CR10872A - Compuestos agonistas y antagonistas del receptor de esfingosina-1-fosfato - Google Patents

Compuestos agonistas y antagonistas del receptor de esfingosina-1-fosfato

Info

Publication number: CR10872A
Authority: CR; Costa Rica
Prior art keywords: sphingosine; agonist; antagonist compounds; phosphate receptor; receptor family
Prior art date: 2006-12-21

Application number

CR10872A

Other languages

English (en)

Spanish (es)

Inventor

Grier A Wallace

Eric C Breinlinger

Kevin P Cusack

Shannon R Fix-Senzel

Thomas D Gordon

Adrian D Hobson

Martin E Hayes

Graham K Ansell

Pintipa Grongsaard

Original Assignee

Abbott Lab

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2006-12-21

Filing date

2009-06-19

Publication date

2009-07-23

Family has litigation

First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=39562856&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=CR10872(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.

2009-06-19 Application filed by Abbott Lab filed Critical Abbott Lab

2009-07-23 Publication of CR10872A publication Critical patent/CR10872A/es

Links

102000011011 Sphingosine 1-phosphate receptors Human genes 0.000 title abstract 3
108050001083 Sphingosine 1-phosphate receptors Proteins 0.000 title abstract 3
239000000556 agonist Substances 0.000 title abstract 2
239000005557 antagonist Substances 0.000 title abstract 2
150000001875 compounds Chemical class 0.000 title abstract 2
102000005962 receptors Human genes 0.000 abstract 2
108020003175 receptors Proteins 0.000 abstract 2
230000008484 agonism Effects 0.000 abstract 1
230000008485 antagonism Effects 0.000 abstract 1
239000003795 chemical substances by application Substances 0.000 abstract 1
239000003814 drug Substances 0.000 abstract 1
230000003389 potentiating effect Effects 0.000 abstract 1
229940124597 therapeutic agent Drugs 0.000 abstract 1

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- C07D413/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
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- C07F9/38—Phosphonic acids [RP(=O)(OH)2]; Thiophosphonic acids ; [RP(=X1)(X2H)2(X1, X2 are each independently O, S or Se)]
- C07F9/40—Esters thereof
- C07F9/4003—Esters thereof the acid moiety containing a substituent or a structure which is considered as characteristic
- C07F9/4006—Esters of acyclic acids which can have further substituents on alkyl
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
- C07F9/02—Phosphorus compounds
- C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
- C07F9/6527—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having nitrogen and oxygen atoms as the only ring hetero atoms
- C07F9/653—Five-membered rings
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
- C07F9/02—Phosphorus compounds
- C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
- C07F9/655—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having oxygen atoms, with or without sulfur, selenium, or tellurium atoms, as the only ring hetero atoms
- C07F9/65515—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having oxygen atoms, with or without sulfur, selenium, or tellurium atoms, as the only ring hetero atoms the oxygen atom being part of a five-membered ring
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
- C07F9/02—Phosphorus compounds
- C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
- C07F9/6553—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having sulfur atoms, with or without selenium or tellurium atoms, as the only ring hetero atoms
- C07F9/655345—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having sulfur atoms, with or without selenium or tellurium atoms, as the only ring hetero atoms the sulfur atom being part of a five-membered ring
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C2601/00—Systems containing only non-condensed rings
- C07C2601/02—Systems containing only non-condensed rings with a three-membered ring
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C2601/00—Systems containing only non-condensed rings
- C07C2601/06—Systems containing only non-condensed rings with a five-membered ring
- C07C2601/08—Systems containing only non-condensed rings with a five-membered ring the ring being saturated

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CR10872A 2006-12-21 2009-06-19 Compuestos agonistas y antagonistas del receptor de esfingosina-1-fosfato CR10872A (es)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
US87631806P	2006-12-21	2006-12-21
US87628806P	2006-12-21	2006-12-21

Publications (1)

Publication Number	Publication Date
CR10872A true CR10872A (es)	2009-07-23

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ID=39562856

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
CR10872A CR10872A (es)	2006-12-21	2009-06-19	Compuestos agonistas y antagonistas del receptor de esfingosina-1-fosfato

Country Status (19)

Country	Link
EP (1)	EP2120575A4 (pt)
JP (1)	JP2010513532A (pt)
KR (1)	KR20090095659A (pt)
AR (1)	AR064650A1 (pt)
AU (1)	AU2007338700A1 (pt)
BR (1)	BRPI0720478A2 (pt)
CA (1)	CA2672727A1 (pt)
CL (1)	CL2007003784A1 (pt)
CO (1)	CO6180436A2 (pt)
CR (1)	CR10872A (pt)
DO (1)	DOP2009000149A (pt)
EC (1)	ECSP099435A (pt)
MX (1)	MX2009006751A (pt)
NO (1)	NO20092376L (pt)
PE (1)	PE20081561A1 (pt)
RU (1)	RU2009128062A (pt)
TW (1)	TW200838497A (pt)
UY (1)	UY30829A1 (pt)
WO (1)	WO2008079382A1 (pt)

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TWI522361B (zh)	2010-07-09	2016-02-21	艾伯維公司	作為s1p調節劑的稠合雜環衍生物
WO2012040532A1 (en)	2010-09-24	2012-03-29	Bristol-Myers Squibb Company	Substituted oxadiazole compounds and their use as s1p1 agonists
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JP6617702B2 (ja)	2013-07-15	2019-12-11	ザリージェンツオブザユニバーシティオブカリフォルニア	Ｆｔｙ７２０のアザサイクリック拘束アナログ
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2007
- 2007-12-21 CA CA002672727A patent/CA2672727A1/en not_active Abandoned
- 2007-12-21 TW TW096149594A patent/TW200838497A/zh unknown
- 2007-12-21 EP EP07863237A patent/EP2120575A4/en not_active Withdrawn
- 2007-12-21 JP JP2009542960A patent/JP2010513532A/ja not_active Withdrawn
- 2007-12-21 WO PCT/US2007/026263 patent/WO2008079382A1/en not_active Ceased
- 2007-12-21 AR ARP070105818A patent/AR064650A1/es not_active Application Discontinuation
- 2007-12-21 KR KR1020097015385A patent/KR20090095659A/ko not_active Withdrawn
- 2007-12-21 BR BRPI0720478-7A patent/BRPI0720478A2/pt not_active Application Discontinuation
- 2007-12-21 MX MX2009006751A patent/MX2009006751A/es not_active Application Discontinuation
- 2007-12-21 RU RU2009128062/04A patent/RU2009128062A/ru not_active Application Discontinuation
- 2007-12-21 UY UY30829A patent/UY30829A1/es not_active Application Discontinuation
- 2007-12-21 AU AU2007338700A patent/AU2007338700A1/en not_active Abandoned
- 2007-12-21 CL CL200703784A patent/CL2007003784A1/es unknown
2008
- 2008-01-02 PE PE2008000051A patent/PE20081561A1/es not_active Application Discontinuation
2009
- 2009-06-02 CO CO09056803A patent/CO6180436A2/es not_active Application Discontinuation
- 2009-06-15 EC EC2009009435A patent/ECSP099435A/es unknown
- 2009-06-19 DO DO2009000149A patent/DOP2009000149A/es unknown
- 2009-06-19 CR CR10872A patent/CR10872A/es not_active Application Discontinuation
- 2009-06-22 NO NO20092376A patent/NO20092376L/no not_active Application Discontinuation

Also Published As

Publication number	Publication date
CO6180436A2 (es)	2010-07-19
CA2672727A1 (en)	2008-07-03
MX2009006751A (es)	2009-06-30
TW200838497A (en)	2008-10-01
RU2009128062A (ru)	2011-01-27
JP2010513532A (ja)	2010-04-30
DOP2009000149A (es)	2010-05-15
ECSP099435A (es)	2009-07-31
EP2120575A1 (en)	2009-11-25
PE20081561A1 (es)	2008-10-30
WO2008079382A1 (en)	2008-07-03
NO20092376L (no)	2009-06-22
BRPI0720478A2 (pt)	2014-01-14
AR064650A1 (es)	2009-04-15
KR20090095659A (ko)	2009-09-09
EP2120575A4 (en)	2011-04-27
UY30829A1 (es)	2008-07-31
CL2007003784A1 (es)	2008-06-27
AU2007338700A1 (en)	2008-07-03

Legal Events

Date	Code	Title	Description
2011-02-07	FA	Abandonment or withdrawal (granting procedure)

Publication	Publication Date	Title
DOP2009000149A (es)	2010-05-15	Compuestos agonistas y antagonistas del receptor de esfingosina-1-fosfato
HN2010001563A (es)	2013-07-22	Compuestos
GT201000153A (es)	2012-04-27	Agonistas novedosos de los receptores de glucocorticoides
CO7400870A2 (es)	2015-09-30	Compuestos derivadios de quinuclidina con actividad antagonista de los receptores muscarínicos y actividad agonista del receptor beta2 adrenérgico
ECSP088989A (es)	2009-01-30	(aza)ciclohexanos carboxilados nuevos como ligandos de receptores de dopamina d3
CR20110455A (es)	2012-01-10	Derivados de indol como antagonistas del receptor crth2
CR20110250A (es)	2011-08-26	Antagonistas de los receptores de la melacortina
NI201300043A (es)	2013-07-01	Antagonistas del receptor del cgrp de piperidinona carboxamida azaindano
ECSP11011019A (es)	2011-05-31	Antagonistas del receptor de orexina de isonicotinamida
UY35177A (es)	2014-06-30	Novedosos derivados de bencimidazol como antagonistas de ep4
UY32926A (es)	2010-11-30	Compuestos como antagonistas de los receptores de ácido lisofosfatídico
CO2017008031A2 (es)	2017-11-10	Compuestos con actividad antagonista de los receptores muscarínicos y actividad agonista del receptor beta2 adrenérgico
CL2008002450A1 (es)	2009-07-31	Compuestos derivados de fenil-pirrolidin-eter, con actividad antagonista de los receptores nk3; procedimientos para su preparacion; composicion farmaceutica; y el uso de los compuestos en el tratamiento de depresion, dolor, psicosis, entre otras.
UY32734A (es)	2010-11-30	Compuestos agonistas del receptor esfingosina 1-fosfato
UY32675A (es)	2010-12-31	Nuevos agonistas del receptor de glucocorticoides
ECSP14002542A (es)	2015-12-31	Nuevos 2hindazoles como antagonistas del receptor ep2
ECSP099573A (es)	2009-12-28	Derivados heterocíclicos como receptores muscarínicos m3
CL2008002310A1 (es)	2009-05-29	Compuestos derivados de benzoil-piperidinas, moduladores del receptor de dopamina d3 y de serotonina 5-ht2a; y uso en el tratamiento y/o prevencion de enfermedades tales como trastornos cognitivos, adiccion a farmacos, depresion y ansiedad.
CR9923A (es)	2008-06-27	Compuestos triciclicos utiles como agonistas de receptores de oxitocina
CO6300937A2 (es)	2011-07-21	Derivados de 3-carboxipropil-aminotetralina y compuestos relacionados como antagonistas de receptores opioides mu
MX2017015047A (es)	2018-04-11	Compuestos que tienen actividad antagonista del receptor muscarinico y actividad agonista del receptor beta2 adrenergico.
UY31931A (es)	2010-01-29	Compuestos de diarilo y uso de los mismos
MX2011008458A (es)	2011-09-01	Metodos para preparar agonistas y antagonistas del receptor s1p.
UY32718A (es)	2010-11-30	Compuestos derivados de 1, 3, 4-tiadiazol, útiles como agonistas del receptor de esfingosina 1-fosfato
CU23534B7 (es)	2010-06-17	Nuevos derivados de 4-bencilidenpiperidina