BRPI0920895A2 - compostos antibióticos de oxazolidinona tricíclica - Google Patents

compostos antibióticos de oxazolidinona tricíclica

Info

Publication number
BRPI0920895A2
BRPI0920895A2 BRPI0920895A BRPI0920895A BRPI0920895A2 BR PI0920895 A2 BRPI0920895 A2 BR PI0920895A2 BR PI0920895 A BRPI0920895 A BR PI0920895A BR PI0920895 A BRPI0920895 A BR PI0920895A BR PI0920895 A2 BRPI0920895 A2 BR PI0920895A2
Authority
BR
Brazil
Prior art keywords
antibiotic compounds
oxazolidinone antibiotic
tricyclic
tricyclic oxazolidinone
compounds
Prior art date
Application number
BRPI0920895A
Other languages
English (en)
Inventor
Christian Hubschwerlen
Cornelia Zumbrunn Acklin
Daniel Ritz
Georg Rueedi
Jean-Philippe Surivet
Original Assignee
Actelion Pharmaceuticals Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=41402623&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=BRPI0920895(A2) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Actelion Pharmaceuticals Ltd filed Critical Actelion Pharmaceuticals Ltd
Publication of BRPI0920895A2 publication Critical patent/BRPI0920895A2/pt
Publication of BRPI0920895A8 publication Critical patent/BRPI0920895A8/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/06—Peri-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47—Quinolines; Isoquinolines
    • A61K31/4738—Quinolines; Isoquinolines ortho- or peri-condensed with heterocyclic ring systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/12—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains three hetero rings
    • C07D471/16—Peri-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/06—Peri-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D519/00—Heterocyclic compounds containing more than one system of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring system not provided for in groups C07D453/00 or C07D455/00

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Plural Heterocyclic Compounds (AREA)
BRPI0920895A 2008-10-07 2009-10-06 Compostos antibióticos de oxazolidinona tricíclica BRPI0920895A8 (pt)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
IB2008054109 2008-10-07
IB2009051059 2009-03-13
IB2009052843 2009-06-30
PCT/IB2009/054357 WO2010041194A1 (en) 2008-10-07 2009-10-06 Tricyclic oxazolidinone antibiotic compounds

Publications (2)

Publication Number Publication Date
BRPI0920895A2 true BRPI0920895A2 (pt) 2015-12-22
BRPI0920895A8 BRPI0920895A8 (pt) 2017-12-26

Family

ID=41402623

Family Applications (1)

Application Number Title Priority Date Filing Date
BRPI0920895A BRPI0920895A8 (pt) 2008-10-07 2009-10-06 Compostos antibióticos de oxazolidinona tricíclica

Country Status (25)

Country Link
US (3) US8618092B2 (pt)
EP (1) EP2344495B1 (pt)
JP (1) JP4833385B1 (pt)
KR (1) KR101294962B1 (pt)
CN (3) CN104151316B (pt)
AR (1) AR073774A1 (pt)
AU (1) AU2009302075B2 (pt)
BR (1) BRPI0920895A8 (pt)
CA (1) CA2739373C (pt)
CY (1) CY1116155T1 (pt)
DK (1) DK2344495T3 (pt)
ES (1) ES2533217T3 (pt)
HR (1) HRP20150370T1 (pt)
IL (1) IL212139A (pt)
MA (1) MA32768B1 (pt)
MX (1) MX2011003370A (pt)
MY (1) MY158520A (pt)
NZ (1) NZ592642A (pt)
PL (1) PL2344495T3 (pt)
PT (1) PT2344495E (pt)
RU (1) RU2530884C2 (pt)
SI (1) SI2344495T1 (pt)
TW (1) TWI415853B (pt)
WO (1) WO2010041194A1 (pt)
ZA (1) ZA201103332B (pt)

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TW201833120A (zh) 2017-02-17 2018-09-16 瑞士商愛杜西亞製藥有限公司 芳基噁唑啶酮抗生素化合物
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Also Published As

Publication number Publication date
US20110195961A1 (en) 2011-08-11
US9346804B2 (en) 2016-05-24
RU2011117412A (ru) 2012-11-20
CN104151315A (zh) 2014-11-19
CN104151316A (zh) 2014-11-19
ES2533217T3 (es) 2015-04-08
KR20110063836A (ko) 2011-06-14
CN102164925A (zh) 2011-08-24
HRP20150370T1 (hr) 2015-05-08
US8618092B2 (en) 2013-12-31
WO2010041194A1 (en) 2010-04-15
MY158520A (en) 2016-10-14
MA32768B1 (fr) 2011-11-01
MX2011003370A (es) 2011-04-28
EP2344495A1 (en) 2011-07-20
AR073774A1 (es) 2010-12-01
ZA201103332B (en) 2012-10-31
US20160237088A1 (en) 2016-08-18
EP2344495B1 (en) 2014-12-31
PT2344495E (pt) 2015-04-01
SI2344495T1 (sl) 2015-03-31
US9822114B2 (en) 2017-11-21
CY1116155T1 (el) 2017-02-08
CN102164925B (zh) 2015-04-08
DK2344495T3 (en) 2015-02-02
KR101294962B1 (ko) 2013-08-12
IL212139A (en) 2016-07-31
TW201018697A (en) 2010-05-16
BRPI0920895A8 (pt) 2017-12-26
JP4833385B1 (ja) 2011-12-07
US20140142093A1 (en) 2014-05-22
CN104151316B (zh) 2016-06-15
JP2012505199A (ja) 2012-03-01
PL2344495T3 (pl) 2015-06-30
RU2530884C2 (ru) 2014-10-20
HK1159611A1 (en) 2012-08-03
AU2009302075A1 (en) 2010-04-15
TWI415853B (zh) 2013-11-21
NZ592642A (en) 2012-11-30
CN104151315B (zh) 2017-01-11
AU2009302075B2 (en) 2015-04-16
CA2739373A1 (en) 2010-04-15
IL212139A0 (en) 2011-06-30
CA2739373C (en) 2017-01-24

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Legal Events

Date Code Title Description
B25A Requested transfer of rights approved

Owner name: IDORSIA PHARMACEUTICALS LTD (CH)

B25L Entry of change of name and/or headquarter and transfer of application, patent and certificate of addition of invention: publication cancelled

Owner name: ACTELION PHARMACEUTICALS LTD (CH)

B25C Requirement related to requested transfer of rights

Owner name: ACTELION PHARMACEUTICALS LTD (CH)

B07D Technical examination (opinion) related to article 229 of industrial property law [chapter 7.4 patent gazette]
B06F Objections, documents and/or translations needed after an examination request according [chapter 6.6 patent gazette]
B25A Requested transfer of rights approved

Owner name: IDORSIA PHARMACEUTICALS LTD (CH)

B07E Notification of approval relating to section 229 industrial property law [chapter 7.5 patent gazette]

Free format text: NOTIFICACAO DE ANUENCIA RELACIONADA COM O ART 229 DA LPI

B06U Preliminary requirement: requests with searches performed by other patent offices: procedure suspended [chapter 6.21 patent gazette]
B11B Dismissal acc. art. 36, par 1 of ipl - no reply within 90 days to fullfil the necessary requirements