BRPI9915208A - preparados farmacêutico e de comprimido para a aplicação oral compreendendo moxifloxacina e seu processo de preparação. - Google Patents

preparados farmacêutico e de comprimido para a aplicação oral compreendendo moxifloxacina e seu processo de preparação.

Info

Publication number
BRPI9915208A
BRPI9915208A BRPI9915208A BRPI9915208A BRPI9915208A BR PI9915208 A BRPI9915208 A BR PI9915208A BR PI9915208 A BRPI9915208 A BR PI9915208A BR PI9915208 A BRPI9915208 A BR PI9915208A BR PI9915208 A BRPI9915208 A BR PI9915208A
Authority
BR
Brazil
Prior art keywords
moxifloxacin
pharmaceutical
oral application
preparation process
tablet preparations
Prior art date
Application number
BRPI9915208A
Other languages
English (en)
Inventor
Patrick Bosche
Hans Friedrich Mahler
Claus Weisemann
Original Assignee
Bayer Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=7889824&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=BRPI9915208(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Bayer Ag filed Critical Bayer Ag
Publication of BRPI9915208A publication Critical patent/BRPI9915208A/pt
Publication of BRPI9915208B1 publication Critical patent/BRPI9915208B1/pt
Publication of BRPI9915208B8 publication Critical patent/BRPI9915208B8/pt

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/28Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2806Coating materials
    • A61K9/2833Organic macromolecular compounds
    • A61K9/286Polysaccharides, e.g. gums; Cyclodextrin
    • A61K9/2866Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47Quinolines; Isoquinolines
    • A61K31/4709Non-condensed quinolines and containing further heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2013Organic compounds, e.g. phospholipids, fats
    • A61K9/2018Sugars, or sugar alcohols, e.g. lactose, mannitol; Derivatives thereof, e.g. polysorbates
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2022Organic macromolecular compounds
    • A61K9/205Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2054Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical & Material Sciences (AREA)
  • Epidemiology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Molecular Biology (AREA)
  • Biophysics (AREA)
  • Organic Chemistry (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Saccharide Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)

Abstract

patente de invenção: <b>"preparado farmacêutico de moxifloxacina"<d>. a presente invenção refere-se a um preparado farmacêutico para a aplicação oral, que contém moxifloxacina, seu sal e/ou hidrato, bem como lactose um processo para a sua preparação, em como o emprego deste preparado para o combate de infecções bacterianas no homem ou nos animais.
BRPI9915208 1998-11-10 1999-10-29 preparados farmacêutico e de comprimido para a aplicação oral compreendendo moxifloxacina e seu processo de preparação. BRPI9915208B8 (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE19855758 1998-11-10
PCT/EP1999/008230 WO2000027398A1 (de) 1998-11-10 1999-10-29 Pharmazeutische zubereitung von moxifloxacin

Publications (3)

Publication Number Publication Date
BRPI9915208A true BRPI9915208A (pt) 2001-07-31
BRPI9915208B1 BRPI9915208B1 (pt) 2011-11-01
BRPI9915208B8 BRPI9915208B8 (pt) 2021-07-06

Family

ID=7889824

Family Applications (2)

Application Number Title Priority Date Filing Date
BR9915208-8A BR9915208A (pt) 1998-11-10 1999-10-29 Preparado farmacêutico de moxifloxacina
BRPI9915208 BRPI9915208B8 (pt) 1998-11-10 1999-10-29 preparados farmacêutico e de comprimido para a aplicação oral compreendendo moxifloxacina e seu processo de preparação.

Family Applications Before (1)

Application Number Title Priority Date Filing Date
BR9915208-8A BR9915208A (pt) 1998-11-10 1999-10-29 Preparado farmacêutico de moxifloxacina

Country Status (41)

Country Link
US (1) US6610327B1 (pt)
EP (1) EP1128831B1 (pt)
JP (1) JP4809978B2 (pt)
KR (1) KR100650489B1 (pt)
CN (1) CN1149993C (pt)
AR (1) AR021074A1 (pt)
AT (1) ATE279193T1 (pt)
AU (1) AU745282B2 (pt)
BG (1) BG64974B1 (pt)
BR (2) BR9915208A (pt)
CA (1) CA2349161C (pt)
CO (1) CO5070571A1 (pt)
CU (1) CU23260B7 (pt)
CZ (1) CZ292069B6 (pt)
DE (1) DE59910858D1 (pt)
DK (1) DK1128831T3 (pt)
EE (1) EE04418B1 (pt)
ES (1) ES2229786T3 (pt)
HK (1) HK1042245B (pt)
HN (1) HN1999000183A (pt)
HR (1) HRP20010332B1 (pt)
HU (1) HU229065B1 (pt)
ID (1) ID29089A (pt)
IL (2) IL142642A0 (pt)
MA (1) MA26757A1 (pt)
MY (1) MY121114A (pt)
NO (1) NO319342B1 (pt)
NZ (1) NZ511554A (pt)
PE (1) PE20001304A1 (pt)
PL (1) PL194020B1 (pt)
PT (1) PT1128831E (pt)
RU (1) RU2230555C9 (pt)
SI (1) SI1128831T1 (pt)
SK (1) SK283936B6 (pt)
SV (1) SV1999000194A (pt)
TR (1) TR200101310T2 (pt)
TW (1) TW580388B (pt)
UA (1) UA72483C2 (pt)
UY (1) UY25792A1 (pt)
WO (1) WO2000027398A1 (pt)
ZA (1) ZA200103141B (pt)

Families Citing this family (32)

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Publication number Priority date Publication date Assignee Title
DE19937116A1 (de) * 1999-08-06 2001-02-08 Bayer Ag Moxifloxacin Kochsalzformulierung
GB0209265D0 (en) 2002-04-23 2002-06-05 Novartis Ag Organic compounds
DE10337191A1 (de) * 2003-08-13 2005-03-17 Bayer Healthcare Ag Neue Verwendung von Chinolon-Antibiotika
WO2005020998A1 (en) * 2003-09-03 2005-03-10 Ranbaxy Laboratories Limited Pharmaceutical compositions of moxifloxacin and processes for their preparation
CN1330306C (zh) * 2004-08-11 2007-08-08 深圳市天一时科技开发有限公司 莫西沙星明胶胶囊剂及其制备方法
WO2006015545A1 (fr) * 2004-08-11 2006-02-16 Shenzhen Tys R & D Co., Ltd. Capsule de gelatine de moxifloxacin et procede pour sa preparation
WO2007033522A1 (fr) * 2005-09-21 2007-03-29 Shenzhen Tys R & D Co., Ltd. Formulation de gélule contenant de la moxifloxacine et son procédé de préparation
WO2007033515A1 (fr) * 2005-09-21 2007-03-29 Shenzhen Tys R & D Co., Ltd. Formulation orale contenant de la moxifloxacine et son procédé de préparation
CN100363001C (zh) * 2005-09-21 2008-01-23 深圳市天一时科技开发有限公司 一种莫西沙星胶囊剂及其制备方法
ES2391132T3 (es) * 2008-10-09 2012-11-21 Abdi Ibrahim Ilac Sanayi Ve Ticaret Anonim Sirketi Uso de disolventes orgánicos en la granulación húmeda de moxifloxacino
WO2010066385A1 (de) 2008-12-08 2010-06-17 Ratiopharm Gmbh Kompaktiertes moxifloxacin
TR200907227A2 (tr) * 2009-09-18 2011-04-21 Bi̇lgi̇ç Mahmut Çözünürlüğü yüksek stabil mikronize granüller.
CN101890169B (zh) * 2009-11-16 2013-09-11 江苏亚邦强生药业有限公司 莫西沙星口服制剂及其制备方法
WO2011086577A2 (en) * 2010-01-12 2011-07-21 Msn Laboratories Limited Pharmaceutical composition of moxifloxacin and its pharmaceutically acceptable salts
CN102247313A (zh) * 2010-06-11 2011-11-23 北京润德康医药技术有限公司 一种以莫西沙星为活性成分的口服缓释固体制剂
CN102247314A (zh) * 2011-01-12 2011-11-23 北京润德康医药技术有限公司 一种以莫西沙星为活性成分的口服固体制剂
EP2510929A1 (en) * 2011-04-11 2012-10-17 Innocoll Technologies Limited Methods for treating bacterial infection
MX2011004759A (es) 2011-05-04 2012-11-21 Senosiain S A De C V Lab Nuevas formas solidas de antibioticos.
RU2466718C1 (ru) * 2011-10-14 2012-11-20 Закрытое акционерное общество "Брынцалов-А" Фармацевтический препарат моксифлоксацина
EP2770985A4 (en) 2011-10-25 2015-01-21 U S Phytotherapy Inc ARTEMISININE AND BERBERINE COMPOSITIONS AND METHOD FOR THE PRODUCTION THEREOF
WO2013063271A1 (en) * 2011-10-25 2013-05-02 U.S. Phytotherapy, Inc. Artemisinin and berberine compositions and methods of making
US9675582B2 (en) 2011-10-25 2017-06-13 U.S. Phytotherapy, Inc. Alternative ACT with natural botanical active GRAS ingredients for treatment and prevention of the Zika virus
US9358261B2 (en) 2011-10-25 2016-06-07 U.S. Phytotherapy, Inc. Additional artemisinin and berberine compositions and methods of making
RU2633477C2 (ru) * 2011-11-30 2017-10-12 Тояма Кемикал Ко., Лтд. Таблетка, содержащая гидрат метансульфоната 1-циклопропил-8-(дифторметокси)-7-[(1r)-1-метил-2, 3-дигидро-1н-изоиндол-5-ил]-4-оксо-1, 4-дигидрохинолин-3-карбоновой кислоты
BRPI1106900A2 (pt) 2011-12-26 2013-11-05 Ems Sa Composição farmacêutica sólida compreendendo antibótico da familia das quinolonas e processo de sua obtenção
CN102525982A (zh) * 2012-02-21 2012-07-04 天津市汉康医药生物技术有限公司 一种稳定的盐酸莫西沙星药物组合物
CN102600093B (zh) * 2012-04-11 2013-06-05 南京优科生物医药有限公司 一种莫西沙星片剂及其制备方法
FR2992218B1 (fr) 2012-06-22 2015-01-23 Rivopharm Sa Composition pharmaceutique de chlorhydrate de moxifloxacine et procede de preparation
CN103768063B (zh) * 2012-10-19 2016-04-20 深圳信立泰药业股份有限公司 一种盐酸莫西沙星药物组合物及其制备方法
RU2561037C2 (ru) * 2013-02-07 2015-08-20 Открытое акционерное общество "Химико-фармацевтический комбинат "АКРИХИН" (ОАО "АКРИХИН") Антибактериальная фармацевтическая композиция и способ ее получения
WO2015093669A1 (ko) * 2013-12-20 2015-06-25 씨제이헬스케어 주식회사 목시플록사신 수성 제형 및 이의 제조방법
RU2558932C1 (ru) * 2014-05-22 2015-08-10 Открытое Акционерное Общество "Татхимфармпрепараты" Фармацевтическая композиция моксифлоксацина и способ ее приготовления

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DE3601566A1 (de) * 1986-01-21 1987-07-23 Bayer Ag Pharmazeutische zubereitungen von ciprofloxacin
US5286754A (en) 1986-01-21 1994-02-15 Bayer Aktiengesellschaft Pharmaceutical formulations of ciprofloxacin
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JPH01175936A (ja) * 1987-12-28 1989-07-12 Kyorin Pharmaceut Co Ltd 6.8−ジフルオロ−1−(2−フルオロエチル)−1,4−ジヒドロ−7−(4−メチル−1−ピペラジニル)−4−オキソ−3−キノリンカルボン酸を有効成分とする錠剤
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Also Published As

Publication number Publication date
SK283936B6 (sk) 2004-05-04
AR021074A1 (es) 2002-06-12
SV1999000194A (es) 2000-10-16
PL348112A1 (en) 2002-05-06
TW580388B (en) 2004-03-21
SI1128831T1 (en) 2005-04-30
RU2230555C9 (ru) 2006-02-27
DE59910858D1 (de) 2004-11-18
UA72483C2 (en) 2005-03-15
MY121114A (en) 2005-12-30
EE04418B1 (et) 2005-02-15
CN1149993C (zh) 2004-05-19
CN1325306A (zh) 2001-12-05
PT1128831E (pt) 2005-01-31
NO20012248D0 (no) 2001-05-07
EP1128831A1 (de) 2001-09-05
AU745282B2 (en) 2002-03-21
NZ511554A (en) 2003-07-25
CZ292069B6 (cs) 2003-07-16
IL142642A0 (en) 2002-03-10
ZA200103141B (en) 2002-05-07
CZ20011652A3 (cs) 2001-08-15
NO319342B1 (no) 2005-07-18
KR100650489B1 (ko) 2006-11-28
BG64974B1 (bg) 2006-11-30
TR200101310T2 (tr) 2001-10-22
ATE279193T1 (de) 2004-10-15
MA26757A1 (fr) 2004-12-20
WO2000027398A1 (de) 2000-05-18
AU1267400A (en) 2000-05-29
HK1042245B (zh) 2005-03-11
EE200100259A (et) 2002-12-16
BRPI9915208B1 (pt) 2011-11-01
CU23260B7 (es) 2008-01-24
PL194020B1 (pl) 2007-04-30
SK6102001A3 (en) 2001-12-03
HN1999000183A (es) 1999-11-01
BRPI9915208B8 (pt) 2021-07-06
HRP20010332A2 (en) 2002-06-30
CA2349161C (en) 2008-01-29
KR20010089424A (ko) 2001-10-06
UY25792A1 (es) 2001-08-27
RU2230555C2 (ru) 2004-06-20
HUP0104762A3 (en) 2002-10-28
ID29089A (id) 2001-07-26
IL142642A (en) 2006-10-05
BR9915208A (pt) 2001-07-31
CA2349161A1 (en) 2000-05-18
PE20001304A1 (es) 2000-12-30
JP2002529415A (ja) 2002-09-10
ES2229786T3 (es) 2005-04-16
JP4809978B2 (ja) 2011-11-09
DK1128831T3 (da) 2005-01-17
HK1042245A1 (en) 2002-08-09
HU229065B1 (en) 2013-07-29
US6610327B1 (en) 2003-08-26
NO20012248L (no) 2001-06-06
BG105459A (en) 2001-12-29
HUP0104762A2 (hu) 2002-05-29
HRP20010332B1 (hr) 2011-01-31
EP1128831B1 (de) 2004-10-13
CO5070571A1 (es) 2001-08-28

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