BRPI1009090A2 - composto, pró-droga, medicamento, métodos, e, uso do composto - Google Patents

composto, pró-droga, medicamento, métodos, e, uso do composto

Info

Publication number
BRPI1009090A2
BRPI1009090A2 BRPI1009090A BRPI1009090A BRPI1009090A2 BR PI1009090 A2 BRPI1009090 A2 BR PI1009090A2 BR PI1009090 A BRPI1009090 A BR PI1009090A BR PI1009090 A BRPI1009090 A BR PI1009090A BR PI1009090 A2 BRPI1009090 A2 BR PI1009090A2
Authority
BR
Brazil
Prior art keywords
compound
prodrug
medicine
methods
compound use
Prior art date
Application number
BRPI1009090A
Other languages
English (en)
Inventor
Haruyuki Nishida
Ikuo Fujimori
Original Assignee
Takeda Pharmaceutical
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Takeda Pharmaceutical filed Critical Takeda Pharmaceutical
Publication of BRPI1009090A2 publication Critical patent/BRPI1009090A2/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/4439—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
BRPI1009090A 2009-03-26 2010-03-25 composto, pró-droga, medicamento, métodos, e, uso do composto BRPI1009090A2 (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP2009077078 2009-03-26
PCT/JP2010/055257 WO2010110378A1 (ja) 2009-03-26 2010-03-25 ピラゾール化合物

Publications (1)

Publication Number Publication Date
BRPI1009090A2 true BRPI1009090A2 (pt) 2016-03-01

Family

ID=42781069

Family Applications (1)

Application Number Title Priority Date Filing Date
BRPI1009090A BRPI1009090A2 (pt) 2009-03-26 2010-03-25 composto, pró-droga, medicamento, métodos, e, uso do composto

Country Status (25)

Country Link
US (1) US8895588B2 (pt)
EP (1) EP2412713B1 (pt)
JP (1) JP5552481B2 (pt)
KR (1) KR101656906B1 (pt)
CN (1) CN102448953B (pt)
AU (1) AU2010228220B2 (pt)
BR (1) BRPI1009090A2 (pt)
CA (1) CA2756086A1 (pt)
CL (1) CL2011002351A1 (pt)
CO (1) CO6460700A2 (pt)
CR (1) CR20110533A (pt)
DO (1) DOP2011000296A (pt)
EA (1) EA019853B1 (pt)
EC (1) ECSP11011419A (pt)
GE (1) GEP20156222B (pt)
IL (1) IL215235A (pt)
MA (1) MA33214B1 (pt)
MX (1) MX2011009943A (pt)
NZ (1) NZ595890A (pt)
PE (1) PE20120618A1 (pt)
SG (1) SG174476A1 (pt)
TN (1) TN2011000474A1 (pt)
UA (1) UA107457C2 (pt)
WO (1) WO2010110378A1 (pt)
ZA (1) ZA201107435B (pt)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP6216338B2 (ja) 2012-06-27 2017-10-18 武田薬品工業株式会社 塩により安定化されたアミンおよび有機酸の液状製剤
CN111419845A (zh) 2012-09-27 2020-07-17 阿莱塔纳治疗学股份有限公司 应用控制食欲不振的化合物的组合物和方法
US9700591B2 (en) 2015-01-28 2017-07-11 Aratana Therapeutics, Inc. Compositions and methods for chronic use of a weight-gaining compound
CN105067814A (zh) * 2015-07-24 2015-11-18 中国科学院成都生物研究所 解旋酶水解atp活性测定方法
KR20210156235A (ko) * 2020-06-17 2021-12-24 일동제약(주) 신규한 산 분비 억제제 및 이의 용도

Family Cites Families (21)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3285991A (en) 1963-03-26 1966-11-15 Union Carbide Corp Polyepoxides cured with the reaction product of a dihydroxydiphenylsul-fone, an amine, and an aldehyde
US4847289A (en) 1987-06-08 1989-07-11 Merck & Co., Inc. Thiophene sulfonamide antiglaucoma agents
CN1071924A (zh) 1991-10-29 1993-05-12 纳幕尔杜邦公司 除草的三唑羧酸酰胺
DE69532245T2 (de) 1994-09-26 2004-09-16 Shionogi & Co., Ltd. Imidazolderivat
JPH0948778A (ja) 1995-08-04 1997-02-18 Sagami Chem Res Center 2−置換−3−アルコキシ−5−(ピロール−2−イル)フラン誘導体
WO1997017070A1 (en) 1995-11-06 1997-05-15 University Of Pittsburgh Inhibitors of protein isoprenyl transferases
CN1246847A (zh) 1996-12-23 2000-03-08 杜邦药品公司 作为Xa因子抑制剂的含氮杂芳族化合物
AU1918299A (en) 1998-02-23 1999-09-06 Warner-Lambert Company Substituted quinoxaline derivatives as interleukin-8 receptor antagonists
AU2003254282A1 (en) 2002-08-01 2004-02-23 Nitromed, Inc. Nitrosated proton pump inhibitors, compositions and methods of use
US7417152B2 (en) 2003-05-02 2008-08-26 Elan Pharmaceuticals, Inc. 4-bromo-5-(2-chloro-benzoylamino)-1H-pyrazole-3-carboxylic acid amide derivatives and related compounds as bradykinin B1 receptor antagonists for the treatment of inflammatory diseases
WO2004103968A1 (en) 2003-05-26 2004-12-02 Aponetics Ag Sulfopyrroles
AU2004259012C1 (en) 2003-07-23 2012-08-02 Exelixis, Inc. Anaplastic lymphoma kinase modulators and methods of use
EP2336107B1 (en) 2004-09-30 2015-09-23 Takeda Pharmaceutical Company Limited Proton pump inhibitors
EP2327692B9 (en) 2005-08-30 2014-06-04 Takeda Pharmaceutical Company Limited 1-heterocyclylsulfonyl, 2-aminomethyl, 5-(hetero-)aryl substituted 1-H-pyrrole derivatives as acid secretion inhibitors
EP2005957B1 (en) 2006-03-31 2012-05-30 Takeda Pharmaceutical Company Limited Acid secretion inhibitor
US8933105B2 (en) * 2007-02-28 2015-01-13 Takeda Pharmaceutical Company Limited Pyrrole compounds
JP2009077078A (ja) 2007-09-19 2009-04-09 Brother Ind Ltd 位置検出システム
EP2196459B1 (en) 2007-09-28 2016-11-02 Takeda Pharmaceutical Company Limited 5-membered heterocyclic compound
PE20090709A1 (es) 2007-09-28 2009-07-15 Takeda Pharmaceutical Compuestos heterociclico de 5 miembros
PE20091846A1 (es) 2008-05-19 2009-12-16 Plexxikon Inc DERIVADOS DE PIRROLO[2,3-d]-PIRIMIDINA COMO MODULADORES DE CINASAS
MX2011000460A (es) 2008-07-18 2011-03-15 Takeda Pharmaceutical Derivados de benzazepina y su uso como antagonistas de histamina h3.

Also Published As

Publication number Publication date
GEP20156222B (en) 2015-01-26
TN2011000474A1 (en) 2013-03-27
IL215235A0 (en) 2011-12-29
EA201171168A1 (ru) 2012-05-30
AU2010228220A1 (en) 2011-11-17
JPWO2010110378A1 (ja) 2012-10-04
EA019853B1 (ru) 2014-06-30
SG174476A1 (en) 2011-10-28
EP2412713B1 (en) 2016-11-30
ECSP11011419A (es) 2011-11-30
KR20110130483A (ko) 2011-12-05
CR20110533A (es) 2012-02-13
DOP2011000296A (es) 2011-10-15
PE20120618A1 (es) 2012-06-05
CL2011002351A1 (es) 2012-07-13
AU2010228220B2 (en) 2015-05-21
NZ595890A (en) 2013-09-27
WO2010110378A1 (ja) 2010-09-30
AU2010228220A2 (en) 2011-11-24
UA107457C2 (uk) 2015-01-12
CO6460700A2 (es) 2012-06-15
KR101656906B1 (ko) 2016-09-12
US8895588B2 (en) 2014-11-25
JP5552481B2 (ja) 2014-07-16
MX2011009943A (es) 2011-10-06
CA2756086A1 (en) 2010-09-30
US20120095057A1 (en) 2012-04-19
MA33214B1 (fr) 2012-04-02
EP2412713A1 (en) 2012-02-01
CN102448953A (zh) 2012-05-09
EP2412713A4 (en) 2014-04-02
CN102448953B (zh) 2014-05-07
IL215235A (en) 2014-07-31
ZA201107435B (en) 2012-08-29

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Legal Events

Date Code Title Description
B08F Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette]
B08K Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette]
B350 Update of information on the portal [chapter 15.35 patent gazette]