-10-01 Publication of BRPI0715199A2 publication Critical patent/BRPI0715199A2/pt

Links

125000005214 aminoheteroaryl group Chemical group 0.000 title 1
230000001225 therapeutic effect Effects 0.000 title 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D213/72—Nitrogen atoms
- C07D213/74—Amino or imino radicals substituted by hydrocarbon or substituted hydrocarbon radicals
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
- A61K31/4439—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A61P17/04—Antipruritics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A61P17/06—Antipsoriatics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/22—Anxiolytics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
- A61P31/20—Antivirals for DNA viruses
- A61P31/22—Antivirals for DNA viruses for herpes viruses
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
- C07D403/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Life Sciences & Earth Sciences (AREA)
Medicinal Chemistry (AREA)
Pharmacology & Pharmacy (AREA)
Veterinary Medicine (AREA)
Public Health (AREA)
General Health & Medical Sciences (AREA)
Animal Behavior & Ethology (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Neurology (AREA)
Neurosurgery (AREA)
Biomedical Technology (AREA)
Diabetes (AREA)
Dermatology (AREA)
Virology (AREA)
Pain & Pain Management (AREA)
Obesity (AREA)
Endocrinology (AREA)
Hematology (AREA)
Emergency Medicine (AREA)
Rheumatology (AREA)
Oncology (AREA)
Psychiatry (AREA)
Immunology (AREA)
Biotechnology (AREA)
Molecular Biology (AREA)
Ophthalmology & Optometry (AREA)
Reproductive Health (AREA)
Communicable Diseases (AREA)
Pulmonology (AREA)
Urology & Nephrology (AREA)
Epidemiology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Plural Heterocyclic Compounds (AREA)

BRPI0715199-3A2A 2006-07-31 2007-07-30 derivados de n-(amino-hetero aril)-1h-indol-2-carboxamida, o respectivo preparo e a respectiva aplicaÇço em terapÊutica BRPI0715199A2 (pt)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
FR0606988A FR2904316B1 (fr)	2006-07-31	2006-07-31	Derives de n-(amino-heteroaryl)-1h-indole-2-carboxamides, leur preparation et leur application en therapeutique.
PCT/FR2007/001316 WO2008015335A1 (fr)	2006-07-31	2007-07-30	Derives de n-(amino-heteroaryl)-1h-indole-2-carboxamides, leur preparation et leur application en therapeutique

Publications (1)

Publication Number	Publication Date
BRPI0715199A2 true BRPI0715199A2 (pt)	2013-10-01

Family

ID=37806631

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
BRPI0715199-3A2A BRPI0715199A2 (pt)	2006-07-31	2007-07-30	derivados de n-(amino-hetero aril)-1h-indol-2-carboxamida, o respectivo preparo e a respectiva aplicaÇço em terapÊutica

Country Status (36)

Country	Link
US (2)	US7786104B2 (pt)
EP (1)	EP2049525B1 (pt)
JP (1)	JP5306201B2 (pt)
KR (1)	KR20090033885A (pt)
CN (1)	CN101511819B (pt)
AR (1)	AR062143A1 (pt)
AT (1)	ATE453637T1 (pt)
AU (1)	AU2007280326B2 (pt)
BR (1)	BRPI0715199A2 (pt)
CA (1)	CA2658799C (pt)
CL (1)	CL2007002169A1 (pt)
CO (1)	CO6150179A2 (pt)
CY (1)	CY1109944T1 (pt)
DE (1)	DE602007004119D1 (pt)
DK (1)	DK2049525T3 (pt)
EA (1)	EA017375B1 (pt)
ES (1)	ES2338610T3 (pt)
FR (1)	FR2904316B1 (pt)
HR (1)	HRP20100121T1 (pt)
IL (1)	IL196571A0 (pt)
JO (1)	JO2644B1 (pt)
MA (1)	MA30695B1 (pt)
ME (1)	ME00590A (pt)
MX (1)	MX2009001222A (pt)
MY (1)	MY145031A (pt)
NO (1)	NO20090952L (pt)
NZ (1)	NZ574345A (pt)
PE (1)	PE20080688A1 (pt)
PL (1)	PL2049525T3 (pt)
PT (1)	PT2049525E (pt)
RS (1)	RS51235B (pt)
SI (1)	SI2049525T1 (pt)
TW (1)	TW200813023A (pt)
UY (1)	UY30518A1 (pt)
WO (1)	WO2008015335A1 (pt)
ZA (1)	ZA200900505B (pt)

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EP2025674A1 (de)	2007-08-15	2009-02-18	sanofi-aventis	Substituierte Tetrahydronaphthaline, Verfahren zu ihrer Herstellung und ihre Verwendung als Arzneimittel
FR2926554B1 (fr) *	2008-01-22	2010-03-12	Sanofi Aventis	Derives de carboxamides azabicycliques, leur preparation et leur application en therapeutique
FR2926556B1 (fr) *	2008-01-22	2010-02-19	Sanofi Aventis	Derives de carboxamides n-azabicycliques, leur preparation et leur application en therapeutique
FR2926553B1 (fr) *	2008-01-23	2010-02-19	Sanofi Aventis	Derives d'indole-2-carboxamides et d'azaindole-2- carboxamides substitues par un groupe silanyle, leur preparation et leur application en therapeutique
AU2010232729A1 (en)	2009-03-31	2011-10-20	Arqule, Inc.	Substituted indolo-pyridinone compounds
EP2794565B1 (en)	2011-12-21	2017-07-26	Novira Therapeutics Inc.	Hepatitis b antiviral agents
CA2881057C (en)	2012-08-28	2020-10-27	Janssen Sciences Ireland Uc	Sulfamoyl-arylamides and the use thereof as medicaments for the treatment of hepatitis b
JP6466348B2 (ja)	2013-02-28	2019-02-06	ヤンセン・サイエンシズ・アイルランド・アンリミテッド・カンパニー	スルファモイル−アリールアミドおよびｂ型肝炎を処置するための医薬品としてのその使用
HUE033542T2 (en)	2013-04-03	2017-12-28	Janssen Sciences Ireland Uc	Their use as medicaments for the treatment of N-phenylcarboxamide derivatives and hepatitis B
TW202126620A (zh)	2013-05-17	2021-07-16	愛爾蘭商健生科學愛爾蘭無限公司	胺磺醯基吡咯醯胺衍生物及其作為用於治療ｂ型肝炎藥物的用途
HUE040446T2 (hu)	2013-05-17	2019-03-28	Janssen Sciences Ireland Uc	Szulfamoiltiofenamid-származékok és gyógyszerként történõ alkalmazásuk hepatitis B kezelésére
WO2015011281A1 (en)	2013-07-25	2015-01-29	Janssen R&D Ireland	Glyoxamide substituted pyrrolamide derivatives and the use thereof as medicaments for the treatment of hepatitis b
MX368158B (es)	2013-10-23	2019-09-20	Janssen Sciences Ireland Uc	Derivados de carboxamida y su uso como medicamentos para el tratamiento de la hepatitis b.
US9169212B2 (en)	2014-01-16	2015-10-27	Novira Therapeutics, Inc.	Azepane derivatives and methods of treating hepatitis B infections
US10392349B2 (en)	2014-01-16	2019-08-27	Novira Therapeutics, Inc.	Azepane derivatives and methods of treating hepatitis B infections
JP6553059B2 (ja)	2014-02-05	2019-07-31	ノヴィラ・セラピューティクス・インコーポレイテッド	Ｈｂｖ感染の治療のための併用療法
PL3102572T3 (pl)	2014-02-06	2019-04-30	Janssen Sciences Ireland Uc	Pochodne sulfamoilopirolamidu i ich zastosowanie jako leki do leczenia wirusowego zapalenia wątroby typu B
EP3271019A1 (en)	2015-03-19	2018-01-24	Novira Therapeutics Inc.	Azocane and azonane derivatives and methods of treating hepatitis b infections
US10875876B2 (en)	2015-07-02	2020-12-29	Janssen Sciences Ireland Uc	Cyclized sulfamoylarylamide derivatives and the use thereof as medicaments for the treatment of hepatitis B
AR106192A1 (es)	2015-09-29	2017-12-20	Novira Therapeutics Inc	Formas cristalinas de un agente antiviral contra la hepatitis b
WO2017181141A2 (en)	2016-04-15	2017-10-19	Novira Therapeutics, Inc.	Combinations and methods comprising a capsid assembly inhibitor
WO2017210545A1 (en)	2016-06-02	2017-12-07	Cadent Therapeutics, Inc.	Potassium channel modulators
EP3571193B1 (en)	2017-01-23	2021-12-01	Cadent Therapeutics, Inc.	Potassium channel modulators
SG11202007097QA (en)	2018-03-14	2020-08-28	Janssen Sciences Ireland Unlimited Co	Capsid assembly modulator dosing regimen
MX2021004647A (es)	2018-10-22	2021-08-16	Novartis Ag	Formas cristalinas de moduladores de los canales de potasio.
AU2020223865A1 (en)	2019-02-22	2021-07-15	Janssen Sciences Ireland Unlimited Company	Amide derivatives useful in the treatment of HBV infection or HBV-induced diseases
BR112021021454A2 (pt)	2019-05-06	2021-12-21	Janssen Sciences Ireland Unlimited Co	Derivados de amida úteis no tratamento da infecção por hbv ou doenças induzidas por hbv

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FR2832148B1 (fr) *	2001-11-14	2004-05-21	Oreal	Nouvelles bases d'oxydation 2,5-diaminopyridine utiles pour la teinture des fibres keratiniques
MY141521A (en)	2002-12-12	2010-05-14	Hoffmann La Roche	5-substituted-six-membered heteroaromatic glucokinase activators
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GB0314136D0 (en)	2003-06-18	2003-07-23	Astrazeneca Ab	Therapeutic agents
GB0322016D0 (en)	2003-09-19	2003-10-22	Merck Sharp & Dohme	New compounds
JP2007505888A (ja)	2003-09-22	2007-03-15	ファイザーインコーポレイテッド	オキシトシン拮抗薬としての置換トリアゾール誘導体
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GB0326633D0 (en) *	2003-11-14	2003-12-17	Merck Sharp & Dohme	Therapeutic agents
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FR2880625B1 (fr) *	2005-01-07	2007-03-09	Sanofi Aventis Sa	Derives de n-(heteroaryl)-1h-indole-2-carboxamides, leur preparation et leur application en therapeutique
US20080221107A1 (en)	2005-07-15	2008-09-11	Astrazeneca Ab	Therapeutic Agents
BRPI0619052A2 (pt) *	2005-11-28	2011-09-20	Hoffmann La Roche	compostos, processo para a sua preparação, composições farmacêuticas que os compreendem, método para o tratamento terapêutico e/ou profilático de enfermidades que são moduladas por inibidores de diacilglicerol aciltransferase, e seu uso

2006
- 2006-07-31 FR FR0606988A patent/FR2904316B1/fr not_active Expired - Fee Related
2007
- 2007-07-20 TW TW096126658A patent/TW200813023A/zh unknown
- 2007-07-24 CL CL200702169A patent/CL2007002169A1/es unknown
- 2007-07-26 PE PE2007000976A patent/PE20080688A1/es not_active Application Discontinuation
- 2007-07-30 BR BRPI0715199-3A2A patent/BRPI0715199A2/pt not_active IP Right Cessation
- 2007-07-30 JP JP2009522302A patent/JP5306201B2/ja not_active Expired - Fee Related
- 2007-07-30 DK DK07823371.5T patent/DK2049525T3/da active
- 2007-07-30 AR ARP070103358A patent/AR062143A1/es not_active Application Discontinuation
- 2007-07-30 NZ NZ574345A patent/NZ574345A/en not_active IP Right Cessation
- 2007-07-30 ME MEP-30/09A patent/ME00590A/xx unknown
- 2007-07-30 KR KR1020097002074A patent/KR20090033885A/ko not_active Ceased
- 2007-07-30 ZA ZA200900505A patent/ZA200900505B/xx unknown
- 2007-07-30 HR HR20100121T patent/HRP20100121T1/hr unknown
- 2007-07-30 DE DE602007004119T patent/DE602007004119D1/de active Active
- 2007-07-30 AU AU2007280326A patent/AU2007280326B2/en not_active Ceased
- 2007-07-30 JO JO2007310A patent/JO2644B1/en active
- 2007-07-30 SI SI200730186T patent/SI2049525T1/sl unknown
- 2007-07-30 ES ES07823371T patent/ES2338610T3/es active Active
- 2007-07-30 RS RSP-2010/0139A patent/RS51235B/sr unknown
- 2007-07-30 PT PT07823371T patent/PT2049525E/pt unknown
- 2007-07-30 CA CA2658799A patent/CA2658799C/fr active Active
- 2007-07-30 AT AT07823371T patent/ATE453637T1/de active
- 2007-07-30 WO PCT/FR2007/001316 patent/WO2008015335A1/fr not_active Ceased
- 2007-07-30 CN CN200780032445.6A patent/CN101511819B/zh not_active Expired - Fee Related
- 2007-07-30 EP EP07823371A patent/EP2049525B1/fr active Active
- 2007-07-30 MX MX2009001222A patent/MX2009001222A/es active IP Right Grant
- 2007-07-30 MY MYPI20090381A patent/MY145031A/en unknown
- 2007-07-30 EA EA200970171A patent/EA017375B1/ru not_active IP Right Cessation
- 2007-07-30 PL PL07823371T patent/PL2049525T3/pl unknown
- 2007-07-31 UY UY30518A patent/UY30518A1/es not_active Application Discontinuation
2009
- 2009-01-18 IL IL196571A patent/IL196571A0/en unknown
- 2009-01-26 US US12/359,468 patent/US7786104B2/en not_active Expired - Fee Related
- 2009-01-29 CO CO09008274A patent/CO6150179A2/es unknown
- 2009-02-13 MA MA31642A patent/MA30695B1/fr unknown
- 2009-03-02 NO NO20090952A patent/NO20090952L/no not_active Application Discontinuation
2010
- 2010-03-22 CY CY20101100268T patent/CY1109944T1/el unknown
- 2010-07-19 US US12/838,771 patent/US8586573B2/en not_active Expired - Fee Related

Also Published As

Publication number	Publication date
CL2007002169A1 (es)	2008-03-07
CO6150179A2 (es)	2010-04-20
AU2007280326A1 (en)	2008-02-07
DK2049525T3 (da)	2010-05-03
EA017375B1 (ru)	2012-12-28
JO2644B1 (en)	2012-06-17
ME00590A (en)	2011-12-20
CY1109944T1 (el)	2014-09-10
ES2338610T3 (es)	2010-05-10
PL2049525T3 (pl)	2010-07-30
JP5306201B2 (ja)	2013-10-02
EA200970171A1 (ru)	2009-06-30
ZA200900505B (en)	2010-04-28
MX2009001222A (es)	2009-02-13
PT2049525E (pt)	2010-03-23
KR20090033885A (ko)	2009-04-06
TW200813023A (en)	2008-03-16
CA2658799C (fr)	2014-10-07
AU2007280326B2 (en)	2012-11-29
MA30695B1 (fr)	2009-09-01
NZ574345A (en)	2011-11-25
JP2009545574A (ja)	2009-12-24
RS51235B (sr)	2010-12-31
WO2008015335A1 (fr)	2008-02-07
CA2658799A1 (fr)	2008-02-07
MY145031A (en)	2011-12-15
AR062143A1 (es)	2008-10-15
DE602007004119D1 (de)	2010-02-11
IL196571A0 (en)	2009-11-18
CN101511819A (zh)	2009-08-19
UY30518A1 (es)	2008-02-29
PE20080688A1 (es)	2008-07-24
NO20090952L (no)	2009-04-23
FR2904316B1 (fr)	2008-09-05
EP2049525A1 (fr)	2009-04-22
CN101511819B (zh)	2014-04-23
ATE453637T1 (de)	2010-01-15
US20100286119A1 (en)	2010-11-11
HRP20100121T1 (hr)	2010-04-30
US20090156573A1 (en)	2009-06-18
SI2049525T1 (sl)	2010-04-30
EP2049525B1 (fr)	2009-12-30
US8586573B2 (en)	2013-11-19
FR2904316A1 (fr)	2008-02-01
US7786104B2 (en)	2010-08-31

Legal Events

Date	Code	Title	Description
2018-04-17	B07D	Technical examination (opinion) related to article 229 of industrial property law [chapter 7.4 patent gazette]
2018-04-24	B06F	Objections, documents and/or translations needed after an examination request according [chapter 6.6 patent gazette]
2019-05-28	B08F	Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette]	Free format text: REFERENTE A 12A ANUIDADE.
2019-09-17	B08K	Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette]	Free format text: EM VIRTUDE DO ARQUIVAMENTO PUBLICADO NA RPI 2525 DE 28-05-2019 E CONSIDERANDO AUSENCIA DE MANIFESTACAO DENTRO DOS PRAZOS LEGAIS, INFORMO QUE CABE SER MANTIDO O ARQUIVAMENTO DO PEDIDO DE PATENTE, CONFORME O DISPOSTO NO ARTIGO 12, DA RESOLUCAO 113/2013.

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IL196571A0 (en)	2009-11-18	N-(aminoheteroaryl)-1h-indole-2-carboxamide derivatives, and preparation and therapeutic application thereof
ZA200900228B (en)	2010-03-31	N-(aminoheteroaryl)-1H-indole-2-carboxamide derivatives, preparation thereof and therapeutic use thereof
BRPI0906567A2 (pt)	2015-07-07	Derivados de ureia de tetra-hidroquinoxalina, o respectivo preparo e a respectiva aplicação em terapêutica j
BRPI0907381A2 (pt)	2015-07-14	Derivados de carboxamidas azabicíclicos, o respectivo preparo e a respectiva aplicação em terapêutica.
DE602007010981D1 (de)	2011-01-13	Cycloalkylaminsubstituierte isochinolin- und isochinolinonderivate
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FR2911604B1 (fr)	2009-04-17	Derives de n-(heteroaryl-1h-indole-2-carboxamides, leur preparation et leur application en therapeutique
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ATE507223T1 (de)	2011-05-15	N-cycloalkyl-carboxamid-, thiocarboxamid- und n- substitutierte carboximidamid-derivate als fungizide
BRPI0715342A2 (pt)	2015-03-24	Derivados de 6-carboxi-normorfinano, síntese e usos dos mesmos
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BRPI0814177A2 (pt)	2015-01-20	Derivados de 1-oxo-1,2-di-hidroisoquinoleína-5-carboxamidas e de 4-oxo-3,4-di-hidroquinazolina-8-carboxamidas, sua preparação e sua aplicação em terapêutica
FR2917413B1 (fr)	2009-08-21	Derives de 7-alkynyl-1,8-naphthyridones, leur preparation et leur application en therapeutique
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