BRPI0718436A2 - Novos derivados de benzamida como antagonistas da bradicina - Google Patents

Novos derivados de benzamida como antagonistas da bradicina

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Publication number
BRPI0718436A2
BRPI0718436A2 BRPI0718436-0A2A BRPI0718436A BRPI0718436A2 BR PI0718436 A2 BRPI0718436 A2 BR PI0718436A2 BR PI0718436 A BRPI0718436 A BR PI0718436A BR PI0718436 A2 BRPI0718436 A2 BR PI0718436A2
Authority
BR
Brazil
Prior art keywords
bradicine
antagonists
benzamide derivatives
new benzamide
new
Prior art date
Application number
BRPI0718436-0A2A
Other languages
English (en)
Inventor
Istvan Vago
Gyula Beke
Eva Bozo
Sandor Farkas
Katalin Hornok
Gyoergy Keserue
Eva Schmidt
Eva Szentirmay
Monika Vastag
Original Assignee
Richter Gedeon Nyrt
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Richter Gedeon Nyrt filed Critical Richter Gedeon Nyrt
Publication of BRPI0718436A2 publication Critical patent/BRPI0718436A2/pt
Publication of BRPI0718436B1 publication Critical patent/BRPI0718436B1/pt
Publication of BRPI0718436B8 publication Critical patent/BRPI0718436B8/pt

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    • C07D295/16—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms
    • C07D295/18—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms by radicals derived from carboxylic acids, or sulfur or nitrogen analogues thereof
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BRPI0718436A 2006-10-27 2007-10-27 compostos antagonistas do receptor b1 da bradicinina derivados de fenilsulfamoilbenzamida, processo para preparar os mesmos, uso dos mesmos e composição farmacêutica BRPI0718436B8 (pt)

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TWI901650B (zh) 2020-03-26 2025-10-21 匈牙利商羅特格登公司 啶及吡啶并〔３，４－ｃ〕嗒衍生物
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HU231691B1 (hu) 2021-09-29 2025-10-28 Richter Gedeon Nyrt GABAA ALFA5 receptor modulátor hatású biciklusos aminszármazékok

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